CymitQuimica logo
Metabolismo

Metabolismo

Os inibidores do metabolismo são compostos que interferem nas vias metabólicas, alterando a produção e utilização de energia dentro das células. Esses inibidores são usados para estudar a regulação do metabolismo, o papel das vias metabólicas em doenças como o câncer e o diabetes, e para desenvolver novas estratégias terapêuticas. Os inibidores do metabolismo podem direcionar várias enzimas e processos envolvidos na glicólise, na oxidação de ácidos graxos e em outras funções metabólicas. Na CymitQuimica, oferecemos uma ampla gama de inibidores do metabolismo de alta qualidade para apoiar sua pesquisa em bioquímica, distúrbios metabólicos e desenvolvimento de medicamentos.

Subcategorias de "Metabolismo"

Exibir 34 mais subcategorias

Foram encontrados 8595 produtos de "Metabolismo"

Ordenar por

Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
produtos por página.
  • Ensifentrine

    CAS:
    <p>Ensifentrine (Ensifentrinum) is a PDE3/4 inhibitor, although its affinity for PDE3(IC50: 0.4 nM) is 3,440 times higher than that for PDE4(IC50: 1479 nM), that</p>
    Fórmula:C26H31N5O4
    Pureza:99.76% - 99.94%
    Cor e Forma:Solid
    Peso molecular:477.56
  • SR1001

    CAS:
    <p>SR 1001 is an inverse agonist for RORα/RORγ (Kis: 172/111 nM).</p>
    Fórmula:C15H13F6N3O4S2
    Pureza:98.93%
    Cor e Forma:Solid
    Peso molecular:477.4
  • Sildenafil Mesylate

    CAS:
    <p>Sildenafil Mesylate is a mesylate form of Sildenafil, an inhibitor of Phosphodiesterase 5.</p>
    Fórmula:C22H30N6O4S·xCH4O3S
    Pureza:99.84%
    Cor e Forma:Solid
    Peso molecular:570.68
  • PQ-10

    CAS:
    <p>PQ-10 (A-844337) is a PDE-10 inhibitor. PQ-10 induces brain glucose metabolism patterns, which may be a potential translational biomarker.</p>
    Fórmula:C22H21N5O3
    Pureza:99.86%
    Cor e Forma:Solid
    Peso molecular:403.43
  • Phenidone

    CAS:
    <p>Phenidone inhibits COX/LOX, reducing rat autoimmune paralysis and lowering blood pressure in hypertensive rats.</p>
    Fórmula:C9H10N2O
    Pureza:97.24%
    Cor e Forma:White Solid Solid Crystalline
    Peso molecular:162.19
  • Obafistat

    CAS:
    <p>Obafistat is a potent inhibitor of aldo-keto reductase AKR1C3 with an IC50 of 1.2 nM for human AKR1C3.</p>
    Fórmula:C15H16FN5O3S
    Pureza:99.71%
    Cor e Forma:Solid
    Peso molecular:365.38
  • TETRAHYDROPIPERINE

    CAS:
    <p>Tetrahydropiperine (Cosmoperine) is a natural product derived from piperine, can be used to treat convulsion, epilepsy, relieve pain, and control insects.</p>
    Fórmula:C17H23NO3
    Pureza:98.04% - 99.61%
    Cor e Forma:Off-White Low Melting Solid With Characteristic Odour
    Peso molecular:289.37
  • 7-Hydroxy-3,4-dihydro-2(1H)-quinolinone

    CAS:
    7-Hydroxy-3,4-dihydro-2(1H)-quinolinone is a weak MAO-A inhibitor(with an IC50 of 183 μM) .
    Fórmula:C9H9NO2
    Pureza:99.20%
    Cor e Forma:Solid
    Peso molecular:163.17
  • Bocidelpar

    CAS:
    <p>Bocidelpar is a modulator of PPARδ with an EC50 of 7.80 nM and improves mitochondrial biogenesis and function in Duchenne Muscular Dystrophy muscle cells.</p>
    Fórmula:C25H27F3N2O3
    Pureza:97.77%
    Cor e Forma:Solid
    Peso molecular:460.49
  • Torcetrapib

    CAS:
    <p>Torcetrapib (CP-529414), a CETP inhibitor, curbs cholesteryl ester movement from HDL to LDL/VLDL; failed Phase III trials due to mortality increase.</p>
    Fórmula:C26H25F9N2O4
    Pureza:98% - 99.59%
    Cor e Forma:Lipid
    Peso molecular:600.47
  • N-(p-amylcinnamoyl) Anthranilic Acid

    CAS:
    <p>N-(p-amylcinnamoyl) Anthranilic Acid (ACA) is a broad spectrum Phospholipase A2 (PLA2) inhibitor and TRP channel blocker.</p>
    Fórmula:C21H23NO3
    Pureza:99.35% - 99.67%
    Cor e Forma:Solid
    Peso molecular:337.41
  • Azumolene

    CAS:
    <p>Azumolene (EU4093 free base)</p>
    Fórmula:C13H9BrN4O3
    Pureza:98.1% - 98.35%
    Cor e Forma:Solid
    Peso molecular:349.14
  • Soticlestat

    CAS:
    <p>Soticlestat (OV935) is a potent, selective and orally active cholesterol 24-hydroxylase (CYP46A1) inhibitor.</p>
    Fórmula:C23H23N3O2
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:373.45
  • CVT-12012

    CAS:
    <p>CVT-12012 is an orally bioavailable inhibitor of stearoyl-CoA desaturase (SCD; IC50 = 6.1 nM in HepG2 cells).</p>
    Fórmula:C21H21F3N4O3
    Pureza:99.56%
    Cor e Forma:Solid
    Peso molecular:434.41
  • Pentamidine

    CAS:
    <p>Pentamidine is an antifungal and antiprotozoal agent, interacting directly with the pathogen genome by binding to AT-rich regions of duplex DNA and the minor</p>
    Fórmula:C19H24N4O2
    Pureza:98.64% - 99.67%
    Cor e Forma:Crystallizes As Colorless Plates From Water Solid
    Peso molecular:340.42
  • BW-A 78U

    CAS:
    <p>BW-A 78U is a PDE4 inhibitor (IC50: 3 μM). It is not inhibition on the lipopolysaccharide (LPS)-induced TNF-α release.</p>
    Fórmula:C13H12FN5
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:257.27
  • AKBA

    CAS:
    <p>AKBA (3-O-Acetyl-11-keto-beta-boswellic acid), a natural component from frankincense, is a novel activator of Nrf2.</p>
    Fórmula:C32H48O5
    Pureza:97.85% - 99.77%
    Cor e Forma:Solid
    Peso molecular:512.72
  • CP-640186

    CAS:
    <p>CP-640186 is an isozyme-nonselective ACCase inhibitor. The IC50s of CP-640186 is 53 nM and 61 nM for rat liver ACC1 and rat skeletal muscle ACC2 respectively.</p>
    Fórmula:C30H35N3O3
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:485.62
  • D159687

    CAS:
    <p>D159687 is a selective PDE4D inhibitor,had a procognitive profile as it improved memory in the novel object recognition test but had no antidepressant benefit.</p>
    Fórmula:C21H19ClN2O2
    Pureza:97.57%
    Cor e Forma:Solid
    Peso molecular:366.84
  • NS-638

    CAS:
    <p>NS-638 is a Ca2+-channel blocker. It can block K+-stimulated intracellular Ca2+-elevation (IC50: 3.4 μM).</p>
    Fórmula:C15H11ClF3N3
    Pureza:98.44%
    Cor e Forma:Solid
    Peso molecular:325.72
  • p-Fluoro-L-phenylalanine

    CAS:
    <p>p-Fluoro-L-phenylalanine: TH substrate, studies enzyme regulation, binds E. coli L-leucine receptor, KD 0.26μM.</p>
    Fórmula:C9H10FNO2
    Pureza:99.63%
    Cor e Forma:White To Off-White Powder
    Peso molecular:183.18
  • Tienilic Acid

    CAS:
    <p>Tienilic Acid is a uricosuric diuretic with certain hepatotoxicity</p>
    Fórmula:C13H8Cl2O4S
    Pureza:99.55%
    Cor e Forma:Solid
    Peso molecular:331.17
  • GSK805

    CAS:
    <p>GSK805 is a potent, orally bioavailable and CNS-penetrant RORγt inhibitor.Cost-effective and quality-assured.</p>
    Fórmula:C23H18Cl2F3NO4S
    Pureza:98% - ≥95%
    Cor e Forma:Solid
    Peso molecular:532.36
  • PF-06282999

    CAS:
    <p>PF-06282999 is a potent and selective myeloperoxidase inhibitor which is potentially useful for the treatment of cardiovascular diseases.</p>
    Fórmula:C13H12ClN3O3S
    Pureza:98.15% - 98.28%
    Cor e Forma:Solid
    Peso molecular:325.77
  • 2-Bromo-4'-hydroxyacetophenone

    CAS:
    <p>2-Bromo-4'-hydroxyacetophenone(PTP Inhibitor I) is a cell-permeable, PTP inhibitor that covalently blocks the catalytic domain of the SHP-1(ΔSH2).</p>
    Fórmula:C8H7BrO2
    Pureza:98.64%
    Cor e Forma:Clear Colorless To Light Yellow Liquid
    Peso molecular:215.04
  • Telaglenastat

    CAS:
    <p>Telaglenastat (CB 839) (IC50 of 24 nM), an effective, specific, and oral inhibitor, which is bioavailable glutaminase, for recombinant human GAC.</p>
    Fórmula:C26H24F3N7O3S
    Pureza:97.57% - 99.89%
    Cor e Forma:Solid
    Peso molecular:571.57
  • SU0268

    CAS:
    <p>SU0268 is a potent and specific 8-Oxoguanine DNA glycosylase 1 (OGG1) inhibitor.</p>
    Fórmula:C26H25N3O4S
    Pureza:99.97% - 99.98%
    Cor e Forma:Solid
    Peso molecular:475.56
  • Pargyline

    CAS:
    <p>Pargyline (Pargylamine) is a monoamine oxidase inhibitor with antihypertensive properties.</p>
    Fórmula:C11H13N
    Pureza:95.64% - 97.21%
    Cor e Forma:Solid
    Peso molecular:159.23
  • PfDHODH-IN-2

    CAS:
    <p>PfDHODH-IN-2: powerful antimalarial, blocks PfDHODH (IC50: 1.11 μM), for malaria research.</p>
    Fórmula:C13H12ClNO3S
    Pureza:98.9%
    Cor e Forma:Solid
    Peso molecular:297.76
  • Pentamidine isethionate

    CAS:
    <p>Pentamidine isethionate (Pentamidine diisethionate) is a synthetic amidine derivative, Pentamidine Isethionate is an antiprotozoal and antifungal agent.</p>
    Fórmula:C23H36N4O10S2
    Pureza:98% - 99.83%
    Cor e Forma:Slight Butyric Odor Very Bitter Taste Ph (5% Aqueous Solution) 4 5-6 5 (Ntp 1992)
    Peso molecular:592.68
  • Linrodostat

    CAS:
    <p>Linrodostat (BMS-986205) is a selective indoleamine 2, 3-dioxygenase 1 (IDO1) inhibitor.</p>
    Fórmula:C24H24ClFN2O
    Pureza:99.54% - 99.71%
    Cor e Forma:Solid
    Peso molecular:410.91
  • L-Cysteinesulfinic acid monohydrate

    CAS:
    <p>L-Cysteinesulfinic acid monohydrate activates rat mGluR1/2/4/5/6/8 with pEC50s of 3.92, 3.9, 2.7, 4.6, 4.0, 3.94 respectively.</p>
    Fórmula:C3H9NO5S
    Pureza:≥98%
    Cor e Forma:Solid
    Peso molecular:171.17
  • FG-2216

    CAS:
    <p>FG-2216 (YM-311) is a HIF-prolyl hydroxylase inhibitor for the PDH2 enzyme; orally bioavailable and induced reversible and significant Epo induction in vivo.</p>
    Fórmula:C12H9ClN2O4
    Pureza:97.1% - >99.99%
    Cor e Forma:Solid
    Peso molecular:280.66
  • JZL 184

    CAS:
    <p>JZL 184 is a potent and selective inhibitor of MAGL with IC50 of 8 nM and 4 μM for inhibition of MAGL and FAAH in mouse brain membranes respectively.</p>
    Fórmula:C27H24N2O9
    Pureza:97.56% - 99.31%
    Cor e Forma:Solid
    Peso molecular:520.49
  • S18-000003

    CAS:
    <p>S18-000003: Oral retinoic acid receptor gamma-t inhibitor, IC50 29 nM, reduces IL-17 production.</p>
    Fórmula:C26H25F3N2O4S
    Pureza:99.24% - 99.31%
    Cor e Forma:Solid
    Peso molecular:518.55
  • Difluprednate

    CAS:
    <p>Difluprednate (Myser)(Durezol) is a corticosteroid, approved for the treatment of post-operative ocular inflammation and pain.</p>
    Fórmula:C27H34F2O7
    Pureza:99.23% - 99.86%
    Cor e Forma:Solid
    Peso molecular:508.55
  • RGX-104

    CAS:
    <p>RGX-104 (RGX-104 free Acid) free Acid is an agonist of potent liver-X nuclear hormone receptor (LXR)</p>
    Fórmula:C34H33ClF3NO3
    Pureza:98.79% - 99.53%
    Cor e Forma:Solid
    Peso molecular:596.08
  • THP104c

    CAS:
    <p>THP104c is an inhibitor of mitochondrial fission.</p>
    Fórmula:C20H16N4O2S
    Pureza:99.33%
    Cor e Forma:Solid
    Peso molecular:376.43
  • KPT9274

    CAS:
    <p>KPT9274 (PAK4-IN-1) is a non-competitive dual inhibitor of PAK4 and NAMPT(IC50= ~120 nM). It is an orally bioavailable small molecule.</p>
    Fórmula:C35H29F3N4O3
    Pureza:99.75% - 99.93%
    Cor e Forma:Solid
    Peso molecular:610.62
  • LOX-IN-3 dihydrochloride

    CAS:
    <p>LOX-IN-3 dihydrochloride is an inhibitor of lysyl oxidase (LOX).</p>
    Fórmula:C13H15Cl2FN2O2S
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:353.24
  • Cobicistat

    CAS:
    <p>Cobicistat (GS-9350): A carbamate, thiazole derivative, and CYP3A inhibitor used to boost anti-HIV drugs for treating HIV.</p>
    Fórmula:C40H53N7O5S2
    Pureza:97.36% - 99.62%
    Cor e Forma:Solid
    Peso molecular:776.02
  • S-(2-Carboxypropyl)cysteine

    CAS:
    <p>S-(2-Carboxypropyl)cysteine is a urinary metabolite of S-(2-Carboxypropyl)glutathione.</p>
    Fórmula:C7H13NO4S
    Pureza:≥98%
    Cor e Forma:Solid
    Peso molecular:207.25
  • (E/Z)-Teriflunomide

    CAS:
    <p>(E/Z)-Teriflunomide (Aubagio), a orally-available Pyrimidine Synthesis Inhibitor, is used to treat relapsing multiple sclerosis.</p>
    Fórmula:C12H9F3N2O2
    Pureza:99.49% - 99.76%
    Cor e Forma:White Solid
    Peso molecular:270.21
  • Toloxatone

    CAS:
    <p>Toloxatone (MD 69276) is a reversible monoamine oxidase A (MAOA) inhibitor.</p>
    Fórmula:C11H13NO3
    Pureza:98.58%
    Cor e Forma:Solid
    Peso molecular:207.23
  • Glycerol 3-phosphate biscyclohexylammonium salt

    CAS:
    <p>Glycerol 3-phosphate biscyclohexylammonium salt is an endogenous metabolite produced by cytosolic glycerol 3-phosphate dehydrogenase pathway.</p>
    Fórmula:C15H35N2O6P
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:370.42
  • Fmoc-Ser(O-α-D-GalNAc(OAc)3)-OH

    CAS:
    <p>Fmoc-Ser(O-α-D-GalNAc(OAc)3)-OH (Fmoc-Ser(Ac3AcNH-α-Gal)-OH) is an anti-tumor drug</p>
    Fórmula:C32H36N2O13
    Pureza:98% - ≥98%
    Cor e Forma:Solid
    Peso molecular:656.63
  • TM5275 sodium

    CAS:
    <p>TM5275 sodium (TM5275 sodium salt) is an inhibitor of plasminogen activator inhibitor 1 (PAI-1).</p>
    Fórmula:C28H27ClN3NaO5
    Pureza:98.8% - 99.74%
    Cor e Forma:Solid
    Peso molecular:543.98
  • ARM1

    CAS:
    <p>ARM1 is a potent inhibitor of aminopeptidase and epoxide hydrolase. The IC50 values are 7.61 µM for aminopeptidase and 12.4 µM for epoxide hydrolase.</p>
    Fórmula:C16H14N2S
    Pureza:99.36%
    Cor e Forma:Solid
    Peso molecular:266.36
  • D-Pantothenic acid

    CAS:
    <p>D-Pantothenic acid (B5): water-soluble, antioxidant, in all living tissues, part of CoA &amp; B2 complex, needed for metabolism &amp; synthesizing cholesterol, etc.</p>
    Fórmula:C9H17NO5
    Pureza:99.85% - 99.92%
    Cor e Forma:Yellow Viscous Oil Solid
    Peso molecular:219.24
  • (±)-Amiflamine

    CAS:
    <p>(±)-Amiflamine (2-dimethylphenethylamine) is an inhibitor of reversible MAO-A.</p>
    Fórmula:C12H20N2
    Pureza:97.24%
    Cor e Forma:Solid
    Peso molecular:192.3
  • Cecropin P1, porcine acetate


    <p>Cecropin P1, porcine acetate is an antibacterial peptide found in Hyalophora cecropia and pig intestine.</p>
    Fórmula:C149H257N45O45
    Pureza:95.4% - 98%
    Cor e Forma:Solid
    Peso molecular:3398.91
  • Bempedoic acid

    CAS:
    <p>Bempedoic acid (ETC1002) is an orally available, once-daily LDL-C lowering small molecule designed to lower elevated levels of LDL-C.</p>
    Fórmula:C19H36O5
    Pureza:99.85% - 99.94%
    Cor e Forma:Solid
    Peso molecular:344.49
  • Efonidipine hydrochloride monoethanolate

    CAS:
    <p>Efonidipine HCl monoethanolate is a calcium blocker, boosts dehydroepiandrosterone sulfate in NCI-H295R cells.</p>
    Fórmula:C36H45ClN3O8P
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:714.18
  • Nitrofurazone

    CAS:
    <p>Nitrofurazone (Furacilin) is a topical anti-infective agent effective against gram-negative and gram-positive bacteria.</p>
    Fórmula:C6H6N4O4
    Pureza:99.87%
    Cor e Forma:Pale Yellow Needles Solution) 6 0 - 6 5 Alkaline Solutions Are Dark Orange (Ntp 1992)
    Peso molecular:198.14
  • 1-Ethynylpyrene

    CAS:
    <p>1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and 2B1(IC50 = 0.04 μM).</p>
    Fórmula:C18H10
    Pureza:98.48%
    Cor e Forma:Solid
    Peso molecular:226.27
  • Suvecaltamide

    CAS:
    <p>Suvecaltamide (MK-8998) as potent inhibitors of T-type calcium channels.</p>
    Fórmula:C20H23F3N2O2
    Pureza:99.29% - 99.70%
    Cor e Forma:Solid
    Peso molecular:380.4
  • Diflubenzuron

    CAS:
    <p>Diflubenzuron (Larvakil) is a benzoyl-urea insecticide, found to be a potent inhibitor of melanosome synthesis in mouse melanoma cells.</p>
    Fórmula:C14H9ClF2N2O2
    Pureza:99.58% - 99.96%
    Cor e Forma:Colorless Crystals Diflubenzuron Is A Colorless To Yellow Crystals Used As A Selective Insecticide
    Peso molecular:310.68
  • PF-04457845

    CAS:
    <p>PF-04457845 is a greatly and effctive FAAH inhibitor, and for hFAAH(IC50=7.2±0.63 nM) and rFAAH(IC50=7.4±0.62 nM).</p>
    Fórmula:C23H20F3N5O2
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:455.43
  • BRL-50481

    CAS:
    <p>BRL-50481 is a novel and selective inhibitor of PDE7 with IC50s of 0.15, 12.1, 62 and 490 μM for PDE7A, PDE7B, PDE4 and PDE3, respectively.</p>
    Fórmula:C9H12N2O4S
    Pureza:99.66%
    Cor e Forma:Solid
    Peso molecular:244.27
  • NCT-501

    CAS:
    <p>NCT-501 is a potent and selective inhibitor of Aldehyde Dehydrogenase 1A1 (ALDH1A1) with IC50 of 40 nM.</p>
    Fórmula:C21H32N6O3
    Pureza:99.19%
    Cor e Forma:Solid
    Peso molecular:416.52
  • Telotristat

    CAS:
    <p>Telotristat, active metabolite of LX1606, is an oral tryptophan hydroxylase inhibitor with potential antiserotonergic effects.</p>
    Fórmula:C25H22ClF3N6O3
    Pureza:99.70%
    Cor e Forma:Solid
    Peso molecular:546.93
  • Pinaverium bromide

    CAS:
    <p>Pinaverium bromide is an calcium channel blocker with Antispasmodic and effectively relieves pain, diarrhea and intestinal discomfort.</p>
    Fórmula:C26H41Br2NO4
    Pureza:99.52%
    Cor e Forma:White Crystalline Powder
    Peso molecular:591.42
  • GSK1016790A

    CAS:
    <p>GSK1016790A (GSK101) (GSK101) is a novel, potent activator of TRPV4 (transient receptor potential vanilloid 4) with EC50 of 34 nM in choroid plexus epithelial</p>
    Fórmula:C28H32Cl2N4O6S2
    Pureza:97.37% - 99.38%
    Cor e Forma:Solid
    Peso molecular:655.61
  • AMG-208

    CAS:
    <p>AMG-208 is a highly selective c-Met inhibitor with IC50 of 9 nM. Phase 1.</p>
    Fórmula:C22H17N5O2
    Pureza:98.56%
    Cor e Forma:Solid
    Peso molecular:383.4
  • ASP-9521

    CAS:
    <p>ASP-9521 is a selective, potent and orally active indole-based AKR1C3 inhibitor with an IC50 of 11 nM for human AKR1C3.Cost-effective and quality-assured.</p>
    Fórmula:C19H26N2O3
    Pureza:95.11% - 96.96%
    Cor e Forma:Solid
    Peso molecular:330.42
  • Glycylsarcosine

    CAS:
    <p>Glycylsarcosine (GLYCYL-SARCOSINE) is a dipeptide obtained by formal condensation of the carboxy group of glycine with the amino group of sarcosine</p>
    Fórmula:C5H10N2O3
    Pureza:98.47%
    Cor e Forma:Solid
    Peso molecular:146.14
  • TOFA

    CAS:
    <p>TOFA (MDL14514) is an allosteric inhibitor of acetyl-CoA carboxylase-α (ACCA).</p>
    Fórmula:C19H32O4
    Pureza:97.52% - 98.98%
    Cor e Forma:Solid
    Peso molecular:324.45
  • GNE-617 hydrochloride

    CAS:
    <p>GNE-617 hydrochloride is a specific inhibitor of NAMPT and inhibits NAMPT activity (IC50: 5 nM).</p>
    Fórmula:C21H16ClF2N3O3S
    Cor e Forma:Solid
    Peso molecular:463.88
  • DHBP dibromide

    CAS:
    <p>DHBP dibromide (1,1'-DI-N-HEPTYL-4,4'-BIPYRIDINIUM DIBRO) is calcium release and a muscle relaxant inhibitor.</p>
    Fórmula:C24H38Br2N2
    Pureza:99.73%
    Cor e Forma:Yellow To Yellow-Green Powder Or Flakes
    Peso molecular:514.38
  • Pentamidine dimesylate

    CAS:
    <p>Pentamidine dimesylate blocks (Ca)S100B-p53, aiding p53 activity against melanoma.</p>
    Fórmula:C20H28N4O5S
    Cor e Forma:Solid
    Peso molecular:436.53
  • Liquiritin

    CAS:
    <p>Liquiritin (Liquiritigenin-4'-O-glucoside) (LIQ) is a main component among the licorice flavonoids, and possesses anti-inflammatory and anti-cancer abilities.</p>
    Fórmula:C21H22O9
    Pureza:98.16% - 98.66%
    Cor e Forma:Solid
    Peso molecular:418.39
  • (Rac)-LB-100

    CAS:
    <p>LB-100, a novel Protein Phosphatase 2A (PP2A) inhibitor, sensitizes malignant meningioma cells to the therapeutic effects of radiation</p>
    Fórmula:C13H20N2O4
    Pureza:97.11% - 99.77%
    Cor e Forma:Solid
    Peso molecular:268.31
  • ML-298

    CAS:
    <p>ML-298 (CID53393915) is a potent, specific inhibitor of Phospholipase D2 (PLD2, IC50 of 355 nM).</p>
    Fórmula:C22H23F3N4O2
    Pureza:99.35%
    Cor e Forma:Solid
    Peso molecular:432.44
  • Calcium D-saccharate tetrahydrate

    CAS:
    <p>Calcium D-saccharate tetrahydrate (Calcium D-saccharate tetrahydrate) is an oxidized non-cyclic hexose sugar.</p>
    Fórmula:C6H16CaO12
    Pureza:98%
    Cor e Forma:White Solid
    Peso molecular:320.26
  • Balipodect

    CAS:
    <p>Balipodect (TAK063) is a highly effective and selective PDE10A inhibitor (IC50: 0.30 nM); Its selectivity is &gt;15000-fold over other PDEs.</p>
    Fórmula:C23H17FN6O2
    Pureza:98% - 99.79%
    Cor e Forma:Solid
    Peso molecular:428.42
  • 6-Hydroxy-4-methylcoumarin

    CAS:
    <p>6-Hydroxy-4-methylcoumarin (6-Hydroxy-4-Methyl-2H-Chromen-2-One) is a secondary metabolite of coumarin, which has anticancer effects.</p>
    Fórmula:C10H8O3
    Pureza:98.93%
    Cor e Forma:Solid
    Peso molecular:176.17
  • Pep 2-8 ammonium salt(1541011-97-5 free base)


    <p>Pep 2-8 ammonium salt inhibits PCSK9-LDL receptor binding (IC50 = 0.8 μM), boosting LDL uptake in HepG2 cells.</p>
    Fórmula:C83H113N17O24
    Pureza:95.76% - 99.87%
    Cor e Forma:Solid
    Peso molecular:1732.91
  • 1-Cyclohexyl-3-dodecyl urea

    CAS:
    <p>1-Cyclohexyl-3-dodecyl urea (NCND) is a highly selective soluble epoxide hydrolase (sEH) inhibitor.</p>
    Fórmula:C19H38N2O
    Pureza:99.59%
    Cor e Forma:Solid
    Peso molecular:310.52
  • EAAT2 activator 1

    CAS:
    <p>EAAT2 activator 1 (3-[(2-Chloro-6-fluorobenzyl)thio]-6-pyridin-2-ylpyridazine) is a thiopyridazine derivative that has been found to increase EAAT2 protein</p>
    Fórmula:C16H11ClFN3S
    Pureza:98.86%
    Cor e Forma:Solid
    Peso molecular:331.8
  • HA130

    CAS:
    <p>HA130 is a selective ATX (autotaxin) inhibitor.</p>
    Fórmula:C24H19BFNO5S
    Pureza:98.26% - ≥95%
    Cor e Forma:Solid
    Peso molecular:463.29
  • 2,5-Di-tert-butylhydroquinone

    CAS:
    <p>2,5-Di-tert-butylhydroquinone (BHQ) is an effective and selective endoplasmic reticulum Ca2+-ATPase inhibitor.</p>
    Fórmula:C14H22O2
    Pureza:97.11%
    Cor e Forma:Pelletslargecrystals
    Peso molecular:222.32
  • Tipifarnib

    CAS:
    <p>Tipifarnib (IND 58359), a quinolinone, inhibits farnesyl transferase, blocks Ras activation, arrests cell growth, and curbs angiogenesis.</p>
    Fórmula:C27H22Cl2N4O
    Pureza:97.1% - 99.22%
    Cor e Forma:Off-White To Pale Beige Solid
    Peso molecular:489.4
  • kb NB 142-70

    CAS:
    <p>kb NB 142-70 is a selective protein kinase D (PKD) inhibitor (IC50 values are 28.3, 58.7 and 53.2 nM for PKD1, 2 and 3 respectively).</p>
    Fórmula:C11H9NO2S2
    Pureza:98.15% - ≥95%
    Cor e Forma:Solid
    Peso molecular:251.32
  • AGN 193109

    CAS:
    <p>AGN 193109, a retinoid analog, is a potent and specific antagonist of RARs (Kds: 2 nM, 2 nM, and 3 nM for RARα, RARβ, and RARγ).</p>
    Fórmula:C28H24O2
    Pureza:99.87% - 99.89%
    Cor e Forma:Solid
    Peso molecular:392.49
  • Indoximod

    CAS:
    <p>Indoximod (NLG-8189) is a methylated tryptophan that inhibits IDO to boost T cell function by preventing tryptophan depletion.</p>
    Fórmula:C12H14N2O2
    Pureza:97.82% - 99.55%
    Cor e Forma:Solid
    Peso molecular:218.25
  • D-Valine

    CAS:
    <p>D-Valine (H-D-Val-OH) is the enantiomer of L-Valine.</p>
    Fórmula:C5H11NO2
    Pureza:99.93%
    Cor e Forma:White Crystals
    Peso molecular:117.15
  • GSK2033

    CAS:
    <p>GSK2033 is an antagonist of LXR (pIC50s: 7 and 7.4 for LXRα or LXRβ, respectively).</p>
    Fórmula:C29H28F3NO5S2
    Pureza:99.70%
    Cor e Forma:Solid
    Peso molecular:591.66
  • Efonidipine

    CAS:
    Efonidipine (NZ-105)(NZ-105) is a dihydropyridine calcium channel blocker, blocking both T-type and L-type calcium channels.
    Fórmula:C34H38N3O7P
    Pureza:98.35% - 99.47%
    Cor e Forma:Solid
    Peso molecular:631.66
  • IDO5L

    CAS:
    <p>IDO5L (INCB024360 analogue) is an effective IDO1 inhibitor(IC50=10 nM).</p>
    Fórmula:C9H7ClFN5O2
    Pureza:99.49% - 99.75%
    Cor e Forma:Solid
    Peso molecular:271.64
  • Tedizolid

    CAS:
    <p>Tedizolid (DA-7157)is a novel oxazolidinone-class antibiotic that inhibits bacterial protein synthesis by binding to the 23S ribosomal RNA of the 50S subunit of</p>
    Fórmula:C17H15FN6O3
    Pureza:96.97% - 99.89%
    Cor e Forma:Solid
    Peso molecular:370.34
  • MPO-IN-28

    CAS:
    <p>MPO-IN-28 is a novel potent, irreversible Myeloperoxidase (MPO) inhibitor with IC50 of 44 nM.</p>
    Fórmula:C11H13N5O
    Pureza:98.04%
    Cor e Forma:Solid
    Peso molecular:231.25
  • BPTES

    CAS:
    <p>BPTES(IC50 of 0.16 μM) is an effective and specific GlutamiN/Ase GLS1 (KGA) inhibitor.</p>
    Fórmula:C24H24N6O2S3
    Pureza:95.83% - 99.64%
    Cor e Forma:Solid
    Peso molecular:524.68
  • Edoxaban hydrochloride

    CAS:
    <p>Edoxaban (DU-176b) HCl: Oral, selective Factor Xa inhibitor, Ki 0.561 nM; prevents thromboembolic disease.</p>
    Fórmula:C24H31Cl2N7O4S
    Cor e Forma:Solid
    Peso molecular:584.52
  • Lazabemide hydrochloride

    CAS:
    <p>Lazabemide hydrochloride (N-(2-Aminoethyl)-5-chlor-2-pyridincarbox) is a reversible and selective mao-b inhibitor(Ki:7.9nM).</p>
    Fórmula:C8H11Cl2N3O
    Pureza:98.65%
    Cor e Forma:Solid
    Peso molecular:236.098
  • Pimecrolimus

    CAS:
    <p>Pimecrolimus, a calcineurin inhibitor, binds FKBP-12, blocking calcium-dependent signals.</p>
    Fórmula:C43H68ClNO11
    Pureza:99.53% - 99.87%
    Cor e Forma:White Crystalline Powder
    Peso molecular:810.45
  • GW 4064

    CAS:
    <p>GW 4064 is an effective farnesoid X receptor (FXR) agonist (EC50 =65 nM).</p>
    Fórmula:C28H22Cl3NO4
    Pureza:98% - 99.94%
    Cor e Forma:Solid
    Peso molecular:542.84
  • SI-113

    CAS:
    <p>SI-113 is a potent and selective inhibitor of SGK1, a serine/threonine protein kinase, that modulates several oncogenic signaling cascades.</p>
    Fórmula:C23H24N6O
    Pureza:98.93%
    Cor e Forma:Solid
    Peso molecular:400.48
  • GSK 2830371

    CAS:
    <p>GSK 2830371 is an orally active, allosteric Wip1 phosphatase inhibitor with IC50 of 6 nM.</p>
    Fórmula:C23H29ClN4O2S
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:461.02
  • PNU-100440

    CAS:
    <p>PNU-100440 is a biologically active compound. It is an intermediate in the synthesis of linezolid dimers, an impurity of the antibacterial agent Linezolid.</p>
    Fórmula:C14H17FN2O4
    Pureza:99.09%
    Cor e Forma:Solid
    Peso molecular:296.29
  • G6PDi-1

    CAS:
    <p>G6PDi-1 is an effective G6PD inhibitor. It depletes NADPH and decreases inflammatory cytokine production.</p>
    Fórmula:C14H12N4OS
    Pureza:98.69%
    Cor e Forma:Solid
    Peso molecular:284.34