GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(942 products)
- Adenosine Receptor(242 products)
- Adrenergic Receptor(2,949 products)
- Bombesin Receptor(30 products)
- Bradykinin Receptor(59 products)
- CXCR(149 products)
- CaSR(32 products)
- Cannabinoid Receptor(195 products)
- Dopamine Receptor(410 products)
- Endothelin Receptor(75 products)
- GNRH Receptor(73 products)
- GPCR19(31 products)
- GRK(32 products)
- GTPase(21 products)
- Glucagon Receptor(166 products)
- Hedgehog/Smoothened(45 products)
- Histamine Receptor(359 products)
- LPA Receptor(21 products)
- Melatonin Receptor(24 products)
- OX Receptor(40 products)
- Opioid Receptor(298 products)
- PAFR(11 products)
- PKA(49 products)
- S1P Receptor(17 products)
- SGLT(30 products)
- Sigma receptor(46 products)
Show 18 more subcategories
Found 5378 products of "GPCR/G-Protein"
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LAS190792
CAS:<p>LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.</p>Formula:C39H43ClN4O9S2Color and Shape:SolidMolecular weight:811.36Latanoprost lactone diol
CAS:Latanoprost lactone diol, a key intermediate for synthesizing Latanoprost (a prostaglandin F2α analogue), lowers IOP by activating FP receptors.Formula:C18H24O4Purity:98%Color and Shape:White Or Almost White Crystalline PowderMolecular weight:304.38BMS-196085
CAS:<p>BMS-196085 is an effective and selective human β( 3) All agonists of adrenergic receptors, in β( 1) Partial agonist activity was 45%.</p>Formula:C24H26F2N2O5SColor and Shape:SolidMolecular weight:492.54ELA-11(human) TFA
<p>ELA-11(human) TFA: apelin receptor agonist, K i =14 nM, inhibits cAMP, stimulates β-arrestin, from ELA-32 fragment.</p>Formula:C60H91F3N16O15S2Color and Shape:SolidMolecular weight:1397.58BAY-747
CAS:<p>BAY-747: oral, brain-penetrant sGC stimulator; improves rat memory, cognition, lowers blood pressure, aids Duchenne muscular dystrophy.</p>Formula:C22H26F2N4O2Color and Shape:SolidMolecular weight:416.464-Chloromethamphetamine hydrochloride
CAS:<p>4-Chloromethamphetamine hydrochloride is a novel psychoactive substance belonging to the amphetamine class.</p>Formula:C10H15Cl2NColor and Shape:SolidMolecular weight:220.14BMS-604992 dihydrochloride
CAS:<p>BMS-604992 dihydrochloride is a selective GHSR agonist with high affinity (Ki=2.3 nM) and potent activity (EC50=0.4 nM), stimulating rodent appetite.</p>Formula:C24H33Cl2N7O5Color and Shape:SolidMolecular weight:570.47L-796,778 acetate
<p>L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for sst1, sst2, sst4 and sst5, IC50 is >1000nM.</p>Formula:C31H44N6O9Purity:98%Color and Shape:SoildMolecular weight:644.72PACAP (1-27), human, ovine, rat
CAS:PACAP (1-27) (the N-terminal fragment of PACAP-38) is a novel neuropeptides originally isolated from bovine hypothalamus, also found in humans and rats.Formula:C142H224N40O39SPurity:98%Color and Shape:SolidMolecular weight:3147.66Upidosin
CAS:<p>Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.</p>Formula:C31H33N3O4Purity:99.66%Color and Shape:SolidMolecular weight:511.61TT-OAD2 free base
CAS:<p>TT-OAD2 free base, a non-peptide GLP-1 receptor agonist, can treat diabetes; has an EC50 of 5 nM.</p>Formula:C50H47Cl2N3O6Purity:98%Color and Shape:SolidMolecular weight:856.83NPC 567
CAS:<p>NPC 567 is an antagonist of the bradykinin receptor.</p>Formula:C60H87N19O13Purity:98%Color and Shape:SolidMolecular weight:1282.48Meluadrine tartrate
CAS:<p>Meluadrine tartrate is an endogenous metabolite.</p>Formula:C16H24ClNO8Purity:98%Color and Shape:SolidMolecular weight:393.82A3AR modulator 1
<p>MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.</p>Formula:C23H25IN4Color and Shape:SolidMolecular weight:484.38Mosliciguat
CAS:<p>Mosliciguat is a guanylate cyclase activator.</p>Formula:C41H36ClF3N2O5Color and Shape:SolidMolecular weight:729.19SRA880 malonate
CAS:<p>SRA880: non-peptide sst(1) antagonist, low affinity for other sst receptors, binds dopamine D4, boosts SRIF, antidepressant-like effects.</p>Formula:C29H36N4O8Purity:98%Color and Shape:SolidMolecular weight:568.62SR-140603
CAS:<p>SR-140603, the less potent enantiomer of SR 140333, is used as the negative control.</p>Formula:C37H45Cl3N2O2Purity:98%Color and Shape:SolidMolecular weight:656.12palm11-PrRP31
<p>Palm11-PrRP31 is a lipid-modified analog of the endogenous appetite-suppressing neuropeptide (PrRP). It functions as a potent dual agonist for GPR10 (EC50 = 39 pM) and NPFF-R2. By mimicking the natural activity of PrRP, palm11-PrRP31 binds to these receptors to reduce food intake. It has potential applications as an anti-obesity agent and is useful in studying neuropeptide and receptor interactions.</p>Formula:C181H289N55O46SMolecular weight:4001.16865SYD5115
<p>SYD5115 is an orally active TSH-R antagonist.</p>Formula:C22H32F2N4O3Molecular weight:438.24425Dehydro Aripiprazole (hydrochloride)
CAS:<p>Dehydro aripiprazole, an active atypical antipsychotic metabolite of aripiprazole, is formed by CYP3A4 and CYP2D6.</p>Formula:C23H26Cl3N3O2Color and Shape:SolidMolecular weight:482.83
