GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,018 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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ABT-299
CAS:ABT-299 is a prodrug of A-85783.Formula:C32H28ClFN4O4SColor and Shape:SolidMolecular weight:619.11PPTN Mesylate
CAS:PPTN Mesylate is an effective and highly selective antagonist of the P2Y14 receptor.Formula:C30H28F3NO5SPurity:98%Color and Shape:SolidMolecular weight:571.61MRS1067
CAS:MRS1067 is an antagonist of A3 adenosine receptor.Formula:C19H16Cl2O3Color and Shape:SolidMolecular weight:363.23MM-22
CAS:biotinylated anandamide analog acts as a probe for visualizing the accumulation and intracellular trafficking of anandamideFormula:C36H60N4O5SPurity:98%Color and Shape:SolidMolecular weight:660.95Ifoxetine sulfate
CAS:Ifoxetine sulfate, an atypical 5-HT inhibitor, may show unique therapeutic effects and side-effects.Formula:C13H19NO2H2O4SPurity:98%Color and Shape:SolidMolecular weight:270.34Butaclamol free base
CAS:Butaclamol is a typical antipsychotic which was never marketed. It also acts as a dopamine receptor antagonist.Formula:C25H31NOPurity:98%Color and Shape:SolidMolecular weight:361.52Tranterol hydrochloride
CAS:Tranterol, a β2-adrenergic receptor agonist, is used potentially for the treatment of asthma.Formula:C13H19Cl2F3N2OPurity:98%Color and Shape:SolidMolecular weight:347.2S(-)-8-Hydroxy-DPAT hydrobromide
CAS:S(-)-8-Hydroxy-DPAT hydrobromide is an agonist of 5-HT1A serotonin receptor.Formula:C16H26BrNOPurity:98%Color and Shape:SolidMolecular weight:328.29PD 118440
CAS:PD 118440 is a Dopamine antagonist. PD 118440 is an orally active dopamine (DA) agonists with pronounced central nervous system effects.Formula:C11H17N3SPurity:98%Color and Shape:SolidMolecular weight:223.34GW-876167
CAS:GW-876167, a 5-HT2C agonist, is used potentially for the treatment of obesity and glaucoma.Formula:C16H21N5O2Purity:98%Color and Shape:SolidMolecular weight:315.37MK-0249
CAS:MK-0249 is a potent antagonist of histamine H3 receptor (human H3, Ki : 1.7 nM).
Formula:C23H24F3N3O2Purity:99.90%Color and Shape:SolidMolecular weight:431.45Tulopafant
CAS:Tulopafant (RP 59227) is a potent platelet-activating factor (PAF) antagonist that increases capillary patency and prolongs allograft heart survival.Formula:C25H19N3O2SPurity:99.38%Color and Shape:SolidMolecular weight:425.5Isoproterenol-d7 HCl
CAS:Isoproterenol-d7: internal standard for GC/LC-MS. β1-/β2-AR agonist, not for β3. Lowers blood pressure, tackles bradydysrhythmias, asthma.Formula:C11H18ClNO3Color and Shape:SolidMolecular weight:254.76(4E)-SUN9221
CAS:(4E)-SUN9221 is a potent dual α1-adrenergic receptor and 5-HT2 receptor antagonist that shows antihypertensive and antiplatelet aggregation activity inFormula:C25H31FN4O3Purity:97.79%Color and Shape:SolidMolecular weight:454.54L-771688
CAS:L-771688 (SNAP 6383) is a novel potent and selective α1A-adrenoceptor antagonist with a Ki value of 0.43±0.02 nM.L-771688 KE is used for the treatment of benignFormula:C28H33F2N5O5Purity:94.15%Color and Shape:SolidMolecular weight:557.59ONO4057
CAS:ONO4057 is a potent and orally active Leukotriene B4 receptor antagonist with an IC50 value of 0.7±0.3 μM.Formula:C27H34O7Purity:>99.99%Color and Shape:SolidMolecular weight:470.55CP-66948
CAS:CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.Formula:C13H20N6SPurity:99.14%Color and Shape:SolidMolecular weight:292.4Indanidine
CAS:Indanidine is a highly selective and potent α-adrenergic agonist with antihypertensive activity.Indanidine is an α-adrenergic antagonist that can be used in theFormula:C11H13N5Purity:>99.99%Color and Shape:SolidMolecular weight:215.25RS-601
CAS:RS-601 is a potent dual leukotriene D4/thromboxane A2 inhibitor that inhibits antigen-induced airway hyperresponsiveness (AHR) and shows asthmatic effects in aFormula:C22H23F6NO4SPurity:99.31%Color and Shape:SolidMolecular weight:511.48TD-5471 hydrochloride
CAS:TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (Formula:C32H32ClN3O4Purity:99.57%Color and Shape:SolidMolecular weight:558.07Odapipam
CAS:Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).Formula:C19H20ClNO2Purity:98%Color and Shape:SolidMolecular weight:329.82PF-03654764
CAS:PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with Fexofenadine for allergic rhinitis.Formula:C20H28F2N2OPurity:>99.99%Color and Shape:SolidMolecular weight:350.45Methdilazine Hydrochloride
CAS:Methdilazine Hydrochloride (Bristaline) is a histamine H1 receptor antagonist for dermatologic conditions and relief of itching by allergies or rhinitis.Formula:C18H21ClN2SColor and Shape:Light-Tan Crystalline Powder 4 8-6 (Ntp 1992)Molecular weight:332.89Norfenefrine HCl
CAS:Norfenefrine HCl is an α1-adrenergic receptor agonist, an endogenous neurotransmitter and sympathomimetic drug for hypotension,glycerol adipose.Formula:C8H12ClNO2Purity:99.44%Color and Shape:SolidMolecular weight:189.64Propiomazine HCl
CAS:Propiomazine HCl is an analgesia adjunct.Formula:C20H25ClN2OSColor and Shape:SolidMolecular weight:376.94Trimopam
CAS:Trimopam is a dopamine receptor agonist of the benzazepine group.Formula:C19H23NO2Color and Shape:SolidMolecular weight:297.39Daledalin tosylate
CAS:Daledalin tosylate is an antidepressant.Formula:C26H32N2O3SColor and Shape:SolidMolecular weight:452.61SKF-80723 HBr
CAS:SKF-80723 HBr is a potent D1 agonist enhancing quinpirole-induced circling in 6-OHDA lesioned rats.Formula:C16H16BrNO2Purity:98%Color and Shape:SolidMolecular weight:334.21Trebenzomine
CAS:Trebenzomine is apsychotropic agent with potential as an antidepressant and an antipsychotic.Formula:C12H17NOPurity:98%Color and Shape:SolidMolecular weight:191.27VL-0395
CAS:VL-0395 is an antagonist of CCK1 receptor.Formula:C25H21N3O4Purity:98%Color and Shape:SolidMolecular weight:427.45Mabuterol, (S)-
CAS:Mabuterol, a β2 adrenoreceptor agonist, lowers rat blood pressure and boosts guinea pig heart rate/force, not affecting other receptors.Formula:C13H18ClF3N2OColor and Shape:SolidMolecular weight:310.74Dacemazine
CAS:Dacemazine is used to treat depression.Formula:C16H16N2OSColor and Shape:SolidMolecular weight:284.38Ambucetamide
CAS:Ambucetamide is an antispasmodic, it may inhibit or diminish the spontaneous rhythmical activity of the human myometrium.Formula:C17H28N2O2Color and Shape:SolidMolecular weight:292.42BAY-386
CAS:BAY-386 is a PAR1 receptor inhibitor which suppresses activation of thrombin and platelet activity.Formula:C22H25F3N4O5SColor and Shape:SolidMolecular weight:514.52F-15599 tosylate
CAS:F-15599 tosylate is a selective 5-HT(1A) agonist.Formula:C26H29ClF2N4O4SColor and Shape:SolidMolecular weight:567.05VUF14738
CAS:VUF14738 is a robust and fatigue-resistant photoswitchable GPCR antagonist.Formula:C25H32N4O2Color and Shape:SolidMolecular weight:420.55Albuterol adipate
CAS:Albuterol adipate, a β2-AR agonist salt, treats asthma/COPD, with high selectivity for pulmonary over cardiac receptors.Formula:C32H52N2O10Color and Shape:SolidMolecular weight:624.77Levomepromazine Maleate
CAS:Levomepromazine Maleate: TCA and SNRI with antihistamine, antiadrenergic, and anticholinergic properties.Formula:C23H28N2O5SColor and Shape:SolidMolecular weight:444.546ZD7114 free base
CAS:ZD7114 (ICI-D7114) selectively activates brown fat, boosts thermogenesis, and aids in obesity and metabolic disorders.Formula:C22H30N2O6Color and Shape:SolidMolecular weight:418.48Ricinelaidic Acid
CAS:Ricinelaidic acid blocks LTB4 receptors; hampers human neutrophil responses; reduces rat bronchoconstriction by 46% at 1 mg/kg i.v.Formula:C18H34O3Color and Shape:SolidMolecular weight:298.46Darbufelone
CAS:Darbufelone (CI-1004) is a non-competitive dual inhibitor of PGF2α and LTB4.Formula:C18H24N2O2SPurity:99.72%Color and Shape:SolidMolecular weight:332.46Ref: TM-T10960
1mg42.00€5mg82.00€10mg124.00€25mg264.00€50mg386.00€100mg532.00€500mg1,063.00€1mL*10mM (DMSO)104.00€VRX 03011 Potassium salt
CAS:VRX 03011, a 5-HT4 partial agonist, is used potentially for the treatment of Alzheimer's disease.Formula:C19H27KN3O3SPurity:98%Color and Shape:SolidMolecular weight:416.6Quinpirole
CAS:Quinpirole is a dopamine D2/D3 receptor agonist.Formula:C13H21N3Color and Shape:SolidMolecular weight:219.33Isoetharine hydrochloride
CAS:Isoetharine HCl, a selective, short-acting oral β-agonist, is used as a bronchodilator for inhalation therapy.Formula:C13H22ClNO3Color and Shape:SolidMolecular weight:275.77Ro 23-3423
CAS:Ro 23-3423 is a specific inhibitor of thromboxane synthetase.Formula:C23H22N4O2Color and Shape:SolidMolecular weight:386.45Bitolterol
CAS:Bitolterol is a new beta 2-adrenergic agonist and classified as a pro-drug.Formula:C28H31NO5Color and Shape:SolidMolecular weight:461.55Glucagon Receptor Antagonist I
CAS:Glucagon antagonist I blocks the GCGR (IC50=181 nM), stops glucagon-induced glycogenolysis, and lowers glucose in glucagon-treated humanized mice.Formula:C20H30N2OSColor and Shape:SolidMolecular weight:346.53VER-3323
CAS:VER-3323 is a selective agonist for the 5-HT2B and 5-HT2C serotonin receptor with potent anorectic effects in animal studies.Formula:C11H15BrN2Purity:98%Color and Shape:SolidMolecular weight:255.15U 101958
CAS:U 101958 is a putative antipsychotic agent It is also a highly selective dopamine D4 receptor antagonist.Formula:C20H27N3OColor and Shape:SolidMolecular weight:325.45Fonazine hydrochloride
CAS:Fonazine hydrochloride is a phenothiazine drug used for the treatment of migraine. It is a serotonin antagonist and histamine antagonist.Formula:C19H26ClN3O2S2Color and Shape:SolidMolecular weight:428.01
