GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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(±)5-iPF2α-VI
CAS:Isoprostanes are prostaglandin (PG)-like products of free-radical induced lipid peroxidation.Formula:C20H34O5Color and Shape:SolidMolecular weight:354.487AM-0466
CAS:AM-0466 has a wide range of applications in life science related research.Formula:C27H19F3N4O4SColor and Shape:SolidMolecular weight:552.52HTR2A antagonist 1
HTR2A antagonist 1 (Compound 15f) is an HTR2A antagonist with an IC50 of 42.79 nM. It induces sub-G1 cell cycle arrest and apoptosis in colorectal cancer cells by activating the p53/p21/caspase 3 signaling pathway. HTR2A antagonist 1 exhibits good liver microsomal stability and is useful for colorectal cancer research.Formula:C35H43Cl2F2N5O4Color and Shape:SolidMolecular weight:706.65L803
CAS:L803 is a selective somatostatin receptor type 4 (SST4) agonist that can inhibit L-type calcium channel currents (ICa). It holds potential for research into degenerative diseases of retinal ganglion cells (RGC), such as glaucoma.Formula:C50H80N13O19PColor and Shape:SolidMolecular weight:1198.22mPGES-1/sEH-IN-1
mPGES-1/sEH-IN-1 (compound 1f) is an sEH inhibitor with an IC50 value of 5 μM. It also exhibits antitumor activity by inhibiting mPGES-1, with an IC50 value of 25 µM.Formula:C20H16F3N3O2Color and Shape:SolidMolecular weight:387.355Yohimbic acid, ethyl ester
CAS:Yohimbic acid, ethyl ester is a biochemical with possible effects on reserpine action.Formula:C22H28N2O3Color and Shape:SolidMolecular weight:368.47SRA880 free base
CAS:SRA880: sst1-receptor antagonist, low affinity for other somatostatin receptors, binds to dopamine D4, may enhance antidepressant effects.Formula:C26H32N4O4Color and Shape:SolidMolecular weight:464.56Moxilubant HCl
CAS:Moxilubant HCl: small molecule LTB4R antagonist for immune, skin, musculoskeletal disorders, and research in psoriasis, arthritis.Formula:C26H38ClN3O4Purity:99.94%Color and Shape:SoildMolecular weight:492.05CAY10580
CAS:CAY10580 is a potent and selective prostaglandin EP 4 receptor agonist ( K i =35 nM).Formula:C19H35NO4Color and Shape:SolidMolecular weight:341.49L-703606 oxalate hydrate
L-703606 oxalate hydrate is an effective, selective NK1 receptor antagonist. It is utilized in research related to gastric acid secretion.Color and Shape:Odour SolidY1 receptor antagonist 1 formic
H 409-22 isomer formic, a formate salt of Y1 receptor antagonist 1, is an antagonist of the neuropeptide Y1 receptor (neuropeptide Y1 receptor). This compound effectively blocks the actions of the receptor, playing a crucial role in modulating physiological responses.Formula:C29H35N5O5Color and Shape:SolidMolecular weight:533.629-deoxy-9-methylene-16,16-dimethyl Prostaglandin E2
CAS:Meteneprost is a strong, long-lasting Prostaglandin E2 analog effective in ending early monkey pregnancies without causing fever or GI issues.Formula:C23H38O4Color and Shape:SolidMolecular weight:378.553WB4-24
CAS:WB4-24 is a GLP-1 receptor agonist that enhances the release of β-endorphin in microglia. It exhibits antiallodynic, anti-inflammatory, and analgesic effects in mouse models of inflammation induced by formalin, carrageenan, and CFA.Formula:C52H48N4O14S2Color and Shape:SolidMolecular weight:1017.09MLS1082
CAS:MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.Formula:C24H23N3O2Purity:99.53%Color and Shape:SolidMolecular weight:385.46Protease-Activated Receptor-1 antagonist 2
CAS:Orally active PAR-1 antagonist with 7 nM IC50; potential for CVD research.Formula:C24H23F2N3O2Color and Shape:SolidMolecular weight:423.46NN1213
NN1213 (Peptide 21) is a long-acting human amylin peptide analogue that functions as a selective amylin receptor agonist. It has an EC50 of 0.177 nM for hAMY3R and 0.262 nM for rAMY3R. In both rat and dog models, NN1213 significantly reduces appetite and is utilized in anti-obesity research.Color and Shape:Odour SolidCCR2 antagonist 1
CAS:CCR2 antagonist 1 is a high-affinity and long-residence-time antagonist of CCR2 (Ki: 2.4 nM).Formula:C28H32BrF3N2OColor and Shape:SolidMolecular weight:549.47YM 218
CAS:YM 218 is a novel, potent, selective antagonist of nonpeptide vasopressin V1A receptor.Formula:C35H38F2N4O4Color and Shape:SolidMolecular weight:616.7Prolactin Releasing Peptide (1-31), human acetate
Prolactin Releasing Peptide (1-31), human (acetate), is a potent GPR10 ligand with high affinity, eliciting prolactin secretion.Formula:C162H26N56O44SColor and Shape:SolidMolecular weight:3724.17Cannabinol methyl ether
CAS:Cannabinol methyl ether, a phytocannabinoid, serves as an analytical reference standard. This compound can be obtained through isolation from Cannabis plants, derived from cannabinol, or synthesized. The physiological and toxicological properties of cannabinol methyl ether remain unknown. It is designed exclusively for research and forensic applications.Formula:C22H28O2Color and Shape:SolidMolecular weight:324.5
