GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,023 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5985 products of "GPCR/G-Protein"
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AL-37350A
CAS:AL-37350A is a 5-HT2 receptor-selective agonist with ocular hypotensive activity.Formula:C14H18N2OColor and Shape:SolidMolecular weight:230.31ADX-10061
CAS:ADX-10061 is a dopamine D1 receptor antagonist.Formula:C19H20N2O4Color and Shape:SolidMolecular weight:340.37Levomoprolol
CAS:Levomoprolol, (S)-enantiomer of the moprololis, is a beta adrenergic antagonist.Formula:C13H21NO3Purity:98%Color and Shape:SolidMolecular weight:239.31RP5063 Hydrochloride
CAS:RP5063 Hydrochloride is a modulator of multimodal serotonin receptors.Formula:C22H26Cl3N3O3Purity:98%Color and Shape:SolidMolecular weight:486.82Dacemazine hydrochloride
CAS:Dacemazine is a phenothiazine derivative that acts as a histamine antagonist at the H1 subtype. It was also assessed as a possible anticancer drug.Formula:C16H17ClN2OSPurity:98%Color and Shape:SolidMolecular weight:320.84BW-A 575C
CAS:BW-A 575C is an inhibitor of ACE.Formula:C29H43N5O8Purity:98%Color and Shape:SolidMolecular weight:589.68Aplysamine-1
CAS:Aplysamine-1 is an antagonist of histamine H3 receptor.Formula:C15H24Br2N2OPurity:98%Color and Shape:SolidMolecular weight:408.17L 368935
CAS:L 368935 is an antagonist of the cholecystokinin receptor.Formula:C27H26N8O2Purity:98%Color and Shape:SolidMolecular weight:494.55Nor-SCH-12679 Maleate
CAS:Nor-SCH-12679 Maleate is a D1-dopamine receptor antagonist.Formula:C22H25NO6Purity:98%Color and Shape:SolidMolecular weight:399.44Clothixamide
CAS:Clothixamide（Clotixamide） is a thioxanthene derivative with antipsychotic activity.Formula:C24H28ClN3OSPurity:95.51%Color and Shape:SolidMolecular weight:442.02Dipiproverine
CAS:Dipiproverine is an alpha-amino acid ester, an antispasmodic compound. It is used as an anticholinergic drug.Formula:C20H30N2O2Color and Shape:SolidMolecular weight:330.46Ipramidil
CAS:Ipramidil (C80-1324) reveals marked dilator activity in the coronary circulation of isolated working hearts.Formula:C10H16N4O4Purity:98%Color and Shape:SolidMolecular weight:256.26CI-943
CAS:CI-943 is a novel potential antipsychotic drug that does not bind to dopamine (DA) receptors and has some developmental neurotoxicity.Formula:C12H17N5Purity:98%Color and Shape:SolidMolecular weight:231.3Meseclazone
CAS:Meseclazone has anti-inflammatory, analgesic, and antipyretic activity. Meseclazone shows inhibitory potency of secondary phase ADP aggregation.Formula:C11H10ClNO3Purity:98%Color and Shape:SolidMolecular weight:239.65L 657925
CAS:L 657925 is an antagonist of the thromboxane A2 receptor.Formula:C21H21ClFNO2Purity:98%Color and Shape:SolidMolecular weight:373.85E55888
CAS:E55888 is a potent and selective full agonist of the 5HT7 serotonin receptor.Formula:C16H23N3Color and Shape:SolidMolecular weight:257.37Etoperidone hydrochloride
CAS:Etoperidone hydrochloride is an antidepressant agent.Formula:C19H29Cl2N5OColor and Shape:SolidMolecular weight:414.37MRS1067
CAS:MRS1067 is an antagonist of A3 adenosine receptor.Formula:C19H16Cl2O3Color and Shape:SolidMolecular weight:363.23Ifoxetine sulfate
CAS:Ifoxetine sulfate, an atypical 5-HT inhibitor, may show unique therapeutic effects and side-effects.Formula:C13H19NO2H2O4SPurity:98%Color and Shape:SolidMolecular weight:270.34Tranterol hydrochloride
CAS:Tranterol, a β2-adrenergic receptor agonist, is used potentially for the treatment of asthma.Formula:C13H19Cl2F3N2OPurity:98%Color and Shape:SolidMolecular weight:347.2GW-876167
CAS:GW-876167, a 5-HT2C agonist, is used potentially for the treatment of obesity and glaucoma.Formula:C16H21N5O2Purity:98%Color and Shape:SolidMolecular weight:315.37Tilisolol HCl
CAS:Tilisolol, a nonselective beta-blocker, dilates dog coronary arteries via ATP-sensitive K(+) channels.Formula:C17H25ClN2O3Purity:98%Color and Shape:SolidMolecular weight:340.85Isoproterenol-d7 HCl
CAS:Isoproterenol-d7: internal standard for GC/LC-MS. β1-/β2-AR agonist, not for β3. Lowers blood pressure, tackles bradydysrhythmias, asthma.Formula:C11H18ClNO3Color and Shape:SolidMolecular weight:254.76L-771688
CAS:L-771688 (SNAP 6383) is a novel potent and selective α1A-adrenoceptor antagonist with a Ki value of 0.43±0.02 nM.L-771688 KE is used for the treatment of benignFormula:C28H33F2N5O5Purity:94.15%Color and Shape:SolidMolecular weight:557.59Masupirdine mesylate
CAS:Masupirdine mesylate (SUVN-502 mesylate) is a 5-HT6 receptor antagonist.Masupirdine mesylate is used to study neurological disorders such as Alzheimer's diseaseFormula:C23H32BrN3O9S3Purity:99.57%Color and Shape:SolidMolecular weight:670.61Odapipam
CAS:Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).Formula:C19H20ClNO2Purity:98%Color and Shape:SolidMolecular weight:329.82Napitane
CAS:napitane (A 75200) is a novel catecholamine uptake inhibitor with inhibitory effects on α-adrenergic receptors and potential antidepressant activity for the
Formula:C22H25NO2Purity:99.77% - 99.89%Color and Shape:SolidMolecular weight:335.44Methdilazine Hydrochloride
CAS:Methdilazine Hydrochloride (Bristaline) is a histamine H1 receptor antagonist for dermatologic conditions and relief of itching by allergies or rhinitis.Formula:C18H21ClN2SColor and Shape:Light-Tan Crystalline Powder 4 8-6 (Ntp 1992)Molecular weight:332.89RP73870
CAS:RP73870 is a gastrin/cholecystokinin-B receptor antagonist and H2 receptor antagonist with potent anti-ulcer activity.Formula:C27H30N4O7SPurity:98%Color and Shape:SolidMolecular weight:554.61PD 118717
CAS:PD 118717: a piperazinyl benzopyranone dopamine agonist with potential antipsychotic properties and no neurological side effects in tests.Formula:C20H22N4O3Purity:98%Color and Shape:SolidMolecular weight:366.41VL-0395
CAS:VL-0395 is an antagonist of CCK1 receptor.Formula:C25H21N3O4Purity:98%Color and Shape:SolidMolecular weight:427.45Ambenoxan hydrochloride
CAS:Ambenoxan hydrochloride is a centrally acting skeletal muscle relaxant.Formula:C14H22ClNO4Color and Shape:SolidMolecular weight:303.78VRX 03011 Potassium salt
CAS:VRX 03011, a 5-HT4 partial agonist, is used potentially for the treatment of Alzheimer's disease.Formula:C19H27KN3O3SPurity:98%Color and Shape:SolidMolecular weight:416.6Quinpirole
CAS:Quinpirole is a dopamine D2/D3 receptor agonist.Formula:C13H21N3Color and Shape:SolidMolecular weight:219.33Trimethaphan camsylate
CAS:Trimethaphan camsylate is a nicotinic antagonist that has been used as a ganglionic blocker in hypertension.Formula:C32H40N2O5S2Color and Shape:SolidMolecular weight:596.801DH-97
CAS:DH-97 is a potent MT2 melatonin receptor antagonist (pKi value = 8.03).Formula:C22H26N2OColor and Shape:SolidMolecular weight:334.45Glucagon Receptor Antagonist I
CAS:Glucagon antagonist I blocks the GCGR (IC50=181 nM), stops glucagon-induced glycogenolysis, and lowers glucose in glucagon-treated humanized mice.Formula:C20H30N2OSColor and Shape:SolidMolecular weight:346.53Toreforant
CAS:Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).Formula:C23H32N6Purity:98%Color and Shape:SolidMolecular weight:392.54TISCH
CAS:TISCH is a potent and selective iodinated ligand for CNS D1 dopamine receptor.Formula:C17H17ClINOColor and Shape:SolidMolecular weight:413.68A-971432
CAS:A-971432: selective S1P5 agonist, IC50 = 0.006 µM. Enhances blood-brain barrier, reduces Huntington’s symptoms in mice at 0.1 mg/kg.Formula:C18H17Cl2NO3Color and Shape:SolidMolecular weight:366.24(R)-Bambuterol
CAS:Bambuterol is a β2-agonist prodrug for asthma and COPD, taken daily, with a good safety profile and reduces plasma LDL-C and cholesterol.Formula:C18H29N3O5Color and Shape:SolidMolecular weight:367.44Thromboxane B2
CAS:Thromboxane B2 is a prostaglandin derivative that is released during anaphylaxis. Thromboxane B2 induces platelet aggregation and arterial contraction.Formula:C20H34O6Color and Shape:SolidMolecular weight:370.48YM-430
CAS:YM-430: β1 blocker & Ca²⁺ channel antagonist; antianginal & antihypertensive; IC50: 59.2 nM (rhythmic contractions), 36.6 mg/kg in rats (ST depression).Formula:C29H35N3O8Purity:98%Color and Shape:SolidMolecular weight:553.6RX821002
CAS:RX821002: potent α2-adrenoceptor antagonist, selective for α2D (pKd 9.7) over α2A (pKd 8.2), low affinity for imidazoline.Formula:C12H14N2O3Purity:98%Color and Shape:SolidMolecular weight:234.25(R)-Azelastine
CAS:(R)-Azelastine, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Formula:C22H24ClN3OColor and Shape:SolidMolecular weight:381.9Metitepine
CAS:Metitepine is a serotonin receptor antagonist in the CNS used as an antipsychotic.Formula:C20H24N2S2Color and Shape:SolidMolecular weight:356.555-OxoETE methyl ester
CAS:5-OxoETE methyl ester is a 5-oxoETE ester, an OXER1 agonist with stronger β-arrestin response, EC50 = 1.54 μM.Formula:C21H32O3Color and Shape:SolidMolecular weight:332.48GBR-13069 dimethanesulfonate
CAS:GBR-13069 dimethanesulfonate is a dopamine reuptake inhibitor.Formula:C30H38F2N2O7S2Color and Shape:SolidMolecular weight:640.76Oxypertine
CAS:Oxypertine, an indole-derived antipsychotic, treats psychoses like mania, schizophrenia, and severe anxiety, akin to chlorpromazine.Formula:C23H29N3O2Color and Shape:SolidMolecular weight:379.5Way 100135
CAS:WAY-100135: research drug, phenylpiperazine, potent 5-HT1A antagonist, partial 5-HT1D agonist, minor 5-HT1B activity.Formula:C24H33N3O2Color and Shape:SolidMolecular weight:395.54
