Inhibitors
Inhibitors are molecules that bind to enzymes, receptors, or other proteins to reduce or block their biological activity. These compounds are widely used in research to study biological pathways, understand disease mechanisms, and develop therapeutic drugs. Inhibitors play a crucial role in the treatment of various diseases, including cancer, cardiovascular diseases, and infections. At CymitQuimica, we provide a diverse range of high-quality inhibitors to support your research in biochemistry, cell biology, and pharmaceutical development.
Subcategories of "Inhibitors"
- Angiogenesis(2,687 products)
- Apoptosis(6,097 products)
- Cell Cycle/Checkpoint(4,691 products)
- Chromatin/Epigenetics(2,376 products)
- Cytoskeletal Signaling(1,472 products)
- DNA Damage/DNA Repair(2,921 products)
- Endocrinology/Hormones(3,611 products)
- Enzyme(3,655 products)
- GPCR/G-Protein(8,755 products)
- Immunology and Inflammation(3,765 products)
- Influenza Virus(298 products)
- JAK/STAT signaling(407 products)
- MAPK Signaling(1,230 products)
- Membrane Transporter/Ion Channel(2,947 products)
- Metabolism(9,940 products)
- Microbiology/Virology(7,347 products)
- Neuroscience(10,240 products)
- Other Inhibitors(36,533 products)
- Oxidation-Reduction(43 products)
- PI3K/Akt/mTOR Signaling(1,437 products)
- Proteases/Proteasome(1,675 products)
- Stem Cell and Derivatives(830 products)
- Tyrosine Kinase/Adaptors(2,028 products)
- Ubiquitination(1,682 products)
Show 16 more subcategories
Found 66582 products of "Inhibitors"
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U 19052
CAS:U 19052 is a Leukotriene D4 antagonist.Formula:C31H42O6SColor and Shape:SolidMolecular weight:542.73ROCK2-IN-6 hydrochloride
CAS:<p>ROCK2-IN-6 hydrochloride (Comp A)为一种选择性ROCK2抑制剂，适用于研究ROCK介导的疾病、自身免疫性病症与炎症。</p>Formula:C26H22ClF2N7OPurity:98%Color and Shape:SolidMolecular weight:521.95GNE-490
CAS:GNE-490 is an effective inhibitor of pan-PI3K with IC50s of 3.5 nM, 25 nM, 5.2 nM, 15 nM for PI3Kα, PI3Kβ, PI3Kδ and PI3Kγ, respectively.Formula:C18H22N6O2SPurity:99.77%Color and Shape:SolidMolecular weight:386.47KAT modulator-1
CAS:<p>KAT modulator-1 (Compound 3), an epigenetics research tool, selectively interacts with the full-length p300 protein but not its catalytic domain [1].</p>Formula:C20H36O2Purity:98%Color and Shape:SolidMolecular weight:308.5Naamidine A
CAS:Naamidine A is a marine alkaloid with a selective ability to inhibit epidermal growth factor receptor (EGFR)-dependent cellular proliferation.Formula:C23H23N5O4Color and Shape:SolidMolecular weight:433.46L-690488
CAS:L-690488 has more effective cell penetration than L-690330. L-690488 is a prodrug of L-690330 and is a selective inositol monophosphatase (IMPase) inhibitor.Formula:C32H52O16P2Purity:98%Color and Shape:SolidMolecular weight:754.69Anticancer agent 95
CAS:Quinazolinone Compound 95, also known as Compound 24, exhibits anticancer properties [1].Formula:C30H32ClN5O3Color and Shape:SolidMolecular weight:546.06Fosthiazate
CAS:<p>Fosthiazate is a broad-spectrum nematicide that combats a range of plant parasitic nematodes such as Meloidogyne spp., Globodera spp., and Pratylenchus spp., by</p>Formula:C9H18NO3PS2Purity:97.78%Color and Shape:SolidMolecular weight:283.35PHD-IN-2
CAS:<p>PHD-IN-2 (Compound 91), a potent PHD antagonist with an IC50 of less than 5 nM, effectively stimulates erythropoietin synthesis in HEP3B cells with an EC50 of</p>Formula:C26H27N7O4Purity:98%Color and Shape:SolidMolecular weight:501.54LY3154885
CAS:LY3154885 is an orally active dopamine D1 receptor orthosteric modulator (PAM) that reduces the risk of drug-drug interactions (DDI).Formula:C23H23Cl2N3O2Color and Shape:SolidMolecular weight:444.35Bioethanomethrin
CAS:Bioethanomethrin is a biochemical.Formula:C24H28O3Color and Shape:SolidMolecular weight:364.485-HT3-In-1
CAS:5-HT3-In-1 (compound example 8) exhabits with 5-HT3 inhibition activity.Formula:C16H21ClN4O3Purity:98%Color and Shape:SolidMolecular weight:352.82Cyclopropavir
CAS:<p>Cyclopropavir (Filociclovir; MBX-400) is a broad-spectrum anti-herpes drug effective against CMV and HHV-6/8 (EC50: 0.7-8 μM).</p>Formula:C11H13N5O3Purity:98%Color and Shape:SolidMolecular weight:263.25Amogastrin
CAS:Amogastrin can be used in conjunction with pertechnetate for gastric scintigraphy.Formula:C35H46N6O8SColor and Shape:SolidMolecular weight:710.84GX-395
CAS:GX-395 is a novel Nav1.7 inhibitor.Formula:C21H17ClF2N6O3S2Purity:98%Color and Shape:SolidMolecular weight:538.98Famitinib malate
CAS:Famitinib malate (SHR1020) is a potent oral kinase inhibitor targeting c-kit, VEGFR-2, and PDGFRβ, with IC50s 2.3, 4.7, 6.6 nM, useful for cancer research.Formula:C27H33FN4O7Color and Shape:SolidMolecular weight:544.57ISPA-28
CAS:ISPA-28: reversible PSAC antagonist via direct CLAG3 binding.Formula:C21H24N6O3Color and Shape:SolidMolecular weight:408.45KM05382
CAS:<p>KM05382 inhibits CDK9 and the transcription of GAPDH.</p>Formula:C20H19ClN2O3S2Color and Shape:SolidMolecular weight:434.96Nampt-IN-10 TFA
CAS:Nampt-IN-10 TFA, a NAMPT inhibitor, shows potency in A2780 (IC50: 5 nM) and CORL23 (IC50: 19 nM), suitable for ADC payloads.Formula:C29H29F4N5O4Color and Shape:SolidMolecular weight:587.21557SN38-PAB-Lys(MMT)-oxydiacetamide-PEG8-N3
CAS:<p>"SN38-PAB-Lys(MMT)-oxydiacetamide-PEG8-N3 is a drug-linker conjugate for antibody-drug conjugates (ADCs), consisting of the anti-cancer agent SN38 linked to Lys</p>Formula:C78H95N9O20Color and Shape:SolidMolecular weight:1478.64Pregnanolone sulfate (pyridinium)
CAS:<p>Pregnanolone sulfate pyridinium, an endogenous neurosteroid, inhibits NMDA receptors and exhibits neuroprotective properties [1].</p>Formula:C26H39NO5SPurity:98%Color and Shape:SolidMolecular weight:477.66SR11237
CAS:<p>SR11237 is a Pan retinoid X receptor (RXR) agonist.</p>Formula:C24H28O4Purity:98.79%Color and Shape:SolidMolecular weight:380.48DORA 42
CAS:DORA 42 is a dual antagonist of the orexin receptor OX1R and OX2R.Formula:C22H24N8OSPurity:98%Color and Shape:SolidMolecular weight:448.54DQP-997-74
CAS:Dihydroquinoline-pyrazoline DQP-997-74 (compound 2i) is a selective N-methyl-d-aspartate receptor (NMDAR) inhibitor that preferentially targets GluN2C/DFormula:C28H19Cl2F2N3O4Color and Shape:SolidMolecular weight:570.373-Hydroxyxanthone
CAS:<p>3-Hydroxyxanthone (3-Hydroxy-xanthen-9-one), a xanthone derivative, exhibits inhibitory effects on NADPH-catalyzed lipid peroxidation in human umbilical vein</p>Formula:C13H8O3Purity:98%Color and Shape:SolidMolecular weight:212.2NTE-122
CAS:NTE-122 is a competitive Acyl-CoA:cholesterol acyltransferase (ACAT) inhibitor.Formula:C38H59ClN6O2Purity:98%Color and Shape:SolidMolecular weight:667.38PTC725
CAS:PTC725 is a selective HCV 1b replicons inhibitor. It has been shown to target the nonstructural protein 4B.Formula:C23H18F4N6O2SPurity:98%Color and Shape:SolidMolecular weight:518.49FK 33-824
CAS:FK 33-824, a stable synthetic analog of methionine enkephalin, reversible with naloxone.Formula:C29H41N5O7SPurity:98%Color and Shape:SolidMolecular weight:603.73ICMT-IN-22
CAS:ICMT-IN-22 (compound 62) acts as an ICMT inhibitor with an IC50 value of 0.63 μM [1].Formula:C22H28ClNO2Color and Shape:SolidMolecular weight:373.92Glucocorticoid receptor agonist-1 phosphate Gly-Glu TFA
CAS:Glucocorticoid Receptor Agonist-1 Phosphate Gly-Glu (TFA) serves as a cleavable linker for the synthesis of Antibody-Drug Conjugates (ADCs).Formula:C44H51F3N3O15PColor and Shape:SolidMolecular weight:949.86LX-1031
CAS:LX-1031 is an effective inhibitor of tryptophan 5-hydroxylase. LX-1031 decreases serotonin (5-HT) synthesis peripherally.Formula:C28H25F3N4O4Purity:97.123% - 98.97%Color and Shape:SolidMolecular weight:538.52AP-C1
CAS:AP-C1 is a potent inhibitor of cGMP-dependent protein kinase II (cGKII), exhibiting a pIC50 value of 6.5, yet it only weakly inhibits cGKII-dependent anionFormula:C24H23N3O2Color and Shape:SolidMolecular weight:385.46IRAK4-IN-28
CAS:<p>IRAK4-IN-28 (compound 42), an orally-active IRAK4 inhibitor (IC50=8.9 nM), exhibits strong binding affinity with a Kd of 0.58 nM for the target enzyme.</p>Formula:C27H31N9O3Purity:98%Color and Shape:SolidMolecular weight:529.59AP-C7
CAS:AP-C7 is a selective inhibitor of cGMP-dependent protein kinase II (cGKII) with a pIC50 value of 5.0, demonstrating only weak inhibition of cGKII-dependentFormula:C18H15N5OColor and Shape:SolidMolecular weight:317.34AZD 4017
CAS:AZD 4017 is an inhibitor of 11β-Hydroxysteroid Dehydrogenase Type 1(11β-HSD1) (IC50: 7 nM).Formula:C22H33N3O3SPurity:99.61%Color and Shape:SolidMolecular weight:419.58GS-6201
CAS:GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor.Formula:C21H21F3N6O2Purity:99.78% - 99.94%Color and Shape:SolidMolecular weight:446.43MET kinase-IN-3
CAS:MET kinase-IN-3 is a potent, orally active MET inhibitor (IC50: 9.8 nM) that exhibits good broad-spectrum anti-proliferative effects on cancer cells.Formula:C25H16ClF2N5O2Color and Shape:SolidMolecular weight:491.88MAO-B-IN-26
CAS:MAO-B-IN-26 (Compound IC9) serves as both a MAO-B and acetylcholinesterase inhibitor.Formula:C17H12BrNOPurity:98%Color and Shape:SolidMolecular weight:326.19BRD4 Inhibitor-18
CAS:BRD4 Inhibitor-18: potent (IC50: 110 nM), impairs MV-4-11 cell growth, disrupts G0/G1 phase, and induces apoptosis.Formula:C26H26ClN3O3SColor and Shape:SolidMolecular weight:496.02A-357300
CAS:A-357300: potent reversible MetAP2 inhibitor, IC50=0.12 uM; promising for neuroblastoma treatment.Formula:C15H22ClN3O3SColor and Shape:SolidMolecular weight:359.87Pentixafor
CAS:<p>Pentixafor is a peptide that selectively targets the CXCR4 receptor and can be labeled with Gallium-68 (68Ga) for visualization using positron emission</p>Formula:C60H80N14O14Purity:98%Color and Shape:SolidMolecular weight:1221.36Leteprinim
CAS:<p>Leteprinim (AIT 082 acid) is an hypoxanthine derivative that stimulates in vitro neurite outgrowth and the production of adenosine and neurotrophins from</p>Formula:C15H13N5O4Purity:99.08%Color and Shape:SolidMolecular weight:327.29ICL-CCIC-0019
CAS:<p>ICL-CCIC-0019 inhibits ChoKα, causes G1 arrest, ER stress, and cancer cell apoptosis.</p>Formula:C26H44Br2N4Purity:99.54%Color and Shape:SolidMolecular weight:572.46(Rac)-BRD0705
CAS:<p>(Rac)-BRD0705 is a less active racemate of BRD0705. BRD0705 is an effective and selective inhibitor of GSK3α.</p>Formula:C20H23N3OPurity:99.7%Color and Shape:SolidMolecular weight:321.42NV-354
CAS:Mitochondria Modulator-1, a mitochondrial regulator, enhances ATP production in mitochondria.Formula:C9H15NO4SColor and Shape:SolidMolecular weight:233.29H-Gly-Leu-Phe-OH
CAS:<p>GLF (H-Gly-Leu-Phe-OH), a tripeptide isolated from α-lactalbumin with immunostimulatory properties, prevents alopecia, epidermal thickening, and adipocyte layer</p>Formula:C17H25N3O4Color and Shape:SolidMolecular weight:335.4KN-93 Phosphate
CAS:KN-93 (Phosphate) can competitively block the binding of calmodulin to the corresponding kinase.Cost-effective and quality-assured.Formula:C26H32ClN2O8PSPurity:99.58% - 99.93%Color and Shape:SolidMolecular weight:599.03Antituberculosis agent-6
CAS:<p>Antituberculosis agent-6: potent against M. tuberculosis (MIC 3.49 μM), antifungal (MIC 62.5 μM), high GI absorption.</p>Formula:C27H20F2N2O3Color and Shape:SolidMolecular weight:458.46GSK3491943
CAS:GSK3491943 is a potent TRPV4 inhibitor with IC50 = 3.2 nM. GSK3491943 is a potential agent for the treatment of heart failure and respiratory diseases.Formula:C18H16Cl2N2O5SColor and Shape:SolidMolecular weight:443.3Sampatrilat
CAS:Sampatrilat, an oral vasopeptidase inhibitor, more potently blocks C-domain ACE (Ki=13.8 nM) over N-domain (Ki=171.9 nM).Formula:C26H40N4O9SPurity:98%Color and Shape:SolidMolecular weight:584.68eeAChE-IN-2
CAS:eeAChE-IN-2 is a potent inhibitor of eeAChE, exhibiting inhibitory potency with an IC50 of 2 nM.Formula:C37H40N8O5SColor and Shape:SolidMolecular weight:708.83HIF-2α-IN-6
CAS:HIF-2α-IN-6 (117) is a HIF-2α inhibitor [1].Formula:C15H13F4NO3SColor and Shape:SolidMolecular weight:363.33Maropitant citrate anhydrous
CAS:Maropitant citrate anhydrous is a neurokinin (NK1) receptor antagonist.Formula:C38H48N2O8Color and Shape:SolidMolecular weight:660.8O-allyl-AP
O-allyl-AP is a neuroprotective and proliferative agent with significantly higher stimulatory effect than that of allopregnanolone.Formula:C24H38O2Color and Shape:SolidMolecular weight:358.57Bocodepsin hydrochloride
CAS:Bocodepsin hydrochloride (OKI-179) is a selective HDAC inhibitor with antitumor properties, efficacious via oral administration.Formula:C26H40ClN5O6S2Purity:98%Color and Shape:SolidMolecular weight:618.21Zabofloxacin
CAS:Zabofloxacin inhibits bacterial topoisomerases II/IV, effectively targeting gram-positive pathogens like S. aureus and S. pneumoniae.Formula:C19H20FN5O4Purity:98%Color and Shape:SolidMolecular weight:401.39HCV-IN-44
CAS:HCV-IN-44 (compound 28) is an inhibitor of the HCV NS5B protein, efficacious in suppressing HCV virus replication and useful for researching HCV infection [1].Formula:C24H26FN3O5SColor and Shape:SolidMolecular weight:487.54MC-VA-PABC-MMAE
CAS:MC-VA-PABC-MMAE is a conjugate consisting of the ADC linker peptide MC-VA-PABC and the cytotoxic agent monomethyl auristatin E (MMAE), a powerful inhibitor ofFormula:C65H99N9O14Color and Shape:SolidMolecular weight:1230.53Tuberculosis inhibitor 7
CAS:Tuberculosis inhibitor 7 (compound 2d), a 3-methoxy-2-phenylimidazo[1,2-b]pyridazine derivative, exhibits potent activity against Mycobacterium tuberculosis andFormula:C21H18FN3O2SColor and Shape:SolidMolecular weight:395.45Cholesterol 24-hydroxylase-IN-2
CAS:<p>Cholesterol 24-hydroxylase-IN-2 is a potent inhibitor of cholesterol 24-hydroxylase (CH24H or CYP46A1), exhibiting an IC50 value of 5.4 nM, and has potential</p>Formula:C20H23FN4OColor and Shape:SolidMolecular weight:354.42S1p receptor agonist 2
CAS:<p>S1P5-selective agonist; less so for S1P1/S1P3; useful for CNS disorders.</p>Formula:C24H23ClN2O4Color and Shape:SolidMolecular weight:438.9Atecegatran metoxil
CAS:Atecegatran Metoxil (AZD0837), an oral thrombin inhibitor in development for stroke prevention in atrial fibrillation, is well-tolerated with favorable PK.Formula:C22H23ClF2N4O5Color and Shape:SolidMolecular weight:496.89Mps1-IN-10
CAS:<p>Mps1-IN-6 (Compound 9) is a highly effective Mps1 inhibitor with an IC50 value of 6.4 nM and exhibits significant anti-proliferation and anti-tumor effects on</p>Formula:C24H27N7O2Color and Shape:SolidMolecular weight:445.52NBD-09027
CAS:NBD-09027 is an inhibitor of HIV-1 entry.Formula:C19H23ClN4O3SPurity:98%Color and Shape:SolidMolecular weight:422.93Antitumor agent-101
CAS:Antitumor agent-101 is a selective, covalent inhibitor targeting lysine methyltransferases G9a/GLP, demonstrating IC50 values of 8.5 nM for G9a and 5.5 nM forFormula:C26H38N6O3Purity:98%Color and Shape:SolidMolecular weight:482.62Borofalan(10B)
CAS:Borofalan(10B) (L-4-Boronophenylalanine) echibits antineoplastic effects.Formula:C9H12BNO4Purity:98.96% - 99.81%Color and Shape:SolidMolecular weight:208.21CD73-IN-11
CAS:CD73-IN-11 is a potent inhibitor used to prepare medication for cancer by blocking adenosine production, which fosters tumor growth.Formula:C14H10F3N5O2Color and Shape:SolidMolecular weight:337.26IDP-73152
CAS:IDP-73152 is a peptide deformylase inhibitor.Formula:C28H41F3N4O4Color and Shape:SolidMolecular weight:554.64PF-02575799
CAS:PF-02575799 is an inhibitor of microsomal triglyceride transfer protein (MTP) (IC50: 0.77±0.29 nM).Formula:C42H37FN4O4Purity:98%Color and Shape:SolidMolecular weight:680.77Ethaverine HBr
CAS:Ethaverine HBr is the parasympathetic nervous system actions inhibitor.Formula:C24H30BrNO4Color and Shape:SolidMolecular weight:476.40Leucettinib-92
CAS:<p>Leucettinib-92 (compound 92) is a kinase inhibitor selective for DYRK/CLK families, displaying IC50 values of 147 nM (CLK1), 39 nM (CLK2), 5.2 nM (CLK4), 0.8 μM</p>Formula:C21H22N4OSPurity:98%Color and Shape:SolidMolecular weight:378.494'-Azidothymidine 5'-triphosphate
CAS:4'-Azidothymidine 5'-triphosphate targets HIV-1 reverse transcriptase and human DNA polymerases alpha & beta.Formula:C10H16N5O14P3Color and Shape:SolidMolecular weight:523.18SAFit1
CAS:SAFit1 is an inhibitor of FK506 binding protein 51 (FKBP51)-specific (Ki: 4±0.3 nM).Formula:C42H53NO11Purity:98%Color and Shape:SolidMolecular weight:747.87S07-1066
CAS:S07-1066, an aldo-keto reductase 1C3 (AKR1C3) inhibitor, enhances doxorubicin (DOX) cytotoxicity by selectively inhibiting AKR1C3-mediated reduction of DOX andFormula:C16H11Cl2FO2Purity:98%Color and Shape:SolidMolecular weight:325.16Sonepiprazole
CAS:Sonepiprazole (PNU-101387G) is a chemical compound known for its selective antagonistic properties toward D4 dopamine receptors, exhibiting dissociationFormula:C21H27N3O3SPurity:99.81%Color and Shape:SolidMolecular weight:401.52CAY10410
CAS:CAY10410 is a PGD2/PGJ2 analog, modified for enhanced PPARγ activity and metabolic stability, non-toxic to SH-SY5Y cells at ≤25μM.Formula:C20H30O3Color and Shape:SolidMolecular weight:318.45BMS-538203
CAS:BMS-538203 is a novel HIV integrase inhibitor.Formula:C12H12FNO5Purity:98%Color and Shape:SolidMolecular weight:269.23FK-143
CAS:<p>FK-143 is a 5-alpha reductase inhibitor.</p>Formula:C40H44N2O3Color and Shape:SolidMolecular weight:600.79CCG-63802
CAS:CCG-63802 is a reversible small-molecule inhibitor of regulator of G protein signaling (RGS) proteins.Formula:C26H18N4O2SPurity:90%Color and Shape:SolidMolecular weight:450.51EHT 5372
CAS:EHT 5372 inhibits DYRK kinases; IC50: 0.22-221 nM for DYRK1A/B, DYRK2/3, CLK1/2/4, GSK-3α/β.Formula:C17H11Cl2N5OSColor and Shape:SolidMolecular weight:404.27Nitro-coronene
CAS:Nitro-coronene-derived carbon dots can serve as lysosome-targeting agents for near-infrared light-induced photothermal cancer therapy research.Formula:C24H8N4O8Color and Shape:SolidMolecular weight:480.34ICMT-IN-50
CAS:ICMT-IN-50 (compound 3) serves as an inhibitor of ICMT with an IC50 value of 0.31 µM [1].Formula:C27H31NO3Color and Shape:SolidMolecular weight:417.54α-HNJNAc
CAS:<p>α-HNJNAc is a potent, competitive hexosaminidases inhibitor that does not interfer with other glycosidases [1].</p>Formula:C9H18N2O5Color and Shape:SolidMolecular weight:234.25Arrhythmias-Targeting Compound 1
CAS:Arrhythmias-Targeting Compound 1 is a compound. It is used in the research of arrhythmias.Formula:C22H32N4O2Purity:98%Color and Shape:SolidMolecular weight:384.52HDAC8-IN-4
CAS:<p>HDAC8-IN-4 is a selective HDAC8 inhibitor, exhibiting inhibitory activity with IC50 values of 0.15 μM for HDAC8 and 12 μM for HDAC3 [1].</p>Formula:C17H14N2O2S2Purity:98%Color and Shape:SolidMolecular weight:342.44O-Demethyl apixaban sulfate
CAS:O-Demethyl apixaban sulfate, a metabolite of the factor Xa inhibitor Apixaban, is in development for treating thrombotic diseases.Formula:C24H23N5O7SColor and Shape:SolidMolecular weight:525.53Ono-RS 347
CAS:Ono-RS 347 is a leukotriene antagonists with the activity of SRS-A antagonist.Formula:C26H25N5O4Purity:98%Color and Shape:SolidMolecular weight:471.51Firuglipel
CAS:<p>Firuglipel is an orally available and selective agonist of GPR119.</p>Formula:C25H26FN3O5Purity:98%Color and Shape:SolidMolecular weight:467.49A81988
CAS:A81988 is an antagonist of angiotensin AT1 receptors.Formula:C23H22N6O2Purity:98%Color and Shape:SolidMolecular weight:414.46NHS-SS-Ph
CAS:NHS-SS-Ph, a cleavable linker utilized in antibody-drug conjugate (ADC) synthesis, facilitates the release of therapeutic agents under specific intracellularFormula:C16H17NO7S2Color and Shape:SolidMolecular weight:399.44ATR-IN-5
CAS:ATR-IN-5 is a potent inhibitor of ATR, a member of the PIKK family of proteins involved in genome stability and DNA damage repair.Formula:C27H32F3N9OColor and Shape:SolidMolecular weight:555.6GPi 688
CAS:glycogen phosphorylase inhibitorFormula:C19H18ClN3O4SPurity:98%Color and Shape:SolidMolecular weight:419.882′,3′-cGMP triethylamine
CAS:Guanosine 2',3'-cyclic phosphate triethylamine, commonly known as 2′,3′-cGMP triethylamine, is an active compound utilizable in numerous research investigationsFormula:C16H27N6O7PColor and Shape:SolidMolecular weight:446.4RO116-9132/238
CAS:<p>RO116-9132/238 is a bioactive chemical.</p>Formula:C28H40Cl2N3O4Color and Shape:SolidMolecular weight:553.54Eleven-Nineteen-Leukemia Protein IN-2
CAS:Eleven-Nineteen-Leukemia Protein IN-2 (compound 23), an ENL inhibitor, exhibits an IC50 of 10.7 nM and is utilized for leukemia research [1].Formula:C22H23N5O2Purity:98%Color and Shape:SolidMolecular weight:389.45ICMT-IN-14
CAS:ICMT-IN-14 (compound 50) serves as an inhibitor of isoprenylcysteine carboxyl methyltransferase (ICMT), exhibiting potent activity with an IC50 of 0.025 μM [1].Formula:C21H25ClFNOColor and Shape:SolidMolecular weight:361.88WAY-606376
CAS:WAY-606376 具有潜在的抗肿瘤活性，可用于研究免疫疾病。Formula:C18H13N3O2SPurity:99.48%Color and Shape:SolidMolecular weight:335.38AU1235
CAS:<p>AU1235 is a Mycobacterium tuberculosis inhibitor.</p>Formula:C17H19F3N2OPurity:99.54% - 99.87%Color and Shape:SolidMolecular weight:324.34GSK761
GSK761 inhibits SP140 (IC50: 77.79 nM), hinders monocyte-to-macrophage differentiation, and prompts CD206+ regulatory macrophages.Formula:C40H46N4O4Color and Shape:SolidMolecular weight:646.82β3-AR agonist 2
CAS:β3-AR agonist 2 is a potent and selective agonist of β3-adrenergic receptor (β3-AR with an EC50 of 8 nM).Formula:C27H38N4O7SPurity:98%Color and Shape:SolidMolecular weight:562.68Lepadin H
CAS:Lepadin H, a marine alkaloid and ferroptosis inducer, exhibits significant cytotoxicity by promoting p53 expression, escalating ROS production, and enhancingFormula:C26H45NO3Purity:98%Color and Shape:SolidMolecular weight:419.64GNE 220
CAS:GNE-220 is a potent and selective inhibitor of MAP4K4 (IC50: 7 nM).Formula:C25H26N8Purity:98%Color and Shape:SolidMolecular weight:438.53E1R
CAS:E1R is a positive sigma-1 receptor (Sig1R PAM) allosteric modulator. It has a cognition-enhancing activity.Formula:C13H16N2O2Color and Shape:SolidMolecular weight:232.28E2072
CAS:E2072 is a potent and selective thiol-based Glutamate Carboxypeptidase II (GCP-II) inhibitor.Formula:C16H14O4SColor and Shape:SolidMolecular weight:302.35mTOR inhibitor-11
CAS:<p>mTOR inhibitor-11 (Compound 9) is a brain-penetrant compound capable of inhibiting mTOR with an IC50 of 21 nM for pS6.</p>Formula:C21H26N6O2Purity:98%Color and Shape:SolidMolecular weight:394.47CD73-IN-4
CAS:CD73-IN-4 is a potent and selective methylenephosphonic acid CD73 inhibitorFormula:C16H23ClN5O7PPurity:98.61%Color and Shape:SolidMolecular weight:463.81ROCK2-IN-2
CAS:ROCK2-IN-2 is a selective inhibitor of ROCK2 (IC50 of <1 μM).Formula:C18H12N6OSPurity:99.65%Color and Shape:SolidMolecular weight:360.39HSP70/SIRT2-IN-2
CAS:<p>HSP70/SIRT2-IN-2 (Compounds 1a), a dual inhibitor of SIRT2 and HSP70, exhibits an IC50 of 45.1±5.0 μM against SIRT2 and demonstrates antitumor activity [1].</p>Formula:C17H13N3S3Purity:98%Color and Shape:SolidMolecular weight:355.5Cynandione A
CAS:Cynandione A is an acetophenone derived from Cynanchum wilfordii with anti-inflammatory activity.Formula:C16H14O6Purity:99.62%Color and Shape:SolidMolecular weight:302.28Anticancer agent 166
CAS:Compound 166, also referred to as compound 3, exhibits potent anticancer properties, demonstrating significant inhibitory activity against Caco-2 cells with anFormula:C19H14OSColor and Shape:SolidMolecular weight:290.38CGP 64213
CAS:CGP 64213 is a GABAb receptor agonist.Formula:C26H36IN2O7PPurity:98%Color and Shape:SolidMolecular weight:646.45YM-08
CAS:<p>YM-08 (Compound 7a), a brain-penetrant SIRT2 inhibitor, exhibits an IC50 of 19.9 μM. Additionally, it acts as an inhibitor of Hsp70 [1].</p>Formula:C19H17N3OS2Purity:98%Color and Shape:SolidMolecular weight:367.49Duocarmycin MB
CAS:<p>Duocarmycin MB, an ADC toxin and DNA alkylating agent, combats multi-drug resistant cells.</p>Formula:C27H26ClN3O4Purity:98%Color and Shape:SolidMolecular weight:491.97DY-46-2
CAS:DY-46-2 is a DNMT3A inhibitor (IC50: 0.39 ± 0.23 μM) with anticancer activity and is used in cancer and tumor research.Formula:C19H22N6O5SPurity:99.12% - 99.12%Color and Shape:SolidMolecular weight:446.48Du011
CAS:Du011 is a biogenesis inhibitor of the E.Formula:C20H15F2NO4SColor and Shape:SolidMolecular weight:403.4Anticancer agent 127
CAS:<p>Anticancer agent 127 (142D6), an IAP inhibitor, covalently binds to the BIR3 domains of XIAP, cIAP1, and cIAP2, with IC50 values of 12 nM, 14 nM, and 9 nM,</p>Formula:C26H37FN4O6SPurity:98%Color and Shape:SolidMolecular weight:552.66SOS1-IN-14
CAS:SOS1-IN-14 是选择性的、有效的、口服具有活力的 SOS1 抑制剂 (IC50: 3.9 nM)。SOS1-IN-14 能够利用 P-糖蛋白介导的外排机制在肠道内被吸收。SOS1-IN-14 能够用于 KRAS 突变的癌症的研究，且抑瘤效果比 BI-3406 好。Formula:C29H29F3N6O2Color and Shape:SolidMolecular weight:550.57BRD5648
CAS:BRD5648 ((R)-BRD0705) is an inactive (R)-enantiomer of BRD0705.Formula:C20H23N3OPurity:99.89%Color and Shape:SolidMolecular weight:321.42S1P1 agonist 6 hemicalcium
CAS:<p>Compound I (S1P1 agonist 6 hemicalcium) is an S1P1 agonist that diminishes autoimmune activity by inhibiting lymphocyte trafficking, and serves as an</p>Formula:C25H26F3NO3CaPurity:98%Color and Shape:SolidMolecular weight:465.51Fervenulin
CAS:<p>Fervenulin, from Streptomyces sp. CMU-MH021, halts egg hatch (MIC: 30 μg/mL) and kills J2 larvae (MIC: 120 μg/mL) of M. incognita.</p>Formula:C7H7N5O2Purity:99.75%Color and Shape:SolidMolecular weight:193.16(Rac)-AMG8379
CAS:<p>(Rac)-AMG8379 ((Rac)-AMG8380) is a racemate of AMG8379 which is an orally active and selective sulfonamide NaV1.7 antagonist.</p>Formula:C25H16ClF2N3O5SPurity:99.6%Color and Shape:SolidMolecular weight:543.93RIP2 kinase inhibitor 1
CAS:Potent RIP2 kinase inhibitor with 0.03 μM IC50, selective for autoimmune disease treatment.Formula:C17H17N5O2SPurity:98%Color and Shape:SolidMolecular weight:355.41Biricodar
CAS:<p>Biricodar is a P-glycoprotein and MRP-1 modulator.</p>Formula:C34H41N3O7Purity:98%Color and Shape:SolidMolecular weight:603.71CS-526
CAS:CS-526 is a reversible proton pump inhibitor targeting the K+ site on H+,K+-ATPase, reducing gastric acid secretion and preventing mucosal lesions.Formula:C20H22FN3OColor and Shape:SolidMolecular weight:339.41TZP-102
CAS:TZP-102 is a potent, oral, ghrelin receptor agonist that has been shown to improve diabetic gastroparesis symptoms.Formula:C28H44N4O4Color and Shape:SolidMolecular weight:500.67Alatrofloxacin
CAS:Alatrofloxacin is a prodrug of trovafloxacin.Formula:C26H25F3N6O5Color and Shape:SolidMolecular weight:558.51TIE-2/VEGFR-2 kinase-IN-5
CAS:TIE-2/VEGFR-2 kinase-IN-5 is a TIE-2 and VEGFR-2 tyrosine kinase receptor inhibitor commonly used in biomedical research related to angiogenesis.Formula:C21H13F6N5O2Purity:99.79%Color and Shape:SolidMolecular weight:481.35A1AT modulator 1
CAS:A1AT Modulator 1 potently inhibits Z α1-antitrypsin (A1AT) polymerization, exhibiting a pIC50 of 8.3 [1].Formula:C21H23FN2O3Color and Shape:SolidMolecular weight:370.42Simotinib
CAS:Simotinib (AL-6802) is an EGFR tyrosine kinase inhibitor (IC50 : 19.9 nM) with antitumour activity for the study of non-small cell lung cancer.Formula:C25H26ClFN4O4Purity:99.7%Color and Shape:SolidMolecular weight:500.95Acetylaleuritolic acid
CAS:<p>Acetylaleuritolic acid, a pentacyclic triterpenoid from Garcinia miniata leaves, inhibits P-388 leukemia.</p>Formula:C32H50O4Color and Shape:SolidMolecular weight:498.74Laninamivir Octanoate Monohydrate
CAS:Laninamivir Octanoate Monohydrate is a neuraminidase inhibitor.Formula:C21H38N4O9Purity:98%Color and Shape:SolidMolecular weight:490.55AKB-6899
CAS:<p>AKB-6899 is an inhibitor of prolyl hydroxylase domain 3 (PHD3) and increases the soluble form of the VEGF receptor (sVEGFR-1) production from GM-CSF-treated</p>Formula:C14H11FN2O4Purity:97.87%Color and Shape:SolidMolecular weight:290.25L 663581
CAS:L 663581 is the benzodiazepine receptor partial agonist.Formula:C17H16ClN5O2Purity:98%Color and Shape:SolidMolecular weight:357.79Deacylketoconazole
CAS:Deacylketoconazole (Deacyl ketoconazole) is a Ketoconazole derivative and is also an antifungal agent.Formula:C24H26Cl2N4O3Purity:98.35%Color and Shape:SolidMolecular weight:489.395-HT2A&5-HT2C agonist-1
CAS:<p>5-HT2A&5-HT2C agonist-1 (Example 2) is a dual-acting agent targeting the 5-HT2A and 5-HT2C receptors with respective IC50 values of 196 nM and 0.9 nM.</p>Formula:C14H20N2OPurity:98%Color and Shape:SolidMolecular weight:232.32NBI 35965 methanesulfonate
CAS:NBI 35965 hydrochloride is a CRF1 antagonist.Formula:C22H26Cl2N4O3SPurity:98%Color and Shape:SolidMolecular weight:497.44Glucocorticoid receptor agonist-1 phosphate Gly-Glu-Br
CAS:Glucocorticoid Receptor Agonist-1 Phosphate (Gly-Glu-Br) is an antibody-drug conjugate (ADC) linker utilized in the synthesis of ABBV-154, ABBV-927, ABBV-368,Formula:C44H51BrN3O14PColor and Shape:SolidMolecular weight:956.77ICAM-1-IN-1
CAS:<p>ICAM-1-IN-1 is a potent and selective E-selectin(IC50 = 7 nM) and ICAM-1(IC50 = 5 nM) inhibitor.</p>Formula:C15H11BrN2O2SPurity:99.67%Color and Shape:SolidMolecular weight:363.23L 708286
CAS:L 708286 is an agent of peptide-based phenethylcarbamoyldifluoromethylene. It is a slow-binding inhibitor of human leucocyte elastase (HLE).Formula:C25H34F2N4O5Purity:98%Color and Shape:SolidMolecular weight:508.56Acifluorfen-methyl
CAS:Acifluorfen-methyl, a photobleaching herbicide [1], functions as an inhibitor of the enzyme protoporphyrinogen oxidase (Protox), which is crucial for heme andFormula:C15H9ClF3NO5Purity:98%Color and Shape:SolidMolecular weight:375.68PZ-II-029
CAS:<p>PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.</p>Formula:C18H15N3O3Purity:99.79%Color and Shape:SolidMolecular weight:321.33KRAS G12C inhibitor 41
CAS:<p>KRAS G12C inhibitor 41 targets a key signaling protein, potentially aiding cancer research.</p>Formula:C36H37ClFN9O2Color and Shape:SolidMolecular weight:682.19PPO-IN-2
CAS:PPO-IN-2 is a protoporphyrinogen IX oxidase inhibitor, exhibiting a Ki value of 16 nM [1].Formula:C17H15ClFN3O2S2Color and Shape:SolidMolecular weight:411.9A 77003
CAS:<p>A 77003 is a HIV-1 protease inhibitor. A77003 impairs HIV-1 protease-mediated Gag processing.</p>Formula:C44H58N8O6Color and Shape:SolidMolecular weight:794.98BRD7-IN-1
CAS:BRD7-IN-1, a BI7273 derivative, forms PROTAC VZ185, targeting BRD7/9 with DC50s of 4.5/1.8 nM via VHL ligand linkage.Formula:C22H28Cl2N4O3Purity:98.95%Color and Shape:SolidMolecular weight:467.39Oxycodegol phosphate
CAS:Oxycodegol phosphate is a mu-opioid agonist used in the treatment of Moderate to Severe Chronic Low Back PainFormula:C31H50NO13PColor and Shape:SolidMolecular weight:675.71Mal-EGGGG-PEG8-amide-bis(deoxyglucitol)
CAS:<p>Mal-EGGGG-PEG8-amide-bis(deoxyglucitol) is a cleavable linker utilized in antibody-drug conjugates (ADCs).</p>Formula:C55H94N10O31Color and Shape:SolidMolecular weight:1391.38CKD-519
CAS:CKD-519: A CETP inhibitor with an IC50 of 2.3 nM, blocking cholesteryl ester transfer in serum.Formula:C31H34F7NO3Color and Shape:SolidMolecular weight:601.6NGD 98-2 hydrochloride
corticotropin-releasing factor receptor 1 (CRF1) antagonistFormula:C19H24F3N3O3·HClPurity:98%Color and Shape:SolidMolecular weight:435.873-O-Acetyl-20-Hydroxyecdysone
CAS:3-O-Acetyl-20-Hydroxyecdysone, a steroid extracted from the roots of Cyanotis arachnoidea C.B.Clark, is characterized by its unique structural modifications.Formula:C29H46O8Purity:99.54%Color and Shape:SolidMolecular weight:522.67JNJ4796
CAS:JNJ4796 is an oral fusion inhibitor that neutralizes influenza A group 1 by blocking HA-mediated fusion, mimicking bnAbs.Formula:C28H27N9O3Purity:98%Color and Shape:SolidMolecular weight:537.57NIBR-1282
CAS:<p>NIBR-1282 is a CCR5 antagonist.</p>Formula:C30H37N5O2Color and Shape:SolidMolecular weight:499.65Avarofloxacin
CAS:Avarofloxacin (JNJ-Q2) is a fluoroquinolone for treating bacterial skin infections and pneumonia.Formula:C21H23F2N3O4Color and Shape:SolidMolecular weight:419.42SARS-CoV-2-IN-66
CAS:<p>SARS-CoV-2-IN-66 (1), a derivative of vitamin K, functions as an inhibitor of SARS-CoV-2, exhibiting an effective concentration (EC50) of 70.8 μM in VeroE6/</p>Formula:C28H30O2Purity:98%Color and Shape:SolidMolecular weight:398.54BVDU 5′-Triphosphate
CAS:<p>BVDU 5′-Triphosphate is an antiviral agent labeled with 5′-Triphosphate that specifically targets viral DNA polymerase.</p>Formula:C11H16BrN2O14P3Purity:98%Color and Shape:SolidMolecular weight:573.08Cisd2 agonist 2
CAS:<p>Cisd2 agonist 2 (compound 6), with an EC50 of 191 nM, is an orally active activator of Cisd2, a protein whose levels are associated with nonalcoholic fatty</p>Formula:C14H14N2O4SColor and Shape:SolidMolecular weight:306.34YM348
CAS:YM348 is an effective and orally active 5-HT2C receptor agonist. YM348 also shows a high affinity for the cloned human 5-HT2C receptor (Ki: 0.89 nM).Formula:C14H17N3OPurity:98%Color and Shape:SolidMolecular weight:243.3Brepocitinib
CAS:Brepocitinib (PF-06700841) is a potent dual JAK1/TYK2 inhibitor (IC50s: 17 nM/23 nM). Brepocitinib also inhibits JAK2/3 (IC50s: 77 nM/6.49 μM).Formula:C18H21F2N7OPurity:99.82%Color and Shape:SolidMolecular weight:389.4Physachenolide C
CAS:<p>Physachenolide C, a selective BET inhibitor, induces apoptosis and arrests the cell cycle at the G0-G1 phase, exhibiting antitumor activity [1].</p>Formula:C30H40O9Purity:98%Color and Shape:SolidMolecular weight:544.63Lalioside
CAS:<p>Lalioside is a potent accelerator of neurite outgrowth.</p>Formula:C14H18O10Color and Shape:SolidMolecular weight:346.29PU-48
CAS:PU-48 is a potent inhibitor of urea transporters A (UT-A) with an IC50 value of 0.32 μM, exhibiting a significant diuretic effect in mouse models withoutFormula:C14H12N2O3SColor and Shape:SolidMolecular weight:288.32GPR119 agonist 2
CAS:GPR119 agonist 2 (compound 43), an orally active agonist of GPR119, exhibits favorable pharmacokinetic properties in rodents and has demonstrated efficacy inFormula:C23H24FN5O4S2Color and Shape:SolidMolecular weight:517.6NT-0796
CAS:<p>NT-0796 is an inflammasome NLRP3 inhibitor that inhibits NLRP3 activation.NT-0796 is a potential NDT-19795 delivery vector.</p>Formula:C23H27N3O4Purity:99.67%Color and Shape:SolidMolecular weight:409.48p-NH2-CHX-A"-DTPA
CAS:<p>p-NH2-CHX-A"-DTPA is a bifunctional chelating agent [1].</p>Formula:C25H36N4O10Color and Shape:SolidMolecular weight:552.57Melafolone
CAS:Melafolone: natural COX-2/EGFR inhibitor, enhances PD-1 therapy by normalizing tumor vessels, lowers PD-L1.Formula:C22H24O7Color and Shape:SolidMolecular weight:400.42CGC 11093
CAS:<p>CGC 11093: A polyamine analog inhibiting human prostate tumor growth in mice; may help regress choroidal neovascularization.</p>Formula:C17H42Cl4N4Color and Shape:SolidMolecular weight:444.35TCS 21311
CAS:<p>TCS 21311 (NIBR3049) selectively inhibits JAK3 (IC50: 8 nM) and PKCα/θ & GSK3β; >100x selective over JAK1, JAK2, TYK2.</p>Formula:C27H25F3N4O4Purity:99.39% - ≥98%Color and Shape:SolidMolecular weight:526.51Proteasome-IN-4
Proteasome-IN-4, a potent non-covalent inhibitor (IC50=8.39nM), halts cancer cell growth, useful for oncology studies.Formula:C44H58N6O5Color and Shape:SolidMolecular weight:750.97Teropavimab
CAS:<p>Teropavimab (3BNC117-LS), an antibody, is utilized in the research of HIV infection [1].</p>Color and Shape:LiquidDuostatin 5
CAS:<p>Duostatin 5 (Duo-5) is a sea hare toxin analog commonly used in the synthesis of ADC compounds.</p>Formula:C40H69N9O6Purity:96.98%Color and Shape:SolidMolecular weight:772.03Inogatran
CAS:Inogatran is a synthetic thrombin inhibitor, developed for the possible treatment and prophylaxis of venous and arterial thrombotic diseases.Formula:C21H38N6O4Purity:98%Color and Shape:SolidMolecular weight:438.56JNJ-46281222
CAS:JNJ-46281222: mGlu2-selective, potent PAM, Kd = 1.7 nM, pEC50 = 7.71.Formula:C23H25F3N4Color and Shape:SolidMolecular weight:414.47BMS-962212
CAS:BMS-962212: reversible, selective FXIa blocker, well-tolerated, quick PD effect, rapid clearance, alters clotting time/activity.Formula:C32H28ClFN8O5Purity:98%Color and Shape:SolidMolecular weight:659.07MLN-3897
CAS:MLN-3897 is an oral CCR1 antagonist, Ki 2.3 nM, blocks 125I-MIP-1α binding, and inhibits Akt signaling in MM cells.Formula:C30H31ClN2O4Purity:98.62%Color and Shape:SolidMolecular weight:519.032-Methoxyestrone
CAS:2-Methoxyestrone is a methoxylated catechol estrogen and the principal metabolite of 2-hydroxyestrone, a nonuterotropic metabolite of estradiol.Formula:C19H24O3Purity:97.07% - 99.18%Color and Shape:SolidMolecular weight:300.39MDL-19744A
CAS:<p>MDL-19744A is an alpha 1-adrenergic receptor antagonist and renal vasodilator.</p>Formula:C21H25NO3SColor and Shape:SolidMolecular weight:371.49Taragarestrant
CAS:Taragarestrant (D-0502), an oral estrogen receptor degrader, combats ER+ breast cancer in research.Formula:C25H25Cl2FN2O2Color and Shape:SolidMolecular weight:475.38L-739758
CAS:<p>L-739758 is a glycoprotein IIb/IIIa inhibitor.</p>Formula:C22H26N4O5S3Color and Shape:SolidMolecular weight:522.66CPUY201112
CAS:<p>CPUY201112, a novel inhibitor of heat shock protein Hsp90, induces p53-mediated apoptosis in MCF-7 cells.</p>Formula:C19H23N3O4Color and Shape:SolidMolecular weight:357.4CAL-130 Racemate
CAS:CAL-130 Racemate is the racemate of CAL-130. CAL-130 is a PI3Kδ and PI3Kγ inhibitor (IC50s: 1.3 and 6.1 nM).Formula:C23H22N8OPurity:98%Color and Shape:SolidMolecular weight:426.47BDW568
CAS:BDW568, a prodrug of BDW-OH, serves as a stimulator of interferon genes (STING) agonist.Formula:C12H12N4O2S2Color and Shape:SolidMolecular weight:308.38Zika virus-IN-3
CAS:Zika virus-IN-3 (Compd 7) is a Zika virus inhibitor, with an EC 50 of 3.4 μM [1].Formula:C23H20ClN3OColor and Shape:SolidMolecular weight:389.88CDD-1819
CAS:<p>CDD-1819, a non-covalent and non-peptide compound, serves as a potent SARS-CoV-2 Mpro inhibitor, exhibiting a K i value of 5 nM.</p>Formula:C35H31N5O2Purity:98%Color and Shape:SolidMolecular weight:553.65sPLA2 inhibitor 1
CAS:KH064 is a sPLA2-IIA inhibitor of oral activity.Formula:C31H37NO4Color and Shape:SolidMolecular weight:487.63Ilepatril
CAS:Ilepatril, also known as AVE-7688, is a vasopeptidase inhibitor for the treatment of hypertension.Formula:C22H28N2O5SColor and Shape:SolidMolecular weight:432.53N-type calcium channel blocker-1
CAS:N-type calcium channel blocker-1 is an orally active analgesic agent,shows high affinity to functionally block N-type calcium channels.Formula:C31H47N3Purity:98%Color and Shape:SolidMolecular weight:461.73K-Ras G12C-IN-1
CAS:K-Ras G12C-IN-1 is a novel and irreversible inhibitor of mutant K-ras G12C.Formula:C22H23Cl2N3O3Color and Shape:SolidMolecular weight:448.34ATM-IN-1
CAS:<p>ATM-IN-1 is a potent inhibitor of ATM. ATM-IN-1 has shown research potential in cancer and neurological diseases.</p>Formula:C30H36N6O3Color and Shape:SolidMolecular weight:528.65BMS-194449
CAS:BMS-194449 is a full beta 3 agonist.Formula:C24H24F4N2O6SColor and Shape:SolidMolecular weight:544.52Licostinel
CAS:<p>Licostinel (CGP 63446) is a glutamate receptor antagonist. Licostinel protects against permanent focal cerebral ischemia.</p>Formula:C8H3Cl2N3O4Purity:98.02%Color and Shape:SolidMolecular weight:276.03CCG-232964
CAS:<p>CCG-232964 is an orally active Rho/MRTF/SRF inhibitor that suppresses LPA-induced CTGF gene expression [1].</p>Formula:C15H15ClN2O3SPurity:98%Color and Shape:SolidMolecular weight:338.81Quercetin 7-glucuronide
CAS:<p>Quercetin 7-glucuronide (Quercetin 7-O-β-glucuronide), a Quercetin metabolite found in Madagascarian Uncarina species, has the capability to inhibit LDL</p>Formula:C21H18O13Purity:98%Color and Shape:SolidMolecular weight:478.36(+)-Carbovir
CAS:(+)-Carbovir is a nucleoside analog with increased chemical stability and increased metabolic stability.Formula:C11H13N5O2Color and Shape:SolidMolecular weight:247.25Crisdesalazine
CAS:Crisdesalazine (AAD 2004) is an inhibitor of microsomal prostaglandin E2 synthase-1 (mPGES-1).Formula:C16H14F3NO3Purity:98.96%Color and Shape:SolidMolecular weight:325.282-Chloroadenosine-5'-O-diphosphate sodium
CAS:<p>2-Chloroadenosine-5'-O-diphosphate, a purine nucleotide adenosine 5'diphosphate (ADP) derivative, demonstrates multiple biological activities.</p>Formula:C10H11ClN5O10P2·3NaColor and Shape:SolidMolecular weight:527.59BMS-695735
CAS:BMS-695735: benzimidazole, inhibits IGF-1 receptor, broad antitumor effects, affects CYP3A4, low solubility, binds plasma proteins.Formula:C26H31ClFN7OColor and Shape:SolidMolecular weight:512.02M5N36
CAS:M5N36: selective Cdc25C inhibitor, IC50: 0.15µM A, 0.19µM B, 0.06µM C; halts cell growth, boosts p-CDK1/2.Formula:C20H16ClN5O3Color and Shape:SolidMolecular weight:409.83O-Benzoylhydroxylamine
CAS:<p>O-Benzoyl hydroxylamine exhibits properties as a dipeptidyl peptidase-IV (DPP-IV) inhibitor and demonstrates antidiabetic effects[1].</p>Formula:C7H7NO2Color and Shape:SolidMolecular weight:137.14JAK2-IN-4
CAS:JAK2-IN-4 is a selective JAK2/JAK3 inhibitor, with IC50 values of 0.7 nM and 23.2 nM for JAK2 and JAK3, respectively.Formula:C23H27N5O4SPurity:98%Color and Shape:SolidMolecular weight:469.56SHP2/CDK4-IN-1
CAS:<p>SHP2/CDK4-IN-1: dual inhibitor, oral, potent (IC50: SHP2 4.3 nM, CDK4 18.2 nM), hinders TNBC growth, strong antitumor effects in mice.</p>Formula:C33H35ClF2N10OSColor and Shape:SolidMolecular weight:693.21
