GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,018 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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ADX-10061
CAS:ADX-10061 is a dopamine D1 receptor antagonist.Formula:C19H20N2O4Color and Shape:SolidMolecular weight:340.37Albuterol adipate
CAS:Albuterol adipate, a β2-AR agonist salt, treats asthma/COPD, with high selectivity for pulmonary over cardiac receptors.Formula:C32H52N2O10Color and Shape:SolidMolecular weight:624.77CP 96345
CAS:CP 96345 is a NK1 receptor antagonist.Formula:C28H32N2OPurity:98%Color and Shape:SolidMolecular weight:412.57Gastrazole free acid
CAS:Gastrazole is a CCK2 receptor antagonist potentially. It also used for the treatment of pancreatic cancer.Formula:C34H34FN5O7Purity:98%Color and Shape:SolidMolecular weight:643.66Levomoprolol
CAS:Levomoprolol, (S)-enantiomer of the moprololis, is a beta adrenergic antagonist.Formula:C13H21NO3Purity:98%Color and Shape:SolidMolecular weight:239.31GAT228
CAS:GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].Formula:C22H18N2O2Color and Shape:SolidMolecular weight:342.39mCPBG
CAS:mCPBG is a potent high affinity agonist of 5-HT3 receptor.Formula:C8H10ClN5Color and Shape:SolidMolecular weight:211.65L-771688 dihydrochloride
CAS:L-771688 is an α1A-adrenoceptor antagonist potentially for the treatment of benign prostatic hyperplasia.Formula:C28H35Cl2F2N5O5Purity:98%Color and Shape:SolidMolecular weight:630.51SNAP 5089
CAS:α1A-adrenoceptor antagonistFormula:C36H40N4O5Purity:98%Color and Shape:SolidMolecular weight:608.73Dacopafant
CAS:Dacopafant is an antagonist of platlet activationg factor receptor.Formula:C12H11N3OSColor and Shape:SolidMolecular weight:245.3ChemR23-IN-2
CAS:ChemR23-IN-2 is a potent, orally active inhibitor of ChemR23 (IC50: 3.2 nM).Formula:C29H26N4O5Color and Shape:SolidMolecular weight:510.54BN 50341
CAS:BN 50341 is an inhibitor of antithrombotic platelet activating factor.Formula:C32H41ClN2O4Purity:98%Color and Shape:SolidMolecular weight:553.13PD 81723
CAS:Allosteric potentiator at the adenosine A1 receptorFormula:C14H12F3NOSPurity:98%Color and Shape:SolidMolecular weight:299.31TP-680
CAS:TP-680 is a antagonist of cholecystokininA receptor.Formula:C35H33N5O4SPurity:98%Color and Shape:SolidMolecular weight:619.73SKF 86466 hydrochloride
CAS:SKF 86466 hydrochloride is an α2-adrenoceptor antagonist.Formula:C11H15Cl2NPurity:98%Color and Shape:SolidMolecular weight:232.15Nor-SCH-12679 Maleate
CAS:Nor-SCH-12679 Maleate is a D1-dopamine receptor antagonist.Formula:C22H25NO6Purity:98%Color and Shape:SolidMolecular weight:399.44SB 258585 hydrochloride
CAS:SB 258585 hydrochloride is a 5-HT6 receptor antagonist.Formula:C18H23ClIN3O3SPurity:98%Color and Shape:SolidMolecular weight:523.82Impromidine
CAS:Impromidine is a highly potent and specific agonist of the histamine H2 receptor.Formula:C14H23N7SPurity:98%Color and Shape:SolidMolecular weight:321.44DR-4004
CAS:DR-4004 is a selective serotonin 5-HT7 receptor antagonist.Formula:C26H30N2OColor and Shape:SolidMolecular weight:386.53Dipiproverine
CAS:Dipiproverine is an alpha-amino acid ester, an antispasmodic compound. It is used as an anticholinergic drug.Formula:C20H30N2O2Color and Shape:SolidMolecular weight:330.46Ipramidil
CAS:Ipramidil (C80-1324) reveals marked dilator activity in the coronary circulation of isolated working hearts.Formula:C10H16N4O4Purity:98%Color and Shape:SolidMolecular weight:256.26Fertirelin acetate
CAS:Fertirelin acetate is a gonadotropin-releasing hormone (GnRH) agonist.Formula:C55H74N16O13Color and Shape:SolidMolecular weight:1167.29SKF-82958
CAS:SKF 82958 is a D1/D5 receptor full agonist.Formula:C19H20ClNO2Purity:98%Color and Shape:SolidMolecular weight:329.82AZD-1678
CAS:AZD-1678 is a potent CCR4 receptor antagonist.Formula:C11H8Cl2FN3O3SColor and Shape:SolidMolecular weight:352.17CI-943
CAS:CI-943 is a novel potential antipsychotic drug that does not bind to dopamine (DA) receptors and has some developmental neurotoxicity.Formula:C12H17N5Purity:98%Color and Shape:SolidMolecular weight:231.3Metitepine
CAS:Metitepine is a serotonin receptor antagonist in the CNS used as an antipsychotic.Formula:C20H24N2S2Color and Shape:SolidMolecular weight:356.55VUF8507
CAS:Vuf8507 is an allosteric regulator of adenosine receptor.Formula:C21H15N3OColor and Shape:SolidMolecular weight:325.36L 646462
CAS:L 646462 is an antidopaminergic agent.Formula:C27H27N3O4Purity:98%Color and Shape:SolidMolecular weight:457.52Umespirone
CAS:Umespirone is a potential antipsychotic/anxiolytic drug of the azapirone class. It possesses anxiolytic and antipsychotic properties.Formula:C28H40N4O5Purity:98%Color and Shape:SolidMolecular weight:512.64SNAP-5089
CAS:SNAP-5089 is a highly selective alpha1A-adrenoceptor antagonist.Formula:C36H41ClN4O5Color and Shape:SolidMolecular weight:645.2L 641953
CAS:L 641953 is an antagonist of the thromboxane receptor.Formula:C15H9FO3SColor and Shape:SolidMolecular weight:288.29Pancopride
CAS:Pancopride（LAS 30451） is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen mustard and dacarbazine-inducedFormula:C18H24ClN3O2Purity:93.64%Color and Shape:SolidMolecular weight:349.86Piclozotan
CAS:Piclozotan (anhydrous), a 5-HT1A receptor agonist, demonstrated significant neuroprotective activity in a transient middle cerebral artery occlusion (t-MCAO)Formula:C23H24ClN3O2Purity:98.59%Color and Shape:SolidMolecular weight:409.91RS 79948 hydrochloride
CAS:α2-adrenoreceptor antagonistFormula:C19H29ClN2O3SPurity:98%Color and Shape:SolidMolecular weight:400.96Hedgehog Antagonist VIII
CAS:Hh antagonist VIII is a quinazolinyl-urea that inhibits Gli transcription in the Hh pathway, linked to cancer, with an IC50 of 70 nM.Formula:C23H15ClF4N4O2Color and Shape:SolidMolecular weight:490.84CAY10397
CAS:CAY10397, a selective inhibitor of 15-hydroxy PGDH, significantly suppresses endogenous 11-oxo-ETE production with a corresponding increase in 11(R)-HETE.Formula:C17H16N2O5Color and Shape:SolidMolecular weight:328.32SC-41930
CAS:SC-41930 is a potent and selective antagonist of leukotriene B4 receptor.Formula:C28H36O7Color and Shape:SolidMolecular weight:484.58LEK 8841
CAS:LEK 8841 is an ergoline derivative that is a potential antipsychotic.Formula:C21H24BrN3O4SPurity:98%Color and Shape:SolidMolecular weight:494.4(R)-(+)-8-Hydroxy-DPAT hydrobromide
CAS:5-HT1A serotonin receptor agonistFormula:C16H26BrNOPurity:98%Color and Shape:SolidMolecular weight:328.29SKF 77434 hydrobromide
CAS:SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.Formula:C19H22BrNO2Purity:98%Color and Shape:SolidMolecular weight:376.29L 659989
CAS:L 659989 is an antagonist of the Platelet-activating factor receptor.Formula:C24H32O8SPurity:98%Color and Shape:SolidMolecular weight:480.57Isothipendyl hydrochloride
CAS:Isothipendyl hydrochloride is a 1st generation H1 antagonist.Formula:C16H20ClN3SColor and Shape:SolidMolecular weight:321.87CB2R agonist 1
CAS:CB2R agonist 1 selectively binds human CB2R, EC50 of 0.56 µM, modulates inflammatory cytokines.Formula:C22H32N2OColor and Shape:SolidMolecular weight:340.5CP19
CAS:CP19 blocks histamine receptors; inhibits EBOV and MARV with IC50s of 3.4 μM and 29.5 μM, respectively; antiviral [1].Formula:C26H30N2O5Color and Shape:SolidMolecular weight:450.53S-14671
CAS:S-14671: 5-HT1A agonist (pKi 9.3), potent in vivo; 5-HT2A/2C antagonist (pKi 7.8).Formula:C22H25N3O2SColor and Shape:SolidMolecular weight:395.52Napamezole
CAS:Napamezole: α2 adrenergic receptor antagonist, blocks α1 in rat vas deferens (Kb 135 nM), reverses clonidine effects on twitch height.Formula:C14H16N2Purity:98%Color and Shape:SolidMolecular weight:212.29Flestolol sulfate
CAS:Flestolol sulfate is an anti-adrenergic beta-receptor.Formula:C15H24FN3O8SColor and Shape:SolidMolecular weight:425.43Phenindamine Tartrate
CAS:Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.Formula:C23H25NO6Color and Shape:SolidMolecular weight:411.45412(S)-hydroxy-16-Heptadecynoic Acid
CAS:The compound is a mechanism-based inhibitor of cytochrome P450 ω-hydroxylase.Formula:C17H30O3Purity:98%Color and Shape:SolidMolecular weight:282.42Loratadine N-oxide
CAS:Loratadine N-oxide is a metabolite of the histamine H1 receptor inverse agonist loratadine.Formula:C22H23ClN2O3Color and Shape:SolidMolecular weight:398.88
