GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5972 products of "GPCR/G-Protein"
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Nebokitug
Nebokitug is a humanized IgG1κ antibody targeting CCL24, with HumanIgG1kappa, Isotype Control serving as its corresponding isotype control.Color and Shape:Odour LiquidMRS 4062 triethylammonium salt
CAS:MRS 4062 triethylammonium salt is a selective P2Y4 receptor agonist (EC50 values are 23, 640, and 740 nM for hP2Y4, hP2Y2 and hP2Y6 respectively).Formula:C42H86N7O15P3Color and Shape:SolidMolecular weight:1022.105Alverine hydrochloride
CAS:Alverine hydrochloride is a parasympatholytic.Formula:C20H28ClNColor and Shape:SolidMolecular weight:317.9Rubraxanthone
CAS:Rubraxanthone is a PAF inhibitor isolated from Garcinia parvifolia Miq.Formula:C24H26O6Color and Shape:SolidMolecular weight:410.466LHRH, Ala(6)-
CAS:LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.Formula:C56H77N17O13Color and Shape:SolidMolecular weight:1196.32JMV-1645
CAS:JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.Formula:C49H69N13O12SPurity:98%Color and Shape:SolidMolecular weight:1064.23RS 18286
CAS:RS 18286 is a LHRH antagonist.Formula:C74H101Cl2N17O14Color and Shape:SolidMolecular weight:1523.6Abediterol napadisylate
CAS:Abediterol napadisylate is a novel long-acting β2-agonist in persistent asthma that is efficacy, safe, and tolerable.Formula:C60H68F4N4O14S2Purity:98%Color and Shape:SolidMolecular weight:1209.32Vapiprost
CAS:Vapiprost is an antagonist of the thromboxane receptor and a prostaglandin receptor.Formula:C30H39NO4Purity:98%Color and Shape:SolidMolecular weight:477.64A 76154
CAS:A 76154 is an antagonist of leutenizing hormone releasing hormone (LHRH).Formula:C70H93FN12O12Color and Shape:SolidMolecular weight:1313.584Glucagon receptor antagonists-1
CAS:Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.Formula:C29H34FNO2Purity:98%Color and Shape:SolidMolecular weight:447.58A71378
CAS:A71378 is a high potency, selectivity CCK-A receptors agonist.Formula:C48H62N8O13SPurity:98%Color and Shape:SolidMolecular weight:991.12Enuvaptan
CAS:Enuvaptan is a vasopressin receptor antagonist and has the potential for research into renal and cardiovascular diseases.Formula:C21H15ClF6N8O3Color and Shape:SolidMolecular weight:576.84I-BOP
CAS:I-BOP is an agonist (KD=0.61 nM) at the thromboxane A2 receptor (TP).Formula:C23H29IO5Color and Shape:SolidMolecular weight:512.384Tetrahydro-β-carboline
CAS:Compound Fr12161, with CAS No. 16502-01-5, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound Fr12161 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formula:C11H12N2Purity:96.31%Color and Shape:Tan SolidMolecular weight:172.2264Guanylin(human)
CAS:Peptide that activates gut guanylyl cyclase, secreted by GI mucosa, regulates water and electrolytes in gut and kidneys.Formula:C58H87N15O21S4Purity:98%Color and Shape:SolidMolecular weight:1458.65M40
CAS:Potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in ratFormula:C94H145N23O24Purity:98%Color and Shape:SolidMolecular weight:1981.33R 396
CAS:R 396 (Acleu-asp-gln-trp-phe-glynh2) is a linear hexapeptide and is also an NK-2 tachykinin receptor antagonist.Formula:C39H51N9O10Purity:98%Color and Shape:SolidMolecular weight:805.8817-phenyl trinor Prostaglandin E2 ethyl amide
CAS:17-phenyl trinor PGE2 ethyl amide, an EP1/EP3 agonist (Ki: 14-54 nM), enhances lipid solubility and tissue uptake, is a potent antifertility agent.Formula:C25H35NO4Color and Shape:SolidMolecular weight:413.55NSC380324
<p>NSC380324 is a P2Y12 receptor antagonist with antiplatelet properties, which can be employed in research on atherosclerotic cardiovascular diseases.</p>Formula:C31H24N4O4Color and Shape:SolidMolecular weight:516.55Edg-2 receptor inhibitor 1
CAS:Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).Formula:C27H27NO5Purity:99.47%Color and Shape:SolidMolecular weight:445.51Ref: TM-T4521
1mg97.00€2mg170.00€5mg274.00€10mg426.00€25mg663.00€50mg947.00€100mg1,264.00€1mL*10mM (DMSO)288.00€[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P
CAS:Broad-spectrum inverse agonist; potent at ghrelin receptor (EC50=5.2 nM); blocks other neuropeptide receptors; induces apoptosis; inhibits tumor growth.Formula:C79H109N19O12Purity:98%Color and Shape:SolidMolecular weight:1516.85RC-3095 TFA
CAS:RC-3095 TFA (RC-3095 (TFA)) is a bombesin/gastrin-releasing peptide (BN/GRP) antagonist with potential anticancer activity.Formula:C58H80F3N15O11Purity:98%Color and Shape:SolidMolecular weight:1220.34Mesoridazine Besylate
CAS:Mesoridazine Besylate (Serentil), a piperidine antipsychotic and phenothiazine, treats schizophrenia; it's a thioridazine metabolite.Formula:C27H32N2O4S3Purity:98.87%Color and Shape:SolidMolecular weight:544.75Phendioxan
CAS:Phendioxan is a biochemcial.Formula:C25H27NO5Color and Shape:SolidMolecular weight:421.49EP4-IN-1
CAS:EP4-IN-1: Potent EP4 receptor inhibitor with anti-tumor, anti-inflammatory, and analgesic properties.Formula:C27H24N2O4Purity:99.94%Color and Shape:SoildMolecular weight:440.49Pirepemat
CAS:Pirepemat (IRL752) is a cortical-preferring catecholamine agent that enhances cognition. It is utilized in the investigation of Parkinson's disease.Formula:C11H13F2NOColor and Shape:SolidMolecular weight:213.22Nesiritide acetate
CAS:Nesiritide, a 32-amino acid natriuretic peptide and recombinant form of human brain natriuretic peptide, enhances vasorelaxation ex vivo in porcine hearts from an acute coronary occlusion model when given as a 2 µg/kg bolus dose followed by a 0.01 µg/kg per minute infusion, facilitated by the calcium ionophore A23187. Formulations containing nesiritide have been utilized in managing congestive heart failure.Formula:C143H244N50O42S4C2H4O2Color and Shape:SolidMolecular weight:3524.1LP 12 hydrochloride
CAS:LP 12 hydrochloride is a selective 5-HT7 receptor agonist (Ki=0.13 nM).Formula:C32H40ClN3OColor and Shape:SolidMolecular weight:518.14SR 142948 TFA
SR 142948 TFA is an orally active, selective non-peptide neurotensin receptor (NT) antagonist, displaying IC50 values of 1.19 nM in h-NTR1-CHO cells, 0.32 nM in HT-29 cells, and 3.96 nM in adult rat brain. In HT-29 cells, it counteracts NT-induced inositol monophosphate formation with an IC50 of 3.9 nM. It blocks NT-induced hypothermia, analgesia, and turning behavior in vivo and can cross the blood-brain barrier, making it useful for research in psychiatric disorders.Color and Shape:Odour Solid3-Deoxyglucosone
CAS:3-Deoxyglucosone(3-Deoxy-D-glucosone) is synthesized by the intermediate pathway of the melad and polyol reactions.3-Deoxyglucosone reacts rapidly with proteinFormula:C6H10O5Purity:95%Color and Shape:SolidMolecular weight:162.14LY86057
CAS:LY86057 is a bioactive chemical.Formula:C20H26N2O3Color and Shape:SolidMolecular weight:342.439Colulintide
CAS:Colulintide is an analog of amylin, utilized in obesity research.Color and Shape:SolidΔ9-THCH
CAS:Δ9-THCH, a phytocannabinoid analytical reference standard, is present in a Cannabis variety cultivated for medicinal use. In the United States, it is classified as a Schedule I compound. This product is designated for research and forensic applications.Formula:C22H32O2Color and Shape:SolidMolecular weight:328.49CB1-IN-3
CB1-IN-3 (Compound 6i) is a potent inhibitor of the cannabinoid receptor type 1 (CB1). It holds potential for research in obesity, inflammation, and neurological disorders.Color and Shape:Odour SolidCannabinol methyl ether
CAS:Cannabinol methyl ether, a phytocannabinoid, serves as an analytical reference standard. This compound can be obtained through isolation from Cannabis plants, derived from cannabinol, or synthesized. The physiological and toxicological properties of cannabinol methyl ether remain unknown. It is designed exclusively for research and forensic applications.Formula:C22H28O2Color and Shape:SolidMolecular weight:324.5Maceneolignan H
CAS:Maceneolignan H, a neolignane from Myristica fragrans, selectively blocks CCR3 (EC50=1.4μM) with allergy research potential.Formula:C24H30O7Color and Shape:SolidMolecular weight:430.49Prostaglandin F2α methyl ester
CAS:Prostaglandin F2α methyl ester is a highly lipid-soluble PGF2α analog used to maintain low intraocular pressure.Formula:C21H36O5Color and Shape:SolidMolecular weight:368.5113,14-dihydro-15-keto Prostaglandin F1α
CAS:<p>13,14-dihydro-15-keto Prostaglandin F1α (13,14-dihydro-15-keto PGF1α) is a metabolite of PGF1α that has been reported in the rat stomach.</p>Formula:C20H36O5Color and Shape:SolidMolecular weight:356.5Losulazine
CAS:<p>Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.</p>Formula:C27H22F4N4O3SPurity:98.83%Color and Shape:SolidMolecular weight:558.55S33084
CAS:S33084 is a potent, selective and competitive antagonist of dopamine D(3)-receptors.Formula:C29H29N3O2Purity:98%Color and Shape:SolidMolecular weight:451.56Xanthine amine congener trihydrochloride
CAS:Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.Formula:C21H29ClN6O4Purity:98.81%Color and Shape:SolidMolecular weight:464.95Berobenatide
CAS:Berobenatide is a glucagon-like peptide-1 (GLP-1) receptor agonist.Color and Shape:Solid2,3-dinor Thromboxane B1
CAS:TXB2 released from platelets becomes 11-dehydro and 2,3-dinor TXB2. Rats excrete 2,3-dinor TXB1, a reliable thromboxane biosynthesis marker.Formula:C18H32O6Color and Shape:SolidMolecular weight:344.448Neuromedin S (human)
CAS:Neuromedin S (human) is a 33-amino acid neuropeptide identified as an endogenous ligand for the orphan G-protein coupled receptor (GPCR) FM-4/TGR-1, acting onProstaglandin F2α isopropyl ester
CAS:PGF2α isopropyl ester is an ester prodrug of PGF2α with enhanced lipid solubility.Formula:C23H40O5Color and Shape:SolidMolecular weight:396.568Secretin, canine TFA
Secretin, canine TFA, is an endocrine hormone that stimulates the secretion of pancreatic fluid rich in bicarbonate. Additionally, Secretin, canine TFA, can regulate the primary cell functions and paracellular permeability of gastric monolayer cells through an Src kinase-dependent pathway.Color and Shape:Odour SolidGalanin (2-29) (rat)
CAS:Peptide agonist for galanin receptorsFormula:C139H208N42O40Purity:98%Color and Shape:SolidMolecular weight:3107.45-HT6 inverse agonist 1
CAS:5-HT6 inverse agonist 1 (Compound 33) is an antagonist of the 5-HT6 receptor with a Ki of 23 nM and a Kb of 6.62 nM. This compound can inhibit 5-HT6R-mediated Cdk5 and mTOR signaling pathways and reduce tactile allodynia induced by spinal nerve ligation (SNL) in rat models.Formula:C22H22Cl2FN3O3SColor and Shape:SolidMolecular weight:498.4Urocortin II, human acetate
Urocortin II, human acetate, is a selective endogenous peptide agonist of type 2 corticotropin-releasing factor (CRF2) receptors, used to study the role of CRF2 receptors in feeding behavior.Color and Shape:Odour Solid
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