GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,030 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(196 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(55 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5985 products of "GPCR/G-Protein"
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Haloperidol D4
CAS:Haloperidol D4 is deuterium-labeled haloperidol.Formula:C21H23ClFNO2Purity:98%Color and Shape:SolidMolecular weight:379.89Uroguanylin (human) TFA
Uroguanylin (human) (TFA) is the natural ligand for the guanylate cyclase C (GCC) receptor expressed in metastatic colorectal cancer tumors. In animal models of human colon cancer, Uroguanylin (human) (TFA) demonstrates antitumor activity.Color and Shape:Odour SolidAntibacterial agent 189
Antibacterialagent 189 (compound 3a) is a potent antibacterial agent with high binding affinity to the target proteins OMPA/exo-1,3-β-glucanase. It demonstrates effective antibacterial activity against Escherichia coli, Pseudomonas aeruginosa, Staphylococcus aureus, Bacillus subtilis, Candida albicans, and Aspergillus flavus. Additionally, Antibacterialagent 189 exhibits strong binding affinity to the target proteins SMO and SUFU/GLI-1.Formula:C37H28N4OMolecular weight:544.22631Calcitonin-13C6,15N4 TFA
Calcitonin-13CIC6,15NIC4(salmon) (Salmon calcitonin-13CIC6,15NIC4) TFA is a version of calcitonin(salmon) labeled with carbon-13 and nitrogen-15. This hormone regulates calcium and acts dualistically as an agonist to both amylin and calcitonin receptors, promoting bone formation while inhibiting bone resorption.Formula:C1401C5H240N4315NO48S2·5C2HF3O2Color and Shape:SolidMolecular weight:4007.93FLLRN
CAS:FLLRN is a biologically active peptide serving as a PAR1-specific antagonist.Formula:C31H51N9O7Color and Shape:SolidMolecular weight:661.79T-10430
T-10430 is a potent and orally active agonist of the leukotriene B4 receptor 2 (BLT2). It shows potential for use in psoriasis research.Formula:C17H22N6OColor and Shape:SolidMolecular weight:326.396A 31472
CAS:A 31472 is a tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Formula:C22H22ClNColor and Shape:SolidMolecular weight:335.87[Pro34]Neuropeptide Y, porcine
CAS:[Pro34]Neuropeptide Y, porcine functions as a selective agonist for the NPY (Y1) receptor and induces vasoconstriction in the guinea pig's caval vein [1].Formula:C190H286N54O56Color and Shape:SolidMolecular weight:4222.63Prostaglandin F2α isopropyl ester
CAS:PGF2α isopropyl ester is an ester prodrug of PGF2α with enhanced lipid solubility.Formula:C23H40O5Color and Shape:SolidMolecular weight:396.568CRL-42872 free base
CAS:CRL-42872 free base is a bioactive chemical.Formula:C22H26N6O6SColor and Shape:SolidMolecular weight:502.54GLP-1R agonist 29
GLP-1R agonist 29 (Compound 20) is a GLP-1R agonist that induces hGLP-1R-mediated cAMP stimulation with an EC50 of 0.018 nM. It exhibits favorable pharmacokinetic properties and shows good in vivo exposure, with an AUC0-∞,sc of 77688 ng·h/mL.Color and Shape:Odour SolidHemokinin 1, human
CAS:Endogenous P-like compound, NK1 receptor agonist; IC50: NK1-1.8 nM, NK3-370 nM, NK2-480 nM; boosts B-cell growth, antiapoptotic, lowers blood pressure in vivo.Formula:C54H84N14O14SPurity:98%Color and Shape:SolidMolecular weight:1185.4Antidepressant agent 3
Agent 3: orally active, antidepressant, anxiolytic, boosts performance and cognition.Formula:C17H30ClN5O2SColor and Shape:SolidMolecular weight:403.97AP 811
CAS:AP 811: Selective NPR3 antagonist, Ki of 0.48 nM, >20,000x selective over NPR1, blocks ANP-induced pump stimulation.Formula:C46H66N12O8Color and Shape:SolidMolecular weight:915.11Corticotropin-releasing factor (human) acetate
Corticotropin-releasing factor (human) acetate stimulates to synthesize and secret adrenocorticotropin in the anterior pituitary.Purity:98.30%Color and Shape:Liquid19(R)-HETE
CAS:19(R)-HETE is a renal artery vasodilator and can be used to study angiotensin II-induced cardiac hypertrophy.Formula:C20H32O3Color and Shape:SolidMolecular weight:320.47Atenolol
CAS:Atenolol (Tenormin) is a selective β1 receptor antagonist.Formula:C14H22N2O3Purity:99.07% - 99.95%Color and Shape:White Crystalline Powder SolidMolecular weight:266.34Xenin-8
CAS:neurotensin-like peptide that modulate pancreatic insulin and glucagon secretion/effectsFormula:C51H79N15O9Purity:98%Color and Shape:SolidMolecular weight:1046.27LCKLSL
CAS:LCKLSL, an N-terminal hexapeptide, inhibits AnxA2 and tPA binding, reduces plasmin, and exhibits anti-angiogenic effects.Formula:C30H57N7O8SMolecular weight:675.89BPP-2
BPP-2 is a GHSR ligand containing the element F. By labeling BPP-2 with the isotope 18F, a PET probe targeting GHSR can be produced. The binding affinity (Ki) of 18F-BPP-2 for GHSR is 274 nM.Formula:C27H28FN5O2Molecular weight:473.2227
