GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(251 products)
- Adrenergic Receptor(3,025 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(218 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(36 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 6011 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Protokylol
CAS:Protokylol is a β-adrenergic receptor agonist.Formula:C18H21NO5Purity:98%Color and Shape:SolidMolecular weight:331.36Reversan
CAS:Reversan(CBLC4H10) is a potent, nontoxic, and glioblastoma-associated inhibitor of multidrug resistance-associated protein 1 (MRP1) and P-glycoprotein (Pgp).Formula:C26H27N5O2Purity:99.05%Color and Shape:SolidMolecular weight:441.53Ref: TM-T12714
1mg44.00€1mL*10mM (DMSO)92.00€5mg93.00€10mg130.00€25mg250.00€50mg401.00€100mg640.00€200mg884.00€hGPR91 antagonist 3
CAS:hGPR91 antagonist 3 is an hGPR91 antagonist. hGPR91 antagonist 3 can be used to study diseases in hypertension and retinal angiogenesis.Formula:C23H18F4N4O2Purity:98.82% - 99.347%Color and Shape:SolidMolecular weight:458.41Ref: TM-T62858
1mg123.00€5mg295.00€1mL*10mM (DMSO)299.00€10mg490.00€25mg792.00€50mg1,071.00€100mg1,468.00€200mg1,972.00€FR 139317
CAS:highly potent and selective ETA endothelin receptor antagonistFormula:C33H44N6O5Purity:98%Color and Shape:SolidMolecular weight:604.74ASP1126
CAS:ASP1126 is a selective and orally active sphingosine-1-phosphate (S1P) agonist (EC50s: 7.12 nM, 517 nM for hS1P1 and hS1P3).Formula:C26H26ClF6NO5Purity:98%Color and Shape:SolidMolecular weight:581.93Butaclamol HCl
CAS:Butaclamol (AY-23,028), an unmarketed typical antipsychotic, is a research chemical that inhibits dopamine receptors.Formula:C25H32ClNOColor and Shape:SolidMolecular weight:397.98KY 234
CAS:KY 234 is a thromboxane synthetase antagonist.Formula:C33H35N5O2Color and Shape:SolidMolecular weight:533.676PNU-142633
CAS:PNU-142633: anti-migraine, selective 5-HT1D agonist, Ki=6 nM; >18,000 nM for 5-HT1B.Formula:C24H30N4O3Purity:98%Color and Shape:SolidMolecular weight:422.52APC-3316 tosylate
CAS:APC-3316 tosylate is a vinyl sulfone cysteine protease inhibitor and selective CCR4 antagonist.Formula:C39H46N4O7S2Color and Shape:SolidMolecular weight:746.94Benzoctamine
CAS:Benzoctamine: oral psychoactive with tranquillizing effects; boosts catecholamine turnover; enhances rat heart [3H]noradrenaline uptake.Formula:C18H19NColor and Shape:SolidMolecular weight:249.35Efpeglenatide
CAS:Efpeglenatide is a long-acting GLP-1 receptor agonist that improves insulin sensitivity, lowers blood glucose, delays weight gain, and supports metabolic disease research.Purity:100% - 100%Color and Shape:SolidVPC12249
CAS:VPC12249, a lysophosphatidic acid receptor type 1 (LPA1) antagonist, plays a functional role in osteoclast differentiation and bone resorption activity.Formula:C34H52NO6PColor and Shape:SolidMolecular weight:601.75A2AAR antagonist 1
CAS:Compound 21a, A2AAR antagonist with 20 nM Ki, useful in neurodegenerative disease study.Formula:C12H8BrN3OColor and Shape:SolidMolecular weight:290.12Alprenolol hydrochloride, (S)-
CAS:Alprenolol hydrochloride, (S)- is a nonselective β-blocker. It is also a serotonin 5HT1A receptor antagonist.Formula:C15H24ClNO2Color and Shape:SolidMolecular weight:285.81Carboprost
CAS:Carboprost (15(S)-15-Methyl Prostaglandin F2α) is a synthetic prostaglandin analogue of PGF2α which has the effect of oxytocic.Formula:C21H36O5Purity:98.18%Color and Shape:White Or Almost White PowderMolecular weight:368.51Ref: TM-T22285
1mg43.00€5mg110.00€1mL*10mM (DMSO)122.00€10mg166.00€25mg290.00€50mg425.00€100mg577.00€200mg778.00€Bifeprunox
CAS:Bifeprunox: potent antipsychotic, partial agonist at D2-like/5-HT1A receptors; treats schizophrenia.Formula:C24H23N3O2Purity:98%Color and Shape:SolidMolecular weight:385.46Apricoxib
CAS:Apricoxib: oral NSAID with antiangiogenic, antineoplastic properties; inhibits COX-2, may reduce tumor growth and angiogenesis.Formula:C19H20N2O3SColor and Shape:SolidMolecular weight:356.44S-22153
CAS:S22153 is an antagonist of melatonin receptor.Formula:C14H17NOSColor and Shape:SolidMolecular weight:247.36(1R,1'S,3'R/1R,1'R,3'S)-L-054,264
CAS:somatostatin sst2 receptor agonistFormula:C33H41N5O2Purity:98%Color and Shape:SolidMolecular weight:539.71(R)-(-)-α-Methylhistamine dihydrobromide
CAS:(R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).Formula:C6H13Br2N3Purity:99.98%Color and Shape:SolidMolecular weight:287GR 128107
CAS:GR 128107 is an antagonist of melatonin receptor.Formula:C16H20N2O2Color and Shape:SolidMolecular weight:272.34AZ-GHS-22
CAS:AZ-GHS-22, an inverse agonist for GHS-R1a (ghrelin receptor), binds with 0.77 nM IC50, cutting mice food intake by 54% at 100 mg/kg.Formula:C27H33ClN6O5S2Color and Shape:SolidMolecular weight:621.17Butaxamine
CAS:Butaxamine is a beta-2 selective adrenergic antagonist used mostly in animal and tissue experiments to characterize BETA-2 adrenergic receptors.Formula:C15H25NO3Purity:98%Color and Shape:SolidMolecular weight:267.36Trifluperidol HCl
CAS:Trifluperidol, a dopamine D2-receptor antagonist, is used to treat schizophrenia.Formula:C22H24ClF4NO2Color and Shape:SolidMolecular weight:445.88UK-9040
CAS:UK-9040 inhibits gastric secretory.Formula:C23H31NSPurity:98%Color and Shape:SolidMolecular weight:353.56Protokylol hydrochloride
CAS:Protokylol hydrochloride is a β-adrenergic agonist and bronchodilator, marketed as Asmetil, Caytine, Palison, Ventaire.Formula:C18H22ClNO5Color and Shape:SolidMolecular weight:367.83NBI-27914 hydrochloride
CAS:corticotropin-releasing factor1 (CRF1) receptor antagonistFormula:C18H21Cl5N4Purity:98%Color and Shape:SolidMolecular weight:470.65Midodrine (hydrochloride)
CAS:Midodrine hydrochloride ((±)-Midodrine hydrochloride) is an α1-receptor agonist used in the treatment of dysautonomia and orthostatic hypotension.Formula:C12H19ClN2O4Molecular weight:290.74SR-31747
CAS:SR-31747 blocks cell proliferation by inhibiting sterol isomerase. SR-31747 is a sigma ligand. It has immunosuppressive and anti-inflammatory properties.Formula:C23H35Cl2NPurity:98%Color and Shape:SolidMolecular weight:396.44AB-MECA
CAS:AB-MECA is a high affinity A3 adenosine receptor agonist. It has high affinity for recombinant A1 and A3 receptors.Formula:C18H21N7O4Purity:98%Color and Shape:SolidMolecular weight:399.4Landiolol
CAS:Landiolol is used as a highly cardioselective ultra short-acting beta-blocker.Formula:C25H39N3O8Purity:98%Color and Shape:White Crystalline PowderMolecular weight:509.59SV293
CAS:SV293 is a selective antagonist of D2 dopamine receptor.Formula:C22H26N2O2SPurity:98%Color and Shape:SolidMolecular weight:382.52(R)-DOI hydrochloride
CAS:(R)-DOI hydrochloride is the salt form of 2,5-Dimethoxy-4-iodoamphetamine (DOI), a potent 5-HT2A and 5-HT2C receptor agonist, orally active and hallucinogenic.Formula:C11H17ClINO2Purity:99.88% - >99.99%Color and Shape:SolidMolecular weight:357.62Bambuterol
CAS:long acting beta-adrenoceptor agonistFormula:C18H29N3O5Purity:98%Color and Shape:Off-White PowderMolecular weight:367.44SK1-I hydrochloride
CAS:SK1-I hydrochloride is a selective and competitive SphK1 inhibitor and sphingosine analog ,anti-leukemic to inhibit tumor cell growth and promote apoptosis.Formula:C17H28ClNO2Purity:99.80%Color and Shape:SolidMolecular weight:313.86TMPPAA
CAS:TMPPAA is an allosteric agonist of 5-HT3 receptor.Formula:C15H21NO2Purity:98%Color and Shape:SolidMolecular weight:247.33LY320135
CAS:CB1 receptor antagonist/inverse agonistFormula:C24H17NO4Purity:98%Color and Shape:SolidMolecular weight:383.4HAMI 3379
CAS:HAMI 3379 (HAMI3379) is a CysLT2 antagonist that attenuates brain damage and inhibits microglia inflammation following focal cerebral ischemia in rats.Formula:C34H45NO8Purity:99.75%Color and Shape:SolidMolecular weight:595.72RBI-257 Maleate
CAS:RBI-257 Maleate is a highly potent selective ligand of dopamine D4 receptor.Formula:C25H32IN3O5Color and Shape:SolidMolecular weight:581.44KUL-7211 racemate
CAS:KUL 7211, a selective β-adrenoceptor agonist, exists as a racemate, referred to as KUL 7211 racemate, which is the mixture of its enantiomers.Formula:C19H23NO5Purity:98%Color and Shape:SolidMolecular weight:345.39EA-230
CAS:Ea-230 is an immunomodulator that may be used in the treatment of renal failure.Formula:C15H27N5O6Color and Shape:SolidMolecular weight:373.4Adriforant hydrochloride
CAS:Adriforant hydrochloride is an antagonist of histamine H4 receptor.Formula:C13H25Cl3N6Purity:98%Color and Shape:SolidMolecular weight:371.74Amosulalol, (-)-
CAS:Amosulalol, (-)-, is an adrenergic agent.Formula:C18H24N2O5SColor and Shape:SolidMolecular weight:380.462-Arachidonoylglycerol
CAS:In the central nervous system, 2-Arachidonoylglycerol is a second endogenous cannabinoid ligandFormula:C23H38O4Purity:95%Color and Shape:LiquidMolecular weight:378.55Benzamide Derivative 1
CAS:Benzamide Derivative 1 Benzamide derivative with gastrokinetic activity.Benzamide Derivative 1 can be used in the study of gastrointestinal diseases.Formula:C22H34ClN3O3Purity:>99.99%Color and Shape:SolidMolecular weight:423.98PNU-96415E
CAS:dopamine D4 and serotonergic 5-HT2A receptor antagonistFormula:C21H27Cl2FN2OPurity:98%Color and Shape:SolidMolecular weight:413.36ZD 7114 hydrochloride
CAS:β3-adrenoceptor agonistFormula:C22H31ClN2O6Purity:98%Color and Shape:SolidMolecular weight:454.94Clenproperol
CAS:Clenproperol is a β2-adrenergic agonist.Formula:C11H16Cl2N2OColor and Shape:SolidMolecular weight:263.16Efaroxan hydrochloride
CAS:Efaroxan hydrochloride a selective, oral α2-adrenoceptor antagonist significantly potentiates adrenaline-induced increases in insulin levels.Formula:C13H17ClN2OPurity:98%Color and Shape:SolidMolecular weight:252.74BPIPP
CAS:guanylyl cyclase (GC) and adenylyl cyclase (AC) inhibitorFormula:C22H16BrN3O3Purity:98%Color and Shape:SolidMolecular weight:450.28
