
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,994 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5963 products of "GPCR/G-Protein"
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ABT-702
CAS:ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.Formula:C22H19BrN6OPurity:99.57%Color and Shape:SoildMolecular weight:463.33Astressin
CAS:Astressin is a truncated CRF analog; binds strongly to receptor's extracellular domain, likely acting as a neutral competitive antagonist.Formula:C161H269N49O42Purity:98%Color and Shape:SolidMolecular weight:3563.16GR 64349
CAS:Potent NK2 agonist, EC50=3.7 nM in rat colon; >1000x selectivity over NK1, >300x over NK3; effective in vivo.Formula:C42H68N10O11SPurity:98%Color and Shape:SolidMolecular weight:921.12NTRC-824
CAS:NTRC-824: NTS2 antagonist, 150x more selective than NTS1; IC50: 38 nM, Ki: 202 nM; nonpeptide, neurotensin-like.Formula:C25H26F3N3O6SPurity:98%Color and Shape:SolidMolecular weight:553.55GLP-1R agonist 14
CAS:GLP-1R agonist 14, also known as Compound 14, is a potent agonist of the GLP-1 receptor, demonstrating an EC50 range of 0-20 nM against human GLP-1 [1].Formula:C45H42F2N10O5Color and Shape:SolidMolecular weight:840.8811-deoxy Prostaglandin F1α
CAS:11-deoxy PGF1α is a synthetic analog of PGF1α.Formula:C20H36O4Color and Shape:SolidMolecular weight:340.504Hemopressin (human, mouse)
CAS:Endogenous peptide, inhibits ep24.15/24.16/ACE with Ki of 27.76/3.43/1.87 μM. Lowers blood pressure, CB1 inverse agonist, reduces pain in vivo.Formula:C50H79N13O12Purity:98%Color and Shape:SolidMolecular weight:1054.26CCR6 antagonist 2
CCR6 antagonist2 (Compound 20c) acts as a CCR6 antagonist with a Ki of 1.1 nM. It inhibits CCL20-induced calcium influx with an IC50 of 4.9 nM and suppresses the chemotactic migration of CCR6+ T cells with an IC50 of 190 nM.Formula:C19H24N4O4Color and Shape:SolidMolecular weight:372.42Ribupatide
CAS:Ribupatide is a dual agonist of gastric inhibitory polypeptide (GIP) and glucagon-like peptide 1 (GLP-1) receptors and can be utilized in antidiabetic research.Color and Shape:SolidRFRP-3(human)
CAS:NPFF1 receptor agonist, IC50 0.7 nM, blocks cAMP by forskolin. A GnIH homolog, it inhibits GnRH neuron activity.Formula:C45H72N14O10Purity:98%Color and Shape:SolidMolecular weight:969.15PG106
CAS:Selective hMC3 receptor antagonist (IC50 = 210 nM). Exhibits no activity at hMC4 receptors and hMC5 receptors.Formula:C51H69N13O9Purity:98%Color and Shape:SolidMolecular weight:1008.19Beraprost
CAS:Beraprost is a stable prostacyclin analog.Formula:C24H30O5Color and Shape:SolidMolecular weight:398.49LGnRH-III, lamprey
CAS:GnRH III triggers luteinizing and follicle-stimulating hormone release, part of the conserved GnRH family.Formula:C59H74N18O14Purity:98%Color and Shape:SolidMolecular weight:1259.33Spantide acetate
Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.
Formula:C77H112N20O15Purity:98.9200%Color and Shape:SolidMolecular weight:1557.8411-deoxy Prostaglandin E1
CAS:11-deoxy Prostaglandin E1 is a prostaglandin E1 analogue that has bronchodilator activity and can inhibit histamine-induced bronchoconstriction and causeFormula:C20H34O4Color and Shape:SolidMolecular weight:338.48Antibiotic Sch 60057
CAS:Antibiotic Sch 60057 is a useful organic compound for research related to life sciences. The catalog number is T125403 and the CAS number is 203061-35-2.Formula:C45H84O6Color and Shape:SolidMolecular weight:721.161BRD9 ligand-6
CAS:BRD9 ligand-6 serves as a ligand for the target protein in PROTAC applications. It is utilized in the synthesis of FHD-609.Formula:C21H21N3O4Color and Shape:SolidMolecular weight:379.41Cortistatin-8
CAS:ghrelin receptor antagonistFormula:C47H68N12O9S2Purity:98%Color and Shape:SolidMolecular weight:1009.25Prostaglandin F1α
CAS:Prostaglandin F1α (PGF1α) is a lipid mediator and an endogenous metabolite of prostacyclin, regulate smooth muscle contraction.Formula:C20H36O5Color and Shape:SolidMolecular weight:356.5Sch 202596
CAS:Sch 202596 is a selective non-peptide antagonist of GAL-1 receptor.Formula:C25H22Cl2O12Color and Shape:SolidMolecular weight:585.34

