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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5963 products of "GPCR/G-Protein"

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  • ABT-702

    CAS:
    ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.
    Formula:C22H19BrN6O
    Purity:99.57%
    Color and Shape:Soild
    Molecular weight:463.33

    Ref: TM-T4668L

    1mg
    70.00€
    5mg
    150.00€
    10mg
    235.00€
    25mg
    445.00€
    50mg
    660.00€
    100mg
    932.00€
  • Astressin

    CAS:
    Astressin is a truncated CRF analog; binds strongly to receptor's extracellular domain, likely acting as a neutral competitive antagonist.
    Formula:C161H269N49O42
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3563.16

    Ref: TM-TP1448

    500µg
    1,459.00€
  • GR 64349

    CAS:
    Potent NK2 agonist, EC50=3.7 nM in rat colon; >1000x selectivity over NK1, >300x over NK3; effective in vivo.
    Formula:C42H68N10O11S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:921.12

    Ref: TM-TP2023

    1mg
    1,575.00€
  • NTRC-824

    CAS:
    NTRC-824: NTS2 antagonist, 150x more selective than NTS1; IC50: 38 nM, Ki: 202 nM; nonpeptide, neurotensin-like.
    Formula:C25H26F3N3O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:553.55

    Ref: TM-T16358

    50mg
    4,474.00€
  • GLP-1R agonist 14

    CAS:
    GLP-1R agonist 14, also known as Compound 14, is a potent agonist of the GLP-1 receptor, demonstrating an EC50 range of 0-20 nM against human GLP-1 [1].
    Formula:C45H42F2N10O5
    Color and Shape:Solid
    Molecular weight:840.88

    Ref: TM-T74608

    5mg
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    50mg
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  • 11-deoxy Prostaglandin F1α

    CAS:
    11-deoxy PGF1α is a synthetic analog of PGF1α.
    Formula:C20H36O4
    Color and Shape:Solid
    Molecular weight:340.504

    Ref: TM-T36771

    1mg
    185.00€
    5mg
    797.00€
    10mg
    1,359.00€
  • Hemopressin (human, mouse)

    CAS:
    Endogenous peptide, inhibits ep24.15/24.16/ACE with Ki of 27.76/3.43/1.87 μM. Lowers blood pressure, CB1 inverse agonist, reduces pain in vivo.
    Formula:C50H79N13O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1054.26

    Ref: TM-TP1900

    1mg
    156.00€
  • CCR6 antagonist 2


    CCR6 antagonist2 (Compound 20c) acts as a CCR6 antagonist with a Ki of 1.1 nM. It inhibits CCL20-induced calcium influx with an IC50 of 4.9 nM and suppresses the chemotactic migration of CCR6+ T cells with an IC50 of 190 nM.
    Formula:C19H24N4O4
    Color and Shape:Solid
    Molecular weight:372.42

    Ref: TM-T205072

    10mg
    To inquire
    50mg
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  • Ribupatide

    CAS:
    Ribupatide is a dual agonist of gastric inhibitory polypeptide (GIP) and glucagon-like peptide 1 (GLP-1) receptors and can be utilized in antidiabetic research.
    Color and Shape:Solid

    Ref: TM-TP3817

    10mg
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    50mg
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  • RFRP-3(human)

    CAS:
    NPFF1 receptor agonist, IC50 0.7 nM, blocks cAMP by forskolin. A GnIH homolog, it inhibits GnRH neuron activity.
    Formula:C45H72N14O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:969.15

    Ref: TM-TP1936

    1mg
    642.00€
  • PG106

    CAS:
    Selective hMC3 receptor antagonist (IC50 = 210 nM). Exhibits no activity at hMC4 receptors and hMC5 receptors.
    Formula:C51H69N13O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1008.19

    Ref: TM-TP1952

    1mg
    264.00€
  • Beraprost

    CAS:
    Beraprost is a stable prostacyclin analog.
    Formula:C24H30O5
    Color and Shape:Solid
    Molecular weight:398.49

    Ref: TM-T30426

    25mg
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    50mg
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    100mg
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  • LGnRH-III, lamprey

    CAS:
    GnRH III triggers luteinizing and follicle-stimulating hormone release, part of the conserved GnRH family.
    Formula:C59H74N18O14
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1259.33

    Ref: TM-TP1700

    100mg
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    500mg
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  • Spantide acetate


    Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.

    Formula:C77H112N20O15
    Purity:98.9200%
    Color and Shape:Solid
    Molecular weight:1557.84

    Ref: TM-T20413L

    1mg
    129.00€
    5mg
    329.00€
    10mg
    525.00€
    25mg
    848.00€
    50mg
    1,159.00€
    100mg
    1,568.00€
    500mg
    3,117.00€
  • 11-deoxy Prostaglandin E1

    CAS:
    11-deoxy Prostaglandin E1 is a prostaglandin E1 analogue that has bronchodilator activity and can inhibit histamine-induced bronchoconstriction and cause
    Formula:C20H34O4
    Color and Shape:Solid
    Molecular weight:338.48

    Ref: TM-T36770

    1mg
    212.00€
    5mg
    874.00€
    10mg
    1,510.00€
    500µg
    118.00€
  • Antibiotic Sch 60057

    CAS:
    Antibiotic Sch 60057 is a useful organic compound for research related to life sciences. The catalog number is T125403 and the CAS number is 203061-35-2.
    Formula:C45H84O6
    Color and Shape:Solid
    Molecular weight:721.161

    Ref: TM-T125403

    1mg
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    5mg
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  • BRD9 ligand-6

    CAS:
    BRD9 ligand-6 serves as a ligand for the target protein in PROTAC applications. It is utilized in the synthesis of FHD-609.
    Formula:C21H21N3O4
    Color and Shape:Solid
    Molecular weight:379.41

    Ref: TM-T201762

    10mg
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    50mg
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  • Cortistatin-8

    CAS:
    ghrelin receptor antagonist
    Formula:C47H68N12O9S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1009.25

    Ref: TM-TP2236

    1mg
    216.00€
  • Prostaglandin F1α

    CAS:
    Prostaglandin F1α (PGF1α) is a lipid mediator and an endogenous metabolite of prostacyclin, regulate smooth muscle contraction.
    Formula:C20H36O5
    Color and Shape:Solid
    Molecular weight:356.5

    Ref: TM-T37919

    1mg
    269.00€
  • Sch 202596

    CAS:
    Sch 202596 is a selective non-peptide antagonist of GAL-1 receptor.
    Formula:C25H22Cl2O12
    Color and Shape:Solid
    Molecular weight:585.34

    Ref: TM-T28705

    25mg
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    50mg
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    100mg
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