GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5985 products of "GPCR/G-Protein"
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Adrenomedullin (16-31), human TFA
Human adrenomedullin (16-31) TFA, fragment 16-31, binds CGRP1 receptor, raises rat blood pressure, not cats’.Formula:C84H130F3N25O23S2Color and Shape:SolidMolecular weight:1979.21Alosetron-d3
CAS:Alosetron D3 (GR 68755 D3) is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.Formula:C17H18N4OPurity:98%Color and Shape:SolidMolecular weight:297.3715(S)-HpEPE
CAS:15(S)-HpEPE, a monohydroperoxy fatty acid, forms when 15-lipoxygenase acts on EPA, with expected biological activities akin to 15(S)-HpETE.Formula:C20H30O4Color and Shape:SolidMolecular weight:334.456Rhazimine
CAS:Rhazimine is an indole alkaloid. It is a dual inhibitor of arachidonic acid metabolism and platelet activating factor-induced platelet aggregation.Formula:C21H22N2O3Color and Shape:SolidMolecular weight:350.418Des His1, Glu8 Exendin-4
Des His1, Glu8 Exendin-4 is a glucagon-like peptide-1 receptor (GLP1R) antagonist that regulates blood glucose and is used in the study of diabetes and obesity.Formula:C179H277N47O59SPurity:99.92%Color and Shape:SolidMolecular weight:4063.46Oxmetidine
CAS:Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular system and is used in the study of duodenal ulcers.Formula:C19H21N5O3SPurity:99.67%Color and Shape:SolidMolecular weight:399.47Ref: TM-T68122
1mg358.00€5mg848.00€10mg1,153.00€25mg1,693.00€50mg2,313.00€100mg3,115.00€500mg6,255.00€Mosliciguat
CAS:Mosliciguat is a guanylate cyclase activator.Formula:C41H36ClF3N2O5Color and Shape:SolidMolecular weight:729.19Octodrine
CAS:Octodrine (2-Amino-6-methylheptane) is primarily used as a pharmaceutical intermediate for Octamylamine; it also functions as a local anesthetic and vasoconstrictor.Formula:C8H19NPurity:99.98%Color and Shape:Clear Colorless To Light Yellow LiquidMolecular weight:129.24BIMU 8
CAS:BIMU 8 is a selective agonist of 5-HT4 with EC50s of 18 nM, 77 nM, and 540 nM for wild-type 5HT4 receptor, T3.36A, and W6.48A mutant 5-HT4.Formula:C19H27ClN4O2Purity:99.87%Color and Shape:SolidMolecular weight:378.9Ref: TM-T21946
1mg85.00€5mg168.00€1mL*10mM (DMSO)175.00€10mg235.00€25mg394.00€50mg582.00€100mg827.00€500mg1,674.00€Neurokinin A(4-10)
CAS:Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .Formula:C34H54N8O10SPurity:98%Color and Shape:SolidMolecular weight:766.91GLP-1R agonist 27
GLP-1R agonist 27 (compound 21) is a potent and orally active GLP-1R agonist. It enhances the accumulation of cyclic adenosine monophosphate (cAMP), reduces blood glucose levels, and decreases food intake. GLP-1R agonist 27 shows potential for research in obesity and type 2 diabetes mellitus (T2DM).Formula:C32H33N5O4SeColor and Shape:SolidMolecular weight:630.6γ1-MSH
CAS:Endogenous melanocortin MC3 receptor agonist (pKi = 7.46) that displays ~ 40-fold selectivity over MC4.Formula:C72H97N21O14SPurity:98%Color and Shape:SolidMolecular weight:1512.76Vapiprost hydrochloride
CAS:Vapiprost hydrochloride is a biochemicla.Formula:C30H40ClNO4Color and Shape:SolidMolecular weight:514.1Spantide II
CAS:Spantide II is an antagonist of tachykinin.Formula:C86H104Cl2N18O13Purity:98%Color and Shape:SolidMolecular weight:1668.77Bertilimumab
CAS:Bertilimumab (CAT 213; iCo-008), a human monoclonal antibody that targets eotaxin-1 (CCL11), shows promise in the research of allergic disorders [1].Color and Shape:LiquidVatinoxan
CAS:Vatinoxan is a peripheral α2 adrenoreceptor antagonist.Formula:C20H26N4O4SPurity:98%Color and Shape:SolidMolecular weight:418.51CCR4 antagonist 3
CAS:Orally active CCR4 antagonist with piperidinyl-azetidine; IC50: 22 nM (calcium flux), 50 nM (CTX); antitumor effects.Formula:C24H27Cl2N7OColor and Shape:SolidMolecular weight:500.43SC-53116
CAS:SC-53116 HCl can increase the production of serotonin in central nervous system tissues and is a psychoactive agent.Formula:C16H22ClN3O2Color and Shape:SolidMolecular weight:323.82MD01-67
CAS:MD01-67 is a macrocyclic compound selectively targeting the neurotensin 2 receptor (NTS2), with a Ki of 2.9 nM. It exhibits analgesic activity and reduces tactile hypersensitivity in rat models of acute, sustained, and chronic inflammatory pain.Formula:C37H58N8O8Color and Shape:SolidMolecular weight:742.91HTL22562
CAS:HTL22562 is a calcitonin gene-related peptide (CGRP) receptor antagonist for acute treatment of migraine.Formula:C40H49N11O5Color and Shape:SolidMolecular weight:763.904
