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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5985 products of "GPCR/G-Protein"

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  • Haloperidol D4

    CAS:
    Haloperidol D4 is deuterium-labeled haloperidol.
    Formula:C21H23ClFNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:379.89

    Ref: TM-T11535

    1mg
    750.00€
  • Uroguanylin (human) TFA


    Uroguanylin (human) (TFA) is the natural ligand for the guanylate cyclase C (GCC) receptor expressed in metastatic colorectal cancer tumors. In animal models of human colon cancer, Uroguanylin (human) (TFA) demonstrates antitumor activity.
    Color and Shape:Odour Solid

    Ref: TM-TP3207

    10mg
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    50mg
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  • Antibacterial agent 189


    Antibacterialagent 189 (compound 3a) is a potent antibacterial agent with high binding affinity to the target proteins OMPA/exo-1,3-β-glucanase. It demonstrates effective antibacterial activity against Escherichia coli, Pseudomonas aeruginosa, Staphylococcus aureus, Bacillus subtilis, Candida albicans, and Aspergillus flavus. Additionally, Antibacterialagent 189 exhibits strong binding affinity to the target proteins SMO and SUFU/GLI-1.
    Formula:C37H28N4O
    Molecular weight:544.22631

    Ref: TM-T209404

    10mg
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    50mg
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  • Calcitonin-13C6,15N4 TFA


    Calcitonin-13CIC6,15NIC4(salmon) (Salmon calcitonin-13CIC6,15NIC4) TFA is a version of calcitonin(salmon) labeled with carbon-13 and nitrogen-15. This hormone regulates calcium and acts dualistically as an agonist to both amylin and calcitonin receptors, promoting bone formation while inhibiting bone resorption.
    Formula:C1401C5H240N4315NO48S2·5C2HF3O2
    Color and Shape:Solid
    Molecular weight:4007.93

    Ref: TM-T201476

    10mg
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    50mg
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  • FLLRN

    CAS:
    FLLRN is a biologically active peptide serving as a PAR1-specific antagonist.
    Formula:C31H51N9O7
    Color and Shape:Solid
    Molecular weight:661.79

    Ref: TM-T78545

    5mg
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    50mg
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  • T-10430


    T-10430 is a potent and orally active agonist of the leukotriene B4 receptor 2 (BLT2). It shows potential for use in psoriasis research.
    Formula:C17H22N6O
    Color and Shape:Solid
    Molecular weight:326.396

    Ref: TM-T204318

    10mg
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    50mg
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  • A 31472

    CAS:
    A 31472 is a tetracyclic spiro amine that has affinity for dopamine D-2 receptors.
    Formula:C22H22ClN
    Color and Shape:Solid
    Molecular weight:335.87

    Ref: TM-T26415

    25mg
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    50mg
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    100mg
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  • [Pro34]Neuropeptide Y, porcine

    CAS:
    [Pro34]Neuropeptide Y, porcine functions as a selective agonist for the NPY (Y1) receptor and induces vasoconstriction in the guinea pig's caval vein [1].
    Formula:C190H286N54O56
    Color and Shape:Solid
    Molecular weight:4222.63

    Ref: TM-TP2523

    10mg
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    50mg
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  • Prostaglandin F2α isopropyl ester

    CAS:
    PGF2α isopropyl ester is an ester prodrug of PGF2α with enhanced lipid solubility.
    Formula:C23H40O5
    Color and Shape:Solid
    Molecular weight:396.568

    Ref: TM-T38196

    1mg
    233.00€
    5mg
    1,018.00€
    10mg
    1,765.00€
  • CRL-42872 free base

    CAS:
    CRL-42872 free base is a bioactive chemical.
    Formula:C22H26N6O6S
    Color and Shape:Solid
    Molecular weight:502.54

    Ref: TM-T31098

    100mg
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    500mg
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  • GLP-1R agonist 29


    GLP-1R agonist 29 (Compound 20) is a GLP-1R agonist that induces hGLP-1R-mediated cAMP stimulation with an EC50 of 0.018 nM. It exhibits favorable pharmacokinetic properties and shows good in vivo exposure, with an AUC0-∞,sc of 77688 ng·h/mL.
    Color and Shape:Odour Solid

    Ref: TM-T206400

    10mg
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    50mg
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  • Hemokinin 1, human

    CAS:
    Endogenous P-like compound, NK1 receptor agonist; IC50: NK1-1.8 nM, NK3-370 nM, NK2-480 nM; boosts B-cell growth, antiapoptotic, lowers blood pressure in vivo.
    Formula:C54H84N14O14S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1185.4

    Ref: TM-TP1899

    1mg
    145.00€
  • Antidepressant agent 3


    Agent 3: orally active, antidepressant, anxiolytic, boosts performance and cognition.
    Formula:C17H30ClN5O2S
    Color and Shape:Solid
    Molecular weight:403.97

    Ref: TM-T75002

    5mg
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    50mg
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  • AP 811

    CAS:
    AP 811: Selective NPR3 antagonist, Ki of 0.48 nM, >20,000x selective over NPR1, blocks ANP-induced pump stimulation.
    Formula:C46H66N12O8
    Color and Shape:Solid
    Molecular weight:915.11

    Ref: TM-T38641

    5mg
    538.00€
  • Corticotropin-releasing factor (human) acetate


    Corticotropin-releasing factor (human) acetate stimulates to synthesize and secret adrenocorticotropin in the anterior pituitary.
    Purity:98.30%
    Color and Shape:Liquid

    Ref: TM-TP1144L

    1mg
    145.00€
    5mg
    472.00€
    10mg
    710.00€
    25mg
    1,274.00€
    50mg
    1,898.00€
  • 19(R)-HETE

    CAS:
    19(R)-HETE is a renal artery vasodilator and can be used to study angiotensin II-induced cardiac hypertrophy.
    Formula:C20H32O3
    Color and Shape:Solid
    Molecular weight:320.47

    Ref: TM-T36216

    25µg
    502.00€
    50µg
    938.00€
    100µg
    1,795.00€
  • Atenolol

    CAS:
    Atenolol (Tenormin) is a selective β1 receptor antagonist.
    Formula:C14H22N2O3
    Purity:99.07% - 99.95%
    Color and Shape:White Crystalline Powder Solid
    Molecular weight:266.34

    Ref: TM-T0007

    1mL*10mM (DMSO)
    50.00€
  • Xenin-8

    CAS:
    neurotensin-like peptide that modulate pancreatic insulin and glucagon secretion/effects
    Formula:C51H79N15O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1046.27

    Ref: TM-TP2209

    1mg
    283.00€
  • LCKLSL

    CAS:
    LCKLSL, an N-terminal hexapeptide, inhibits AnxA2 and tPA binding, reduces plasmin, and exhibits anti-angiogenic effects.
    Formula:C30H57N7O8S
    Molecular weight:675.89

    Ref: TM-T40614

    25mg
    1,034.00€
  • BPP-2


    BPP-2 is a GHSR ligand containing the element F. By labeling BPP-2 with the isotope 18F, a PET probe targeting GHSR can be produced. The binding affinity (Ki) of 18F-BPP-2 for GHSR is 274 nM.
    Formula:C27H28FN5O2
    Molecular weight:473.2227

    Ref: TM-T209024

    10mg
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    50mg
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