GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,023 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5986 products of "GPCR/G-Protein"
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Cicloprolol hydrochloride
CAS:Cicloprolol hydrochloride is a new potent and selective beta 1-adrenoceptor antagonist with partial agonist activity for the study of coronary heart disease.Formula:C18H30ClNO4Purity:97.26%Color and Shape:SolidMolecular weight:359.89Bamirastine
CAS:Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect onFormula:C31H37N5O3Purity:96.68%Color and Shape:SolidMolecular weight:527.66(4E)-SUN9221
CAS:(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity inFormula:C25H31FN4O3Purity:97.79%Color and Shape:SolidMolecular weight:454.54L-771688
CAS:L-771688 (SNAP 6383) is a novel potent and selective α1A-adrenoceptor antagonist with a Ki value of 0.43±0.02 nM.L-771688 KE is used for the treatment of benignFormula:C28H33F2N5O5Purity:94.15%Color and Shape:SolidMolecular weight:557.59ONO4057
CAS:ONO4057 is a potent and orally active Leukotriene B4 receptor antagonist with an IC50 value of 0.7±0.3 μM.Formula:C27H34O7Purity:>99.99%Color and Shape:SolidMolecular weight:470.55L-803087
CAS:L-803087: potent sst4 receptor agonist, 0.7 nM Ki, 280x selectivity, boosts AMPA responses & seizures in mice.Formula:C25H29F2N5O3Purity:99.37%Color and Shape:SolidMolecular weight:485.53Ref: TM-T11800
1mg50.00€5mg112.00€1mL*10mM (DMSO)126.00€10mg175.00€25mg366.00€50mg585.00€100mg928.00€200mg1,234.00€TD-5471 hydrochloride
CAS:TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (Formula:C32H32ClN3O4Purity:99.57%Color and Shape:SolidMolecular weight:558.07Odapipam
CAS:Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).Formula:C19H20ClNO2Purity:98%Color and Shape:SolidMolecular weight:329.82Napitane
CAS:napitane (A 75200) is a novel catecholamine uptake inhibitor with inhibitory effects on α-adrenergic receptors and potential antidepressant activity for the
Formula:C22H25NO2Purity:99.77% - 99.89%Color and Shape:SolidMolecular weight:335.44Norfenefrine HCl
CAS:Norfenefrine HCl is an α1-adrenergic receptor agonist, an endogenous neurotransmitter and sympathomimetic drug for hypotension,glycerol adipose.Formula:C8H12ClNO2Purity:99.44%Color and Shape:SolidMolecular weight:189.64Propiomazine HCl
CAS:Propiomazine HCl is an analgesia adjunct.Formula:C20H25ClN2OSColor and Shape:SolidMolecular weight:376.94Daledalin tosylate
CAS:Daledalin tosylate is an antidepressant.Formula:C26H32N2O3SColor and Shape:SolidMolecular weight:452.61PD 118717
CAS:PD 118717: a piperazinyl benzopyranone dopamine agonist with potential antipsychotic properties and no neurological side effects in tests.Formula:C20H22N4O3Purity:98%Color and Shape:SolidMolecular weight:366.41SKF-80723 HBr
CAS:SKF-80723 HBr is a potent D1 agonist enhancing quinpirole-induced circling in 6-OHDA lesioned rats.Formula:C16H16BrNO2Purity:98%Color and Shape:SolidMolecular weight:334.21Trebenzomine
CAS:Trebenzomine is apsychotropic agent with potential as an antidepressant and an antipsychotic.Formula:C12H17NOPurity:98%Color and Shape:SolidMolecular weight:191.27Argiprestocin
CAS:Argiprestocin: antidiuretic, regulates osmolality, neurohypophysial hormone, vasoconstrictor.Formula:C43H67N15O12S2Purity:99.34%Color and Shape:SolidMolecular weight:1050.22Mabuterol, (S)-
CAS:Mabuterol, a β2 adrenoreceptor agonist, lowers rat blood pressure and boosts guinea pig heart rate/force, not affecting other receptors.Formula:C13H18ClF3N2OColor and Shape:SolidMolecular weight:310.74Colterol HCl
CAS:Colterol HCl, a β2-adrenoceptor agonist salt, is used for bronchospasm in asthma and COPD.Formula:C12H20ClNO3Color and Shape:SolidMolecular weight:261.75Ambucetamide
CAS:Ambucetamide is an antispasmodic, it may inhibit or diminish the spontaneous rhythmical activity of the human myometrium.Formula:C17H28N2O2Color and Shape:SolidMolecular weight:292.42BAY-386
CAS:BAY-386 is a PAR1 receptor inhibitor which suppresses activation of thrombin and platelet activity.Formula:C22H25F3N4O5SColor and Shape:SolidMolecular weight:514.52VUF14738
CAS:VUF14738 is a robust and fatigue-resistant photoswitchable GPCR antagonist.Formula:C25H32N4O2Color and Shape:SolidMolecular weight:420.55Albuterol adipate
CAS:Albuterol adipate, a β2-AR agonist salt, treats asthma/COPD, with high selectivity for pulmonary over cardiac receptors.Formula:C32H52N2O10Color and Shape:SolidMolecular weight:624.77Aceprometazine
CAS:Aceprometazine (1664CB) is an antipsychotic which is orally active. Aceprometazine can be used in psychiatric disorders research, for example, depression [1].Formula:C19H22N2OSColor and Shape:SolidMolecular weight:326.46GBR-12935 maleate
CAS:GBR-12935: dopamine reuptake inhibitor, used in research for Parkinson's and brain's dopamine pathways.Formula:C32H38N2O5Color and Shape:SolidMolecular weight:530.665Thiothixene hydrochloride
CAS:Thiothixene hydrochloride is an antipsychotic agent that can be used in the study of schizophrenia and bipolar mania.Formula:C23H30ClN3O2S2Color and Shape:SolidMolecular weight:480.08Isoetharine hydrochloride
CAS:Isoetharine HCl, a selective, short-acting oral β-agonist, is used as a bronchodilator for inhalation therapy.Formula:C13H22ClNO3Color and Shape:SolidMolecular weight:275.77Ro 23-3423
CAS:Ro 23-3423 is a specific inhibitor of thromboxane synthetase.Formula:C23H22N4O2Color and Shape:SolidMolecular weight:386.45Dicentrine HCl
CAS:Dicentrine HCl is the salt form of Dicentrine, an alpha 1-adrenoceptor antagonist effective against human hyperplastic prostates.Formula:C20H22ClNO4Color and Shape:SolidMolecular weight:375.85Bitolterol
CAS:Bitolterol is a new beta 2-adrenergic agonist and classified as a pro-drug.Formula:C28H31NO5Color and Shape:SolidMolecular weight:461.555-HT4 antagonist 1
CAS:5-HT4 antagonist 1 is an antagonist of 5-HT4 (pKi = 9.6).Formula:C23H36N4O5SPurity:99.75%Color and Shape:SolidMolecular weight:480.62Sch 44643
CAS:Sch 44643 is an antagonist of platelet activating factor with oral activity.Formula:C25H22ClN3O2Color and Shape:SolidMolecular weight:431.91VER-3323
CAS:VER-3323 is a selective agonist for the 5-HT2B and 5-HT2C serotonin receptor with potent anorectic effects in animal studies.Formula:C11H15BrN2Purity:98%Color and Shape:SolidMolecular weight:255.15U 101958
CAS:U 101958 is a putative antipsychotic agent It is also a highly selective dopamine D4 receptor antagonist.Formula:C20H27N3OColor and Shape:SolidMolecular weight:325.45Toreforant
CAS:Toreforant is an effective and selective histamine H4 receptor antagonist (Ki at the human receptor: 8.4 nM).Formula:C23H32N6Purity:98%Color and Shape:SolidMolecular weight:392.54TISCH
CAS:TISCH is a potent and selective iodinated ligand for CNS D1 dopamine receptor.Formula:C17H17ClINOColor and Shape:SolidMolecular weight:413.68Zimelidine
CAS:Zimelidine, a withdrawn antidepressant, posed Guillain-Barre risk.Formula:C16H17BrN2Purity:98%Color and Shape:SolidMolecular weight:317.22RP-72540
CAS:RP-72540: CCKB receptor blocker, 200x more selective for CCKA, binds to stomach gastrin, limits [3H]pCCK-8 in mouse brain, <0.01% reaches forebrain.Formula:C28H30N4O6Purity:98%Color and Shape:SolidMolecular weight:518.56(R)-Bambuterol
CAS:Bambuterol is a β2-agonist prodrug for asthma and COPD, taken daily, with a good safety profile and reduces plasma LDL-C and cholesterol.Formula:C18H29N3O5Color and Shape:SolidMolecular weight:367.44Carbuterol hydrochloride
CAS:Carbuterol hydrochloride is a short-acting β2 adrenoreceptor agonist.Formula:C13H22ClN3O3Color and Shape:SolidMolecular weight:303.79PF-06412154 HCl
CAS:PF-06412154 HCl is a glucagon receptor antagonist.Formula:C24H28ClN3O3Color and Shape:SolidMolecular weight:441.96Thromboxane B2
CAS:Thromboxane B2 is a prostaglandin derivative that is released during anaphylaxis. Thromboxane B2 induces platelet aggregation and arterial contraction.Formula:C20H34O6Color and Shape:SolidMolecular weight:370.48Amosulalol, (+)-
CAS:Amosulalol, (+)-, is an adrenergic agent.Formula:C18H24N2O5SColor and Shape:SolidMolecular weight:380.46CP-122721
CAS:CP-122721: NK1 receptor blocker, has antidepressant, anti-anxiety, antiemetic effects, and selectively inhibits substance P receptors.Formula:C20H23F3N2O2Color and Shape:SolidMolecular weight:380.4Z-335 sodium
CAS:Z-335 Salt, a thromboxane A2 receptor antagonist, is used potentially for the treatment of arterial occlusive disease.Formula:C18H18ClNNaO4SColor and Shape:SolidMolecular weight:402.84NGD 98-2
CAS:NGD 98-2 is a new generation, topology 2 selective orally active corticotropin releasing factor-1 (CRF-1) receptor antagonist.Formula:C19H24F3N3O3Color and Shape:SolidMolecular weight:399.41Trimazosin hydrochloride
CAS:Trimazosin hydrochloride is used in the treatment of hypertensive patients failing to respond to thiazides.Formula:C20H32ClN5O7Color and Shape:SolidMolecular weight:489.95mCPBG
CAS:mCPBG is a potent high affinity agonist of 5-HT3 receptor.Formula:C8H10ClN5Color and Shape:SolidMolecular weight:211.65ChemR23-IN-2
CAS:ChemR23-IN-2 is a potent, orally active inhibitor of ChemR23 (IC50: 3.2 nM).Formula:C29H26N4O5Color and Shape:SolidMolecular weight:510.54TP-680
CAS:TP-680 is a antagonist of cholecystokininA receptor.Formula:C35H33N5O4SPurity:98%Color and Shape:SolidMolecular weight:619.73Mivazerol
CAS:Mivazerol is an alpha 2-adrenoceptor agonist.Formula:C11H11N3O2Color and Shape:SolidMolecular weight:217.22
