CymitQuimica logo
GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

Show 19 more subcategories

Found 5985 products of "GPCR/G-Protein"

Sort by

Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • Cortistatin-14 acetate


    Cortistatin-14 acetate, a neuropeptide have structural similarity to somatostatin-14, binds and exerts its function via the somatostatin receptors (sst1-sst5).

    Formula:C83H118N20O20S2
    Purity:98.24% - 99.63%
    Color and Shape:Soild
    Molecular weight:1780.08

    Ref: TM-TP1570L

    1mg
    111.00€
    5mg
    415.00€
    10mg
    509.00€
    25mg
    745.00€
    50mg
    1,111.00€
    100mg
    1,501.00€
  • J-115814

    CAS:
    J-115814 is a potent feeding stimulant.
    Formula:C29H38ClN5O3S
    Color and Shape:Solid
    Molecular weight:572.16

    Ref: TM-T32246

    25mg
    1,444.00€
  • LAS190792

    CAS:
    LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.
    Formula:C39H43ClN4O9S2
    Color and Shape:Solid
    Molecular weight:811.36

    Ref: TM-T74709

    5mg
    To inquire
    50mg
    To inquire
  • Linaclotide acetate

    CAS:

    Linaclotide acetate, an oral guanylate cyclase C agonist with 14 amino acids, treats constipation-predominant IBS and chronic constipation.

    Formula:C61H83N15O23S6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1586.79

    Ref: TM-T11852L

    100mg
    To inquire
    500mg
    To inquire
  • [Phe8Ψ(CH-NH)-Arg9]-Bradykinin

    CAS:
    Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage.
    Formula:C50H75N15O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1046.23

    Ref: TM-TP2076

    1mg
    225.00€
  • L-threo Lysosphingomyelin (d18:1)

    CAS:
    L-threo Lysosphingomyelin, a natural S1P receptor agonist, has EC50s: 19.3 nM (hS1P1), 131.8 nM (hS1P3), 313.3 nM (hS1P2).
    Formula:C23H49N2O5P
    Color and Shape:Solid
    Molecular weight:464.62

    Ref: TM-T38452

    5mg
    1,378.00€
  • AR ligand 40


    AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.
    Formula:C21H25N5
    Color and Shape:Solid
    Molecular weight:347.211

    Ref: TM-T207383

    10mg
    To inquire
    50mg
    To inquire
  • PSB 0777 ammonium salt

    CAS:
    adenosine A2A receptor full agonist
    Formula:C18H24N6O7S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:500.55

    Ref: TM-T23196

    10mg
    1,026.00€
    50mg
    4,399.00€
  • β-CGRP (mouse)


    β-CGRP (mouse), a calcitonin gene-related peptide, induces vasodilation and is applicable in research areas including cardiovascular, pro-inflammatory, migraine, and metabolic studies.
    Formula:C165H265N49O55S2
    Color and Shape:Solid
    Molecular weight:3879.29

    Ref: TM-TP2859

    10mg
    To inquire
    50mg
    To inquire
  • Sch 202596

    CAS:
    Sch 202596 is a selective non-peptide antagonist of GAL-1 receptor.
    Formula:C25H22Cl2O12
    Color and Shape:Solid
    Molecular weight:585.34

    Ref: TM-T28705

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • CB2R probe 1

    CAS:

    CB2R Probe 1, a cannabinoid 2 receptor (CB2R) fluorescent probe, exhibits both safety and environmental friendliness, boasting a dissociation constant (K i) of

    Formula:C36H42N4O4
    Color and Shape:Solid
    Molecular weight:594.74

    Ref: TM-T74604

    5mg
    To inquire
    50mg
    To inquire
  • (3R,5R,6S)-Atogepant


    (3R,5R,6S)-Atogepant (MK-8031) is a CGRP antagonist enantiomer used in migraine research.
    Formula:C29H23F6N5O3
    Color and Shape:Solid
    Molecular weight:603.52

    Ref: TM-T73703

    5mg
    To inquire
    50mg
    To inquire
  • Agaridoxin

    CAS:

    Agaridoxin is a mushroom metabolite.

    Formula:C11H14N2O5
    Color and Shape:Solid
    Molecular weight:254.242

    Ref: TM-T29709

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • S 16474

    CAS:
    S 16474 is an antagonist of Neurokinin-1 Receptor.
    Formula:C44H48N6NaO8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:811.892

    Ref: TM-T26169

    25mg
    1,369.00€
  • PG106

    CAS:
    Selective hMC3 receptor antagonist (IC50 = 210 nM). Exhibits no activity at hMC4 receptors and hMC5 receptors.
    Formula:C51H69N13O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1008.19

    Ref: TM-TP1952

    1mg
    264.00€
  • Adrenocorticotropic Hormone (ACTH) (1-39), rat

    CAS:
    ACTH (1-39), rat: potent MC2 agonist, forms fragments in vitro, isolated by HPLC, characterized by amino acids and NH2-terminus.
    Formula:C210H315N57O57S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4582.23

    Ref: TM-TP1249

    1mg
    178.00€
    5mg
    712.00€
  • 15-keto-17-phenyl trinor Prostaglandin F2α

    CAS:
    Bimatoprost is an F-series prostaglandin (PG) analog which has been approved for use as an ocular hypotensive drug.
    Formula:C23H30O5
    Color and Shape:Solid
    Molecular weight:386.488

    Ref: TM-T37934

    1mg
    220.00€
    5mg
    944.00€
    10mg
    1,700.00€
  • Protease-Activated Receptor-1 antagonist 2

    CAS:
    Orally active PAR-1 antagonist with 7 nM IC50; potential for CVD research.
    Formula:C24H23F2N3O2
    Color and Shape:Solid
    Molecular weight:423.46

    Ref: TM-T74266

    5mg
    To inquire
    50mg
    To inquire
  • Fasitibant chloride hydrochloride

    CAS:
    Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.
    Formula:C36H50Cl4N6O6S
    Color and Shape:Solid
    Molecular weight:836.7

    Ref: TM-T31747

    100mg
    To inquire
    500mg
    To inquire
  • tBPC

    CAS:
    Enhances Y4R response to PP, NPY & PYY with EC50 of 0.03, 0.4, 0.5 nM; selective for Y4R over Y1R, Y2R, Y5R.
    Formula:C16H24O2
    Color and Shape:Solid
    Molecular weight:248.36

    Ref: TM-T37528

    10mg
    123.00€
    50mg
    510.00€