
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(993 products)
- Adenosine Receptor(246 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(59 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(212 products)
- Dopamine Receptor(433 products)
- Endothelin Receptor(79 products)
- GNRH Receptor(77 products)
- GPCR19(32 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(182 products)
- Hedgehog/Smoothened(47 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(310 products)
- PAFR(12 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5745 products of "GPCR/G-Protein"
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Urocortin, rat
CAS:<p>Endogenous CRF agonist. Ki values are 13, 1.5 and 0.97 nM for hCRF1, rCRF2α and mCRF2β respectively.</p>Formula:C206H338N62O64Purity:98%Color and Shape:SolidMolecular weight:4707.26Sphingosine-1-phosphate (d16:1)
CAS:<p>C16 S1P binds S1P1/EDG-1 (115%), S1P3/EDG-3 (83%), S1P2/EDG-5 (103%) receptors; elevated in glaucoma.</p>Formula:C16H34NO5PColor and Shape:SolidMolecular weight:351.424HHS-0701
CAS:HHS-0701: SuTEx ligand, strong PTGR2 inhibitor, blocks 15-Keto-PGE2 metabolism.Formula:C20H20N4O3SPurity:97.24%Color and Shape:SoildMolecular weight:396.46HAEGTFTSD acetate(926018-45-3 free base)
HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted fromFormula:C42H61N11O19Purity:98%Color and Shape:SolidMolecular weight:1024.01Kisspeptin-10, human
CAS:<p>Kisspeptin-10, human is an effective vasoconstrictor and inhibitor of angiogenesis.</p>Formula:C63H83N17O14Purity:98%Color and Shape:SolidMolecular weight:1302.46217-trifluoromethylphenyl trinor Prostaglandin F2α
CAS:A number of 17-phenyl trinor prostaglandin F2α (17-phenyl trinor PGF2α) derivatives have been approved for the treatment of glaucoma.Formula:C24H31F3O5Color and Shape:SolidMolecular weight:456.502(S)-Azelastine hydrochloride
CAS:(S)-Azelastine HCl, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Formula:C22H25Cl2N3OPurity:98%Color and Shape:SolidMolecular weight:418.36Pasireotide ditrifluoroacetate
Pasireotide is a stable cyclohexapeptide somatostatin mimic.Formula:C62H68F6N10O13Purity:98%Color and Shape:SolidMolecular weight:1275.25MK-0493 HCl
CAS:MK-0493 is a novel, potent, and selective agonist for melanocortin receptor 4 (MC4R).Formula:C30H39Cl2F2N3O2Color and Shape:SolidMolecular weight:582.55Sarafotoxin S6b
CAS:<p>non-selective endothelin receptor agonist</p>Formula:C110H163N27O34S5Purity:98%Color and Shape:SolidMolecular weight:2567.96Denrakibart
<p>Denrakibart is a humanized IgG2κ antibody targeting CCL17, with HumanIgG2kappa, Isotype Control serving as the corresponding isotype control.</p>Color and Shape:Odour LiquidR 50595
CAS:R 50595 is a selective non-competitive cisapride antagonist.Formula:C30H35Cl2F2N3O3Purity:98%Color and Shape:SolidMolecular weight:594.52AC-178335
CAS:AC-178335: SRIF antagonist, Ki=172 nM, inhibits SRIF's adenylate cyclase effects (IC50=5.1 µM), triggers GH release in rats.Formula:C49H63N13O7Color and Shape:SolidMolecular weight:946.11A 76154
CAS:A 76154 is an antagonist of leutenizing hormone releasing hormone (LHRH).Formula:C70H93FN12O12Color and Shape:SolidMolecular weight:1313.584L-779976
CAS:L-779,976 is an agonist of somatostatin receptor.Formula:C33H43N7O3Color and Shape:SolidMolecular weight:585.74Azirkitug
Azirkitug is a humanized IgG1κ antibody targeting CCR8, with HumanIgG1kappa, Isotype Control serving as its corresponding isotype control.Color and Shape:Odour LiquidOno 3708
CAS:Ono-3708 is a potent antagonist of the thromboxane A2/prostaglandin endoperoxide receptor in vitro and in vivo.Formula:C23H37NO4Purity:98%Color and Shape:SolidMolecular weight:391.54LHRH, Ala(6)-
CAS:LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.Formula:C56H77N17O13Color and Shape:SolidMolecular weight:1196.32TLX agonist 2
<p>TLX agonist 2 (compound 31) is a TLX agonist with an EC50 of 0.1 μM and a Kd of 0.16 μM. This compound enhances transcriptional activity by binding to TLX, thereby boosting the expression of TLX target genes. TLX agonist 2 is utilized in research on neurodegenerative diseases.</p>Color and Shape:Odour SolidFR190997
CAS:FR190997 is an agonist of bradykinin B2 receptor.Formula:C37H33Cl2N5O5Color and Shape:SolidMolecular weight:698.59

