GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,018 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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ICI 192605
CAS:ICI 192605 is a potent thromboxane A2 receptor (TP receptor) antagonist.Formula:C22H23ClO5Color and Shape:SolidMolecular weight:402.87AL-3138
CAS:AL-3138 is a prostaglandin F2alpha (PGF2alpha) analogue which antagonizes FP prostanoid receptor-mediated inositol phosphates generation.Formula:C20H33FO4Color and Shape:SolidMolecular weight:356.47MK-8133
CAS:MK-8133 is an antagonist of orexin-2 selective receptor with favorable development properties.Formula:C23H21N5O2Color and Shape:SolidMolecular weight:399.45Fluprostenol methyl ester
CAS:Fluprostenol, a vet-approved luteolytic, has an isopropyl ester, travoprost, used as an eye pressure reducer. CAY10532 is its methyl ester form.Formula:C24H31F3O6Color and Shape:SolidMolecular weight:472.49SB 207710
CAS:SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.Formula:C19H27IN2O4Color and Shape:SolidMolecular weight:474.33QCC-374
CAS:QCC-374 is a prostanoid agonist. It potentially for the treatment of pulmonary arterial hypertension.Formula:C28H33N3O2Purity:98%Color and Shape:SolidMolecular weight:443.58UK 1745
CAS:UK 1745 is a novel drug of cardiotonic.Formula:C16H23ClN2O2Color and Shape:SolidMolecular weight:310.82LY288513
CAS:Selective CCK2 receptor antagonistFormula:C22H18BrN3O2Purity:98%Color and Shape:SolidMolecular weight:436.3GSK-269984B
CAS:GSK-269984B is a novel antagonist of EP1 receptor.Formula:C20H14Cl2FNO3Purity:98%Color and Shape:SolidMolecular weight:406.23WB403
CAS:WB403 activates TGR5, lowers fasting/postprandial glucose and HbA1c, enhances glucose tolerance, and normalizes pancreatic α/β-cells in diabetic mice.Formula:C19H19BrN2OSPurity:98%Color and Shape:SolidMolecular weight:403.34PD-135666
CAS:PD-135666 is an antagonist of CCK receptor.Formula:C33H39N3O5Purity:98%Color and Shape:SolidMolecular weight:557.68S-777469
CAS:S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.Formula:C23H27FN2O4Color and Shape:SolidMolecular weight:414.47CB2 receptor agonist 3
CAS:GP 2A is a selective agonist of CB2 receptor.Formula:C24H23Cl2N3OColor and Shape:SolidMolecular weight:440.36INCB38579
CAS:INCB38579: Oral, selective H4 antagonist; crosses brain barrier; IC50s - hH4R: 4.8 nM, mH4R: 42 nM, rH4R: 32 nM; anti-inflammatory and antipruritic.Formula:C25H34N6OColor and Shape:SolidMolecular weight:434.58Edivoxetine
CAS:Edivoxetine (LY2216684) is a selective norepinephrine reuptake inhibitor for ADHD and depression.Formula:C18H26FNO4Color and Shape:SolidMolecular weight:339.4ChemR23-IN-1
CAS:ChemR23-IN-1 inhibits human and mouse ChemR23 (IC50: 38 nM, 100 nM) and stops CAL-1 chemotaxis induced by Chemerin in vitro.Formula:C28H29N7O2Color and Shape:SolidMolecular weight:495.58BGC-20-1531 free base
CAS:BGC-20-1531 (PGN 1531) free base is a selective and potent prostaglandin EP4 receptor antagonist (pKB: 7.6) that exhibits potential for migraine research.Formula:C26H24N2O6SColor and Shape:SolidMolecular weight:492.54Bopindolol (malonate)
CAS:Bopindolol is a non-selective β-adrenergic receptor antagonist.Formula:C26H32N2O7Color and Shape:SolidMolecular weight:484.549GPR183-IN-2
CAS:GPR183-IN-2 (compound 23) is an effective, orally active inhibitor of GPR183, displaying an IC50 value of 39.45 nM in Ca2+ mobilization assays. This compound has potential applications in research related to cancer, autoimmune diseases, pain, and osteoporosis.Formula:C19H23BrN2O3Color and Shape:SolidMolecular weight:407.3Iso-SLR 080811
CAS:Iso-SLR 080811 is an isomer of SLR 080811, suitable for relevant research in the life sciences. SLR080811 is a selective SphK2 inhibitor (Ki=1.3 μM).Formula:C21H32ClN5OPurity:98.34%Color and Shape:SolidMolecular weight:405.97CB1R Allosteric modulator 3
CAS:CB1R Allosteric modulator 3 is a CB1R modulator.CB1R Allosteric modulator 3 inhibits cAMP, and can be used for the study of obesity and nicotine addiction.Formula:C22H17ClN2O2Purity:98.18%Color and Shape:SolidMolecular weight:376.84DOV-216,303 Free Base
CAS:DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.Formula:C11H11Cl2NPurity:96.7%Color and Shape:SolidMolecular weight:228.12Nedocromil
CAS:Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).Formula:C19H17NO7Purity:95% - 97.34%Color and Shape:SolidMolecular weight:371.345-Carboxamidotryptamine maleate
CAS:5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.Formula:C15H17N3O5Purity:99.88%Color and Shape:SolidMolecular weight:319.31Mirisetron
CAS:Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.Formula:C24H31N3O2Purity:99.88%Color and Shape:SolidMolecular weight:393.52Iprindole
CAS:Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].Formula:C19H28N2Purity:99.54%Color and Shape:SolidMolecular weight:284.44Ref: TM-T37015
2mg34.00€5mg50.00€10mg75.00€25mg145.00€50mg253.00€100mg432.00€200mg618.00€1mL*10mM (DMSO)79.00€RS 15385-197
CAS:RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.Formula:C18H26N2O3SColor and Shape:SolidMolecular weight:350.48AHR-13268D
CAS:AHR-13268D is a new agent of antiallergic/antihistaminic.Formula:C28H29F2NNaO4Purity:98%Color and Shape:SolidMolecular weight:504.53R 47243
CAS:R 47243 is used as a racemic alpha 2 antagonist.Formula:C22H25N3O2SPurity:98%Color and Shape:SolidMolecular weight:395.52Burimamide
CAS:Burimamide is an antagonist of histamine. It appears to block both H2 and H3 histamine receptors.Formula:C9H16N4SPurity:98%Color and Shape:SolidMolecular weight:212.32FR 121196
CAS:FR 121196, a potential antidementia drug, ameliorates the impaired memory of rat in the Morris water maze.Formula:C12H16FN3O3SColor and Shape:SolidMolecular weight:301.34A23887
CAS:A23887 is a potentially neuroleptic tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Formula:C22H24ClNPurity:98%Color and Shape:SolidMolecular weight:337.89NNC-38-1049
CAS:NNC-38-1049 is a novel selective antagonist of histamine H3.Formula:C19H25ClN2O2Purity:98%Color and Shape:SolidMolecular weight:348.87Dipiproverine hydrochloride
CAS:Dipiproverine hydrochloride is an antispasmodic alpha-amino acid ester used as an anticholinergic.Formula:C20H32Cl2N2O2Purity:98%Color and Shape:SolidMolecular weight:403.39Opiranserin
CAS:Opiranserin is a development as an injectable agent for the treatment of postoperative pain.Formula:C21H34N2O5Purity:98%Color and Shape:SolidMolecular weight:394.51Ro 04-6790 dihydrochloride
CAS:Ro 04-6790 dihydrochloride is an effective and selective antagonist of the serotonin 5-HT6 receptor.Formula:C12H18Cl2N6O2SPurity:98%Color and Shape:SolidMolecular weight:381.28HSR-609
CAS:HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.Formula:C21H21FN2O3Purity:98%Color and Shape:SolidMolecular weight:368.4AS1069562
CAS:AS1069562 inhibits 5-HT/NE reuptake, boosts IGF-1, FGF2 mRNA in dorsal root ganglia, spinal cord.Formula:C20H23NO5SPurity:98%Color and Shape:SolidMolecular weight:389.46Dexnafenodone Hydrochloride
CAS:Dexnafenodone Hydrochloride is an adrenergic receptor antagonist and serotonin uptake inhibitor.Formula:C20H24ClNOColor and Shape:SolidMolecular weight:329.86LY 87130
CAS:LY 87130 is a phenylethanolamine-N-methyltransferase inhibitor.Formula:C12H13NPurity:98%Color and Shape:SolidMolecular weight:171.24FAUC-3019
CAS:FAUC-3019 is a partial agonist of the dopamine D(4) receptor.Formula:C22H24N2OColor and Shape:SolidMolecular weight:332.44Lergotrile
CAS:Lergotrile is used as an enzyme Inhibitor (Prolactin).Formula:C17H18ClN3Purity:98%Color and Shape:SolidMolecular weight:299.8RS 52367
CAS:RS 52367 is a beta-adrenergic antagonist.Formula:C18H34ClN3O3SColor and Shape:SolidMolecular weight:408RGH 1756
CAS:RGH 1756 is an atypical antipsychotic with high affinity to dopamine D(3) receptors that leads to c-Fos induction in a unique pattern.Formula:C26H30N4O2SPurity:98%Color and Shape:SolidMolecular weight:462.61Amthamine dihydrobromide
CAS:H2 agonistFormula:C6H13Br2N3SPurity:98%Color and Shape:SolidMolecular weight:319.06Flerobuterol
CAS:Flerobuterol is a potential antidepressant agent related to beta-adrenergic agonists.Formula:C12H18FNOPurity:98%Color and Shape:SolidMolecular weight:211.28LUF5981
CAS:LUF5981 is a selective agonist of human adenosine A1 receptor.Formula:C24H23N3Color and Shape:SolidMolecular weight:353.46DA 4643
CAS:DA 4643, a histamine H2-receptor antagonist, binds similarly to mifentidine at the receptor.Formula:C12H16Cl2N6SPurity:98%Color and Shape:SolidMolecular weight:347.26CV-3988
CAS:CV-3988 is a specific antagonist of PAF-R (platelet-activating factor receptor)(Ki = 0.872 μM).Formula:C28H53N2O7PSColor and Shape:SolidMolecular weight:592.775-Nonyloxytryptamine oxalate
CAS:5-HT1B agonistFormula:C21H32N2O5Purity:98%Color and Shape:SolidMolecular weight:392.49
