GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,022 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
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Found 5984 products of "GPCR/G-Protein"
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GRK2-IN-1 hydrochloride (2055990-90-2 free base)
GRKs-IN-1 hydrochloride has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: 130 nM) and GRK5 (IC50: 7.1 μM).Formula:C24H26ClFN4O4Purity:98%Color and Shape:SolidMolecular weight:488.94RGS2-Galpha-q interaction-IN-1
RGS2–Galpha-q interaction-IN-1 (Compound AJ-3) is an inhibitor of the RGS2-Galpha-q interaction. It inhibits the growth of cancer cell lines that express RGS2 and has anti-cell migration properties.Formula:C30H30ClN7O3Color and Shape:SolidMolecular weight:572.06Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP (1-7)-GRF (8-27)
CAS:Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP(1-7)-GRF(8-27) is a selective antagonist [1] for the vasoactive intestinal peptide 1 (VIP 1) receptor.Formula:C150H246N44O38Color and Shape:SolidMolecular weight:3273.83Conessine hydrobromide
CAS:Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.Formula:C24H41BrN2Color and Shape:SolidMolecular weight:437.51Apelin-12 acetate
Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.Formula:C66H107N21O16SPurity:98.82%Color and Shape:SolidMolecular weight:1482.75Ref: TM-T39823L
1mg128.00€5mg172.00€10mg269.00€25mg429.00€1mL*10mM (DMSO)430.00€50mg610.00€100mg820.00€LRGILS-NH2
CAS:LRGILS-NH2, reverse sequence of SLIGRL-NH2, is a control peptide for PAR2, affecting gut transit.Formula:C29H56N10O7Purity:98%Color and Shape:SolidMolecular weight:656.82L-770644 dihydrochloride
CAS:L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.Formula:C30H38ClN7O4SColor and Shape:SolidMolecular weight:628.19L 152804
CAS:L 152804: Y5 receptor antagonist, reduces food intake/boosts energy, leads to weight loss in obese mice.Formula:C23H26O4Purity:99.82%Color and Shape:SolidMolecular weight:366.45Ref: TM-T15679
5mg48.00€1mL*10mM (DMSO)49.00€10mg75.00€25mg111.00€50mg170.00€100mg245.00€200mg349.00€15(S)-Latanoprost
CAS:15(S)-Latanoprost, a latanoprost analog with inverted hydroxyl at C-15, has an IC50 of 24 nM and reduces IOP by 1 mmHg at 3 μg.Formula:C26H40O5Color and Shape:SolidMolecular weight:432.59Vapiprost hydrochloride
CAS:Vapiprost hydrochloride is a biochemicla.Formula:C30H40ClNO4Color and Shape:SolidMolecular weight:514.1Spantide II
CAS:Spantide II is an antagonist of tachykinin.Formula:C86H104Cl2N18O13Purity:98%Color and Shape:SolidMolecular weight:1668.77Bertilimumab
CAS:Bertilimumab (CAT 213; iCo-008), a human monoclonal antibody that targets eotaxin-1 (CCL11), shows promise in the research of allergic disorders [1].Color and Shape:LiquidW140 HBr
CAS:[(3S)-3-amino-4-(3-hexylanilino)-4-oxobutyl]phosphonic acid;hydrobromide is a S1P1 antagonist with Ki of 2.84 μM.Formula:C16H28BrN2O4PPurity:99.85%Color and Shape:SoildMolecular weight:423.28Ref: TM-T60204
1mg115.00€2mg172.00€5mg255.00€1mL*10mM (DMSO)284.00€10mg375.00€25mg562.00€50mg787.00€100mg1,074.00€Biotinyl-neuropeptide W-23 (human)
CAS:Biotinyl-neuropeptide W-23 (human) is a biotinylated form of neuropeptide W-23 (human), which functions as an agonist for the NPBW1 (GPR7) and NPBW2 (GPR8)Formula:C129H197N37O30S2Color and Shape:SolidMolecular weight:2810.3Methimepip dihydrobromide
CAS:Methimepip dihydrobromide is a selective H3R agonist.Formula:C10H19Br2N3Color and Shape:SolidMolecular weight:341.091Prolactin Releasing Peptide (1-31), human acetate
Prolactin Releasing Peptide (1-31), human (acetate), is a potent GPR10 ligand with high affinity, eliciting prolactin secretion.Formula:C162H26N56O44SColor and Shape:SolidMolecular weight:3724.17Neuropeptide Y5 receptor ligand-1
CAS:Neuropeptide Y5 receptor ligand-1 (Compound 54), a carbazole derivative, acts as a powerful antagonist to the neuropeptide Y5 (NPY-5) receptor [1].Formula:C19H17N3O2Color and Shape:SolidMolecular weight:319.36GB-110 hydrochloride
GB-110 HCl: potent, nonpeptidic oral PAR2 agonist; triggers Ca2+ release in HT29 cells; EC50 0.28 μM.Formula:C33H49ClN6O5Color and Shape:SolidMolecular weight:645.23Neuropeptide FF
CAS:Endogenous antiopioid peptide and agonist at NPFF1 and NPFF2 receptors (Ki values are 2.82 and 0.21 nM respectively).Formula:C54H76N14O10Purity:98%Color and Shape:SolidMolecular weight:1081.27d[Leu4,Lys8]-VP
CAS:Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.Formula:C47H67N11O11S2Purity:98%Color and Shape:SolidMolecular weight:1026.2
![d[Leu4,Lys8]-VP](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1927.webp&w=3840&q=75)