GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,012 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5981 products of "GPCR/G-Protein"
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Desmethyl Mirtazapine (hydrochloride)
CAS:Desmethyl mirtazapine is a metabolite of the antidepressant mirtazapine.1It is formed from mirtazapine by the cytochrome P450 (CYP) isoform CYP3A4.Formula:C16H18ClN3Color and Shape:SolidMolecular weight:287.79Kisspeptin-54(human)
CAS:Endogenous ligand for KISS1 receptor; Ki values: rat 1.80 nM, human 1.45 nM. Inhibits tumor spread, stimulates gonadotropin release.Formula:C258H401N79O78Purity:98%Color and Shape:SolidMolecular weight:5857.49K-(D-1-Nal)-FwLL-NH2
CAS:Potent ghrelin receptor inverse agonist with Ki of 4.9/31 nM in COS7/HEK293T; blocks Gq/G13 signaling.Formula:C51H67N9O6Purity:98%Color and Shape:SolidMolecular weight:902.13BIIE-0246
CAS:BIIE-0246 is a selective NPY2R antagonist, IC50=15 nM at the rat [125I]PYY3-36 site, reduces NPY-stimulated expression of p-AKT S473 and P-p44/42 MAPK.Formula:C49H57N11O6Purity:98%Color and Shape:SolidMolecular weight:896.05Adrenocorticotropic Hormone (ACTH) (1-39), rat TFA
Adrenocorticotropic Hormone (ACTH) (1-39), rat (TFA) is a potent melanocortin 2 receptor (MC2) agonist.Formula:C212H316F3N57O59SPurity:98%Color and Shape:SolidMolecular weight:4696.18Galanin (1-29)(rat, mouse)
CAS:Non-selective galanin agonist; Ki: GAL1-0.98, GAL2-1.48, GAL3-1.47 nM. Anticonvulsant, stops full seizures in rats.Formula:C141H211N43O41Purity:98%Color and Shape:White Lyophilized PowderMolecular weight:3164.499Bromchlorbuterol hydrochloride
CAS:Bromchlorbuterol HCl, a potent β-agonist, is used to study lung diseases like asthma.Formula:C12H19BrCl2N2OColor and Shape:SolidMolecular weight:358.1[Tyr1]-Somatostatin-14
CAS:[Tyr1]-Somatostatin-14 could binds to SSTR2.Formula:C82H108N18O20S2Molecular weight:1729.995-hydroxy Propranolol
CAS:5-hydroxy Propranolol, a propranolol metabolite, is formed in the liver via P450 2D6.Formula:C16H21NO3Color and Shape:SolidMolecular weight:275.34815(S)-15-methyl Prostaglandin F2α methyl ester
CAS:15(S)-15-methyl Prostaglandin F2α methyl ester can be used in related research in the field of life sciences.Formula:C22H38O5Color and Shape:SolidMolecular weight:382.53Ivabradine-d3 hydrochloride
CAS:Ivabradine HCl: novel If blocker, IC50 2.9 μM, slows heart rate; D3 version is deuterium labeled.Formula:C27H37ClN2O5Purity:98%Color and Shape:SolidMolecular weight:508.071-39-Corticotropin (human)(TFA)
ACTH (1-39) human (TFA) is a melanocortin agonist that boosts adrenal CS production and affects the CNS and immune system.Formula:C207H308N56O58S·C2HF3O2Purity:98%Color and Shape:SolidMolecular weight:4655.16GLP-1 (9-36) amide
CAS:GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.Formula:C140H214N36O43Purity:97%Color and Shape:SolidMolecular weight:3089.41CCG258208 hydrochloride
GRKs-IN-1 HCl (14as) strongly inhibits GRK2 (IC50=130nM) & GRK5 (IC50=7.1μM), is a paroxetine derivative with 100x cardiac boost.
Color and Shape:SolidFR252384
CAS:FR252384 is an antagonist of the neuropeptide Y-Y5 receptor (IC50: 2.3 nM).Formula:C18H17N3Purity:98%Color and Shape:SolidMolecular weight:275.35OXA(17-33)
CAS:Potent and selective peptide orexin OX1 receptor agonist (EC50 values are 8.29 and 187 nM for OX1 and OX2 receptors respectively). Truncated form of orexin A.Formula:C79H125N23O22Purity:98%Color and Shape:SolidMolecular weight:1749Cholecystokinin Octapeptide, desulfated
CAS:Cholecystokinin Octapeptide, desulfated (CCK Octapeptide, non-sulfated) is an octapeptide composed of 8 amino acids from cholecystokinin-8.Formula:C49H62N10O13S2Purity:97.12%Color and Shape:SolidMolecular weight:1063.21Amisulpride hydrochloride
CAS:Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.Formula:C17H28ClN3O4SColor and Shape:SolidMolecular weight:405.9411-deoxy Prostaglandin E2
CAS:11-deoxy PGE2 is a synthetic PGE2 analog, a potent bronchoconstrictor, 5-30x stronger than PGF2α on human respiratory muscles.Formula:C20H32O4Color and Shape:SolidMolecular weight:336.47Mabuterol free base
CAS:Mabuterol: selective β2 agonist, inhibits isoprenaline, affects rat uterus and rabbit jejunum, alters intestinal propulsion.Formula:C13H18ClF3N2OPurity:98%Color and Shape:SolidMolecular weight:310.74
