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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5983 products of "GPCR/G-Protein"

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  • Bz-Dab(nbd)-awfpp-nle-NH2

    CAS:
    Bz-Dab(nbd)-ala-trp-phe-pro-pro-nle-NH2 is a fluorescent NK2 antagonist.
    Formula:C56H65N13O11
    Color and Shape:Solid
    Molecular weight:1096.2

    Ref: TM-T25197

    25mg
    1,369.00€
  • Ramelteon metabolite M-II

    CAS:
    Ramelteon M-II binds MT1/MT2 with IC50s: 208/1470 pM; it's the main metabolite and a melatonin receptor agonist.
    Formula:C16H21NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:275.34

    Ref: TM-T12689

    1mg
    210.00€
    5mg
    620.00€
    10mg
    1,125.00€
  • MR33317


    MR33317 is an inhibitor of acetylcholinesterase with an IC50 value of 41 nM. Additionally, it acts as an agonist for brain 5-HT4 receptors.
    Formula:C22H28ClN3O2
    Molecular weight:401.187

    Ref: TM-T210213

    10mg
    To inquire
    50mg
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  • Prolactin-Releasing Peptide (1-31), bovine


    Prolactin-Releasing Peptide (1-31), bovine, is a fragment of prolactin-releasing peptide (PrRP).
    Formula:C44H80N14O15
    Molecular weight:1044.59276

    Ref: TM-TP3385

    10mg
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    50mg
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  • CI-988 hemihydrate


    CI-988 hemihydrate (PD134308) is a potent and selective orally active CCK2R (cholecystokinin 2 receptor) antagonist, with an IC50 of 1.7 nM for mouse cortical CCK2. It is over 1600 times more selective for CCK2 than for CCK1 receptors. CI-988 hemihydrate exhibits anxiolytic and antitumor properties.
    Formula:C35H42N4O6H2O
    Molecular weight:632.321

    Ref: TM-T208995

    10mg
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    50mg
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  • YM 16638

    CAS:
    YM 16638 is an LT antagonist that can be used to study antigen-induced early and late airway responses in allergic sheep.
    Formula:C18H22N2O5S3
    Purity:99.18%
    Color and Shape:Solid
    Molecular weight:442.57

    Ref: TM-T35258

    1mg
    358.00€
    5mg
    873.00€
    10mg
    1,161.00€
    25mg
    1,755.00€
    50mg
    2,358.00€
    100mg
    3,177.00€
  • JMV 449

    CAS:
    Potent neurotensin agonist; IC50=0.15 nM, EC50=1.9 nM. Causes hypothermia, neuroprotection, analgesia in mice.
    Formula:C38H66N8O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:746.96

    Ref: TM-TP2012

    1mg
    477.00€
  • SRA880 malonate

    CAS:
    SRA880: non-peptide sst(1) antagonist, low affinity for other sst receptors, binds dopamine D4, boosts SRIF, antidepressant-like effects.
    Formula:C29H36N4O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:568.62

    Ref: TM-T26225

    25mg
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    50mg
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    100mg
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  • SR-140603

    CAS:
    SR-140603, the less potent enantiomer of SR 140333, is used as the negative control.
    Formula:C37H45Cl3N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:656.12

    Ref: TM-T26222

    25mg
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    50mg
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    100mg
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  • Upidosin

    CAS:

    Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.

    Formula:C31H33N3O4
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:511.61

    Ref: TM-T9762

    10mg
    47.00€
    25mg
    70.00€
    50mg
    90.00€
    100mg
    136.00€
    200mg
    197.00€
  • (R,R)-Palonosetron Hydrochloride

    CAS:
    (R,R)-Palonosetron Hydrochloride is the active enantiomer of Palonosetron
    Formula:C19H25ClN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.87

    Ref: TM-T13437

    25mg
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    50mg
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    100mg
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  • GLP-1 receptor agonist 4

    CAS:
    GLP-1 receptor agonist 4 targets GLP-1R, EC50 64.5 nM, potential diabetes treatment research.
    Formula:C51H44Cl2N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:879.82

    Ref: TM-T11405

    100mg
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    500mg
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  • GLP-1R agonist 20


    GLP-1R agonist 20 (Compound I-132) is an agonist of the glucagon-like peptide-1 receptor (GLP-1 receptor), with an EC50 value of 0.0162 nM.
    Formula:C31H30Cl2F2N4O5
    Molecular weight:646.15613

    Ref: TM-T209770

    10mg
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    50mg
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  • SPN009


    SPN009 (Sequence 3) is a GLP-1 receptor (GLP-1 Receptor) agonist, with an EC50 of 2.84 nM, and improves type 2 diabetes in DB/DB mouse models.
    Formula:C191H299N45O59
    Molecular weight:4167.17798

    Ref: TM-TP3525

    10mg
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    50mg
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  • PAR-4 Agonist Peptide, amide

    CAS:
    PAR-4 Agonist Peptide, amide (AY-NH2) is an agonist of proteinase-activated receptor-4 (PAR-4).
    Formula:C34H48N8O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:680.79

    Ref: TM-T7623

    1mg
    52.00€
    5mg
    137.00€
    10mg
    195.00€
  • ACT-373898

    CAS:
    ACT-373898 is a metabolite of the endothelin (ET) receptor type A (ETA) and ETBdual antagonist macitentan .1
    Formula:C15H17BrN4O5S
    Color and Shape:Solid
    Molecular weight:445.29

    Ref: TM-T35623

    1mg
    96.00€
    5mg
    261.00€
    10mg
    439.00€
    25mg
    893.00€
  • CYN 154806

    CAS:
    CYN 154806: potent sst2 antagonist; pIC50: 8.58 (sst2), 5.41 (sst1), 6.07 (sst3), 5.76 (sst4), 6.48 (sst5).
    Formula:C56H68N12O14S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1197.34

    Ref: TM-TP1877

    1mg
    1,140.00€
  • 7-Hydroxy-PIPAT maleate

    CAS:
    7-Hydroxy-PIPAT maleate is a D3R agonist.
    Formula:C16H22INO
    Color and Shape:Solid
    Molecular weight:371.262

    Ref: TM-T38188

    10mg
    130.00€
    50mg
    513.00€
  • Atrial natriuretic factor (1-28) (rat) TFA


    ANP (1-28), rat (TFA) inhibits Ang II-induced endothelin-1 secretion; main circulating ANP form in rats.
    Formula:C130H206N45F3O41S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3176.43

    Ref: TM-TP1218

    1mg
    217.00€
    5mg
    770.00€
  • LY 344864 racemate

    CAS:
    LY 344864 racemate is a 5-HT1F receptor agonist.
    Formula:C21H22FN3O
    Purity:99.75%
    Color and Shape:Soild
    Molecular weight:351.42

    Ref: TM-T2344L

    5mg
    43.00€
    10mg
    66.00€
    25mg
    100.00€
    50mg
    166.00€
    100mg
    To inquire
    1mL*10mM (DMSO)
    34.00€