Metabolismo
Os inibidores do metabolismo são compostos que interferem nas vias metabólicas, alterando a produção e utilização de energia dentro das células. Esses inibidores são usados para estudar a regulação do metabolismo, o papel das vias metabólicas em doenças como o câncer e o diabetes, e para desenvolver novas estratégias terapêuticas. Os inibidores do metabolismo podem direcionar várias enzimas e processos envolvidos na glicólise, na oxidação de ácidos graxos e em outras funções metabólicas. Na CymitQuimica, oferecemos uma ampla gama de inibidores do metabolismo de alta qualidade para apoiar sua pesquisa em bioquímica, distúrbios metabólicos e desenvolvimento de medicamentos.
Subcategorias de "Metabolismo"
- AhR(41 produtos)
- Aminopeptidase(67 produtos)
- CETP(18 produtos)
- Anidrase carbónica(178 produtos)
- Caseína quinase(130 produtos)
- DHFR(33 produtos)
- Descarboxilase(4 produtos)
- Desidrogenase(270 produtos)
- FAAH(64 produtos)
- FXR(58 produtos)
- Factor Xa(80 produtos)
- Sintase de Ácidos graxos(33 produtos)
- Ferroptose(215 produtos)
- GR(3 produtos)
- GSNOR(3 produtos)
- Glucoquinase(54 produtos)
- HIF/HIF Prolil-Hidroxilase(142 produtos)
- HMG-CoA Reductase(33 produtos)
- Hidroxilase(30 produtos)
- IDO(82 produtos)
- LDL(8 produtos)
- Lipase(97 produtos)
- Lipídio(59 produtos)
- Lipoxigenase(125 produtos)
- MAO(87 produtos)
- MPO(2 produtos)
- NAMPT(36 produtos)
- P450(6 produtos)
- PAI-1(25 produtos)
- PDE(166 produtos)
- PED(1 produtos)
- PKM(15 produtos)
- PPAR(164 produtos)
- Fosfolipase(82 produtos)
- ROR(42 produtos)
- Receptor de Retinóide(29 produtos)
- SGK(11 produtos)
- Tiorredoxina(12 produtos)
- Transferase(30 produtos)
- Tansportador(42 produtos)
- UGT(4 produtos)
- Inibidores de Xantina Oxidase (XO)(9 produtos)
Exibir 34 mais subcategorias
Foram encontrados 8626 produtos de "Metabolismo"
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Fmoc-Tyr(3-F,tBu)-OH
CAS:<p>Fmoc-Tyr(3-F,tBu)-OH: Cyclic peptide with high permeability, target-specific affinity. Sourced from WO2018225864A1.</p>Fórmula:C28H28FNO5Cor e Forma:SolidPeso molecular:477.53218:0,18:1 PS sodium
CAS:<p>18:0,18:1 PS sodium, a lipid found in synaptic vesicles and cholesterol, serves a role in metabolic research [1].</p>Fórmula:C42H79NNaO10PCor e Forma:SolidPeso molecular:812.04Hydroxycotinine
CAS:<p>Hydroxycotinine is the main nicotine metabolite detected in smokers' urine.</p>Fórmula:C10H12N2O2Pureza:98%Cor e Forma:SolidPeso molecular:192.218Deschloro Cetirizine dihydrochloride
CAS:<p>Deschloro Cetirizine Dihydrochloride: a Cetirizine impurity, second-gen antihistamine, and metabolite of hydroxyzine.</p>Fórmula:C21H28Cl2N2O3Cor e Forma:SolidPeso molecular:427.365PAz-PC
CAS:<p>PAz-PC (Azelaoyl PC) is a truncated phospholipid oxidation product that enhances endothelial barrier disruption caused by HKSA.</p>Fórmula:C33H64NO10PCor e Forma:SolidPeso molecular:665.84CAIX/CAXII-IN-4
<p>CAIX/CAXII-IN-4 (Compound 7h) is an inhibitor of carbonic anhydrase (CA) that binds to CAIX, CA XII, and CAII with Ki values of 1.324 μM, 0.435 μM, and 3.035 μM, respectively. This compound exhibits broad-spectrum anti-tumor activity and inhibits the proliferation of central nervous system tumor cells U251, with a GI50 of 0.361 μM.</p>Fórmula:C23H21N5O3SCor e Forma:SolidPeso molecular:447.51Pyruvate kinase
CAS:<p>Pyruvate kinase is a glycolytic enzyme that catalyzes the conversion of phosphoenolpyruvate and ADP to pyruvate and ATP [1] .</p>Cor e Forma:SolidInosine-5'-monophosphate (sodium salt hydrate)
CAS:<p>substrate of IMP dehydrogenase (IMPDH)</p>Fórmula:C10H29N4Na2O16PPureza:98%Cor e Forma:SolidPeso molecular:538.31Carvedilol metabolite 4-Hydroxyphenyl Carvedilol
CAS:<p>4-Hydroxyphenyl Carvedilol is a metabolite of Carvedilol. Carvedilol is a beta-blocker/alpha-1 blocker.</p>Fórmula:C24H26N2O5Pureza:98%Cor e Forma:SolidPeso molecular:422.47(R,S)-Carvedilol Glucuronide
CAS:<p>(R,S)-Carvedilol glucuronide is a racemic mix, metabolized by UGT1A1, UGT2B4, and UGT2B7.</p>Fórmula:C30H34N2O10Cor e Forma:SolidPeso molecular:582.606Sinbaglustat
CAS:<p>Sinbaglustat (OGT2378), an oral N-alkyl iminosugar, inhibits GCS/GBA2 and treats lysosomal storage and neurodegenerative disorders.</p>Fórmula:C11H23NO4Pureza:99.93%Cor e Forma:SolidPeso molecular:233.3PAPA NONOate
CAS:<p>PAPA NONOate is a pH-regulated NO donor.PAPA NONOate has potential antitumor activity and can be used to study diabetic wound healing disorders.</p>Fórmula:C6H16N4O2Pureza:98%Cor e Forma:SolidPeso molecular:176.22Glycerol kinase
CAS:<p>GyK, a bacterial sugar kinase, initiates glycerol metabolism by converting it into G3P, key for cell uptake.</p>Cor e Forma:SolidArylsulfatase
CAS:<p>Arylsulfatase, a type I sulfatase enzyme found in both prokaryotes and eukaryotes, is frequently utilized in biochemical research [1].</p>Cor e Forma:Solid2',5,6',7-Tetrahydroxyflavone
CAS:<p>2',5,6',7-Tetrahydroxyflavone is a useful organic compound for research related to life sciences.</p>Fórmula:C15H10O6Cor e Forma:SolidPeso molecular:286.2391-Salicylate Glucuronide
CAS:<p>1-Salicylate Glucuronide (Salicylic Acid b-D-O-Glucuronide) is a metabolite of salicylic acid after glucuronidation, promoting excretion.</p>Fórmula:C13H14O9Cor e Forma:SolidPeso molecular:314.25Izilendustat
CAS:<p>Tert-butyl compound inhibits human EGLN-1; confirmed by spectrometry after 20 mins.</p>Fórmula:C22H28ClN3O4Pureza:99.95%Cor e Forma:SolidPeso molecular:433.93b-Cortolone
CAS:<p>b-Cortolone, a metabolite of Cortisol, exhibits relatively lower biological activity.</p>Fórmula:C21H34O5Cor e Forma:SolidPeso molecular:366.49Carboxyaminoimidazole ribotide
CAS:<p>CAIR, an E. coli metabolite, helps identify its PurE active site and aids in fungal purine synthesis.</p>Fórmula:C9H14N3O9PCor e Forma:SolidPeso molecular:339.2Genz-123346
CAS:<p>Genz-123346 is an oral inhibitor of glucosylceramide synthase, blocking ceramide to GL1 conversion, with a 14 nM IC50.</p>Fórmula:C52H82N4O14Pureza:98%Cor e Forma:SolidPeso molecular:987.23Desmethylazelastine
CAS:<p>Desmethylazelastine, Azelastine's metabolite; 97% protein bound; 54-hour half-life; treats allergies, asthma, diabetes, SARS-CoV-2.</p>Fórmula:C21H22ClN3OCor e Forma:SolidPeso molecular:367.87Diglycyl-histidine
CAS:<p>Diglycyl-histidine is a tripeptide complexed with cupric ion designed to mimic specific Cu(II) transport site of ascorbate on albumin molecule.</p>Fórmula:C10H15N5O4Cor e Forma:SolidPeso molecular:269.26ATP ditromethamine
CAS:<p>ATP ditromethamine is key for energy storage, metabolism, and acts as a coenzyme and signaling molecule in immunity and inflammation.</p>Fórmula:C18H38N7O19P3Cor e Forma:SolidPeso molecular:749.45ARL67156 triethylamine
<p>ARL67156, a selective ecto-ATPase inhibitor, blocks NTPDase1, 3, and NPP1; used in calcific valve, asthma research. Ki: 11-18 μM.</p>Fórmula:C15H24Br2N5O12P3·3C6H15N)Cor e Forma:SolidPeso molecular:1154.23N-Desmethyl Bendamustine
CAS:<p>N-DesmethylBendamustine is a metabolite of Bendamustine. It exerts cytotoxic effects on various lymphoma cell lines and peripheral blood lymphocytes.</p>Fórmula:C15H19Cl2N3O2Cor e Forma:SolidPeso molecular:344.24DPPD-Q
CAS:<p>DPPD-Q, an antioxidant and an oxidative derivative of substituted p-phenylenediamine (DPPD), is identified in tire wear particles, rubber debris, particulate matter 2.5 (PM2.5), and wastewater influents and effluents. At a concentration of 5 µM, DPPD-Q inhibits soybean urease by 91.4%.</p>Fórmula:C18H14N2O2Cor e Forma:SolidPeso molecular:290.32ZD-2138
CAS:<p>ZD-2138: Selective 5-LOX inhibitor, eases allergen-induced asthma attacks and airway constriction in guinea pigs.</p>Fórmula:C23H24FNO4Pureza:99.68% - >99.99%Cor e Forma:SolidPeso molecular:397.44Clopidogrel carboxylic acid
CAS:<p>Clopidogrel Related Compound A is a useful organic compound for research related to life sciences.</p>Fórmula:C15H14ClNO2SCor e Forma:SolidPeso molecular:307.79GS-493
CAS:<p>GS-493: Specific SHP2 inhibitor, very potent (IC50=71 nM), 29x affinity vs. SHP1, 45x vs. PTP1B; hinders cancer cell growth/movement.</p>Fórmula:C21H14N6O8SCor e Forma:SolidPeso molecular:510.44HIV-1 inhibitor-58
<p>HIV-1 Inhibitor-58 (Compound 10c) is a non-nucleoside reverse transcriptase inhibitor with broad-spectrum antiviral properties, effective against both wild-type</p>Fórmula:C26H24N6O2Cor e Forma:SolidPeso molecular:452.51Picornain 3C
CAS:<p>Picornain 3C, a protease in picornaviruses, cleaves Gln-Gly bonds in poliovirus polyproteins and similar sites in others.</p>Cor e Forma:Solid11β-HSD1-IN-11
CAS:<p>11β-HSd1-in-11 is a potent and competitive inhibitor of 11-β-hydroxysteroid dehydrogenase 1 (11β-HSD1) IN rats and humans with IC50 values of 0.34 μM and 0.13</p>Fórmula:C15H11F3O3SPureza:99.61%Cor e Forma:SoildPeso molecular:328.31Bifenazate-diazene
CAS:<p>Bifenazate-diazene, a significant degradation product of Bifenazate, is characterized as a selective carbazate acaricide and insecticide [1].</p>Fórmula:C17H18N2O3Cor e Forma:SolidPeso molecular:298.34ERAP1 modulator-1
CAS:<p>ERAP1 modulator-1 (Compound 1) is a regulator of endoplasmic reticulum aminopeptidase 1 (ERAP1) with an IC50 of less than 250 nM.</p>Fórmula:C23H23F3N2O5SCor e Forma:SolidPeso molecular:496.5CCR1/5/8 activator 1
CAS:<p>CCR1/5/8 activator 1 is a cytoplasmic phospholipase A inhibitor with antifungal activity.</p>Fórmula:C10H9NOPureza:>99.99%Cor e Forma:SolidPeso molecular:159.18Doxorubicinol
CAS:<p>Doxorubicinol is the major circulating metabolite of doxorubicin with antineoplastic acitivity.</p>Fórmula:C27H31NO11Cor e Forma:SolidPeso molecular:545.54Cycloechinulin
CAS:<p>Cycloechinulin, a fungal metabolite from A. ochraceus, cuts corn earworm weight gain by 33% at 100 ppm.</p>Fórmula:C20H21N3O3Cor e Forma:SolidPeso molecular:351.4062MD
CAS:<p>2MD, a vitamin D-like oral drug, enhances bone mass/strength and lowers IOP by gene regulation.</p>Fórmula:C27H44O3Cor e Forma:SolidPeso molecular:416.64PROTAC PTPN2 degrader-1
CAS:<p>PROTAC PTPN2 degrader-1, a strong PTPN2 eliminator, may aid cancer/metabolic disease research.</p>Fórmula:C33H27FN6O8SCor e Forma:SolidPeso molecular:686.67Dapagliflozin-3-O-β-D-Glucuronide
CAS:<p>Dapagliflozin-3-O-β-D-glucuronide is a metabolite of dapagliflozin .</p>Fórmula:C27H33ClO12Cor e Forma:SolidPeso molecular:585CD13-IN-1
<p>CD13-IN-1 (Compound 5f) is a CD13 inhibitor with an IC50 value of 1.71 μM. It effectively suppresses the proliferation of various tumor cells, demonstrating antitumor activity.</p>Cor e Forma:Odour SolidDSPE-PEG1000-R9
<p>DSPE-PEG1000-R9 is a PEG compound composed of DSPE and the polyarginine-9 peptide (R9). It can be utilized in drug delivery applications.</p>Cor e Forma:Odour SolidDSPE-PEG5000-THRPPMWSPVWP
<p>DSPE-PEG5000-THRPPMWSPVWP is a PEG compound composed of DSPE and a transferrin receptor (TfR) peptide. The peptide sequence THRPPMWSPVWP binds to the TfR and is subsequently internalized into cells that express the receptor.</p>Cor e Forma:Odour SolidAbiraterone N-oxide
CAS:<p>Abiraterone N-oxide is a metabolite of Abiraterone . Abiraterone is a potent and irreversible CYP17A1 inhibitor with antiandrogen activity [1] .</p>Fórmula:C24H31NO2Cor e Forma:SolidPeso molecular:365.51Uridine 5'-triphosphate tris salt
CAS:<p>Uridine 5'-triphosphate tris salt is an endogenous metabolite .</p>Fórmula:C13H26N3O18P3Cor e Forma:SolidPeso molecular:605.28Seco Rapamycin
CAS:<p>Seco Rapamycin, a ring-opened Rapamycin derivative, does not affect mTOR function.</p>Fórmula:C51H79NO13Cor e Forma:SolidPeso molecular:914.187DSPE-PEG2000-TH
<p>DSPE-PEG2000-TH is a PEG conjugate made from DSPE and a pH-responsive cell-penetrating peptide (TH). In acidic environments—such as the tumor microenvironment—TH becomes activated, allowing for the selective delivery of small molecules, oligonucleotides, and proteins into tumor cells.</p>Cor e Forma:Odour SolidRelzomostat
CAS:<p>Relzomostat inhibits MetAP2, with research potential for obesity and type 2 diabetes.</p>Fórmula:C24H36F2N2O5Cor e Forma:SolidPeso molecular:470.558Phenylpyropene A
CAS:<p>Phenylpyropene A, a P. griseofulvum fungus product, blocks ACAT (IC50=0.8μM) and DGAT, kills M. persicae at 5ppm.</p>Fórmula:C32H38O10Cor e Forma:SolidPeso molecular:582.64Saccharopine hydrochloride
<p>Saccharopine hydrochloride, from lysine degradation, disrupts mitochondria and hinders development.</p>Fórmula:C11H21ClN2O6Cor e Forma:SolidPeso molecular:312.75SCD1 inhibitor-3
CAS:<p>SCD1 inhibitor-3 (ML-270) is a highly effective and orally available compound that inhibits SCD1 with remarkable safety.</p>Fórmula:C19H16FN7O2Pureza:99.5%Cor e Forma:SolidPeso molecular:393.3711,12-DiHETrE
CAS:<p>11,12-DiHETrE: Endogenous P450 eicosanoid, used in preterm labor study and NAFL/NASH differentiation.</p>Fórmula:C20H34O4Cor e Forma:SolidPeso molecular:338.48Diaphorase
CAS:<p>Diaphorase from anaerobic sludge catalyzes RDX biotransformation via denitrification.</p>Cor e Forma:SolidLYP-IN-3
<p>LYP-IN-3 (compound D34) is a selective Lymphoid-tyrosine phosphatase (LYP) inhibitor (Ki=0.93 μM) that modulates the T-cell receptor (TCR) signaling pathway</p>Fórmula:C35H27NO6SPureza:98%Cor e Forma:SolidPeso molecular:589.66Lactosylsphingosine (d18:1)
CAS:<p>Lactosylsphingosine (d18:1) is a sphingolipid with a lactose moiety that can inhibit fMetLeuPhe-induced cell aggregation at a concentration of 1 μm.</p>Fórmula:C30H57NO12Cor e Forma:SolidPeso molecular:623.77Cvs 738
CAS:<p>Cvs 738 is the desmethyl form of CVS 1123, an orally bioavailable inhibitor of thrombin.</p>Fórmula:C23H40N6O6Cor e Forma:SolidPeso molecular:496.6ACAT-IN-6
CAS:<p>ACAT-IN-6, from EP1236468A1 example 200, is a potent ACAT inhibitor that blocks NF-κB transcription.</p>Fórmula:C31H47N3O5SCor e Forma:SolidPeso molecular:573.79Neoechinulin C
CAS:<p>Neoechinulin C, a neuroprotective indolediketopiperazine, guards neurons against paraquat in Parkinson's.</p>Fórmula:C24H27N3O2Cor e Forma:SolidPeso molecular:389.49Chrysophanol triglucoside
CAS:<p>Chrysophanol triglucoside from Cassia obtusifolia, blocks PTP1B (IC50 80.17μM) & α-glucosidase (IC50 197.06μM), may aid diabetes study.</p>Fórmula:C33H40O19Cor e Forma:SolidPeso molecular:740.664Carboxylesterase-IN-1
CAS:<p>Carboxylesterase-IN-1, a pesticide inhibits carboxylesterase at 50 μg/mL, akin to triphenyl phosphate.</p>Fórmula:C30H37BrN2O5Cor e Forma:SolidPeso molecular:585.5396-Azathymine acid
CAS:<p>6-Azathymine is a metabolite of Pymetrozine, an insecticide targeting aphids and whiteflies by disrupting feeding.</p>Fórmula:C4H3N3O4Cor e Forma:SolidPeso molecular:157.08α-Amylase-IN-4
<p>α-Amylase-IN-4 (Compd 10y) exhibits the highest level of amylase inhibition, demonstrating an IC50 value of 17.83 ± 0.14 μg/mL [1].</p>Cor e Forma:Odour SolidIsoglycycoumarin
CAS:<p>Isoglycycoumarin, a flavonoid derived from the roots of Glycyrrhiza uralensis, serves as a highly selective probe for human cytochrome P450 2A6.</p>Fórmula:C21H20O6Pureza:98%Cor e Forma:SolidPeso molecular:368.38(S)-Higenamine
CAS:<p>(S)-Higenamine, a benzylisoquinoline precursor, forms from dopamine and 4-HPAA via NCS.</p>Fórmula:C16H17NO3Cor e Forma:SolidPeso molecular:271.31Garcinone B
CAS:<p>Garcinone B, a xanthone derivative naturally isolated from the pericarp of Mangosteen, serves as a potent inhibitor of ACE2 and Mpro, and is utilized in COVID-</p>Fórmula:C23H22O6Pureza:98%Cor e Forma:SolidPeso molecular:394.42CETP-IN-4
CAS:<p>CETP-IN-4 is a cholesteryl ester transfer protein (CETP) inhibitor.</p>Fórmula:C36H28F9N3O4Cor e Forma:SolidPeso molecular:737.623DSPE-PEG3000-LyP-1
<p>DSPE-PEG3000-LyP-1 is a PEG compound composed of DSPE and a nine-residue peptide (LyP-1). The LyP-1 component specifically targets tumor-associated lymphatics and macrophages.</p>Cor e Forma:Odour SolidPTP1B-IN-22
CAS:<p>PTP1B-IN-22 is a protein tyrosine phosphatase 1B (PTP1B) inhibitor that inhibits glucose uptake in skeletal muscle L6 myotubes.</p>Fórmula:C16H12N2O3S2Pureza:98.35%Cor e Forma:SoildPeso molecular:344.41L-Pyroglutamic acid β-naphthylamide
CAS:<p>L-Pyroglutamic acid β-naphthylamide (PYR) is a derivative of glutamic acid.</p>Fórmula:C15H14N2O2Cor e Forma:SolidPeso molecular:254.28β-1,4-GALT1-IN-1
<p>β-1,4-GALT1-IN-1 (Compound 6) is a β-1,4-GALT1 inhibitor with an IC50 value of 6.2 μM. It is applicable in studying various pathological conditions, including cancer, autoimmune diseases, and viral infections.</p>Fórmula:C29H23NO10Cor e Forma:SolidPeso molecular:545.49416,16-dimethyl Prostaglandin A2
CAS:<p>16,16-dimethyl PGA2, a stable analog of PGA2, greatly reduces Sendai virus growth and helps mice survive influenza and cancer.</p>Fórmula:C22H34O4Cor e Forma:SolidPeso molecular:362.5Ilaprazole sulfone
CAS:<p>Ilaprazole sulfone, main Ilaprazole metabolite, formed mostly by CYP3A4/5, is an oral proton pump inhibitor.</p>Fórmula:C19H18N4O3SCor e Forma:SolidPeso molecular:382.44LYP-IN-4
<p>LYP-IN-4 (compound D14), a reversible and selective lymphotyrosine phosphatase (LYP) inhibitor (Ki=1.34 μM, IC50=3.52μM), regulates TCR signaling, increases PD-</p>Fórmula:C29H21ClN2O8SPureza:98%Cor e Forma:SolidPeso molecular:5936,8-Dihydroxy-1,2,7-trimethoxy-3-methylanthraquinone
CAS:<p>Compound 1, 6,8-Dihydroxy-1,2,7-trimethoxy-3-methylanthraquinone, is an anthraquinone α-glucosidase inhibitor with an IC50 of 185 μM, and it can be isolated</p>Fórmula:C18H16O7Pureza:98%Cor e Forma:SolidPeso molecular:344.32SB-435495 hydrochloride
CAS:<p>SB-435495 hydrochloride is a potent, selective, reversible, non-covalent, and orally active inhibitor of Lp-PLA2, exhibiting an IC50 of 0.06 nM [1] [3].</p>Fórmula:C38H41ClF4N6O2SCor e Forma:SolidPeso molecular:757.28Ethyl 4-chloro-2-oxo-1,2-dihydroquinoline-3-carboxylate
CAS:<p>ethyl 4-chloro-2-oxo-1,2-dihydroquinoline-3-carboxylate inhibits NAD(P)H: quinone oxidoreductase 1.</p>Fórmula:C12H10ClNO3Pureza:99.19%Cor e Forma:SolidPeso molecular:251.67ITH12711
<p>ITH12711, a PP2A ligand, can traverse the blood-brain barrier (BBB) and exerts neuroprotection by restoring PP2A-phosphatase activity [1].</p>Fórmula:C12H20O5Pureza:98%Cor e Forma:SolidPeso molecular:244.28ACAT-IN-4
CAS:<p>ACAT-IN-4 inhibits ACAT and NF-κB-mediated transcription.</p>Fórmula:C32H50N2O5SCor e Forma:SolidPeso molecular:574.823α-Hydroxysteroid dehydrogenase
CAS:<p>3α-Hydroxysteroid dehydrogenase (3α-HSD), encoded by the AKR1C4 gene, is responsible for catalyzing the transformation of 3-ketosteroids into 3α-hydroxy</p>Cor e Forma:SolidDSPE-PEG5000-PP1
<p>DSPE-PEG5000-PP1 is a PEG compound composed of DSPE and the PP1 peptide, which targets inflammatory atherosclerotic plaques. It can be used for drug delivery.</p>Cor e Forma:Odour SolidTerpendole C
CAS:<p>Terpendole C, an indole diterpene from A. yamanashiensis, inhibits ACAT with IC50 of 2.1 μM in rats, 0.46 μM in J774 cells, non-toxic.</p>Fórmula:C32H41NO5Cor e Forma:SolidPeso molecular:519.682Stevisalioside A
<p>Stevisalioside A (Compound 2), isolated from the roots of Stevia serrata, is an orally active antidiabetic agent that inhibits Protein Tyrosine Phosphatase 1B (</p>Fórmula:C35H50O15Pureza:98%Cor e Forma:SolidPeso molecular:710.76Glucuronokinase (AtGlcAK)
CAS:<p>AtGlcAK: GHMP-kinase family, specific for D-glucuronic acid, Km 0.7 mM, converts it with ATP to D-glucuronic-1-phosphate and ADP.</p>Cor e Forma:SolidEnpp-1-IN-15
CAS:<p>Compound 88a (Enpp-1-IN-15) is an inhibitor of Ectonucleotide Pyrophosphatase/Phosphodiesterase 1 (Enpp-1), exhibiting a Ki value of 0.00586 nM [1].</p>Fórmula:C16H20N6O2SCor e Forma:SolidPeso molecular:360.43UDP-sugar pyrophosphorylase (BlUSP)
CAS:<p>BlUSP enzyme turns Glc-1-P into UDP-Glucose, transferring uridyl from UTP and producing PPi.</p>Cor e Forma:SolidACAT-IN-5
CAS:<p>ACAT-IN-5 inhibits ACAT, suppressing NF-κB-mediated transcription.</p>Fórmula:C32H49N3O5SCor e Forma:SolidPeso molecular:587.82Quercetin 3-(6″-caffeoylsophoroside)
CAS:<p>Quercetin 3-(6″-caffeoylsophoroside) is an orally active compound exhibiting α-amylase inhibitory activity, with an IC50 value of 73.66 μg/mL, and demonstrates</p>Fórmula:C27H40N4O7Cor e Forma:SolidPeso molecular:532.63PEG2000-C-DMG
CAS:<p>PEG2000-C-DMG is a pegylated lipid for Onpattro, reducing transthyretin production via RNAi.</p>Fórmula:C126H249NO52Cor e Forma:SolidPeso molecular:2000 (Average)RORγt inverse agonist 31
<p>RORγt inverse agonist 31 (14g) is a potent antagonist of the retinoic acid receptor-related orphan receptor γt (RORγt), exhibiting an inhibitory concentration (</p>Fórmula:C23H15Cl2F3N4O3SPureza:98%Cor e Forma:SolidPeso molecular:555.36D-Erythrose 4-phosphate sodium
CAS:<p>D-erythrose 4-sodium phosphate: sodium salt of monosaccharide, made from erythritol via 3 isomerases.</p>Fórmula:C4H8NaO7PPureza:98%Cor e Forma:SolidPeso molecular:222.07Boc-Ile-Glu-Gly-Arg-AMC
CAS:<p>Boc-IEGR-AMC: fluorogenic substrate for factor Xa and Halocynthia roretzi acrosin.</p>Fórmula:C34H50N8O10Pureza:98%Cor e Forma:White PowderPeso molecular:730.81DSPE-PEG5000-ANG
<p>DSPE-PEG5000-ANG is a PEGylated compound formed by DSPE and the dual-targeting ligand (Angiopep-2, ANG). ANG exhibits high binding efficacy to LRP1 and has been utilized for targeting glioma delivery. DSPE-PEG5000-ANG is applicable in drug delivery.</p>Cor e Forma:Odour SolidROS-IN-2
<p>ROS-IN-2 (compound 85), a seco-lupane triterpenoid derivative, inhibits reactive oxygen species (ROS) production and shields mitochondria from oxidative damage</p>Fórmula:C42H62ClNO8SPureza:98%Cor e Forma:SolidPeso molecular:776.46FS-2
<p>FS-2 is a potent, specific inhibitor of L-type CaV channels, effectively impeding high K+ or glucose-induced L-type Ca2+ influx in RIN beta cells [1].</p>Fórmula:C297H462N92O86S10Pureza:98%Cor e Forma:SolidPeso molecular:7018.06PKM2-IN-4
<p>Compound 5C, referred to as Pkm2-in-4, is a selective PKM2 inhibitor (IC50 = 0.35 µM) that modulates pyruvate-dependent respiration and promotes mitochondrial</p>Fórmula:C15H17BrClNO3SeCor e Forma:SolidPeso molecular:453.62Diadenosine pentaphosphate pentalithium
CAS:<p>Endogenous vasoactive compound, found in platelets and brain cells, part of diadenosine polyphosphates (ApnA, n=2–7).</p>Fórmula:C20H24Li5N10O22P5Cor e Forma:SolidPeso molecular:946.03Ovotransferrin (328-332)
CAS:<p>Ovotransferrin (328-332), with an IC50 of 20 μM, exhibits protective activity against hypertension by inhibiting the Angiotensin-Converting Enzyme (ACE) and</p>Fórmula:C25H46N8O7Pureza:98%Cor e Forma:SolidPeso molecular:570.68MAGL-IN-10
<p>MAGL-IN-10, a reversible monoacylglycerol lipase (MAGL) inhibitor, exhibits favorable ADME properties and low in vivo toxicity.</p>Pureza:98%Cor e Forma:Odour SolidCaptopril EP Impurity B
CAS:<p>Captopril EP Impurity B, an antihypertensive thiol ACE inhibitor with IC50 of 0.025 μM.</p>Fórmula:C9H14BrNO3Cor e Forma:SolidPeso molecular:264.12Sp-cAMPS triethylamine
CAS:<p>Sp-cAMPS triethylamine activates PKA I/II and inhibits PDE3A (Ki 47.6µM), binds PDE10 GAF (EC50 40µM).</p>Fórmula:C16H27N6O5PSCor e Forma:SolidPeso molecular:446.46
