GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,004 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(155 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(192 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5971 products of "GPCR/G-Protein"
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AA 497 HCl
CAS:AA 497, a beta-2 agonist, suppresses Ca spikes.Formula:C14H22ClNO3Color and Shape:SolidMolecular weight:287.78U 67827E
CAS:U 67827E is a long-lasting cholecystokinin agonist. It acts by decreases food intake.Formula:C53H68N10O17SPurity:98%Color and Shape:SolidMolecular weight:1149.24Pasireotide (diaspartate)
CAS:Pasireotide diaspartate (SOM230) has high agonist activity at sst1/2/3/5, less at sst4; it's antiproliferative and proapoptotic.Formula:C66H80N12O17Color and Shape:SolidMolecular weight:1313.41[18F]-Labeled L-dopa precursor
CAS:[18F]-Labeled L-dopa precursor is a precursor for synthesis of 18F-labeled L-dopa[1].Formula:C35H36N2O7Color and Shape:SolidMolecular weight:596.67Denikitug
Denikitug is a chimeric antibody of the IgG1κ type that targets CCR8, with its corresponding isotype control being HumanIgG1kappa, Isotype Control.Color and Shape:Odour LiquidSB 699551
CAS:SB 699551 is a selective 5-HT5A antagonist (Ki=6.31 nM) that enhances 5-HT neuronal function. It inhibits SERT (Ki=25.12 nM),inhibit breast cancer.Formula:C34H45N3OPurity:99.83%Color and Shape:SoildMolecular weight:511.74Ref: TM-T23325L
1mg190.00€5mg471.00€10mg662.00€25mg1,036.00€50mg1,429.00€100mg1,821.00€200mg2,489.00€N6-Benzyl-5'-ethylcarboxamido adenosine
CAS:N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.Formula:C19H22N6O4Color and Shape:SolidMolecular weight:398.42GIP/GLP-1 dual receptor agonist-1
CAS:Compound 4: GIP/GLP-1 agonist for metabolic/fatty liver disease research.Color and Shape:SolidMK-0493 HCl
CAS:MK-0493 is a novel, potent, and selective agonist for melanocortin receptor 4 (MC4R).Formula:C30H39Cl2F2N3O2Color and Shape:SolidMolecular weight:582.55Bamosiran
CAS:Bamosiran, a small interfering RNA (siRNA), specifically targets the β-adrenergic receptor 2 to reduce intraocular pressure.Color and Shape:SolidAMTG-DA1
AMTG-DA1 is a ligand for the gastrin-releasing peptide receptor (GRPR), and it can be utilized in cancer research.Formula:C101H149IN22O25Color and Shape:SolidMolecular weight:2197.0109palm-PrRP31
palm-PrRP31 is a potent dual agonist for GPR10 (EC50=72 pM) and NPFF-R2. It activates downstream signaling pathways by binding to GPR10 and NPFF-R2 receptors, leading to reduced appetite and increased energy expenditure. palm-PrRP31 can be utilized to investigate its mechanism of action in the nervous system, thereby elucidating the complex biological processes involved in the regulation of appetite and energy expenditure.Formula:C176H282N56O43SMolecular weight:3900.1322Neuropeptide Y (human) free acid
CAS:Neuropeptide Y (human) free acid is the deamidated form of Neuropeptide Y (human, rat, mouse). The amidation of the C-terminal tyrosine in Neuropeptide Y is essential for its function, while the non-amidated form cannot initiate G-protein signaling.Formula:C189H284N54O58SMolecular weight:4270.06542A 77636 hydrochloride
CAS:A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).
Formula:C20H28ClNO3Purity:99.57%Color and Shape:SolidMolecular weight:365.89Cyclic AC253
Cyclic AC253 is an amylin receptor antagonist with an IC50 of 0.3 μM. It offers neuroprotective effects against Aβ toxicity and mitigates Aβ-induced impairments in hippocampal long-term potentiation. Additionally, Cyclic AC253 is capable of penetrating the blood-brain barrier.Formula:C126H202N42O40S2Molecular weight:3007.45049palm11-PrRP31
Palm11-PrRP31 is a lipid-modified analog of the endogenous appetite-suppressing neuropeptide (PrRP). It functions as a potent dual agonist for GPR10 (EC50 = 39 pM) and NPFF-R2. By mimicking the natural activity of PrRP, palm11-PrRP31 binds to these receptors to reduce food intake. It has potential applications as an anti-obesity agent and is useful in studying neuropeptide and receptor interactions.Formula:C181H289N55O46SMolecular weight:4001.16865GLP-1R agonist 20
GLP-1R agonist 20 (Compound I-132) is an agonist of the glucagon-like peptide-1 receptor (GLP-1 receptor), with an EC50 value of 0.0162 nM.Formula:C31H30Cl2F2N4O5Molecular weight:646.15613CB2R/FAAH modulator-3
CAS:CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.Formula:C22H31NO2Purity:99.81%Color and Shape:SoildMolecular weight:341.49BPP-2
BPP-2 is a GHSR ligand containing the element F. By labeling BPP-2 with the isotope 18F, a PET probe targeting GHSR can be produced. The binding affinity (Ki) of 18F-BPP-2 for GHSR is 274 nM.Formula:C27H28FN5O2Molecular weight:473.2227Satavaptan
CAS:Satavaptan is a vasopressin V2 receptor antagonist. Satavaptan improves the control of ascites in cirrhosis.Formula:C33H45N3O8SColor and Shape:SolidMolecular weight:643.79
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