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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5980 products of "GPCR/G-Protein"

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  • APJ receptor agonist 4

    CAS:
    <p>Potent, orally active APJ receptor agonist 4; EC50: 0.06 nM, Ki: 0.07 nM; good pharmacokinetics in rodent HF model; safe in studies; boosts cardiac function.</p>
    Formula:C28H28ClFN6O3
    Color and Shape:Solid
    Molecular weight:551.02

    Ref: TM-T39587

    5mg
    1,206.00€
  • I-BOP

    CAS:
    I-BOP is an agonist (KD=0.61 nM) at the thromboxane A2 receptor (TP).
    Formula:C23H29IO5
    Color and Shape:Solid
    Molecular weight:512.384

    Ref: TM-T35585

    1mg
    2,062.00€
    100µg
    283.00€
    500µg
    1,264.00€
  • NPS ALX Compound 4a hydrochloride(1:1)


    NPS ALX Compound 4a hydrochloride(1:1) is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with an IC50 of 7.2 nM and a Ki of 0.2 nM.
    Formula:C25H26ClN3O2S
    Purity:99.84%
    Color and Shape:Soild
    Molecular weight:468.01

    Ref: TM-T12262L1

    1mg
    40.00€
    5mg
    88.00€
    10mg
    119.00€
    25mg
    198.00€
    50mg
    288.00€
    100mg
    393.00€
    200mg
    520.00€
    1mL*10mM (DMSO)
    97.00€
  • Anticancer agent 258

    CAS:
    Anticanceragent 258 is an imidazo[1,2-B][1,2,4]triazole derivative that modulates nuclear receptor activity. It exhibits an EC50 of 63 nM for Nurr in N2A cells and an IC50 of 0.1 pM for Nur77 in HEK293 cells. Anticanceragent 258 is applicable in studies related to cancer, metabolic disorders, and neurological diseases.
    Formula:C17H12F2N4
    Color and Shape:Solid
    Molecular weight:310.3

    Ref: TM-T203128

    10mg
    To inquire
    50mg
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  • AA 497 HCl

    CAS:
    AA 497, a beta-2 agonist, suppresses Ca spikes.
    Formula:C14H22ClNO3
    Color and Shape:Solid
    Molecular weight:287.78

    Ref: TM-T26359L

    25mg
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    50mg
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    100mg
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  • Peptide YY (PYY), human

    CAS:
    PYY: a 36-amino-acid hormone, amidated, part of neuroendocrine control, acts via Neuropeptide Y receptors.
    Formula:C194H295N55O57
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4309.75

    Ref: TM-TP1762

    1mg
    200.00€
    5mg
    752.00€
  • Lanerkitug


    Lanerkitug is a humanized IgG1λ2 antibody that targets CCR8, with HumanIgG1lambda2, Isotype Control serving as its corresponding isotype control.
    Color and Shape:Odour Liquid

    Ref: TM-T9901A-352

    1mg
    To inquire
    5mg
    To inquire
  • Tirzepatide hydrochloride


    Tirzepatide HCl is a dual GIP and GLP-1 receptor agonist.
    Formula:C225H349N48O68Cl
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4849.91

    Ref: TM-TP1110

    1mg
    253.00€
    5mg
    663.00€
  • AC-178335

    CAS:
    AC-178335: SRIF antagonist, Ki=172 nM, inhibits SRIF's adenylate cyclase effects (IC50=5.1 µM), triggers GH release in rats.
    Formula:C49H63N13O7
    Color and Shape:Solid
    Molecular weight:946.11

    Ref: TM-T26536

    25mg
    1,444.00€
  • Osanetant

    CAS:
    Osanetant produces anxiolytic- and antidepressant-like effects. Osanetant is a selective NK3 receptor antagonist. It is researched for schizophrenia.
    Formula:C35H41Cl2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:606.62

    Ref: TM-T16408

    25mg
    2,300.00€
    50mg
    3,022.00€
    100mg
    4,085.00€
  • ADTN

    CAS:
    ADTN is an agonist of the dopamine receptor.
    Formula:C10H13NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:179.22

    Ref: TM-T23643

    5mg
    To inquire
  • Fenoldopam

    CAS:
    Fenoldopam is a selective D1-like dopamine receptor partial agonist (EC50 = 57 nM).
    Formula:C16H16ClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:305.76

    Ref: TM-T22779

    25mg
    To inquire
    50mg
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    100mg
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  • Luteinizing Hormone Releasing Hormone (LH-RH), salmon

    CAS:
    LH-RH: a hypothalamus-made pituitary hormone, key in reproductive control.
    Formula:C60H73N15O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1212.31

    Ref: TM-TP1112

    1mg
    84.00€
    5mg
    172.00€
    10mg
    299.00€
  • RXFP3/4 agonist 1

    CAS:
    RXFP3/4 agonist 1 is a relaxin family peptide 3/4 receptor (RXFP3/4) agonist(EC50s of 82/2 nM, respectivley).
    Formula:C20H22ClN5O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:383.88

    Ref: TM-T12785

    25mg
    2,300.00€
    50mg
    3,022.00€
    100mg
    4,085.00€
  • Sar-[D-Phe8]-des-Arg9-Bradykinin

    CAS:
    Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.
    Formula:C47H66N12O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:975.11

    Ref: TM-TP1917

    1mg
    217.00€
  • Donetidine

    CAS:
    Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.
    Formula:C20H25N5O3S
    Purity:99.32%
    Color and Shape:Solid
    Molecular weight:415.51

    Ref: TM-T68056

    1mg
    60.00€
    5mg
    131.00€
    10mg
    192.00€
    25mg
    314.00€
    50mg
    457.00€
    100mg
    653.00€
    200mg
    884.00€
  • Bombinakinin M

    CAS:
    Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.
    Formula:C100H159N31O24
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2179.55

    Ref: TM-TP2075

    1mg
    220.00€
  • Orexin A (human, rat, mouse)

    CAS:
    Orexin A, a 33 AA neuropeptide in humans, rats, mice, influences various processes, studied in pancreatic function and as an OX1R antagonist.
    Formula:C152H243N47O44S4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3561.1

    Ref: TM-TP1301

    500µg
    2,300.00€
  • Cetirizine D8 dihydrochloride

    CAS:
    Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.
    Formula:C21H26Cl2N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.4

    Ref: TM-T19234

    1mg
    998.00€
    500µg
    527.00€
  • Sarafotoxin S6b

    CAS:
    non-selective endothelin receptor agonist
    Formula:C110H163N27O34S5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2567.96

    Ref: TM-TP2290

    1mg
    To inquire
    100mg
    To inquire
    500mg
    To inquire