GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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MrgprX2 antagonist-4
CAS:MrgprX2 antagonist-4, from patent US20210128561A1, inhibits MrgprX2 receptor; useful for skin inflammation studies.Formula:C16H19N3OColor and Shape:SolidMolecular weight:269.3486α-Prostaglandin I1
CAS:6α-Prostaglandin I1 (6α-PGI1) is a stable Prostaglandin I2 (PGI2) analog resistant to hydrolysis in aqueous solutions.Formula:C20H34O5Color and Shape:SolidMolecular weight:354.487Hemopressin(human, mouse) TFA
CAS:Hemopressin TFA: nonapeptide from hemoglobin, oral CB1 inverse agonist, eases inflammatory pain.Formula:C52H80F3N13O14Purity:98%Color and Shape:SolidMolecular weight:1168.27PEN (human)
CAS:PEN (human) is an Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.Formula:C97H159N27O32Purity:98%Color and Shape:SolidMolecular weight:2215.49Peptide YY (PYY), human
CAS:PYY: a 36-amino-acid hormone, amidated, part of neuroendocrine control, acts via Neuropeptide Y receptors.Formula:C194H295N55O57Purity:98%Color and Shape:SolidMolecular weight:4309.75(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
CAS:Analog of LHRH, stimulates LH and FSH release, controls reproduction.Formula:C59H84N18O14Color and Shape:SolidMolecular weight:1269.41AY 254
CAS:AY 254: Potent PAR2 agonist, ERK1/2 activation (EC50=2 nM), limits caspase 3/8, aids HT29 cell healing, boosts IL-8.
Formula:C30H49N9O6Color and Shape:SolidMolecular weight:631.779YM 16638
CAS:YM 16638 is an LT antagonist that can be used to study antigen-induced early and late airway responses in allergic sheep.Formula:C18H22N2O5S3Purity:99.18%Color and Shape:SolidMolecular weight:442.57Leukotriene B5
CAS:LTB5, an eicosapentaenoic acid metabolite via 5-LO, has varied bioactivities and enhances bullfrog lung strip contraction.Formula:C20H30O4Color and Shape:SolidMolecular weight:334.456H-Ser-Phe-Leu-Leu-Arg-OH
CAS:Thrombin Receptor Activator for Peptide 5 (TRAP-5) is also called Coagulation Factor II Receptor (1-5), used in the research of coronary heart disease (CHD).Formula:C30H50N8O7Purity:98%Color and Shape:SolidMolecular weight:634.77TAK-683 acetate
TAK-683 acetate: potent KISS1R agonist (IC50=170 pM), stable, nonapeptide. Affects GnRH, FSH, LH, testosterone; potential in prostate cancer research.Formula:C66H87N17O15Color and Shape:SolidMolecular weight:1358.5BIIE-0246
CAS:BIIE-0246 is a selective NPY2R antagonist, IC50=15 nM at the rat [125I]PYY3-36 site, reduces NPY-stimulated expression of p-AKT S473 and P-p44/42 MAPK.Formula:C49H57N11O6Purity:98%Color and Shape:SolidMolecular weight:896.05PF-03382792
CAS:PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.Formula:C23H32FN3O4Purity:99.64%Color and Shape:SolidMolecular weight:433.52CAY10734
CAS:CAY10734 has a wide range of applications in life science related research.Formula:C23H25N3O3Color and Shape:SolidMolecular weight:391.471Jmv 179
CAS:Jmv 179 is an antagonist of the cholecystokinin receptor.Formula:C51H67N7O15SColor and Shape:SolidMolecular weight:1050.19Lu AA33810
CAS:Lu AA33810 is a selective neuropeptide Y5 (NPY5) receptor antagonist with an oral activity and BBB permeability, anti-anxiety and antidepressant-like effects.Formula:C19H25N3O2S3Purity:97.92% - 99.61%Color and Shape:SolidMolecular weight:423.62GLP-2(1-33)(human)
CAS:GLP-2(1-33) (human) is an enteroendocrine hormone which stimulates the growth of the intestinal epithelium.Formula:C165H254N44O55SPurity:98%Color and Shape:SolidMolecular weight:3766.19GW-328267
CAS:GW-328267 is an agonist of the adenosine A2 receptor.Formula:C21H26N10O4Color and Shape:SolidMolecular weight:482.5Carazolol-d7
CAS:Carazolol-d7 is the deuterium-labeled isotope of Carazolol, commonly used in pharmacokinetic studies to investigate the metabolic pathways of Carazolol.Formula:C18H22N2O2Color and Shape:SolidMolecular weight:305.42IRAK inhibitor 4 trans
IRAK inhibitor 4 targets and blocks IRAK4 activity; refers to its trans molecular configuration.Formula:C33H35F3N6O3Purity:98%Color and Shape:SolidMolecular weight:620.66
