
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,028 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(61 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6012 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
INCB3344 R-isomer
INCB3344 is a potent CCR2 antagonist. INCB3344 R-isomer is the R-isomer of INCB3344.Formula:C29H34F3N3O6Purity:98%Color and Shape:SolidMolecular weight:577.59[Ala11,D-Leu15]-Orexin B acetate
[Ala11,D-Leu15]-Orexin B acetate is a selective agonist of orexin-2 receptor (OX2) with an EC50 of 0.13 nM, showing 400-fold selectivity over OX1 (52 nM).Formula:C122H210N44O37SPurity:98.18%Color and Shape:SolidMolecular weight:2917.317-Hydroxy-PIPAT maleate
CAS:7-Hydroxy-PIPAT maleate is a D3R agonist.Formula:C16H22INOColor and Shape:SolidMolecular weight:371.262Met-RANTES,human,acetate
Met-RANTES (human) acetate is the acetate salt form of Met-RANTES (human). It acts as an antagonist for CCR1 and CCR5 receptors. This compound inhibits the human chemokines MIP-1α and MIP-1β, with respective IC50 values of 5 and 2 nM. Additionally, Met-RANTES (human) acetate reduces bone destruction and alleviates adjuvant-induced arthritis (AIA) in rats.Color and Shape:Odour Solid5-methoxy-α-Ethyltryptamine
CAS:5-Methoxy-alpha-ethyltryptamine is a psychoactive substance that can cause various effects. It belongs to the tryptamine chemical class and can be used for various psychoactive and stimulant effects.
Formula:C13H18N2OPurity:98.25%Color and Shape:SolidMolecular weight:218.29S1P2 antagonist 1
CAS:S1P2 antagonist 1 is an orally bioavailable S1P2 antagonist against fibrotic diseases.Formula:C23H21ClN4O4Color and Shape:SolidMolecular weight:452.9[Ala1,3,11,15]-Endothelin
CAS:Selective ETB endothelin receptor agonist (IC50 values are 0.33 and 2200 nM for displacing [125I]-ET-1 from ETB and ETA receptors respectively).Formula:C109H163N25O32SPurity:98%Color and Shape:SolidMolecular weight:2368Apelin-36(human)
CAS:Endogenous APJ agonist, EC50=20nM, regulates cardiovascular function, fluid balance, and feeding; blocks certain HIV strains.Formula:C184H297N69O43SPurity:98%Color and Shape:SolidMolecular weight:4195.87Antidepressant agent 3
Agent 3: orally active, antidepressant, anxiolytic, boosts performance and cognition.Formula:C17H30ClN5O2SColor and Shape:SolidMolecular weight:403.97Suntinorexton
CAS:Suntinorexton (TAK 861) is an orexin type 2 receptor (OX2R) agonist used in the study of neurologic disorders.Formula:C23H28F2N2O4SPurity:99.89%Color and Shape:SolidMolecular weight:466.54Ref: TM-T39807
1mg171.00€5mg418.00€1mL*10mM (DMSO)428.00€10mg666.00€25mg1,017.00€50mg1,372.00€100mg1,793.00€200mg2,405.00€Anti-TSHR Antibody (M22)
Anti-TSHR Antibody (M22) is a humanized IgG1 monoclonal antibody targeting the thyroid-stimulating hormone receptor (TSHR). This antibody is capable of inhibiting the interaction between TSH and TSHR.Color and Shape:Odour LiquidJmv 179
CAS:Jmv 179 is an antagonist of the cholecystokinin receptor.Formula:C51H67N7O15SColor and Shape:SolidMolecular weight:1050.19Leukotriene B5
CAS:LTB5, an eicosapentaenoic acid metabolite via 5-LO, has varied bioactivities and enhances bullfrog lung strip contraction.Formula:C20H30O4Color and Shape:SolidMolecular weight:334.456Somatostatin-28 (1-14)
CAS:Somatostatin-28 (1-14) is a truncated neuropeptide from prosomatostatin cleavage.Formula:C61H105N23O21SPurity:98%Color and Shape:SolidMolecular weight:1528.71Kisspeptin-10, rat
CAS:Kisspeptin-10, rat is an Endogenous ligand for the rodent kisspeptin receptor (KISS1, GPR54).Formula:C63H83N17O15Purity:98%Color and Shape:SolidMolecular weight:1318.44Colulintide
CAS:Colulintide is an analog of amylin, utilized in obesity research.Color and Shape:SolidLY-53857 free base
CAS:LY-53857 free base is a bioactive chemical.Formula:C23H32N2O3Color and Shape:SolidMolecular weight:384.51CHS-114
CHS-114 (SRF-114) is a fully human IgG1 antibody targeting the (CCR8) receptor. It shows potential for research in head and neck squamous cell carcinoma (HNSCC). The isotype control for CHS-114 can be referred to as HumanIgG1kappa, Isotype Control.Color and Shape:Odour LiquidPancreatic Polypeptide, bovine
CAS:Agonist at Y4 neuropeptide Y receptors.Formula:C186H287N53O56S2Purity:98%Color and Shape:SolidMolecular weight:4225.78Cortistatin-29 (rat) (trifluoroacetate salt)
CAS:Cortistatin-29, similar to somatostatin-28, derives from preprocortistatin and binds to SST receptors 1-5 with varying IC50 values.Formula:C161H240N46O41S2Color and Shape:SolidMolecular weight:3540.09

