GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,058 products)
- Adenosine Receptor(216 products)
- Adrenergic Receptor(3,265 products)
- Bombesin Receptor(37 products)
- Bradykinin Receptor(63 products)
- CXCR(179 products)
- CaSR(31 products)
- Cannabinoid Receptor(226 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(448 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(89 products)
- GPCR19(40 products)
- GRK(43 products)
- GTPase(26 products)
- Glucagon Receptor(210 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(389 products)
- LPA Receptor(22 products)
- Melatonin Receptor(26 products)
- OX Receptor(57 products)
- Opioid Receptor(337 products)
- PAFR(12 products)
- PKA(57 products)
- S1P Receptor(22 products)
- SGLT(33 products)
- Sigma receptor(49 products)
Show 19 more subcategories
Found 6058 products for "GPCR/G-Protein".
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MDL 29913
CAS:NK2 tachykinin receptor selective antagonist.Formula:C40H56N8O6Purity:98%Color and Shape:SolidMolecular weight:745Neuropeptide S(Mouse) TFA
Neuropeptide S(Mouse) TFA: Endogenous NPSR agonist, EC50 3 nM, boosts Ca2+, activity, wakefulness, and lowers mouse anxiety.Formula:C92H157F3N34O29Color and Shape:SolidMolecular weight:2296.49(Pro34)-Peptide YY (human)
CAS:(Pro34)-Peptide YY (human) is a highly Y 1 -selective full agonist of Peptide YY /neuropeptide Y receptors [1] .Formula:C194H294N54O56Color and Shape:SolidMolecular weight:4278.73Spantide II
CAS:Spantide II is an antagonist of tachykinin.Formula:C86H104Cl2N18O13Purity:98%Color and Shape:SolidMolecular weight:1668.77Neuropeptide Y (13-36), amide, human
CAS:Neuropeptide Y (13-36), amide, human is a neuropeptide Y receptor agonist.Formula:C134H207N41O36SPurity:98%Color and Shape:SolidMolecular weight:3000.4Misoprostol
CAS:Misoprostol, a prostaglandin E1 derivative, has a strong inhibitory effect on gastric acid secretion, while having a contractile effect on pregnancy.Formula:C22H38O5Purity:99.78%Color and Shape:SolidMolecular weight:382.53Uroguanylin (human) TFA
Uroguanylin (human) (TFA) is the natural ligand for the guanylate cyclase C (GCC) receptor expressed in metastatic colorectal cancer tumors. In animal models of human colon cancer, Uroguanylin (human) (TFA) demonstrates antitumor activity.Color and Shape:Odour Solid[Leu13]-Motilin
CAS:[Leu13]-Motilin (KW-5139) is an analogue of the gastrointestinal hormone motilin that induces concentration-dependent contractions in rabbit gastrointestinalFormula:C121H190N34O35Purity:98%Color and Shape:SolidMolecular weight:2681.01EP3 antagonist 4
CAS:EP3 antagonist 4: hEP inhibitor, Ki = 2 nM, low clearance, high oral AUC, good bioavailability in rats, potential for diabetes research.Formula:C22H20Cl3FN4O3S2Purity:98%Color and Shape:SolidMolecular weight:577.91Retrobradykinin
CAS:Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.Formula:C50H73N15O11Color and Shape:SolidMolecular weight:1060.228Neuropeptide Y (3-36) (human, rat)
CAS:Neuropeptide Y (3-36) is a Y2 receptor agonist that limits norepinephrine release, produced by DPP4 from NPY.Formula:C175H269N53O54SColor and Shape:SolidMolecular weight:4011.5(2R,2R)-PF-07258669
CAS:(2R,2R)-PF-07258669' is an antagonist for the MC4R (melanocortin 4 receptor), primarily studied for its role in regulating appetite and energy expenditure.Formula:C25H27FN6O2Color and Shape:SolidMolecular weight:462.52Bz-Dab(nbd)-awfpp-nle-NH2
CAS:Bz-Dab(nbd)-ala-trp-phe-pro-pro-nle-NH2 is a fluorescent NK2 antagonist.Formula:C56H65N13O11Color and Shape:SolidMolecular weight:1096.2Cagrilintide
CAS:Cagrilintide is a long-acting amylin analogue acting as a dual agonist of the amylin receptor and calcitonin receptor, reducing body weight and food intake.Formula:C194H312N54O59S2Purity:98.83% - 99.95%Color and Shape:White SolidMolecular weight:4409.01Peptide YY (PYY) (3-36), porcine TFA
Peptide YY (PYY) (3-36), porcine TFA, functions as a gut hormone that serves as a Y2 receptor agonist, effectively reducing appetite [1].Formula:C176H272N52O54·C2HF3O2Color and Shape:SolidMolecular weight:4094.44TAK-683 acetate
TAK-683 acetate: potent KISS1R agonist (IC50=170 pM), stable, nonapeptide. Affects GnRH, FSH, LH, testosterone; potential in prostate cancer research.Formula:C66H87N17O15Color and Shape:SolidMolecular weight:1358.5Setmelanotide
CAS:Setmelanotide (BIM-22493) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).Formula:C49H68N18O9S2Purity:99.93%Color and Shape:White SolidMolecular weight:1117.31Ref: TM-T12882
1mg50.00€5mg105.00€10mg172.00€1mL*10mM (DMSO)197.00€25mg268.00€50mg401.00€100mg580.00€[D-Trp34]-Neuropeptide Y Acetate
[D-Trp34]-Neuropeptide Y Acetate is a potent Y5 receptor agonist that increases rat food intake; less potent at Y1, Y2, Y4, Y6.Formula:C198H293N55O58Purity:99.73%Color and Shape:SoildMolecular weight:4371.78AY 254
CAS:AY 254: Potent PAR2 agonist, ERK1/2 activation (EC50=2 nM), limits caspase 3/8, aids HT29 cell healing, boosts IL-8.Formula:C30H49N9O6Color and Shape:SolidMolecular weight:631.779CGRP 8-37 (rat)
CAS:CGRP 8-37 (rat) is a CGRP receptor antagonist, a CGRP fragment with potential anti-injury effects that induces arterial relaxation.Formula:C138H224N42O41Purity:98.11% - 99.28%Color and Shape:SolidMolecular weight:3127.51
![[Leu13]-Motilin](https://static.cymitquimica.com/products/TM/thumb-webp/T78563.webp)
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