GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,997 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5958 products of "GPCR/G-Protein"
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VIP(6-28)(human, rat, porcine, bovine)
CAS:VIP(6-28) blocks VIP-induced cAMP signaling in humans, rats, pigs, and cows.Formula:C126H207N37O34SPurity:98%Color and Shape:SolidMolecular weight:2816.28DD202-114
CAS:DD202-114 is an effective and selective agonist of GLP1R. It promotes the accumulation of cAMP, reduces blood glucose levels, and decreases food intake. Additionally, DD202-114 holds potential for research in type 2 diabetes mellitus (T2DM) and obesity studies.Formula:C33H35FN4O5Color and Shape:SolidMolecular weight:586.65Biotinyl-neuropeptide W-23 (human)
CAS:Biotinyl-neuropeptide W-23 (human) is a biotinylated form of neuropeptide W-23 (human), which functions as an agonist for the NPBW1 (GPR7) and NPBW2 (GPR8)Formula:C129H197N37O30S2Color and Shape:SolidMolecular weight:2810.3Contulakin G
CAS:Contulakin G: O-glycosylated neurotensin, weak neurotensin receptor agonist, strong antinociceptive.Formula:C88H140N20O37Molecular weight:2070.17MR 409
CAS:MR 409, a selective growth hormone-releasing hormone (GHRH) agonist, exhibits notable neuroprotective properties by augmenting endogenous neurogenesis inFormula:C153H252N44O43Color and Shape:SolidMolecular weight:3395.91N-Methyl-2-phenylpropan-1-amine hydrochloride
CAS:N-Methyl-2-phenylpropan-1-amine hydrochloride is an analogue of β-methylphenethylamine (BMPEA) and demonstrates neurotransmitter-releasing properties in experiments involving NET and DAT.Formula:C10H16ClNColor and Shape:SolidMolecular weight:185.69Cholecystokinin
CAS:Cholecystokinin, a peptide hormone, functions as a hunger suppressant by inhibiting food intake and promoting the digestion of fat and protein, and is employedColor and Shape:SolidBrain Natriuretic Peptide-45, rat TFA
Brain Natriuretic Peptide-45, rat TFA (BNP-45, rat TFA) is an isoform of rat brain natriuretic peptide extracted from rat heart, exhibiting significantColor and Shape:Odour Solid[D-Pro4,D-Trp7,9,10] Substance P (4-11)
CAS:[D-Pro4,D-Trp7,9,10] Substance P (4-11) serves as a potent antagonist of the tachykinin family of neuropeptides [1].Formula:C62H74N14O10SMolecular weight:1207.4Exendin-3
CAS:Exendin-3, a peptide from Gila monster venom, stimulates pancreatic secretion and belongs to the glucagon family.Formula:C184H282N50O61SPurity:98%Color and Shape:SolidMolecular weight:4202.57Antidepressant agent 10
CAS:Compound PDK0386, with CAS No. 87691-87-0, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0386 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formula:C11H13N3SMolecular weight:219.306Thrombostatin cont-1
CAS:Thrombostatin cont-1, an analogue of the bradykinin metabolite thrombostatin, has been shown to reduce platelet activation in the canine carotid arteryFormula:C87H142N34O29S2Molecular weight:2192.4Endothelin 1 (swine, human) (TFA)
CAS:Synthetic human/swine Endothelin 1 (TFA) peptide; a potent vasoconstrictor acting on ET A and ET B receptors.Formula:C111H160F3N25O34S5Molecular weight:2605.93Neurokinin A TFA
CAS:Neurokinin A TFA (NKA TFA) is a neuropeptide within the neurokinin family, serving as the endogenous ligand and agonist for the NK-2 (Neurokinin 2) receptor.Formula:C52H81F3N14O16SPurity:98.704%Color and Shape:SolidMolecular weight:1247.34Dabelotine, (S)-
CAS:Dabelotine, (S)- is the S-isomer of Dabelotine. Dabelotine is an adrenergic agonist used in the study of dementia.Formula:C15H22N2O2Color and Shape:SolidMolecular weight:262.35Pegapamodutide
CAS:Pegapamodutide (LY-2944876) is a dual glucagon-GLP-1 receptor agonist utilized in research concerning type 2 diabetes and obesity [1].Color and Shape:SolidLiraglutide acetate
CAS:Liraglutide acetate is the acetate salt form of Liraglutide, which is a glucagon-like peptide-1 (GLP-1) receptor agonist, utilized in the study of type 2 diabetes.Formula:C172H265N43O51·xC2H4O2Color and Shape:SolidMolecular weight:3751.20 (free base)Aldioxa
CAS:Aldioxa is a Gastrointestinal Agent.Formula:C4H7AlN4O5Color and Shape:SolidMolecular weight:218.10Urodilatin
CAS:Urodilatin, an analogue of ANF-(99-126), serves as a diuretic-natriuretic regulatory peptide with applications in the study of acute renal failure, congestiveColor and Shape:SolidLipoxin B4 methyl ester
CAS:Lipoxin B4 methyl ester is a lipid-soluble prodrug of LXB4, inhibiting PMN migration/adhesion by LTB4 with IC50 of 0.3 nM.Formula:C21H34O5Color and Shape:SolidMolecular weight:366.498
