GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,027 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
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Carbocyclic Thromboxane A2
CAS:Carbocyclic Thromboxane A2 can be used in related research in the field of life sciences. Its product number is T36548 and CAS number is 74034-56-3.Formula:C22H36O3Color and Shape:SolidMolecular weight:348.527Pasireotide pamoate
CAS:Pasireotide pamoate is a stable cyclohexapeptide somatostatin mimic. Pasireotide pamoate exhibits antisecretory, antiproliferative, and proapoptotic activity.Formula:C81H82N10O15Purity:98%Color and Shape:SolidMolecular weight:1435.58Tirzepatide hydrochloride
Tirzepatide HCl is a dual GIP and GLP-1 receptor agonist.Formula:C225H349N48O68ClPurity:98%Color and Shape:SolidMolecular weight:4849.91α-CGRP(human) TFA
α-CGRP(human) TFA is a 37-amino acid regulatory neuropeptide that is extensively located within the central and peripheral nervous system, functioning as aFormula:C165H268F3N51O51S2Color and Shape:SolidMolecular weight:3903.33Contulakin G
CAS:Contulakin G: O-glycosylated neurotensin, weak neurotensin receptor agonist, strong antinociceptive.Formula:C88H140N20O37Molecular weight:2070.17Brexpiprazole S-oxide D8
CAS:Brexpiprazole S-oxide D8 (DM-3411 D8) is a deuterium-labeled metabolite of Brexpiprazole, a partial agonist at 5-HT1A and dopamine receptors.Formula:C25H19D8N3O3SPurity:98%Color and Shape:SolidMolecular weight:457.61Biotinyl-neuropeptide W-23 (human)
CAS:Biotinyl-neuropeptide W-23 (human) is a biotinylated form of neuropeptide W-23 (human), which functions as an agonist for the NPBW1 (GPR7) and NPBW2 (GPR8)Formula:C129H197N37O30S2Color and Shape:SolidMolecular weight:2810.3DD202-114
CAS:DD202-114 is an effective and selective agonist of GLP1R. It promotes the accumulation of cAMP, reduces blood glucose levels, and decreases food intake. Additionally, DD202-114 holds potential for research in type 2 diabetes mellitus (T2DM) and obesity studies.Formula:C33H35FN4O5Color and Shape:SolidMolecular weight:586.65MD01-67
CAS:MD01-67 is a macrocyclic compound selectively targeting the neurotensin 2 receptor (NTS2), with a Ki of 2.9 nM. It exhibits analgesic activity and reduces tactile hypersensitivity in rat models of acute, sustained, and chronic inflammatory pain.Formula:C37H58N8O8Color and Shape:SolidMolecular weight:742.91BQ-3020 ammonium
BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] ET-1 binding to ET B receptors with an IC50 of 0.2Formula:C96H140N20O25S·xNH3Purity:98%Color and Shape:SolidMolecular weight:2006.32 (free base)VIP(6-28)(human, rat, porcine, bovine)
CAS:VIP(6-28) blocks VIP-induced cAMP signaling in humans, rats, pigs, and cows.Formula:C126H207N37O34SPurity:98%Color and Shape:SolidMolecular weight:2816.28Neuropeptide W-23 (human) (TFA)
Neuropeptide W-23 (human) (NPW-23) TFA, representing the active form of Neuropeptide W, functions as an endogenous agonist for both NPBW1 (GPR7) and NPBW2 (GPR8Color and Shape:Odour SolidTCMCB07 TFA
TCMCB07 TFA is a cyclic nonapeptide and an orally active, brain-penetrating antagonist of the melanocortin receptor 4 (MC4R), playing a significant role inFormula:C63H87N15O11·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:1230.46 (free base)Tabernanthalog
CAS:TBG is a 5-HT2A agonist reducing alcohol/heroin cravings and promoting neuroplasticity with antidepressant effects in rodents.Formula:C14H18N2OPurity:99.82% - 99.89%Color and Shape:SoildMolecular weight:230.31Ref: TM-T60221
1mg175.00€2mg264.00€1mL*10mM (DMSO)344.00€5mg404.00€10mg592.00€25mg888.00€50mg1,243.00€100mg1,701.00€500mg3,402.00€RWJ 676070
CAS:RWJ 676070 is an antagonist of vasopressin V1A/V2 receptor.Formula:C30H26ClFN2O5Color and Shape:SolidMolecular weight:548.99PAMP-12(human, porcine) TFA
PAMP-12(human, porcine) TFA, a significant constituent of immunoreactive (ir)-PAMP, derives from the adrenomedullin precursor and functions as a potentColor and Shape:Odour Solid4-Methylhistamine
CAS:4-Methylhistamine serves as a potent agonist for the histamine 4 receptor (H4R), holding promise for research into immune-related diseases, including cancer andFormula:C6H11N3Purity:98%Color and Shape:SolidMolecular weight:125.17Dapoxetine
CAS:Dapoxetine (Dapoxetina) is a selective serotonin reuptake inhibitor, for the treatment of premature ejaculation.Formula:C21H23NOPurity:99.73%Color and Shape:White To Off-White Crystalline PowderMolecular weight:305.42W140 HBr
CAS:[(3S)-3-amino-4-(3-hexylanilino)-4-oxobutyl]phosphonic acid;hydrobromide is a S1P1 antagonist with Ki of 2.84 μM.Formula:C16H28BrN2O4PPurity:99.85%Color and Shape:SoildMolecular weight:423.28Ref: TM-T60204
1mg115.00€2mg172.00€5mg255.00€1mL*10mM (DMSO)284.00€10mg375.00€25mg562.00€50mg787.00€100mg1,074.00€TCMCB07
CAS:TCMCB07, a cyclic nonapeptide, serves as an orally active, brain-penetrant antagonist of the melanocortin receptor 4 (MC4R), with significant implications inFormula:C63H87N15O11Purity:98%Color and Shape:SolidMolecular weight:1230.46
