GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,023 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5986 products of "GPCR/G-Protein"
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VUF 5681 dihydrobromide
CAS:histamine H3 receptor silent antagonistFormula:C11H21Br2N3Purity:98%Color and Shape:SolidMolecular weight:355.11PF-06412154 HCl
CAS:PF-06412154 HCl is a glucagon receptor antagonist.Formula:C24H28ClN3O3Color and Shape:SolidMolecular weight:441.96L-775,606
CAS:L-775,606 is a selective agonist of 5-hydroxytryptamine 1D.Formula:C25H29FN6Purity:98%Color and Shape:SolidMolecular weight:432.54Bunaprolast
CAS:Bunaprolast (U66858) is a novel and potent leukotriene B4 (LTB4) inhibitor.Bunaprolast exhibits oxidative degradation activity and inhibits lipoxygenase andFormula:C17H20O3Purity:>99.99%Color and Shape:SolidMolecular weight:272.34VUF 8430
CAS:VUF 8430 is a selective agonist for the H4 receptor.Formula:C4H11N5SPurity:98%Color and Shape:SolidMolecular weight:161.23L 741742 hydrochloride
CAS:L 741742 hydrochloride is a selective, high-affinity human D4 receptor antagonist with good oral bioavailability and brain penetration.Formula:C23H26Cl2N2OPurity:99.9%Color and Shape:SolidMolecular weight:417.37Amosulalol, (+)-
CAS:Amosulalol, (+)-, is an adrenergic agent.Formula:C18H24N2O5SColor and Shape:SolidMolecular weight:380.46CP-122721
CAS:CP-122721: NK1 receptor blocker, has antidepressant, anti-anxiety, antiemetic effects, and selectively inhibits substance P receptors.Formula:C20H23F3N2O2Color and Shape:SolidMolecular weight:380.4Protokylol
CAS:Protokylol is a β-adrenergic receptor agonist.Formula:C18H21NO5Purity:98%Color and Shape:SolidMolecular weight:331.36YM-430
CAS:YM-430: β1 blocker & Ca²⁺ channel antagonist; antianginal & antihypertensive; IC50: 59.2 nM (rhythmic contractions), 36.6 mg/kg in rats (ST depression).Formula:C29H35N3O8Purity:98%Color and Shape:SolidMolecular weight:553.6Trimazosin hydrochloride
CAS:Trimazosin hydrochloride is used in the treatment of hypertensive patients failing to respond to thiazides.Formula:C20H32ClN5O7Color and Shape:SolidMolecular weight:489.95mCPBG
CAS:mCPBG is a potent high affinity agonist of 5-HT3 receptor.Formula:C8H10ClN5Color and Shape:SolidMolecular weight:211.65ChemR23-IN-2
CAS:ChemR23-IN-2 is a potent, orally active inhibitor of ChemR23 (IC50: 3.2 nM).Formula:C29H26N4O5Color and Shape:SolidMolecular weight:510.54BRL 44408 Maleate Salt
CAS:BRL 44408 Maleate is an α2A-adrenoceptor antagonist with antidepressant and analgesic activity.Formula:C17H21N3O4Purity:98.71%Color and Shape:SolidMolecular weight:331.37(R)-Azelastine
CAS:(R)-Azelastine, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Formula:C22H24ClN3OColor and Shape:SolidMolecular weight:381.9Metitepine
CAS:Metitepine is a serotonin receptor antagonist in the CNS used as an antipsychotic.Formula:C20H24N2S2Color and Shape:SolidMolecular weight:356.55Butopamine
CAS:Butopamine differs from dobutamine in location of only one hydroxyl group, but is no longer a catecholamine.Formula:C18H23NO3Color and Shape:SolidMolecular weight:301.385-OxoETE methyl ester
CAS:5-OxoETE methyl ester is a 5-oxoETE ester, an OXER1 agonist with stronger β-arrestin response, EC50 = 1.54 μM.Formula:C21H32O3Color and Shape:SolidMolecular weight:332.48Bifeprunox
CAS:Bifeprunox: potent antipsychotic, partial agonist at D2-like/5-HT1A receptors; treats schizophrenia.Formula:C24H23N3O2Purity:98%Color and Shape:SolidMolecular weight:385.46Apricoxib
CAS:Apricoxib: oral NSAID with antiangiogenic, antineoplastic properties; inhibits COX-2, may reduce tumor growth and angiogenesis.Formula:C19H20N2O3SColor and Shape:SolidMolecular weight:356.44Ethiazide
CAS:Ethiazide is a benzothiadiazine sulfonamide derivative belonging to the class of the thiazide diuretics.Formula:C9H12ClN3O4S2Color and Shape:SolidMolecular weight:325.79PF 10040
CAS:PF 10040 is an antagonist of platelet activating factor (PAF).Formula:C20H24ClNO2Color and Shape:SolidMolecular weight:345.86(1R,1'S,3'R/1R,1'R,3'S)-L-054,264
CAS:somatostatin sst2 receptor agonistFormula:C33H41N5O2Purity:98%Color and Shape:SolidMolecular weight:539.71Fertirelin acetate
CAS:Fertirelin acetate is a gonadotropin-releasing hormone (GnRH) agonist.Formula:C55H74N16O13Color and Shape:SolidMolecular weight:1167.29Oxypertine
CAS:Oxypertine, an indole-derived antipsychotic, treats psychoses like mania, schizophrenia, and severe anxiety, akin to chlorpromazine.Formula:C23H29N3O2Color and Shape:SolidMolecular weight:379.5Butaxamine
CAS:Butaxamine is a beta-2 selective adrenergic antagonist used mostly in animal and tissue experiments to characterize BETA-2 adrenergic receptors.Formula:C15H25NO3Purity:98%Color and Shape:SolidMolecular weight:267.36L-694,247
CAS:L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E receptors, and can be used to study neurological diseases.Formula:C20H21N5O3SPurity:98.36%Color and Shape:White SolidMolecular weight:411.48Way 100135
CAS:WAY-100135: research drug, phenylpiperazine, potent 5-HT1A antagonist, partial 5-HT1D agonist, minor 5-HT1B activity.Formula:C24H33N3O2Color and Shape:SolidMolecular weight:395.54Q8 hydrochloride
CAS:Q8 is an antagonist of cysteinyl leukotreine receptor. Q8 inhibits VEGF-independent angiogenesis.Formula:C17H14ClNO2Purity:98%Color and Shape:SolidMolecular weight:299.75UK-9040
CAS:UK-9040 inhibits gastric secretory.Formula:C23H31NSPurity:98%Color and Shape:SolidMolecular weight:353.56AUY-954 free base
CAS:AUY-954 is a selective S1P(1) modulator reducing EAN inflammation and demyelination in rats.Formula:C25H20F3NO2SColor and Shape:SolidMolecular weight:455.49Protokylol hydrochloride
CAS:Protokylol hydrochloride is a β-adrenergic agonist and bronchodilator, marketed as Asmetil, Caytine, Palison, Ventaire.Formula:C18H22ClNO5Color and Shape:SolidMolecular weight:367.83Clopenthixol
CAS:Clopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.Formula:C22H25ClN2OSColor and Shape:SolidMolecular weight:400.96Paltusotine HCl
CAS:Paltusotine, also known as CRN00808, is a somatostatin receptor agonist.Formula:C27H24Cl2F2N4OColor and Shape:SolidMolecular weight:529.41NBI-27914 hydrochloride
CAS:corticotropin-releasing factor1 (CRF1) receptor antagonistFormula:C18H21Cl5N4Purity:98%Color and Shape:SolidMolecular weight:470.65SR-31747
CAS:SR-31747 blocks cell proliferation by inhibiting sterol isomerase. SR-31747 is a sigma ligand. It has immunosuppressive and anti-inflammatory properties.Formula:C23H35Cl2NPurity:98%Color and Shape:SolidMolecular weight:396.44WRC-0571
CAS:WRC-0571 is a highly potent, selective antagonist of A1 adenosine receptors.Formula:C17H26N6OPurity:98%Color and Shape:SolidMolecular weight:330.43Landiolol
CAS:Landiolol is used as a highly cardioselective ultra short-acting beta-blocker.Formula:C25H39N3O8Purity:98%Color and Shape:White Crystalline PowderMolecular weight:509.59Bambuterol
CAS:long acting beta-adrenoceptor agonistFormula:C18H29N3O5Purity:98%Color and Shape:Off-White PowderMolecular weight:367.44ChemR23-IN-4
CAS:ChemR23-IN-4 is a potent inhibitor of orally active ChemR23, capable of acting on human ChemR23 (IC50: 17 nM).Formula:C27H26N6O3Color and Shape:SolidMolecular weight:482.53TMPPAA
CAS:TMPPAA is an allosteric agonist of 5-HT3 receptor.Formula:C15H21NO2Purity:98%Color and Shape:SolidMolecular weight:247.33CM304
CAS:CM304 is a highly selective sigma-1 receptor antagonist.Formula:C18H26ClFN2OSColor and Shape:SolidMolecular weight:372.93Elzasonan
CAS:Elzasonan is a selective 5-hydroxytryptamine 1B receptor antagonist used to treat patients with major depressive disorder and obsessive compulsive disorder.Formula:C22H23Cl2N3OSColor and Shape:SolidMolecular weight:448.41Adriforant hydrochloride
CAS:Adriforant hydrochloride is an antagonist of histamine H4 receptor.Formula:C13H25Cl3N6Purity:98%Color and Shape:SolidMolecular weight:371.74PNU-96415E
CAS:dopamine D4 and serotonergic 5-HT2A receptor antagonistFormula:C21H27Cl2FN2OPurity:98%Color and Shape:SolidMolecular weight:413.36ZD 7114 hydrochloride
CAS:β3-adrenoceptor agonistFormula:C22H31ClN2O6Purity:98%Color and Shape:SolidMolecular weight:454.94GSK-269984A
CAS:GSK-269984A is an antagonist of Prostaglandin E2 Receptor 1 (EP1) (pIC50: 7.9).Formula:C20H14Cl2FNNaO3Purity:98%Color and Shape:SolidMolecular weight:429.22Usmarapride free base
CAS:Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.Formula:C21H29N5O2Purity:99.91% - 99.91%Color and Shape:SolidMolecular weight:383.49Cirazoline (free base)
CAS:Cirazoline: full α1A agonist, partial α1B/D, nonselective α2 antagonist; potential vasoconstrictor.Formula:C13H16N2OColor and Shape:SolidMolecular weight:216.28ST-836
CAS:ST-836 is a dopamine receptor ligand; Antiparkinsonian agent .Formula:C23H34N4OSPurity:98%Color and Shape:SolidMolecular weight:414.61
