GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,024 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5990 products of "GPCR/G-Protein"
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Kisspeptin-10, rat
CAS:Kisspeptin-10, rat is an Endogenous ligand for the rodent kisspeptin receptor (KISS1, GPR54).Formula:C63H83N17O15Purity:98%Color and Shape:SolidMolecular weight:1318.44Colulintide
CAS:Colulintide is an analog of amylin, utilized in obesity research.Color and Shape:SolidACTH (1-14)
CAS:ACTH (1-14) is a pituitary hormone fragment that controls cortisol and androgen levels.Formula:C77H109N21O20SPurity:98%Color and Shape:SolidMolecular weight:1680.88TCMCB07
CAS:TCMCB07, a cyclic nonapeptide, serves as an orally active, brain-penetrant antagonist of the melanocortin receptor 4 (MC4R), with significant implications inFormula:C63H87N15O11Purity:98%Color and Shape:SolidMolecular weight:1230.46RFRP-1(human)
CAS:Endogenous NPFF agonist with EC50 of 0.0011 nM (NPFF2) and 29 nM (NPFF1); reduces cardiac function and raises prolactin in rats. GnIH homolog.Formula:C67H101N19O14SPurity:98%Color and Shape:SolidMolecular weight:1428.72CAY10734
CAS:CAY10734 has a wide range of applications in life science related research.Formula:C23H25N3O3Color and Shape:SolidMolecular weight:391.4711-(4-Fluorobenzyl)-1H-indazole-3-carboxylic acid
CAS:1-(4-Fluorobenzyl)-1H-indazole-3-carboxylic acid (Compound 31) is a metabolite of AB-FUBINACA. It acts as an MRGPRX4 antagonist with an IC50 greater than 2.5 μM.Formula:C15H11FN2O2Color and Shape:SolidMolecular weight:270.26Sigma-1 receptor antagonist 5
Sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic action on sigma receptorsFormula:C26H27N3OPurity:98%Color and Shape:SolidMolecular weight:397.51ent-Prostaglandin E2
CAS:Enzymatic PGE2 is optically pure; radical peroxidation makes it racemic. In oxidative stress, rac-PGE2 forms via 15-E2t-isoprostane.Formula:C20H32O5Color and Shape:SolidMolecular weight:352.471Gemeprost
CAS:Gemeprost treats obstetric bleeding and induces abortion up to 24 weeks when used with mifepristone.Formula:C23H38O5Purity:98%Color and Shape:SolidMolecular weight:394.545-methoxy-α-Ethyltryptamine
CAS:5-Methoxy-alpha-ethyltryptamine is a psychoactive substance that can cause various effects. It belongs to the tryptamine chemical class and can be used for various psychoactive and stimulant effects.
Formula:C13H18N2OPurity:98.25%Color and Shape:SolidMolecular weight:218.29MCUF-651
CAS:MCUF-651 is a guanylyl cyclase A receptor positive allosteric modulators, EC50=0.45 μM.Formula:C17H22F2N4OSPurity:99.83%Color and Shape:SoildMolecular weight:368.44Ref: TM-T67734
1mg56.00€5mg118.00€1mL*10mM (DMSO)126.00€10mg178.00€25mg344.00€50mg557.00€100mg790.00€Neurokinin B (TFA)
CAS:Neurokinin B TFA, a tachykinin, targets NK1R, NK2R, nk3r GPCRs, modulating effects.Formula:C59H81F6N13O18S2Purity:98%Color and Shape:SolidMolecular weight:1438.475-OMe-UDP trisodium salt
CAS:Potent P2Y6 agonistFormula:C10H16N2O13P2Purity:98%Color and Shape:SolidMolecular weight:434.19GPR55 agonist 4
GPR55 agonist 4 (Compound 28), with an EC50 of 131 nM for hGPR55 and 1.41 nM for rGPR55, effectively induces β-arrestin recruitment to human GPR55 [1].Formula:C19H16FN5O2Color and Shape:SolidMolecular weight:365.36Calcitonin (8-32), salmon
CAS:Calcitonin (8-32), salmon: selective amylin receptor antagonist, regulates calcium/phosphorus, thyroid origin, 32-aa peptide.Formula:C119H198N36O37Purity:98%Color and Shape:SolidMolecular weight:2725.06tcY-NH2
CAS:Selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.Formula:C40H49N7O7Purity:98%Color and Shape:SolidMolecular weight:739.87Lysophosphatidic acid
CAS:Lysophosphatidic acid is a bioactive chemical.Formula:C21H41O7PColor and Shape:SolidMolecular weight:436.52CB2R agonist 2
CB2R agonist 2 (cis-17-para) is a CB2R agonist [1].Purity:98%Color and Shape:Odour SolidCB2R agonist 3
CB2R agonist 3, a potent activator of cannabinoid receptor 2 (CB2R), exhibits an EC50 value of 0.37μM, indicative of its significant role in the immune system [Purity:98%Color and Shape:Odour Solid
