GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
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Subcategories of "GPCR/G-Protein"
5-HT Receptor
Adenosine Receptor
Adrenergic Receptor
Bombesin Receptor
Bradykinin Receptor
CXCR
CaSR
Cannabinoid Receptor
Cholecystokinin
Dopamine Receptor
Endothelin Receptor
GNRH Receptor
GPCR19
GRK
GTPase
Glucagon Receptor
Hedgehog/Smoothened
Histamine Receptor
LPA Receptor
Melatonin Receptor
OX Receptor
Opioid Receptor
PAFR
PKA
S1P Receptor
SGLT
Sigma receptor
Show 19 more subcategories
Products of "GPCR/G-Protein"
Perospirone
CAS:150915-41-6
Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.
Formula:
C23H30N4O2S
Purity:
98.86%
Color and Shape:
White Powder
Molecular weight:
426.57
Ref: TM-T4576
| 5mg | 43.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 107.00 € | ||
| 50mg | 189.00 € | ||
| 100mg | 322.00 € | ||
| 200mg | 451.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Neurokinin A(4-10) TFA(97559-35-8 free base)
Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].
Formula:
C36H55F3N8O12S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
880.93
Ref: TM-TP1385
| 1mg | 47.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 252.00 € | ||
| 25mg | 415.00 € | ||
| 50mg | 582.00 € | ||
| 100mg | 785.00 € | ||
| 200mg | 1,052.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
NPY 5RA972
CAS:439861-56-0
NPY 5RA972 is a neuropeptide Y Y5 receptor antagonist
Formula:
C21H25N3O2
Purity:
99.02%
Color and Shape:
Solid
Molecular weight:
351.44
Ref: TM-T23087
| 1mg | 46.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 135.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
SBI-115
CAS:882366-16-7
SBI-115 is an antagonist of TGR5. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via …
Formula:
C14H13ClN2O4S
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
340.78
Ref: TM-T7428
| 5mg | 52.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 217.00 € | ||
| 100mg | 348.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Litorin acetate(55749-97-8 Free base)
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.
Formula:
C53H72N14O13S
Purity:
97.64%
Color and Shape:
Liquid
Molecular weight:
1145.29
Ref: TM-T20604L
| 1mg | 83.00 € | ||
| 5mg | 207.00 € | ||
| 10mg | 332.00 € | ||
| 25mg | 546.00 € | ||
| 50mg | 801.00 € | ||
| 100mg | 1,100.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Chlorprothixene
CAS:113-59-7
Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first …
Formula:
C18H18ClNS
Purity:
98.77% - 99.69%
Color and Shape:
Pale Yellow Crystals Solid
Molecular weight:
315.86
Ref: TM-T0074
| 1g | 140.00 € | ||
| 100mg | 37.00 € | ||
| 200mg | 53.00 € | ||
| 500mg | 96.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
LY334370
CAS:182563-08-2
LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nM
Formula:
C21H22FN3O
Purity:
98.48%
Color and Shape:
Solid
Molecular weight:
351.42
Ref: TM-T4266
| 5mg | 45.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 187.00 € | ||
| 100mg | 272.00 € | ||
| 200mg | 375.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Sevoflurane
CAS:28523-86-6
Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.
Formula:
C4H3F7O
Purity:
99.78%
Color and Shape:
Less Oil Colorless Oil
Molecular weight:
200.05
Ref: TM-T22425
| 100mg | 234.00 € | ||
| 200mg | 350.00 € | ||
| 500mg | 588.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
CCG215022
CAS:1813527-81-9
CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 …
Formula:
C26H22FN7O3
Purity:
97.46% - 99.69%
Color and Shape:
Solid
Molecular weight:
499.5
Ref: TM-T3498
| 1mg | 94.00 € | ||
| 2mg | 138.00 € | ||
| 5mg | 231.00 € | ||
| 10mg | 369.00 € | ||
| 25mg | 616.00 € | ||
| 50mg | 877.00 € | ||
| 100mg | 1,196.00 € | ||
| 500mg | 2,385.00 € | ||
| 1mL*10mM (DMSO) | 257.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Felypressin
CAS:56-59-7
Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic …
Formula:
C46H65N13O11S2
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
1040.22
Ref: TM-T2568
| 2mg | 37.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 114.00 € | ||
| 50mg | 169.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Geissoschizine methyl ether
CAS:60314-89-8
Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social …
Formula:
C22H26N2O3
Purity:
99.68% - 99.86%
Color and Shape:
Solid
Molecular weight:
366.45
Ref: TM-TN1032
| 1mg | 135.00 € | ||
| 5mg | 395.00 € | ||
| 10mg | 578.00 € | ||
| 25mg | 899.00 € | ||
| 50mg | 1,203.00 € | ||
| 100mg | 1,626.00 € | ||
| 1mL*10mM (DMSO) | 373.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
VUF10460
CAS:1028327-66-3
VUF10460 is a non-imidazole histamine H4 receptor agonist.
Formula:
C15H19N5
Purity:
98.68% - 99.53%
Color and Shape:
Solid
Molecular weight:
269.34
Ref: TM-T3963
| 5mg | 34.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 164.00 € | ||
| 100mg | 247.00 € | ||
| 200mg | 365.00 € | ||
| 1mL*10mM (DMSO) | 39.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Leuphasyl TFA
CAS:67586-27-0
Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.
Formula:
C31H40F3N5O9
Purity:
98.79%
Color and Shape:
Solid
Molecular weight:
683.67
Ref: TM-T20435L
| 1mg | 83.00 € | ||
| 2mg | 107.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 780.00 € | ||
| 200mg | 1,034.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Ansofaxine hydrochloride
CAS:916918-84-8
Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).
Formula:
C24H32ClNO3
Purity:
99.57% - 99.77%
Color and Shape:
Solid
Molecular weight:
417.97
Ref: TM-T5380
| 1mg | 76.00 € | ||
| 5mg | 166.00 € | ||
| 10mg | 258.00 € | ||
| 25mg | 500.00 € | ||
| 50mg | 707.00 € | ||
| 100mg | 916.00 € | ||
| 1mL*10mM (DMSO) | 175.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Treprostinil
CAS:81846-19-7
Treprostinil (Orenitram) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).
Formula:
C23H34O5
Purity:
99.71%
Color and Shape:
Solid
Molecular weight:
390.51
Ref: TM-T5150
| 2mg | 46.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 268.00 € | ||
| 50mg | 448.00 € | ||
| 100mg | 640.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
BA 1 acetate(183241-31-8 free base)
BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer …
Formula:
C59H80N14O13
Purity:
95.3%
Color and Shape:
Solid
Molecular weight:
1193.35
Ref: TM-TP1913L1
| 1mg | 94.00 € | ||
| 5mg | 182.00 € | ||
| 10mg | 274.00 € | ||
| 25mg | 495.00 € | ||
| 50mg | 716.00 € | ||
| 100mg | 994.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Binodenoson
CAS:144348-08-3
Binodenoson (WRC 0470), a selective A2A adenosine receptor agonist, aids in coronary imaging.
Formula:
C17H25N7O4
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
391.42
Ref: TM-T9516
| 1mg | 137.00 € | ||
| 5mg | 282.00 € | ||
| 10mg | 424.00 € | ||
| 25mg | 701.00 € | ||
| 50mg | 937.00 € | ||
| 100mg | 1,319.00 € | ||
| 1mL*10mM (DMSO) | 311.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Nelotanserin
CAS:839713-36-9
Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B …
Formula:
C18H15BrF2N4O2
Purity:
98.01% - 98.42%
Color and Shape:
Solid
Molecular weight:
437.24
Ref: TM-T7350
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | 510.00 € | ||
| 500mg | 1,109.00 € | ||
| 1mL*10mM (DMSO) | 84.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Asapiprant
CAS:932372-01-5
Asapiprant (S-555739) is a potent and selective DP1 receptor antagonist (Ki: 0.44 nM). It exhibited …
Formula:
C24H27N3O7S
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
501.55
Ref: TM-T5386
| 1mg | 41.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 155.00 € | ||
| 25mg | 282.00 € | ||
| 50mg | 446.00 € | ||
| 100mg | 726.00 € | ||
| 200mg | 933.00 € | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy …
Formula:
C61H88N16O14
Purity:
98.1%
Color and Shape:
Solid
Molecular weight:
1269.45
Ref: TM-TP1434L
| 1mg | 75.00 € | ||
| 5mg | 131.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 322.00 € | ||
| 100mg | 487.00 € |
Estimated delivery in United States, on Tuesday 28 Jan 2025
