GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(53 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5980 products of "GPCR/G-Protein"
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Apelin-12 acetate
Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.Formula:C66H107N21O16SPurity:98.82%Color and Shape:SolidMolecular weight:1482.75Ref: TM-T39823L
1mg216.00€5mg304.00€10mg472.00€25mg753.00€50mg1,074.00€100mg1,444.00€1mL*10mM (DMSO)757.00€Cannabinol methyl ether
CAS:Cannabinol methyl ether, a phytocannabinoid, serves as an analytical reference standard. This compound can be obtained through isolation from Cannabis plants, derived from cannabinol, or synthesized. The physiological and toxicological properties of cannabinol methyl ether remain unknown. It is designed exclusively for research and forensic applications.Formula:C22H28O2Color and Shape:SolidMolecular weight:324.5O-2172
CAS:O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).Formula:C14H16Cl2O2Color and Shape:SolidMolecular weight:287.18YM 16638
CAS:YM 16638 is an LT antagonist that can be used to study antigen-induced early and late airway responses in allergic sheep.Formula:C18H22N2O5S3Purity:99.18%Color and Shape:SolidMolecular weight:442.57Urocortin, rat
CAS:Endogenous CRF agonist. Ki values are 13, 1.5 and 0.97 nM for hCRF1, rCRF2α and mCRF2β respectively.Formula:C206H338N62O64Purity:98%Color and Shape:SolidMolecular weight:4707.26PG106
CAS:Selective hMC3 receptor antagonist (IC50 = 210 nM). Exhibits no activity at hMC4 receptors and hMC5 receptors.Formula:C51H69N13O9Purity:98%Color and Shape:SolidMolecular weight:1008.19Hydroxybupropion
CAS:Hydroxybupropion is the major active metabolite of Bupropion and an antagonist of nACh receptor. Hydroxybupropion inhibits norepinephrine uptake (IC50 = 1.7 μM).Formula:C13H18ClNO2Purity:99.73%Color and Shape:Off-White SolidMolecular weight:255.74Ref: TM-T11588
1mg89.00€5mg204.00€10mg331.00€25mg545.00€50mg777.00€100mg1,063.00€1mL*10mM (DMSO)232.00€Spantide acetate
<p>Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.</p>Formula:C77H112N20O15Purity:98.9200%Color and Shape:SolidMolecular weight:1557.84Amylin, amide, rat
CAS:Amylin: peptide, 50% similar to CGRP, found with somatostatin in stomach cells, reduces acid secretion in mice.Formula:C167H272N52O53S2Purity:99.92%Color and Shape:SolidMolecular weight:3920.4411-deoxy Prostaglandin E1
CAS:11-deoxy Prostaglandin E1 is a prostaglandin E1 analogue that has bronchodilator activity and can inhibit histamine-induced bronchoconstriction and causeFormula:C20H34O4Color and Shape:SolidMolecular weight:338.48Mesoridazine Besylate
CAS:Mesoridazine Besylate (Serentil), a piperidine antipsychotic and phenothiazine, treats schizophrenia; it's a thioridazine metabolite.Formula:C27H32N2O4S3Purity:98.87%Color and Shape:SolidMolecular weight:544.75Kisspeptin-10, human
CAS:Kisspeptin-10, human is an effective vasoconstrictor and inhibitor of angiogenesis.Formula:C63H83N17O14Purity:98%Color and Shape:SolidMolecular weight:1302.462PEN (human)
CAS:PEN (human) is an Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.Formula:C97H159N27O32Purity:98%Color and Shape:SolidMolecular weight:2215.49LY86057
CAS:LY86057 is a bioactive chemical.Formula:C20H26N2O3Color and Shape:SolidMolecular weight:342.439Azirkitug
Azirkitug is a humanized IgG1κ antibody targeting CCR8, with HumanIgG1kappa, Isotype Control serving as its corresponding isotype control.Color and Shape:Odour LiquidSch 202596
CAS:Sch 202596 is a selective non-peptide antagonist of GAL-1 receptor.Formula:C25H22Cl2O12Color and Shape:SolidMolecular weight:585.34Lenbelintide
CAS:Lenbelintide is a dual amylin/calcitonin receptor agonist, useful in studies related to obesity.Color and Shape:SolidBerobenatide
CAS:Berobenatide is a glucagon-like peptide-1 (GLP-1) receptor agonist.Color and Shape:SolidOno 3708
CAS:Ono-3708 is a potent antagonist of the thromboxane A2/prostaglandin endoperoxide receptor in vitro and in vivo.Formula:C23H37NO4Purity:98%Color and Shape:SolidMolecular weight:391.54LHRH, Ala(6)-
CAS:LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.Formula:C56H77N17O13Color and Shape:SolidMolecular weight:1196.32
