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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 6012 products of "GPCR/G-Protein"

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  • INCB3344 R-isomer


    INCB3344 is a potent CCR2 antagonist. INCB3344 R-isomer is the R-isomer of INCB3344.
    Formula:C29H34F3N3O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:577.59

    Ref: TM-T11650

    25mg
    2,178.00€
    50mg
    2,862.00€
    100mg
    3,870.00€
  • [Ala11,D-Leu15]-Orexin B acetate


    [Ala11,D-Leu15]-Orexin B acetate is a selective agonist of orexin-2 receptor (OX2) with an EC50 of 0.13 nM, showing 400-fold selectivity over OX1 (52 nM).
    Formula:C122H210N44O37S
    Purity:98.18%
    Color and Shape:Solid
    Molecular weight:2917.31

    Ref: TM-TP1975L

    1mg
    281.00€
    5mg
    637.00€
    10mg
    954.00€
    25mg
    1,720.00€
    50mg
    2,313.00€
  • 7-Hydroxy-PIPAT maleate

    CAS:
    7-Hydroxy-PIPAT maleate is a D3R agonist.
    Formula:C16H22INO
    Color and Shape:Solid
    Molecular weight:371.262

    Ref: TM-T38188

    10mg
    130.00€
    50mg
    513.00€
  • Met-RANTES,human,acetate


    Met-RANTES (human) acetate is the acetate salt form of Met-RANTES (human). It acts as an antagonist for CCR1 and CCR5 receptors. This compound inhibits the human chemokines MIP-1α and MIP-1β, with respective IC50 values of 5 and 2 nM. Additionally, Met-RANTES (human) acetate reduces bone destruction and alleviates adjuvant-induced arthritis (AIA) in rats.
    Color and Shape:Odour Solid

    Ref: TM-T200698

    10mg
    To inquire
    50mg
    To inquire
  • 5-methoxy-α-Ethyltryptamine

    CAS:

    5-Methoxy-alpha-ethyltryptamine is a psychoactive substance that can cause various effects. It belongs to the tryptamine chemical class and can be used for various psychoactive and stimulant effects.

    Formula:C13H18N2O
    Purity:98.25%
    Color and Shape:Solid
    Molecular weight:218.29

    Ref: TM-T9746

    1mL*10mM (DMSO)
    50.00€
    5mg
    51.00€
    10mg
    80.00€
    25mg
    148.00€
    50mg
    268.00€
    100mg
    446.00€
    200mg
    621.00€
  • S1P2 antagonist 1

    CAS:
    S1P2 antagonist 1 is an orally bioavailable S1P2 antagonist against fibrotic diseases.
    Formula:C23H21ClN4O4
    Color and Shape:Solid
    Molecular weight:452.9

    Ref: TM-T39798

    5mg
    873.00€
  • [Ala1,3,11,15]-Endothelin

    CAS:
    Selective ETB endothelin receptor agonist (IC50 values are 0.33 and 2200 nM for displacing [125I]-ET-1 from ETB and ETA receptors respectively).
    Formula:C109H163N25O32S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2368

    Ref: TM-TP2099

    5mg
    452.00€
  • Apelin-36(human)

    CAS:
    Endogenous APJ agonist, EC50=20nM, regulates cardiovascular function, fluid balance, and feeding; blocks certain HIV strains.
    Formula:C184H297N69O43S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4195.87

    Ref: TM-TP2093

    1mg
    1,918.00€
  • Antidepressant agent 3


    Agent 3: orally active, antidepressant, anxiolytic, boosts performance and cognition.
    Formula:C17H30ClN5O2S
    Color and Shape:Solid
    Molecular weight:403.97

    Ref: TM-T75002

    5mg
    To inquire
    50mg
    To inquire
  • Suntinorexton

    CAS:
    Suntinorexton (TAK 861) is an orexin type 2 receptor (OX2R) agonist used in the study of neurologic disorders.
    Formula:C23H28F2N2O4S
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:466.54

    Ref: TM-T39807

    1mg
    171.00€
    5mg
    418.00€
    1mL*10mM (DMSO)
    428.00€
    10mg
    666.00€
    25mg
    1,017.00€
    50mg
    1,372.00€
    100mg
    1,793.00€
    200mg
    2,405.00€
  • Anti-TSHR Antibody (M22)


    Anti-TSHR Antibody (M22) is a humanized IgG1 monoclonal antibody targeting the thyroid-stimulating hormone receptor (TSHR). This antibody is capable of inhibiting the interaction between TSH and TSHR.
    Color and Shape:Odour Liquid

    Ref: TM-T9901A-942

    5mg
    To inquire
    1mg
    175.00€
  • Jmv 179

    CAS:
    Jmv 179 is an antagonist of the cholecystokinin receptor.
    Formula:C51H67N7O15S
    Color and Shape:Solid
    Molecular weight:1050.19

    Ref: TM-T24204

    25mg
    1,369.00€
  • Leukotriene B5

    CAS:
    LTB5, an eicosapentaenoic acid metabolite via 5-LO, has varied bioactivities and enhances bullfrog lung strip contraction.
    Formula:C20H30O4
    Color and Shape:Solid
    Molecular weight:334.456

    Ref: TM-T36423

    25µg
    472.00€
    50µg
    919.00€
    100µg
    1,691.00€
    500µg
    6,621.00€
  • Somatostatin-28 (1-14)

    CAS:
    Somatostatin-28 (1-14) is a truncated neuropeptide from prosomatostatin cleavage.
    Formula:C61H105N23O21S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1528.71

    Ref: TM-TP1823

    1mg
    138.00€
    5mg
    535.00€
    10mg
    827.00€
  • Kisspeptin-10, rat

    CAS:
    Kisspeptin-10, rat is an Endogenous ligand for the rodent kisspeptin receptor (KISS1, GPR54).
    Formula:C63H83N17O15
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1318.44

    Ref: TM-TP1666

    1mg
    178.00€
    5mg
    763.00€
    10mg
    1,170.00€
    25mg
    2,008.00€
  • Colulintide

    CAS:
    Colulintide is an analog of amylin, utilized in obesity research.
    Color and Shape:Solid

    Ref: TM-TP3252

    10mg
    To inquire
    50mg
    To inquire
  • LY-53857 free base

    CAS:
    LY-53857 free base is a bioactive chemical.
    Formula:C23H32N2O3
    Color and Shape:Solid
    Molecular weight:384.51

    Ref: TM-T33018

    100mg
    To inquire
    500mg
    To inquire
  • CHS-114


    CHS-114 (SRF-114) is a fully human IgG1 antibody targeting the (CCR8) receptor. It shows potential for research in head and neck squamous cell carcinoma (HNSCC). The isotype control for CHS-114 can be referred to as HumanIgG1kappa, Isotype Control.
    Color and Shape:Odour Liquid

    Ref: TM-T9901A-769

    1mg
    To inquire
    5mg
    To inquire
  • Pancreatic Polypeptide, bovine

    CAS:
    Agonist at Y4 neuropeptide Y receptors.
    Formula:C186H287N53O56S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4225.78

    Ref: TM-TP1731

    1mg
    244.00€
    5mg
    827.00€
  • Cortistatin-29 (rat) (trifluoroacetate salt)

    CAS:
    Cortistatin-29, similar to somatostatin-28, derives from preprocortistatin and binds to SST receptors 1-5 with varying IC50 values.
    Formula:C161H240N46O41S2
    Color and Shape:Solid
    Molecular weight:3540.09

    Ref: TM-T35663

    1mg
    To inquire