GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(326 products)
- PAFR(13 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5968 products of "GPCR/G-Protein"
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Adrenomedullin (16-31), human TFA
Human adrenomedullin (16-31) TFA, fragment 16-31, binds CGRP1 receptor, raises rat blood pressure, not cats’.Formula:C84H130F3N25O23S2Color and Shape:SolidMolecular weight:1979.21Olcegepant hydrochloride
CAS:Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a selective calcitonin gene-related peptide 1 (CGRP1) receptor antagonist.Formula:C38H48Br2ClN9O5Purity:99.69%Color and Shape:SolidMolecular weight:906.11TAK-448 acetate
CAS:TAK-448 acetate (MVT-602 acetate) is a KISS1R agonist, a synthetic peptide similar to kisspeptin.Formula:C60H84N16O16Purity:99.88%Color and Shape:SolidMolecular weight:1285.41Guanylin (mouse, rat)
CAS:<p>Guanylin (mouse, rat), a peptide consisting of 15 amino acids, acts as an activator of intestinal guanylate cyclase and is utilized in diarrhea research [1].</p>Formula:C60H90N16O22S4Purity:98%Color and Shape:SolidMolecular weight:1515.71[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH
CAS:<p>[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH is a synthetic LHRH analog and a GnRH receptor antagonist.</p>Formula:C67H84N16O13Color and Shape:SolidMolecular weight:1321.48TCMCB07 TFA
TCMCB07 TFA is a cyclic nonapeptide and an orally active, brain-penetrating antagonist of the melanocortin receptor 4 (MC4R), playing a significant role inFormula:C63H87N15O11·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:1230.46 (free base)Spns2-IN-1
Spns2-IN-1 is a potent Spns2 inhibitor, effectively impeding Spns2-dependent S1P transport with an IC50 value of 1.4±0.3 μM, crucial for modulating the immunePurity:98%Color and Shape:Odour SolidBQ-3020 ammonium
BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] ET-1 binding to ET B receptors with an IC50 of 0.2Formula:C96H140N20O25S·xNH3Purity:98%Color and Shape:SolidMolecular weight:2006.32 (free base)15(R)-Pinane Thromboxane A2
CAS:15(R)-PTA2 is an (R)-epimer of PTA2; doesn't inhibit platelet aggregation or gastric tone; less effective than PTA2 at blocking prostaglandin contraction.Formula:C24H40O3Color and Shape:SolidMolecular weight:376.5814-Thiouridine 5′-triphosphate disodium
CAS:4-Thiouridine 5′-triphosphate (4-Thio-UTP) tetrasodium functions as a potent agonist at P2Y 2 and P2Y 4 receptors, with half-maximal effective concentrations (Formula:C9H11N2Na2O14P3SPurity:98%Color and Shape:SolidMolecular weight:546.19NF546 hydrate
NF546 (hydrate), a selective non-nucleotide P2Y11 agonist, exhibits a pEC50 value of 6.27 and induces interleukin-8 secretion from human monocyte-derivedFormula:C47H44N6Na4O17P4·5H2OPurity:98%Color and Shape:SolidMolecular weight:1424.01Sigma-1 receptor antagonist 4
<p>Sigma-1 receptor antagonist 4 (Compound 32) is a potent σ1R antagonist that significantly enhances morphine's analgesic effects and reverses morphine-induced</p>Formula:C22H26N2OColor and Shape:SolidMolecular weight:334.45PACAP (6-38), human, ovine, rat acetate
PACAP (6-38), human, ovine, rat acetate is a potent PACAP receptor antagonist with IC50s of 30, 600, and 40 nM for PACAP type I receptor, PACAP type II receptorFormula:C184H303N55O48SPurity:99.84%Color and Shape:SoildMolecular weight:4085.84L-779976
CAS:L-779,976 is an agonist of somatostatin receptor.Formula:C33H43N7O3Color and Shape:SolidMolecular weight:585.74FK 224
CAS:FK 224 is an antagonist of tachykinin receptor.Formula:C54H72N8O13Color and Shape:SolidMolecular weight:1041.213PSA1 (141-150)
CAS:This Prostate Specific Antigen 1 peptide was used in the immunotherapy of cancer experiments.Formula:C55H93N13O13SPurity:98%Color and Shape:SolidMolecular weight:1176.47Lysophosphatidic acid
CAS:Lysophosphatidic acid is a bioactive chemical.Formula:C21H41O7PColor and Shape:SolidMolecular weight:436.52(Pro34)-Peptide YY (human)
CAS:(Pro34)-Peptide YY (human) is a highly Y 1 -selective full agonist of Peptide YY /neuropeptide Y receptors [1] .Formula:C194H294N54O56Color and Shape:SolidMolecular weight:4278.73isomer-Cilansetron
CAS:isomer-Cilansetron is an isomer of Cilansetron.Formula:C20H21N3OPurity:99.92% - 99.96%Color and Shape:SoildMolecular weight:319.4TGR5 agonist 7
TGR5 agonist 7 (Compound 22-Na) is an intestine-restricted, orally active agonist of the G protein-coupled bile acid receptor TGR5 (GPBAR1 or GPR131) with an EC50 of less than 1 μM. In mouse models, it demonstrates blood glucose-lowering effects, making it useful for diabetes research.Formula:C37H59N2NaO9SColor and Shape:SolidMolecular weight:730.93
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