GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,017 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
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LPA2 antagonist 1
CAS:LPA2 antagonist 1 is a potent LPA2 antagonist.Formula:C20H23Cl2N5O2S2Purity:99.85%Color and Shape:SolidMolecular weight:500.47γ-Linolenic acid ethyl ester
CAS:γ-Linolenic acid ethyl ester (Ethyl γ-linolenate) is a leukotriene B 4 receptor 4 (LTB 4 ) antagonist which has a potential anti-inflammatory effect[1].Formula:C20H34O2Color and Shape:SolidMolecular weight:306.48Benzatropine
CAS:Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.Formula:C21H25NOPurity:98%Color and Shape:SolidMolecular weight:307.43(RS)-Butyryltimolol
CAS:(RS)-Butyryltimolol, a racemic prodrug of Timolol, enhances its corneal absorption and acts as a β-adrenergic blocker.Formula:C17H30N4O4SPurity:98%Color and Shape:SolidMolecular weight:386.51Remoxipride
CAS:Remoxipride is an antipsychotic agent. Remoxipride is specific for dopamine D2 receptors.Formula:C16H23BrN2O3Purity:98%Color and Shape:SolidMolecular weight:371.27PF-4479745
CAS:PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.Formula:C17H22N4Purity:98%Color and Shape:SolidMolecular weight:282.38MRS1186
CAS:MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).Formula:C16H12ClN5O2Purity:98%Color and Shape:SolidMolecular weight:341.75L-Alprenolol
CAS:L-Alprenolol is a non-selective beta-blocker and a 5-HT1A and 5-HT1B receptor antagonist.Formula:C15H23NO2Purity:98%Color and Shape:SolidMolecular weight:249.35Carcinine
CAS:Carcinine ditrifluoroacetate is a H3 receptor antagonist.Formula:C8H14N4OPurity:98%Color and Shape:SolidMolecular weight:182.22Ro 60-0175 fumarate
CAS:5-HT2 receptor agonistFormula:C15H16ClFN2O4Purity:98%Color and Shape:SolidMolecular weight:342.75MRS2298
CAS:MRS2298, a potent antagonists of the P2Y 1 receptor, has antiaggregatory activity in human platelets.Formula:C10H16ClN5O8P2Purity:98%Color and Shape:SolidMolecular weight:431.66MAT2A-IN-1
CAS:MAT2A-IN-1 suppresses MAT2A, key for MTAP-deficient cancer cell growth; studied for gastric, colon, liver, pancreatic cancers.Formula:C29H28F2N6O4Color and Shape:SolidMolecular weight:562.57Carboprost
CAS:Carboprost (15(S)-15-Methyl Prostaglandin F2α) is a synthetic prostaglandin analogue of PGF2α which has the effect of oxytocic.Formula:C21H36O5Purity:98.18%Color and Shape:White Or Almost White PowderMolecular weight:368.51Ref: TM-T22285
1mg43.00€5mg110.00€10mg166.00€25mg290.00€50mg425.00€100mg577.00€200mg778.00€1mL*10mM (DMSO)122.00€HSK0935
CAS:HSK0935 is a highly selective and orally available SGLT2 inhibitor (IC50: 1.3 nM). It has antihyperglycemic activities.Formula:C22H25ClO7Purity:98%Color and Shape:SolidMolecular weight:436.88GW848687X
CAS:GW848687X, a potent and selective prostaglandin EP1 receptor antagonist, is used for the treatment of inflammatory pain.Formula:C24H18ClF2NO3Purity:98%Color and Shape:SolidMolecular weight:441.85Cyclazosin HCl
CAS:Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.Formula:C23H28ClN5O4Purity:99.10%Color and Shape:SolidMolecular weight:473.95GR 196429
CAS:GR 196429: MT1-selective melatonin receptor agonist; induces sleep, alters circadian rhythm, stimulates melatonin in mice.Formula:C14H18N2O2Purity:98%Color and Shape:SolidMolecular weight:246.3CID1792197
CAS:CID1792197 is a selective agonist of GPR55.Formula:C24H23N3O4S2Purity:98%Color and Shape:SolidMolecular weight:481.59Setastine HCl
CAS:Setastine HCl is a potent antagonist of histamine H1-receptor mediated responses.Formula:C22H29Cl2NOColor and Shape:SolidMolecular weight:394.38L-694,247
CAS:L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E receptors, and can be used to study neurological diseases.Formula:C20H21N5O3SPurity:98.36%Color and Shape:White SolidMolecular weight:411.48PM226
CAS:CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.Formula:C22H31NO3Color and Shape:SolidMolecular weight:357.49L-817,818
CAS:somatostatin sst5 receptor agonistFormula:C33H36N4O3Purity:98%Color and Shape:SolidMolecular weight:536.66threo Ifenprodil hemitartrate
CAS:σ receptor agonist and NR2B subunit-selective NMDA receptor antagonistFormula:C21H27NO2C4H6O6Purity:98%Color and Shape:SolidMolecular weight:400.49Vasopressin V2 receptor antagonist 1
CAS:Vasopressin V2 receptor antagonist 1 (Compound 4g) is a vasopressin V2receptor (V2R) antagonist (Ki: 3.8 nM). dominant polycystic kidney disease (ADPKD).Formula:C33H37ClN4O4Color and Shape:SolidMolecular weight:589.12PA-9
CAS:PA-9 is the first small-molecule PAC1 receptor antagonist.Formula:C17H18N6O2Purity:98%Color and Shape:SolidMolecular weight:338.36MRS1177
CAS:MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).Formula:C20H12ClN5O2Purity:98%Color and Shape:SolidMolecular weight:389.79A 49816
CAS:A 49816 is a high-ceiling diuretic.Formula:C18H17Cl2NO5Color and Shape:SolidMolecular weight:398.24Vicagrel
CAS:Vicagrel, an oral antiplatelet, boosts aspirin's effect, targeting P2Y12 and fights clots in heart and vessel diseases.Formula:C18H18ClNO4SPurity:98%Color and Shape:SolidMolecular weight:379.86Ibodutant
CAS:Ibodutant is an effective and selective tachykinin NK2 receptor antagonist (pKi: 10.1).Formula:C37H48N4O4SPurity:98%Color and Shape:SolidMolecular weight:644.87Stresson
CAS:Stresson is a beta-blocking agent bunitrolol.Formula:C14H21ClN2O2Color and Shape:SolidMolecular weight:284.78S20928
CAS:S20928 is an antagonist of melatonin receptor.Formula:C17H19NOColor and Shape:SolidMolecular weight:253.34DV 7028 hydrochloride
CAS:DV 7028 hydrochloride is a 5-HT2A receptor antagonist.Formula:C21H26ClFN4O3Purity:98%Color and Shape:SolidMolecular weight:436.91hA2A/hCA XII modulator 1
CAS:Potent hA2AAR antagonist & hCA XII inhibitor; Ki: hA2AAR 6.4 nM, hCA XII 6.2 nM. Possible cancer research use.Formula:C24H19N7O4SColor and Shape:SolidMolecular weight:501.52Usmarapride free base
CAS:Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.Formula:C21H29N5O2Purity:99.91% - 99.91%Color and Shape:SolidMolecular weight:383.49Carbinoxamine
CAS:Carbinoxamine: antihistamine for hay fever, angioedema, rhinitis, mild urticaria, dermatographism, allergic conjunctivitis; an H1-antagonist.Formula:C16H19ClN2OPurity:98%Color and Shape:LiquidMolecular weight:290.79EGIS-7625
CAS:EGIS-7625 is a selective and competitive antagonist of 5-HT2B receptor.Formula:C18H24Cl2N4O2Purity:98%Color and Shape:SolidMolecular weight:399.32TR4161
CAS:TR4161 is a prostaglandin bronchodilator of low tracheobronchial irritancy.Formula:C20H36O4Color and Shape:SolidMolecular weight:340.5GR-203040 HCl
CAS:GR203040 inhibits cyclophosphamide-induced damage in the rat and ferret bladder. GR-203040 is a selective NK1 receptor antagonist.Formula:C20H26Cl2N6OColor and Shape:SolidMolecular weight:437.37HEMADO
CAS:HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).Formula:C17H23N5O4Purity:98%Color and Shape:SolidMolecular weight:361.4PF-592379
CAS:PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).Formula:C13H21N3OPurity:98%Color and Shape:SolidMolecular weight:235.33Centanafadine
CAS:Centanafadine inhibits NE/DA transporters and serotonin transporter (IC50: NE=6 nM, DA=38 nM, 5-HT=83 nM).Formula:C15H15NPurity:98%Color and Shape:SolidMolecular weight:209.29UCSF678
CAS:UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.Formula:C15H18N2O2SColor and Shape:SolidMolecular weight:290.38S(-)-Bisoprolol
CAS:S(-)-Bisoprolol, a β1-blocker, may aid in researching hypertension and heart diseases.Formula:C18H31NO4Color and Shape:SolidMolecular weight:325.44Spirendolol
CAS:Spirendolol is an antagonist of β adrenergic receptor.Formula:C21H31NO3Purity:98%Color and Shape:SolidMolecular weight:345.48UP202-56
CAS:UP202-56 is an adenosinergic agonist and is an adenosine analog.Formula:C33H37N7O4Purity:98%Color and Shape:SolidMolecular weight:595.69FK-1052 HCl
CAS:FK-1052 HCl is a serotonin 3 & 4 dual receptor antagonist.Formula:C18H20ClN3OColor and Shape:SolidMolecular weight:329.83Savoxepin mesylate
CAS:Savoxepin mesylate, a tetracyclic cyano-dibenzoxepino-azepine derivative, has potent antidopaminergic activity.Formula:C26H30N2O4SPurity:98%Color and Shape:SolidMolecular weight:466.59A331440
CAS:A331440 is an modulator of L-histidine and histamine H3 receptor.Formula:C22H27N3OColor and Shape:SolidMolecular weight:349.47TCS-OX2-29 HCl
CAS:TCS-OX2-29 is a selective orexin-2 receptor antagonist (IC50 = 40 nM), which plays an important role in pain modulation.Formula:C23H32ClN3O3Purity:98%Color and Shape:SolidMolecular weight:433.97
