GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,017 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(158 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(194 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(327 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5983 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Befetupitant
CAS:Befupupitant(Ro67-5930) is a potent and selective tachykinin 1 receptor (NK1R) antagonist for the study of corneal neovascularization.Formula:C29H29F6N3O2Purity:98.72%Color and Shape:SolidMolecular weight:565.55HSR-609
CAS:HSR-609, a histamine H1 receptor antagonist, is used potentially for the treatment of allergic rhinitis.Formula:C21H21FN2O3Purity:98%Color and Shape:SolidMolecular weight:368.4Ro 04-6790 dihydrochloride
CAS:Ro 04-6790 dihydrochloride is an effective and selective antagonist of the serotonin 5-HT6 receptor.Formula:C12H18Cl2N6O2SPurity:98%Color and Shape:SolidMolecular weight:381.28Dipiproverine hydrochloride
CAS:Dipiproverine hydrochloride is an antispasmodic alpha-amino acid ester used as an anticholinergic.Formula:C20H32Cl2N2O2Purity:98%Color and Shape:SolidMolecular weight:403.39NNC-38-1049
CAS:NNC-38-1049 is a novel selective antagonist of histamine H3.Formula:C19H25ClN2O2Purity:98%Color and Shape:SolidMolecular weight:348.87PG 01037 dihydrochloride
CAS:PG 01037 dihydrochloride (PG-01037 2HCl) is a potent and selective dopamine D3 receptor antagonist with a Ki of 0.7 nM.Formula:C26H28Cl4N4OPurity:99.89%Color and Shape:SolidMolecular weight:554.34AHR-14310C
CAS:AHR-14310C is a long-acting and nonsedating H1-antihistamine.Formula:C24H28F2N2O3Purity:98%Color and Shape:SolidMolecular weight:430.49LP44 hydrochloride
CAS:LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.Formula:C27H38ClN3OSPurity:98.06%Color and Shape:SolidMolecular weight:488.13LG 82-4-00
CAS:LG 82-4-00 is an inhibitor of thromboxane.Formula:C10H11ClN2O3SPurity:98%Color and Shape:SolidMolecular weight:274.722-Iodomelatonin
CAS:2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, >5x selective over MT2, used to map melatonin sites in brain/tissues.Formula:C13H15IN2O2Purity:99.7%Color and Shape:SolidMolecular weight:358.17Ref: TM-T10073
10mg43.00€25mg79.00€50mg118.00€100mg178.00€200mg268.00€500mgTo inquire1mL*10mM (DMSO)34.00€AHR-13268D
CAS:AHR-13268D is a new agent of antiallergic/antihistaminic.Formula:C28H29F2NNaO4Purity:98%Color and Shape:SolidMolecular weight:504.53TIK-301
CAS:TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM
Formula:C14H17ClN2O2Purity:98%Color and Shape:SolidMolecular weight:280.75SM-2470
CAS:SM-2470 is an α1-adrenoceptor antagonist with antihypertensive activity and hypocholesterolemic activity that inhibits cholesterol absorption.Formula:C23H30ClN5O3Purity:98.91%Color and Shape:SolidMolecular weight:459.97RS 15385-197
CAS:RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.Formula:C18H26N2O3SColor and Shape:SolidMolecular weight:350.48Usmarapride
CAS:Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.Formula:C23H31N5O6Color and Shape:SolidMolecular weight:473.53RXFP3/4 agonist 2
CAS:RXFP3/4 agonist 2 is a nonpeptide bis-RXFP3/4 agonist used in the study of diseases caused by metabolic abnormalities.Formula:C22H22N6O2Purity:99.82%Color and Shape:SolidMolecular weight:402.45ST3932
CAS:ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).Formula:C12H16N8OPurity:98%Color and Shape:SolidMolecular weight:288.31PRX933 hydrochloride
CAS:PRX933 hydrochloride (GW876167 hydrochloride) is an agonist of 5-HT2C receptor and can be used in studies about hypertension acute treatment.Formula:C16H22ClN5O2Purity:99.51% - 99.89%Color and Shape:SolidMolecular weight:351.84Ref: TM-T12565
1mg338.00€5mg538.00€10mg858.00€25mg1,269.00€50mg1,720.00€100mg2,305.00€1mL*10mM (DMSO)618.00€(±)-Tazifylline
CAS:(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.Formula:C23H32N6O3SPurity:99.54%Color and Shape:SolidMolecular weight:472.6Ref: TM-T10000
1mg140.00€5mg269.00€10mg389.00€25mg610.00€50mg820.00€100mg1,063.00€1mL*10mM (DMSO)350.00€O-2093
CAS:anandamide uptake inhibitorFormula:C34H43Cl2NO3Purity:98%Color and Shape:SolidMolecular weight:584.62PRX-08066 Maleic acid
CAS:PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.Formula:C23H21ClFN5O4SPurity:97.59%Color and Shape:SolidMolecular weight:517.96Ref: TM-T6959
1mg79.00€5mg168.00€10mg220.00€25mg398.00€50mg587.00€100mg835.00€200mg1,134.00€1mL*10mM (DMSO)380.00€Org-12962
CAS:Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).Formula:C10H11ClF3N3Purity:98.34%Color and Shape:SolidMolecular weight:265.66EMDT
CAS:EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.Formula:C15H22N2OPurity:97.66% - 99.78%Color and Shape:SolidMolecular weight:246.35Ref: TM-T11183
1mg87.00€2mg118.00€5mg167.00€10mg202.00€25mg449.00€50mg652.00€100mg888.00€500mg1,783.00€1mL*10mM (DMSO)166.00€AUY-954 free base
CAS:AUY-954 is a selective S1P(1) modulator reducing EAN inflammation and demyelination in rats.Formula:C25H20F3NO2SColor and Shape:SolidMolecular weight:455.49SC 53116 Hydrochloride
CAS:SC 53116 Hydrochloride is selective agonist of the newly identified serotonin 5-HT4 receptor subtype.Formula:C16H23Cl2N3O2Color and Shape:SolidMolecular weight:360.28WRC-0571
CAS:WRC-0571 is a highly potent, selective antagonist of A1 adenosine receptors.Formula:C17H26N6OPurity:98%Color and Shape:SolidMolecular weight:330.43Sch 33303
CAS:Sch 33303 is an antiallergy agents.Formula:C19H16N2O3Color and Shape:SolidMolecular weight:320.34Noberastine maleate
CAS:Noberastine maleate, a fast-acting furan-derived H1 antagonist, peaks at 4 hours with minimal CNS effects and maximal efficacy at 30 mg/day.Formula:C25H29N5O9Color and Shape:SolidMolecular weight:543.53PF 10040
CAS:PF 10040 is an antagonist of platelet activating factor (PAF).Formula:C20H24ClNO2Color and Shape:SolidMolecular weight:345.86CM304
CAS:CM304 is a highly selective sigma-1 receptor antagonist.Formula:C18H26ClFN2OSColor and Shape:SolidMolecular weight:372.93Elzasonan
CAS:Elzasonan is a selective 5-hydroxytryptamine 1B receptor antagonist used to treat patients with major depressive disorder and obsessive compulsive disorder.Formula:C22H23Cl2N3OSColor and Shape:SolidMolecular weight:448.414-Chloro Trazodone hydrochloride
CAS:4-Chloro Trazodone HCl is a Trazodone isomer, an antidepressant for anxiety disorders.Formula:C19H23Cl2N5OColor and Shape:SolidMolecular weight:408.32Naxifylline
CAS:Naxifylline is an A1 adenosine receptor blocker that increases urine and protects kidneys during edema treatment in heart failure.Formula:C18H24N4O3Color and Shape:SolidMolecular weight:344.415-OxoETE methyl ester
CAS:5-OxoETE methyl ester is a 5-oxoETE ester, an OXER1 agonist with stronger β-arrestin response, EC50 = 1.54 μM.Formula:C21H32O3Color and Shape:SolidMolecular weight:332.48Arvanil
CAS:Arvanil (N-Vanillylarachidonamide) is a synthetic capsaicin-amphetamine hybrid that acts as a ligand for VR1 and CB1, offering neuroprotective effects.Formula:C28H41NO3Purity:99.49%Color and Shape:SolidMolecular weight:439.632-Acetylbenzoic acid
CAS:2-Acetylbenzoic acid outperforms 2-propionyloxybenzoic in hindering platelet function and PG synthesis; both similar in blocking PGI2 creation.Formula:C9H8O3Purity:99.62%Color and Shape:Off-White SolidMolecular weight:164.16WAY 629
CAS:WAY 629 is a selective SR-2C agonist that also act as potent 5-HT2C receptor agonists.Formula:C15H18N2Color and Shape:SolidMolecular weight:226.32LPA2 antagonist 1
CAS:LPA2 antagonist 1 is a potent LPA2 antagonist.Formula:C20H23Cl2N5O2S2Purity:99.85%Color and Shape:SolidMolecular weight:500.47CP-809101
CAS:CP-809101 is an effective and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Formula:C15H17ClN4OPurity:98%Color and Shape:SolidMolecular weight:304.77Amibegron
CAS:Amibegron: oral β3 adrenergic agonist, CNS-penetrating, with antidepressant and anxiolytic properties.Formula:C22H26ClNO4Color and Shape:SolidMolecular weight:403.9CP 66713
CAS:CP-66713 is an adenosine A2 receptor antagonist.Formula:C15H10ClN5Color and Shape:SolidMolecular weight:295.73Metitepine
CAS:Metitepine is a serotonin receptor antagonist in the CNS used as an antipsychotic.Formula:C20H24N2S2Color and Shape:SolidMolecular weight:356.55A-65186
CAS:A-65186 is a CCK antagonist used in the study of inflammation and gastrointestinal tract injury.Formula:C25H35N3O4Purity:98.85% - 99.94%Color and Shape:SolidMolecular weight:441.56TP-680
CAS:TP-680 is a antagonist of cholecystokininA receptor.Formula:C35H33N5O4SPurity:98%Color and Shape:SolidMolecular weight:619.73ChemR23-IN-2
CAS:ChemR23-IN-2 is a potent, orally active inhibitor of ChemR23 (IC50: 3.2 nM).Formula:C29H26N4O5Color and Shape:SolidMolecular weight:510.54mCPBG
CAS:mCPBG is a potent high affinity agonist of 5-HT3 receptor.Formula:C8H10ClN5Color and Shape:SolidMolecular weight:211.65Trimazosin hydrochloride
CAS:Trimazosin hydrochloride is used in the treatment of hypertensive patients failing to respond to thiazides.Formula:C20H32ClN5O7Color and Shape:SolidMolecular weight:489.95Cgp 52608
CAS:CGP 52608 is a selective ligand for RAR-associated orphan receptor alpha.Formula:C8H12N4OS2Color and Shape:SolidMolecular weight:244.34VUF8504
CAS:VUF8504 is a novel ligand of adenosine A3 receptor.Formula:C22H17N3O2Color and Shape:SolidMolecular weight:355.39Cannabicitran
CAS:Cannabicitran is a cannabinoid that can decrease rabbits intraocular pressure [1] [2].Formula:C21H30O2Color and Shape:SolidMolecular weight:314.46
