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Metabolismo

Metabolismo

Os inibidores do metabolismo são compostos que interferem nas vias metabólicas, alterando a produção e utilização de energia dentro das células. Esses inibidores são usados para estudar a regulação do metabolismo, o papel das vias metabólicas em doenças como o câncer e o diabetes, e para desenvolver novas estratégias terapêuticas. Os inibidores do metabolismo podem direcionar várias enzimas e processos envolvidos na glicólise, na oxidação de ácidos graxos e em outras funções metabólicas. Na CymitQuimica, oferecemos uma ampla gama de inibidores do metabolismo de alta qualidade para apoiar sua pesquisa em bioquímica, distúrbios metabólicos e desenvolvimento de medicamentos.

Subcategorias de "Metabolismo"

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Foram encontrados 8625 produtos de "Metabolismo"

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  • DSPE-PEG2000-NYZL1


    <p>DSPE-PEG2000-NYZL1 is a PEG compound composed of DSPE and NYZL1. NYZL1 has the ability to specifically bind to bladder cancer tissues and cells. DSPE-PEG2000-NYZL1 is suitable for drug delivery applications.</p>
    Cor e Forma:Odour Solid
  • Osteogenic Growth Peptide, OGP

    CAS:
    <p>OGP, a natural 14-mer serum peptide at μM levels, is crucial for osteogenic response to bone injury.</p>
    Fórmula:C68H110N22O18
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1523.74
  • Sulotroban potassium


    <p>Sulotroban potassium is a small molecule thromboxane A2 receptor (TXA2R) antagonist that can be used to study myocardial infarction and thrombosis.</p>
    Fórmula:C16H16KNO5S
    Pureza:98.02%
    Cor e Forma:Soild
    Peso molecular:373.46
  • (±)14-HDHA

    CAS:
    <p>(±)14-HDHA is an oxidized metabolite of DHA and can be further oxidized to the 14-oxoDHA, 14-HDoHE inhibits LPS-induced IL-6 mRNA expression.</p>
    Fórmula:C22H32O3
    Cor e Forma:Solid
    Peso molecular:344.49
  • 1-Palmitoyl Lysophosphatidic Acid

    CAS:
    <p>1-Palmitoyl Lysophosphatidic Acid boosts antibiotics against P. aeruginosa by binding Ca2+ and Mg2+.</p>
    Fórmula:C19H39O7P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:410.48
  • Perflubutane

    CAS:
    <p>Perfluorobutane is a gas that is colorless.</p>
    Fórmula:C4F10
    Pureza:98%
    Cor e Forma:Colorless Gas Colorless Gas
    Peso molecular:238.03
  • (S)-Higenamine

    CAS:
    <p>(S)-Higenamine, a benzylisoquinoline precursor, forms from dopamine and 4-HPAA via NCS.</p>
    Fórmula:C16H17NO3
    Cor e Forma:Solid
    Peso molecular:271.31
  • Sphingomyelins (buttermilk)

    CAS:
    <p>Sphingomyelins, 2-15% of organ phospholipids, are prevalent in brain and nerve sheaths, regulate cholesterol, and turn into ceramides by hydrolysis.</p>
    Fórmula:C46H93N2O6P(fortricosanoyl)
    Cor e Forma:Solid
    Peso molecular:801.2
  • Terpendole C

    CAS:
    <p>Terpendole C, an indole diterpene from A. yamanashiensis, inhibits ACAT with IC50 of 2.1 μM in rats, 0.46 μM in J774 cells, non-toxic.</p>
    Fórmula:C32H41NO5
    Cor e Forma:Solid
    Peso molecular:519.682
  • Sucunamostat hydrochloride


    <p>Sucunamostat (SCO-792) hydrochloride is an orally active, reversible inhibitor of enteropeptidase, displaying inhibition constants (IC50) of 4.6 nM for rat</p>
    Fórmula:C22H23ClN4O8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:506.89
  • Adrenocorticotropic Hormone (ACTH) (18-39), human

    CAS:
    <p>ACTH (18-39), or Corticotropin-like Peptide, boosts insulin, amylase, and protein secretion dose-dependently.</p>
    Fórmula:C112H165N27O36
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:2465.67
  • Cholesterol esterase

    CAS:
    <p>Cholesterol esterase breaks down cholesterol ester into cholesterol and free fatty acids, aiding absorption.</p>
    Cor e Forma:Solid
  • PKCζ/ι pseudosubstrate inhibitor

    CAS:
    <p>PKCζ/ι pseudosubstrate inhibitor demonstrates comprehensive inhibitory activity across the protein kinase C (PKC) family and is associated with the induction of</p>
    Fórmula:C76H128N30O16
    Cor e Forma:Solid
    Peso molecular:1718.02
  • Quercetin 3-(6″-caffeoylsophoroside)

    CAS:
    <p>Quercetin 3-(6″-caffeoylsophoroside) is an orally active compound exhibiting α-amylase inhibitory activity, with an IC50 value of 73.66 μg/mL, and demonstrates</p>
    Fórmula:C27H40N4O7
    Cor e Forma:Solid
    Peso molecular:532.63
  • L-Pyroglutamic acid β-naphthylamide

    CAS:
    <p>L-Pyroglutamic acid β-naphthylamide (PYR) is a derivative of glutamic acid.</p>
    Fórmula:C15H14N2O2
    Cor e Forma:Solid
    Peso molecular:254.28
  • PLA2-IN-1


    <p>PLA2-IN-1 (Compound 7) is a potent and selective inhibitor of phospholipase A (PLA2) with an IC50 value of 1 nM. It effectively inhibits PLA2-induced coagulation disorders in vitro and shows potential for use as an antidote for snake bites caused by cobra venom.</p>
    Cor e Forma:Odour Solid
  • Ciwujianoside C2

    CAS:
    <p>Ciwujianoside C2 is a useful organic compound for research related to life sciences. The catalog number is T126337 and the CAS number is 114892-56-7.</p>
    Fórmula:C60H94O26
    Cor e Forma:Solid
    Peso molecular:1231.39
  • Antibacterial agent 218


    <p>Antibacterialagent 218 (compound d28) is an orally active inhibitor of sterol 24-C-methyltransferase with an IC50 value of 0.273 μM. It also displays antifungal activity against Candida albicans SC5314, with an IC50 of 0.25 μg/mL.</p>
    Fórmula:C30H24N4OS
    Peso molecular:488.16708
  • N-acetyl Dapsone

    CAS:
    <p>N-acetyl Dapsone is an anti-inflammatory and antimicrobial compound widely used in the treatment of leprosy, malaria, acne and various immune disorders.</p>
    Fórmula:C14H14N2O3S
    Pureza:99.86%
    Cor e Forma:White
    Peso molecular:290.34
  • Olmesartan ethyl ester

    CAS:
    <p>Olmesartan ethyl ester is an impurity of Olmesartan (RNH-6270), an AT1R antagonist for high blood pressure research.</p>
    Fórmula:C26H30N6O3
    Cor e Forma:Solid
    Peso molecular:474.55
  • TRH Precursor Peptide


    <p>Thyrotropin Releasing Hormone Precursor Peptide</p>
    Fórmula:C42H75N19O10
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1006.17
  • α-Glucosidase-IN-49


    <p>α-Glucosidase-IN-49 (compound C23) is a potent inhibitor of α-Glucosidase, with an IC50 of 0.52 μM. This compound exhibits oral bioactivity, effectively lowering blood glucose levels and enhancing glucose tolerance in mice.</p>
    Fórmula:C21H13F3N4O3S3
    Peso molecular:522.01019
  • Abiraterone N-oxide

    CAS:
    <p>Abiraterone N-oxide is a metabolite of Abiraterone . Abiraterone is a potent and irreversible CYP17A1 inhibitor with antiandrogen activity [1] .</p>
    Fórmula:C24H31NO2
    Cor e Forma:Solid
    Peso molecular:365.51
  • C22 Galactosylceramide (d18:1/22:0)

    CAS:
    <p>C22 Galactosylceramide, a CNS sphingolipid, rises in mouse spinal cord on a methionine-restricted diet, found in Alzheimer's hippocampus.</p>
    Fórmula:C46H89NO8
    Cor e Forma:Solid
    Peso molecular:784.20
  • 10-FTHF

    CAS:
    <p>10-FTHF is a donor of formyl groups in anabolism used as a substrate in formyltransferase reactions, which is important in purine biosynthesis.</p>
    Fórmula:C20H23N7O7
    Cor e Forma:Solid
    Peso molecular:473.44
  • D,L-erythro-PDMP

    CAS:
    <p>D,L-erythro-PDMP inhibits growth in rabbit fibroblasts and blocks UDP-glucose: ceramide glucosyltransferase.</p>
    Fórmula:C23H38N2O3
    Cor e Forma:Solid
    Peso molecular:390.568
  • Cirsiliol 4′-glucoside

    CAS:
    <p>Cirsiliol 4′-glucoside, a compound extracted from Ruellia tuberosa L., acts as a free radical scavenger and demonstrates potential anti-diabetic activity [1].</p>
    Fórmula:C23H24O12
    Cor e Forma:Solid
    Peso molecular:492.43
  • hCAIX/XII-IN-14


    <p>hCAIX/XII-IN-14 (Compound 1i) is an inhibitor of hCAIX and hCAXII, with Ki values of 9.4 nM for hCAII, 5.6 nM for hCAIX, and 6.3 nM for hCAXII.</p>
    Fórmula:C16H14F3N3O4S
    Cor e Forma:Solid
    Peso molecular:401.36
  • CAIX/CAXII-IN-4


    <p>CAIX/CAXII-IN-4 (Compound 7h) is an inhibitor of carbonic anhydrase (CA) that binds to CAIX, CA XII, and CAII with Ki values of 1.324 μM, 0.435 μM, and 3.035 μM, respectively. This compound exhibits broad-spectrum anti-tumor activity and inhibits the proliferation of central nervous system tumor cells U251, with a GI50 of 0.361 μM.</p>
    Fórmula:C23H21N5O3S
    Cor e Forma:Solid
    Peso molecular:447.51
  • DSPE-PEG1000-ANG


    <p>DSPE-PEG1000-ANG is a PEG compound composed of DSPE and a dual-targeting ligand (Angiopep-2, ANG). ANG demonstrates high LRP1 binding efficiency and has been utilized for targeting glioma delivery. DSPE-PEG1000-ANG is suitable for drug delivery applications.</p>
    Cor e Forma:Odour Solid
  • 1-Pentadecanoyl-rac-glycerol

    CAS:
    <p>1-Pentadecanoyl-rac-glycerol: a monoacylglycerol with sn-1 pentadecanoic acid, found in wheat bran, rises in fatty liver models.</p>
    Fórmula:C18H36O4
    Cor e Forma:Solid
    Peso molecular:316.482
  • Desoxycarbadox

    CAS:
    <p>Desoxycarbadox, derived from Carbadox, is a quinoxaline-di-N-oxide antibiotic compound.</p>
    Fórmula:C11H10N4O2
    Cor e Forma:Solid
    Peso molecular:230.227
  • DSPE-PEG2000-WYRGRL


    <p>DSPE-PEG2000-WYRGRL is a PEG compound composed of DSPE and the cartilage-targeting peptide (WYRGRL). The peptide WYRGRL can specifically bind to type II collagen α1. DSPE-PEG2000-WYRGRL is utilized for drug delivery.</p>
    Cor e Forma:Odour Solid
  • Lead Ionophore IV

    CAS:
    <p>Lead Ionophore IV, an ion carrier, actively facilitates the transport of metal ions. It is commonly utilized in biological research to investigate the biological effects of lead ions and their impact on cellular functions. Additionally, Lead Ionophore IV is employed in developing drug delivery systems to enhance the bioavailability of compounds.</p>
    Fórmula:C60H84N4O4S4
    Cor e Forma:Solid
    Peso molecular:1053.59
  • NLG802

    CAS:
    <p>NLG802 is a prodrug of indoximod, an orally active indoleamine 2,3-dioxygenase (IDO) inhibitor.</p>
    Fórmula:C20H30ClN3O3
    Pureza:99.61%
    Cor e Forma:Solid
    Peso molecular:395.92
  • DBPR-110

    CAS:
    <p>DBPR-110: NS5A inhibitor, EC50 of 3.9 pM for HCV1b, SI &gt;12.8 million; EC50 of 228.8 pM for HCV2a, SI &gt;173,130.</p>
    Fórmula:C50H48N6O4S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:861.09
  • 5′-Nucleotidase

    CAS:
    <p>5′-Nucleotidase (CD73), an ectoenzyme and intrinsic membrane glycoprotein, catalyzes the hydrolysis of 5-nucleotides into their corresponding nucleosides [1].</p>
    Cor e Forma:Solid
  • TNAP-IN-1

    CAS:
    <p>TNAP-IN-1 is a specific inhibitor of tissue-nonspecific alkaline phosphatase (TNAP) and is utilized in studying diseases related to soft tissue calcification.</p>
    Fórmula:C17H16N2O4S
    Pureza:99.03%
    Cor e Forma:Solid
    Peso molecular:344.39
  • 3'-sulfo Galactosylsphingosine (ammonium salt)

    CAS:
    <p>Sulfatide derivative inhibits cell migration, adhesion, PKC, cytochrome c; accumulates in metachromatic leukodystrophy; used for LC-MS quantification.</p>
    Fórmula:C24H50N2O10S
    Cor e Forma:Solid
    Peso molecular:558.73
  • DSPE-PEG2000-EB1


    <p>DSPE-PEG2000-EB1 is a PEG compound composed of DSPE and the pH-responsive transmembrane peptide (EB1). It is utilized for drug delivery.</p>
    Cor e Forma:Odour Solid
  • Purpactin A

    CAS:
    <p>Purpactin A is a useful organic compound for research related to life sciences. The catalog number is T126026 and the CAS number is 133806-59-4.</p>
    Fórmula:C23H26O7
    Cor e Forma:Solid
    Peso molecular:414.454
  • 6-Azathymine acid

    CAS:
    <p>6-Azathymine is a metabolite of Pymetrozine, an insecticide targeting aphids and whiteflies by disrupting feeding.</p>
    Fórmula:C4H3N3O4
    Cor e Forma:Solid
    Peso molecular:157.08
  • MeIQx

    CAS:
    <p>MeIQx, a carcinogenic compound in cooked fish/meat, triggers DNA-reactive metabolites and rat tumors.</p>
    Fórmula:C11H11N5
    Cor e Forma:Solid
    Peso molecular:213.244
  • Thalifendine chloride

    CAS:
    <p>Thalifendine chloride is a metabolite of berberine,the methoxy group at the C-10 position undergoes demethylation by CYP51. cytotoxicity against P-388 cells.</p>
    Fórmula:C19H16ClNO4
    Cor e Forma:Solid
    Peso molecular:357.79
  • RORγ agonist 1

    CAS:
    <p>RORγ agonist 1 is a highly potent and orally bioavailable compound that activates the RORγ receptor.</p>
    Fórmula:C29H27ClF4N2O4S
    Cor e Forma:Solid
    Peso molecular:611.05
  • 23,25-Dihydroxy-24-oxovitamin D3

    CAS:
    <p>23,25-Dihydroxy-24-oxovitamin D3, a prominent metabolite of 24(R),25-Dihydroxyvitamin D3, holds significant potential for studying metabolic disorders[1].</p>
    Fórmula:C27H42O4
    Cor e Forma:Solid
    Peso molecular:430.629
  • Coumachlor

    CAS:
    <p>Coumachlor, a first-generation anticoagulant rodenticide, blocks the formation of prothrombin and inhibits blood coagulation causing internal haemorrhage.</p>
    Fórmula:C19H15ClO4
    Cor e Forma:Solid
    Peso molecular:342.77
  • Cy3 IRGD-PEG-DSPE


    <p>Cy3 IRGD-PEG-DSPE is a PEG phospholipid containing Cy3 dye, applicable for protein/nucleic acid labeling and fluorescence microscopy. It self-assembles in aqueous solutions to form micelles or lipid bilayers, which are useful for creating liposomes or nanoparticles for the delivery of nutrients, such as mRNA or DNA vaccines.</p>
    Cor e Forma:Odour Solid
  • D-Ribofuranose1-dihydrogenphosphate dicyclohexanamine

    CAS:
    <p>D-Ribofuranose 1-phosphate is used to synthesize 5-fluorouracil via uridine phosphorylase.</p>
    Fórmula:C11H24NO8P
    Cor e Forma:Solid
    Peso molecular:329.28
  • Bifenazate-diazene

    CAS:
    <p>Bifenazate-diazene, a significant degradation product of Bifenazate, is characterized as a selective carbazate acaricide and insecticide [1].</p>
    Fórmula:C17H18N2O3
    Cor e Forma:Solid
    Peso molecular:298.34
  • (±)14(15)-EpEDE

    CAS:
    <p>8,11,14-Eicosatrienoic acid, also known as dihomo-γ-linolenic acid , is a polyunsaturated fatty acid (PUFA) produced from γ-linolenic acid by the action of</p>
    Fórmula:C20H34O3
    Cor e Forma:Solid
    Peso molecular:322.489
  • (-)-Jasmonoyl-L-isoleucine

    CAS:
    <p>(-)-Jasmonoyl-L-isoleucine ((-)-JA-L-Ile), an enantiomer of (+)-JA-L-Ile [1], is an inactive endogenous hormone.</p>
    Fórmula:C18H29NO4
    Cor e Forma:Solid
    Peso molecular:323.43
  • Saccharopine hydrochloride


    <p>Saccharopine hydrochloride, from lysine degradation, disrupts mitochondria and hinders development.</p>
    Fórmula:C11H21ClN2O6
    Cor e Forma:Solid
    Peso molecular:312.75
  • DSPE-PEG2000-RVG29


    <p>DSPE-PEG2000-RVG29 is a PEG compound composed of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 specifically binds to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and can traverse the BBB.</p>
    Cor e Forma:Odour Solid
  • 2-NP-AHD

    CAS:
    <p>2-NP-AHD, derived from AHD/nitrofuran metabolite, indicates illegal nitrofuran use.</p>
    Fórmula:C10H8N4O4
    Cor e Forma:Solid
    Peso molecular:248.20
  • β-1,3-Galactosyltransferase (CgtB)

    CAS:
    <p>CgtB enzyme, needed for GM1-like LOS SIAL, catalyzes galactose addition in biochemical studies.</p>
    Cor e Forma:Solid
  • ARL67156 trisodium salt

    CAS:
    <p>ARL 67156 inhibits NTPDase1, 3, NPP1 (Ki: 11, 18, 12 μM) and ecto-ATPase; it's a trisodium salt.</p>
    Fórmula:C15H21Br2N5Na3O12P3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:785.05
  • Carvedilol metabolite 4-Hydroxyphenyl Carvedilol

    CAS:
    <p>4-Hydroxyphenyl Carvedilol is a metabolite of Carvedilol. Carvedilol is a beta-blocker/alpha-1 blocker.</p>
    Fórmula:C24H26N2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:422.47
  • Liarozole fumarate

    CAS:
    <p>Liarozole fumarate is used as a retinoic acid metabolism blocking agent (RAMBA) and an aromatase inhibitor.</p>
    Fórmula:C17H13ClN4C4H4O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:482.88
  • SHR168442

    CAS:
    <p>SHR168442 is a potent RORγ modulator, exhibiting an IC50 value of 0.035 μM.</p>
    Fórmula:C23H25Cl2F2N3O3S
    Cor e Forma:Solid
    Peso molecular:532.43
  • Cortisol sulfate

    CAS:
    <p>Cortisol sulfate (Cortisol 21-sulfate) is a metabolite of Cortisol . Cortisol sulfate is a specific ligand for intracellular transcortin [1] [2] [3] .</p>
    Fórmula:C21H30O8S
    Cor e Forma:Solid
    Peso molecular:442.52
  • Angiotensin 1/2 (1-9)

    CAS:
    <p>Angiotensin 1/2 (1-9) is containing the amino acids 1-9 that are converted from Angiotensin I/II peptide.</p>
    Fórmula:C56H78N16O13
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1183.32
  • CooP

    CAS:
    <p>CooP is a nonapeptide targeting glioblastoma. It binds to FABP3 for chemotherapy delivery.</p>
    Fórmula:C32H57N9O11S
    Cor e Forma:Solid
    Peso molecular:775.91
  • Mead acid

    CAS:
    <p>Mead acid, a 5,8,11-Eicosatrienoic Omega-9 unsaturated fatty acid, signals essential fatty acid deficiency.</p>
    Fórmula:C20H34O2
    Cor e Forma:Solid
    Peso molecular:306.49
  • DSPE-PEG2000-K237


    <p>DSPE-PEG2000-K237 is a PEG compound consisting of DSPE and the KDR-targeting peptide (K237). K237 functionally disrupts the interaction between VEGF and KDR receptors, resulting in significant biological effects such as inhibition of angiogenesis and tumor growth. DSPE-PEG2000-K237 is applicable in drug delivery.</p>
    Cor e Forma:Odour Solid
  • Cefetamet Hydrochloride

    CAS:
    <p>Cefetamet is a potent antibiotic to treat respiratory and urinary tract infections.</p>
    Fórmula:C14H16ClN5O5S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:433.89
  • Lunine

    CAS:
    <p>Lunine is a bioactive chemical.</p>
    Fórmula:C16H17NO4
    Cor e Forma:Solid
    Peso molecular:287.31
  • ZK53

    CAS:
    <p>ZK53 is a mitochondrial casein hydrolysing protease P (HsClpP) activator that induces apoptosis and inhibits the hydrolysis of alpha-casein by HsClpP.</p>
    Fórmula:C19H20BrF2N3O
    Pureza:97.8% - 99.36%
    Cor e Forma:Soild
    Peso molecular:424.28
  • O-Demethyl Lenvatinib hydrochloride


    <p>O-Demethyl Lenvatinib HCl is a Lenvatinib metabolite; an oral inhibitor targeting VEGFR, FGFR, PDGFR, KIT, RET with antitumor properties.</p>
    Fórmula:C20H18Cl2N4O4
    Cor e Forma:Solid
    Peso molecular:449.29
  • Mevalonic acid 5-pyrophosphate tetralithium

    CAS:
    <p>Mevalonic acid 5-pyrophosphate (also known as 5-Diphosphomevalonic acid) tetralithium is an endogenous metabolite involved in the mevalonate pathway.</p>
    Fórmula:C6H10Li4O10P2
    Cor e Forma:Solid
    Peso molecular:331.85
  • Dextranase

    CAS:
    <p>Dextranase, a glucan hydrolase, breaks down α-(1,6)-glucosidic bonds in dextran, useful in food, sugar modification, medicine, and more.</p>
    Cor e Forma:Solid
  • Carbonic anhydrase inhibitor 31


    <p>Carbonic anhydrase inhibitor31 is an mtCA2 inhibitor (Ki: 5.2 nM) that can be used in antituberculosis research.</p>
    Fórmula:C24H20N6O5S
    Cor e Forma:Solid
    Peso molecular:504.12159
  • Uricosuric agent-1

    CAS:
    <p>Acetic acid, 2-[4-[(2-ethyl-3-benzofuranyl)carbonyl]phenoxy]- is a compound used for antiviral activity determinations.</p>
    Fórmula:C19H16O5
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:324.33
  • HSP90-IN-30


    <p>HSP90-IN-30 (compound 3e) inhibits the activity of the HSP90 molecular chaperone. Under hypoxic conditions, HSP90-IN-30 suppresses HIF-1 transcriptional activity with an IC50 value of 2.16 μM.</p>
    Fórmula:C20H39B12N4O2
    Peso molecular:499.41897
  • β-1,4-GALT1-IN-1


    <p>β-1,4-GALT1-IN-1 (Compound 6) is a β-1,4-GALT1 inhibitor with an IC50 value of 6.2 μM. It is applicable in studying various pathological conditions, including cancer, autoimmune diseases, and viral infections.</p>
    Fórmula:C29H23NO10
    Cor e Forma:Solid
    Peso molecular:545.494
  • DSPE-PEG1000-PP1


    <p>DSPE-PEG1000-PP1 is a PEG compound composed of DSPE and the PP1 peptide. The PP1 peptide targets inflammatory atherosclerotic plaques. DSPE-PEG1000-PP1 is suitable for drug delivery applications.</p>
    Cor e Forma:Odour Solid
  • Vitamin D4

    CAS:
    <p>Vitamin D4 is the active Vitamin D analog.</p>
    Fórmula:C28H46O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:398.66
  • Retinyl glucoside

    CAS:
    <p>Retinyl-β-D-glucoside, a biologically active metabolite of vitamin A, naturally occurs in fish and mammals.</p>
    Fórmula:C26H40O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:448.59
  • (±)10(11)-DiHDPA

    CAS:
    <p>(±)10(11)-DiHDPA is produced from cytochrome P450 epoxygenase action on docosahexaenoic acid .</p>
    Fórmula:C22H34O4
    Cor e Forma:Solid
    Peso molecular:362.51
  • IDO1-IN-24


    <p>IDO1-IN-24 (compound 2c) inhibits the production of IDO1 during cell assays, with an IC50 value of 17 μM.</p>
    Fórmula:C18H22N2O4
    Peso molecular:330.15796
  • Zymostenol

    CAS:
    <p>Zymostenol (5a-Cholest-8-en-3b-ol) is a RORγ agonist with an EC50 of 1 μM.Zymostenol is a late stage precursor of cholesterol biosynthesis.</p>
    Fórmula:C27H46O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:386.65
  • Cytoglobosin C

    CAS:
    <p>Cytoglobosin C, a derivative of cytochalasan, demonstrates significant cytotoxic effects on SGC-7901 and A549 cell lines, with an inhibitory concentration (IC50</p>
    Fórmula:C32H38N2O5
    Cor e Forma:Solid
    Peso molecular:530.65
  • Asundexian

    CAS:
    <p>Asundexian (BAY-2433334) is a potent and orally active inhibitor of the coagulation factor FXIa that directly and reversibly binds to the active site of FXIa,</p>
    Fórmula:C26H21ClF4N6O4
    Pureza:99.89% - 99.90%
    Cor e Forma:Solid
    Peso molecular:592.93
  • Galcuronokinase (AtGalAK)


    <p>AtGalAK, a GHMP kinase, converts d-GalA to GalA-1-P using ATP.</p>
    Cor e Forma:Solid
  • Bacterial α-Amylase

    CAS:
    <p>Bacterial α-Amylase is an enzyme that catalyzes the hydrolysis reaction of starch into smaller sugar molecules such as maltose and glucose.</p>
    Cor e Forma:Solid
  • LDHA-IN-3

    CAS:
    <p>LDHA-IN-3 is a potent selenobenzene-based LDHA inhibitor with a 145.2 nM IC50, useful in cancer research.</p>
    Fórmula:C13H9F3Se
    Pureza:99.71%
    Cor e Forma:Solid
    Peso molecular:301.17
  • N-acetyl Leukotriene E4

    CAS:
    <p>N-acetyl Leukotriene E4 is an endogenous metabolite of Leukotriene E4, less active than Leukotriene E4, causing constriction of the airways.</p>
    Fórmula:C25H39NO6S
    Cor e Forma:Solid
    Peso molecular:481.65
  • A 58365 A

    CAS:
    <p>A 58365 A, an ACE inhibitor from Streptomyces chromofuscus, treats heart failure and hypertension.</p>
    Fórmula:C12H13NO6
    Cor e Forma:Solid
    Peso molecular:267.23
  • BPP

    CAS:
    <p>BPP is a fluorescent microviscosity probe used to image natural HOBr in living cells and zebrafish.</p>
    Fórmula:C13H13NS
    Cor e Forma:Solid
    Peso molecular:215.31
  • (±)20-HDHA

    CAS:
    <p>(±)20-HDHA is an autoxidation product and is a racemic mixture of Docosahexaenoic acid (DHA).</p>
    Fórmula:C22H32O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:344.49
  • Ser-Ala-alloresact acetate


    <p>Ser-Ala-alloresact acetate is a sperm-activating peptide (SAP) that is released by marine invertebrate eggs and plays an important role in fertilization.</p>
    Fórmula:C44H75N13O16S2
    Pureza:99.73%
    Cor e Forma:Solid
    Peso molecular:1106.28
  • 3α-Hydroxysteroid dehydrogenase

    CAS:
    <p>3α-Hydroxysteroid dehydrogenase (3α-HSD), encoded by the AKR1C4 gene, is responsible for catalyzing the transformation of 3-ketosteroids into 3α-hydroxy</p>
    Cor e Forma:Solid
  • Promothiocin A

    CAS:
    <p>Promothiocin A is an antibiotic.</p>
    Fórmula:C36H37N11O8S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:815.88
  • SMS2-IN-1

    CAS:
    <p>SMS2-IN-1: potent SMS2 inhibitor; IC50: 6.5 nM, Kd: 37 nM; 150x selectivity over SMS1.</p>
    Fórmula:C34H37F6N3O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:681.67
  • SGK1-IN-4

    CAS:
    <p>SGK1-IN-4 is a selective inhibitor of SGK1 and can be used in studies about osteoarthritis.</p>
    Fórmula:C23H21ClFN5O4S
    Pureza:97.03%
    Cor e Forma:Solid
    Peso molecular:517.96
  • SBI993

    CAS:
    <p>SBI993, a SBI-477 analog, confirms MondoA gene action in vivo and lowers muscle TAG and liver fat.</p>
    Fórmula:C23H23N3O5S
    Pureza:99.20%
    Cor e Forma:Solid
    Peso molecular:453.51
  • CAY10434

    CAS:
    <p>CAY10434, a potent CYP4A hydroxylase inhibitor, has an IC50 of 8.8 nM and boosts angiotensin II contraction, Emax 6764 mg.</p>
    Fórmula:C17H25N3O
    Pureza:99.85%
    Cor e Forma:Solid
    Peso molecular:287.4
  • PEG2000-C-DMG

    CAS:
    <p>PEG2000-C-DMG is a pegylated lipid for Onpattro, reducing transthyretin production via RNAi.</p>
    Fórmula:C126H249NO52
    Cor e Forma:Solid
    Peso molecular:2000 (Average)
  • γ-Acetylenic GABA hydrochloride

    CAS:
    <p>γ-Acetylenic GABA hydrochloride is a GABA transaminase inhibitor.</p>
    Fórmula:C6H10ClNO2
    Pureza:99.28% - 99.64%
    Cor e Forma:Solid
    Peso molecular:163.6
  • Estriol 16α-(β-D-glucuronide)

    CAS:
    <p>Estriol 16α-(β-D-glucuronide), an endogenous metabolite found in urine, is utilized in pregnancy research [1] [2].</p>
    Fórmula:C24H32O9
    Cor e Forma:Solid
    Peso molecular:464.51
  • Glycodeoxycholic acid monohydrate

    CAS:
    <p>Glycodeoxycholic acid monohydrate is a nuclear receptor ligand.</p>
    Fórmula:C26H45NO6
    Cor e Forma:Solid
    Peso molecular:467.64
  • ACAT-IN-10 dihydrochloride

    CAS:
    <p>ACAT-IN-10 dihydrochloride, from EP1236468A1 example 197, inhibits acyl-CoA: cholesterol acyltransferase and reduces NF-κB transcription.</p>
    Fórmula:C35H58Cl2N4O5S
    Cor e Forma:Solid
    Peso molecular:717.83
  • D-γ-Glutamyl-D-glutamic acid

    CAS:
    D-γ-Glutamyl-D-glutamic acid is a linear polymer with repeating D-glutamic acid units, useful in studies of microbial cell walls and immunological recognition.
    Fórmula:C10H16N2O7
    Pureza:99.41%
    Cor e Forma:Solid
    Peso molecular:276.24
  • Diaphorase

    CAS:
    <p>Diaphorase from anaerobic sludge catalyzes RDX biotransformation via denitrification.</p>
    Cor e Forma:Solid
  • 16(S)-HETE

    CAS:
    <p>16(S)-HETE, a CYP450 byproduct of arachidonic acid, inhibits kidney tubule ATPase by 60% at 2 μM upon angiotensin II trigger.</p>
    Fórmula:C20H32O3
    Cor e Forma:Solid
    Peso molecular:320.473
  • Fellutanine A

    CAS:
    <p>Fellutanine A is a useful organic compound for research related to life sciences. The catalog number is T129801 and the CAS number is 175414-35-4.</p>
    Cor e Forma:Soild
  • Histone acetyltransferase p300 Inhibitor 4c

    CAS:
    <p>2-Amino-4-(4-chlorophenyl)thiazole blocks hCA I/II, AChE, BChE with Ki: ~0.008, 0.124, 0.129, 0.083 µM.</p>
    Fórmula:C9H7ClN2S
    Pureza:99.76%
    Cor e Forma:Solid
    Peso molecular:210.68
  • BSO-07


    <p>BSO-07 is a ROS/JNK activator that exhibits potent anti-cancer properties, demonstrated by an IC50 of 24.81 μM in human breast cancer (BC) cells. The mechanism of action for BSO-07 involves JNK activation and the promotion of increased ROS levels, which lead to the induction of apoptosis (Apoptosis) and tumorigenic apoptosis. This includes enhanced expression of apoptosis-related proteins such as PARP, Bax, phosphorylated p53, ATF4, and CHOP, along with a reduction in the levels of anti-apoptotic proteins (e.g., Bcl-2, Bcl-xL, and Survivin). BSO-07 holds promise for research in the field of breast cancer.</p>
    Cor e Forma:Odour Solid
  • hBChE-IN-3


    <p>hBChE-IN-3 (compound 30) serves as both an activator of carbonic anhydrase (CA) and an inhibitor of cholinesterase (ChE), exhibiting IC50 values of 7.4 nM for AchE and 1.9 nM for BchE. This compound is utilized in the research of neurodegenerative and psychiatric disorders.</p>
    Cor e Forma:Odour Solid
  • CAIX/CAXII-IN-3


    <p>CAIX/CAXII-IN-3 (compound 11) serves as an inhibitor for CAIX/CAXII, exhibiting an IC50 value of less than 65 nM. Additionally, this compound effectively inhibits the proliferation of human melanoma cells.</p>
    Cor e Forma:Odour Solid
  • β-Glucosidase

    CAS:
    <p>β-Glucosidase is a glucoside bond hydrolase involved in glucose metabolism and can be used to study diseases caused by abnormal glucose metabolism.</p>
    Fórmula:C24H44O12
    Cor e Forma:Solid
    Peso molecular:524.6
  • 17(R)-HETE

    CAS:
    <p>Kidney sodium transport is partly controlled by 17-HETE, a CYP450 metabolite of arachidonic acid, with the (S) enantiomer inhibiting ATPase at 2 μM.</p>
    Fórmula:C20H32O3
    Cor e Forma:Solid
    Peso molecular:320.473
  • DSPE-PEG5000-KAA


    <p>DSPE-PEG5000-KAA is a PEG compound composed of DSPE and the CKAAKNK (KAA) peptide. The CKAAKNK peptide specifically targets the tumor vasculature of RIP-Tag2 transgenic mice. DSPE-PEG5000-KAA can be utilized for drug delivery purposes.</p>
    Cor e Forma:Odour Solid
  • IP3RPEP6

    CAS:
    <p>IP3RPEP6 serves as a competitive inhibitor of IP3R. Its IC50 values for IP3R1, IP3R2, and IP3R3 are 9.0 μM, 3.9 μM, and 4.3 μM, respectively. This compound does not affect ryanodine receptors and Cx43 hemichannels, and it is capable of modulating intracellular calcium signaling.</p>
    Fórmula:C49H79N15O24
    Cor e Forma:Solid
    Peso molecular:1262.24
  • DSPE-PEG5000-GRGDS


    <p>DSPE-PEG5000-GRGDS is a PEG compound composed of DSPE and the anti-adhesion peptide (GRGDS). GRGDS can inhibit the binding and adhesion between the extracellular matrix and cell surface integrins. DSPE-PEG5000-GRGDS is applicable for drug delivery.</p>
    Cor e Forma:Odour Solid
  • Pseudoerythromycin A enol ether

    CAS:
    <p>Pseudoerythromycin A enol ether, a non-antibiotic erythromycin degradation product, serves as a standard in stability studies.</p>
    Fórmula:C37H65NO12
    Cor e Forma:Solid
    Peso molecular:715.91
  • Xanthine oxidase-IN-16


    <p>Xanthine oxidase-IN-16 is an effective orally active inhibitor of xanthine oxidase (XO), demonstrating significant therapeutic efficacy in rats with hyperuricemia and an IC50 of 102 nM.</p>
    Cor e Forma:Odour Solid
  • Curcumin monoglucuronide

    CAS:
    <p>Curcumin monoglucuronide, curcumin's in vivo metabolite, useful for metabolic research and cancer study.</p>
    Fórmula:C27H28O12
    Cor e Forma:Solid
    Peso molecular:544.50
  • 20,26-Dihydroxyecdysone

    CAS:
    <p>20,26-Dihydroxyecdysone is a predominant ecdysteroid metabolite [1] .</p>
    Fórmula:C27H44O8
    Cor e Forma:Solid
    Peso molecular:496.63
  • Glycidamide

    CAS:
    <p>Glycidamide is a carcinogen and metabolite of acrylamide that induces DNA adduct formation and mutations.</p>
    Fórmula:C3H5NO2
    Cor e Forma:Solid
    Peso molecular:87.08
  • 13-epi-12-oxo Phytodienoic Acid

    CAS:
    <p>13-epi-12-oxo PDA is a lipoxygenase derivative of α-linolenic acid in green plant leaves, often isomerizing during extraction and storage.</p>
    Fórmula:C18H28O3
    Cor e Forma:Solid
    Peso molecular:292.41
  • α-Glucosidase-IN-67


    α-Glucosidase-IN-67 (compound 5k) is a potent inhibitor of α-glucosidase, exhibiting IC50 values of 0.31 µM for α-glucosidase and 4.51 µM for α-amylase. This compound shows potential for research in type 2 diabetes.
    Fórmula:C24H22BrN3O3S
    Peso molecular:511.05653
  • 1-Myristoyl-2-hydroxy-sn-glycero-3-PE

    CAS:
    <p>Naturally-occurring lysophospholipid raises intracellular calcium and is higher in breast cancer patients.</p>
    Fórmula:C19H40NO7P
    Cor e Forma:Solid
    Peso molecular:425.50
  • 1-Naphthyl 3,5-dinitrobenzoate

    CAS:
    <p>1-Naphthyl 3,5-dinitrobenzoate (JMC-4) is an inhibitor of 5-LOX can be used in studies about inflammatory therapy.</p>
    Fórmula:C17H10N2O6
    Pureza:99.79%
    Cor e Forma:Solid
    Peso molecular:338.27
  • Sarcophine

    CAS:
    <p>Sarcophine is a natural cembranoid from the Red Sea soft coral Sarcophyton glaucum.</p>
    Fórmula:C20H28O3
    Cor e Forma:Solid
    Peso molecular:316.441
  • 5,6-epoxy-13-cis Retinoic Acid

    CAS:
    <p>5,6-epoxy-13-cis Retinoic Acid is a metabolite of 13-cis retinoic acid.</p>
    Fórmula:C20H28O3
    Cor e Forma:Solid
    Peso molecular:316.441
  • SX29


    <p>SX29 is a non-competitive α-glucosidase inhibitor with oral activity, exhibiting an IC50 of 2.12 μM. It possesses hypoglycemic properties; oral administration of SX29 reduces blood glucose levels and enhances glucose tolerance in diabetic mice.</p>
    Cor e Forma:Odour Solid
  • α-Glucosidase-IN-74


    <p>α-Glucosidase-IN-74, a nicotinamide-thiazole derivative, functions as an α-glucosidase (α-glucosidase) inhibitor. It demonstrates antidiabetic activity by reducing blood glucose and triglyceride levels in Streptozotocin-induced diabetic animals.</p>
    Cor e Forma:Odour Solid
  • (±)7(8)-EpDTE

    CAS:
    <p>(±)7(8)-EpDTE is an oxylipin and an oxidative metabolite of docosapentaenoic acid .</p>
    Fórmula:C22H34O3
    Cor e Forma:Solid
    Peso molecular:346.511
  • Prunetin 5-O-β-D-glucopyranoside

    CAS:
    <p>Prunetin 5-O-β-D-glucopyranoside, an isoflavone obtained from Potentilla astracanica extracts, is a potent uncompetitive inhibitor of α-glucosidase (IC 50 = 56.</p>
    Fórmula:C22H22O10
    Cor e Forma:Solid
    Peso molecular:446.408
  • Aromatase-IN-2

    CAS:
    <p>Aromatase-IN-2 has anti-inflammatory, antitumor and antiasthmatic effects.</p>
    Fórmula:C17H22N2O
    Pureza:99.80%
    Cor e Forma:Solid
    Peso molecular:270.37
  • N-Trifluoroacetyladriamycin

    CAS:
    <p>N-Trifluoroacetyladriamycin, Valrubicin's metabolite, treats bladder cancer; it's an analog of doxorubicin, infused into the bladder.</p>
    Fórmula:C29H28F3NO12
    Cor e Forma:Solid
    Peso molecular:639.533
  • DSPE-PEG5000-NGR


    <p>DSPE-PEG5000-NGR is a PEG compound composed of DSPE and the Asn-Gly-Arg (NGR) peptide. The NGR peptide has the capability to target tumor vasculature antigen CD13. DSPE-PEG5000-NGR is applicable in drug delivery.</p>
    Cor e Forma:Odour Solid
  • Phenacaine

    CAS:
    <p>Phenacaine, also known as Holocaine, is a local anesthetic that blocks certain Ca 2+ enzymes in red blood cells, brain, and heart.</p>
    Fórmula:C18H22N2O2
    Cor e Forma:Solid
    Peso molecular:298.38
  • MNI caged kainic acid

    CAS:
    <p>Generates large inward currents at resting membrane potential</p>
    Fórmula:C19H23N3O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:389.40
  • 2-Aminoflubendazole

    CAS:
    <p>2-Aminoflubendazole, a metabolite of benzimidazoles (BZ), belongs to a class of drugs effective against fungi, protozoa, and helminths.</p>
    Fórmula:C14H10FN3O
    Cor e Forma:Solid
    Peso molecular:255.25
  • Mersalyl

    CAS:
    <p>Mersalyl is an organic mercurial diuretic.</p>
    Fórmula:C13H16HgNNaO6
    Cor e Forma:Solid
    Peso molecular:505.854
  • Rubratoxin A

    CAS:
    <p>Rubratoxin A is a classical mycotoxin used as a PP2A-specific inhibitor.</p>
    Fórmula:C26H32O11
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:520.531
  • 8-Demethyl Ivabradine

    CAS:
    <p>8-Demethyl Ivabradine, a metabolite of Ivabradine, is an oral HCN channel blocker.</p>
    Fórmula:C26H34N2O5
    Cor e Forma:Solid
    Peso molecular:454.567
  • 7β,25-Dihydroxycholesterol

    CAS:
    <p>7β,25-Dihydroxycholesterol, an endogenous metabolite, functions as chemoattractants for immune cells that express EBI2 [1].</p>
    Fórmula:C27H46O3
    Cor e Forma:Solid
    Peso molecular:418.65
  • Pectin

    CAS:
    <p>Pectin, a plant cell wall derived heteropolysaccharide, forms nanoparticles for delivery and acts as an antimicrobial adsorbent.</p>
    Cor e Forma:Solid
  • Tacalcitol monohydrate

    CAS:
    <p>Tacalcitol monohydrate(Curatoderm monohydrate), a vitamin D3 analog that promotes bone development by regulating calcium ions, can be used to study psoriasis.</p>
    Fórmula:C27H46O4
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:434.65
  • Calcitetrol

    CAS:
    <p>Calcitetrol is the hormonally active form of vitamin D with three hydroxyl groups.</p>
    Fórmula:C27H44O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:432.64
  • Glycolithocholic acid, sodium salt

    CAS:
    <p>Sodium glycolithocholate is a bile acid salt used to diagnose UC, NASH, and PSC.</p>
    Fórmula:C26H42NNaO4
    Pureza:99.95%
    Cor e Forma:Solid
    Peso molecular:455.61
  • α-Glucosidase-IN-57


    <p>α-Glucosidase-IN-57 (Compound 10c) is a competitive, orally active α-glucosidase inhibitor with an IC50 of 0.180 μM and a Ki of 0.15 μM. It effectively reduces fasting and overall blood glucose levels in mice, making it suitable for antidiabetic research.</p>
    Fórmula:C32H23FN4OS
    Peso molecular:530.15766
  • SF2312 ammonium


    <p>SF2312 ammonium is the ammonium salt of SF2312, a phosphonate antibiotic and enolase inhibitor derived from the actinomycete Micromonospora and active under</p>
    Fórmula:C4H11N2O6P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:214.11
  • Geranyl pyrophosphate triammonium

    CAS:
    <p>Geranyl pyrophosphate, an intermediary for making cholesterol, terpenes, and others, forms from dimethylallyl and isopentenyl pyrophosphates.</p>
    Fórmula:C10H29N3O7P2
    Cor e Forma:Solid
    Peso molecular:365.304
  • Kallikrein

    CAS:
    <p>Kallikrein is capable of forming the kallikrenase kalinin system (KKS) in plasma and tissues, producing bradykinin and kalin peptides , respectively [1] .</p>
    Cor e Forma:Solid
  • 4-hydroxy Nonenal Mercapturic Acid

    CAS:
    <p>Peroxidation of ω-6 PUFAs produces 4-HNE, which is rapidly cleared and excreted, mostly as urine metabolites, within 48h in rats.</p>
    Fórmula:C14H25NO5S
    Cor e Forma:Solid
    Peso molecular:319.42
  • AMK318


    AMK318 (Immobilized cephalexin acylase) is a biocatalyst and a critical enzyme in novel biocatalyst technology. Enzyme engineering focuses on improving enzyme reaction kinetics, substrate selectivity, and activity under harsh conditions (such as low or high pH). By incorporating stimulus responsiveness into these enzyme modifications, dynamic control of activity becomes feasible.
  • Coformycin

    CAS:
    <p>Coformycin is a ribonucleoside antibiotic synergist and adenosine deaminase inhibitor.</p>
    Fórmula:C11H16N4O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:284.27
  • S32826

    CAS:
    <p>S32826, a potent autotaxin inhibitor with an IC50 of 8.8 nM, blocks LPA release and targets α, β, γ isoforms.</p>
    Fórmula:C21H36NO4P
    Cor e Forma:Solid
    Peso molecular:397.496
  • PR280


    <p>PR280 is a potent inhibitor of dihydroceramide desaturase 1 (Des1) with an IC50 of 700 nM. It forms hydrogen bonds with amino acid residues of Des1, while its cyclopropenone group may coordinate with the iron center, stabilizing its binding at Des1's active site. This inhibits the ceramide biosynthesis pathway, preventing dihydroceramide (dhCer) from converting into ceramide. PR280 can be used in research related to sphingolipid metabolism disorders, including cancer and metabolic diseases.</p>
    Fórmula:C27H49NO4
    Peso molecular:451.36616
  • 3α,7α-Dihydroxycoprostanic acid

    CAS:
    3α,7α-Dihydroxycoprostanic acid, an endogenous metabolite and bile acid, serves as the precursor to chenodeoxycholic acid [1].
    Fórmula:C27H46O4
    Peso molecular:434.65
  • GLUT1-IN-1


    <p>GLUT1-IN-1 inhibits GLUT1; cytotoxic to HeLa, A549, HepG2 (IC50: 5.49, 11.14, 8.73 μM); potential in PDT and cancer research.</p>
    Fórmula:C25H31BF2I2N6O7
    Cor e Forma:Solid
    Peso molecular:830.17
  • Mitochondrial respiration-IN-3


    <p>Mitochondrial respiration-IN-3, a cell-permeable fluorine derivative of Dalfopristin, inhibits glioblastoma stem cell translation for cancer research.</p>
    Fórmula:C35H51FN4O7S
    Cor e Forma:Solid
    Peso molecular:690.87
  • Impurity B of Calcitriol

    CAS:
    <p>Impurity B is a byproduct of Calcitriol, the active hormone form of vitamin D3 and VDR activator.</p>
    Fórmula:C27H44O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:416.64
  • 5A2-SC8 TFA


    <p>5A2-SC8 TFA is an ionizable amino lipid used in lipid nanoparticles (LNPs), offering high delivery potential and low in vivo toxicity. It effectively delivers small RNAs, such as siRNA and miRNA, to tumor cells. Moreover, 5A2-SC8 TFA LNPs provide unique delivery paths for RNA within the liver, enhancing therapeutic outcomes in cancer models.</p>
    Cor e Forma:Odour Solid
  • α-Amylase/α-Glucosidase-IN-11


    <p>α-Amylase/α-Glucosidase-IN-11 (Compound 5d) is an isoxazoline-indigo hybrid with notable antidiabetic properties. It acts as a competitive inhibitor of the key digestive enzymes α-amylase (IC50 = 30.39 μM) and α-glucosidase (IC50 = 65.1 μM). Additionally, it does not penetrate the blood-brain barrier.</p>
    Fórmula:C33H40ClN5O5
    Peso molecular:621.2718
  • Myristoyl coenzyme A lithium

    CAS:
    <p>Myristoyl coenzyme A lithium, a compound marked by lithium in its myristoylated form, plays a crucial role in the biochemical mechanism of myristoylation, essential for both viral functionalities and tumor growth in colon epithelial cells. This process is predominantly governed by N-myristoyltransferase (NMT), which exhibits increased activity in colon epithelial tumors compared to normal cells. The activity of NMT is significantly influenced by the reduction of coenzyme A (CoA), a vital regulator that enhances NMT's ability to induce myristoylation, unlike its oxidized form which impedes this process. Consequently, Myristoyl coenzyme A serves as an inhibitor to the demyristoylation activity, showcasing its potential as an anticancer and antiviral agent.</p>
    Fórmula:C35H63LiN7O17P3S
    Cor e Forma:Solid
    Peso molecular:985.3374
  • SGK1-IN-3 hydrochloride


    <p>SGK1-IN-3 hydrochloride (compound 3a) is an efficacious, orally bioavailable SGK1 inhibitor. The serine/threonine kinase SGK1 acts as an activator of the β-catenin pathway and strongly stimulates cartilage degradation, being upregulated under genomic control in diseased osteoarthritic cartilage. SGK1-IN-3 hydrochloride holds potential for osteoarthritis research.</p>
    Fórmula:C23H21Cl3N6O3S
    Peso molecular:566.04614
  • α-Glucosidase-IN-60


    <p>α-Glucosidase-IN-60 (Compound 5k) acts as a competitive inhibitor of α-Glucosidase, with an IC50 of 10.8 μM.</p>
    Fórmula:C23H14N2O5
    Peso molecular:398.09027
  • Berninamycin D

    CAS:
    <p>Berninamycin D, a cyclic peptide derived from Streptomyces bernensis through fermentation, is recognized as a fungal metabolite [1].</p>
    Fórmula:C45H45N13O13S
    Cor e Forma:Solid
    Peso molecular:1007.98
  • BChE-IN-36


    <p>hBChE-IN-4 (compound 40) serves as an effective activator for hCA and an inhibitor for BChE. It demonstrates affinity for various hCA subtypes with affinity constants (KA) of 266 nM for hCA I, 76.9 nM for hCA II, 918 nM for hCA IV, 893 nM for hCA VB, and 98.0 nM for hCA VII. Inhibition concentrations (IC50) for eeAChE and eqBChE are recorded at 72.1 nM and 4.2 nM, respectively. hBChE-IN-4 is non-cytotoxic and has demonstrated potential cognitive enhancement effects. It holds potential for research in neurodegenerative and other neuropsychiatric disorders.</p>
    Cor e Forma:Odour Solid
  • (±)10(11)-EpDPA

    CAS:
    <p>Cytochrome P450 metabolism of polyunsaturated fatty acids produces numerous bioactive epoxide regioisomers.</p>
    Fórmula:C22H32O3
    Cor e Forma:Solid
    Peso molecular:344.495
  • Netupitant metabolite Netupitant N-oxide

    CAS:
    <p>Netupitant N-oxide is a highly selective antagonist of NK1 receptor, is Netupitant metabolite.</p>
    Fórmula:C30H32F6N4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:594.59
  • Calcium 2-oxoglutarate

    CAS:
    <p>Calcium 2-oxoglutarate is an intermediate in the production of GTP or ATP in the Krebs cycle. It is a reversible inhibitor of tyrosinase (IC50: 15 mM).</p>
    Fórmula:C5H8CaO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:188.192
  • (Z)-7-Dodecen-1-ol

    CAS:
    (Z)-7-Dodecen-1-ol counteracts the attractive properties of Z-7-dodecen-1-yl acetate.
    Fórmula:C12H24O
    Peso molecular:184.32
  • Triornicin

    CAS:
    <p>Triornicin is a siderophore and tumor inhibitory factor isolated from Epicoccum purpurascens similar in structure to desferricoprogen.</p>
    Fórmula:C31H50N6O12
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:698.76
  • SDUY817


    <p>SDUY817 is a dual APN/NEP inhibitor with IC50 values of 0.29 μM for APN and 7.4 μM for NEP. It exhibits analgesic effects in a concentration- and time-dependent manner, making it a potential candidate for research in the field of neuropathic pain disorders.</p>
    Fórmula:C18H16IN3O3
    Cor e Forma:Solid
    Peso molecular:449.24
  • Reduced Haloperidol

    CAS:
    <p>Reduced haloperidol, an active metabolite of haloperidol, binds dopamine D2/sigma-1 receptors and inhibits neurotransmitter reuptake.</p>
    Fórmula:C21H25ClFNO2
    Cor e Forma:Solid
    Peso molecular:377.88
  • VDR agonist 2


    <p>VDR agonist 2 (compound 16i), a vitamin D receptor (VDR) agonist, effectively inhibits TGF-β1-induced hepatic stellate cell (HSC) activation, demonstrating</p>
    Fórmula:C20H21F3O3
    Cor e Forma:Solid
    Peso molecular:366.37
  • 1,2,3,6,7,8-Hexachlorodibenzofuran

    CAS:
    <p>1,2,3,6,7,8-Hexachlorodibenzofuran (1,2,3,6,7,8-HxCDF) is a type of polychlorinated dibenzofuran (PCDF). It promotes the expression of aryl hydrocarbon hydroxylase (AHH) and ethoxyresorufin-O-deethylase (EROD) genes in H-4-II-E rat hepatoma cells with EC50 values of 1.47 and 1.24 nM, respectively. 1,2,3,6,7,8-HxCDF also reduces rat body weight, causes thymic atrophy, and induces the expression of cytochrome P450 (CYP) subtype CYP1A1 and 4-chlorobiphenyl hydroxylase genes with EC50 values of 3.2, 0.9, 0.35, and 0.21 µmol/kg.</p>
    Fórmula:C12H2Cl6O
    Cor e Forma:Solid
    Peso molecular:374.86
  • 2-Methoxy-4-propylphenol

    CAS:
    <p>2-Methoxy-4-propylphenol is an inhibitor of human carbonic anhydrase isoenzymes 1/2/9/12 and has antifungal activity.</p>
    Fórmula:C10H14O2
    Cor e Forma:Solid
    Peso molecular:166.22
  • VM4-037

    CAS:
    <p>VM4-037 is a PET imaging agent used for carbonic anhydrase IX.</p>
    Fórmula:C26H29FN6O7S2
    Cor e Forma:Solid
    Peso molecular:620.67
  • C18:1 Ceramide (d18:1/18:1(9Z))

    CAS:
    <p>C18:1 Ceramide (d18:1/18:1(9Z)) is a ceramide, and C18:1-Ceramide levels are elevated in overweight and insulin-resistant , advanced ovarian cancer.</p>
    Fórmula:C36H69NO3
    Pureza:99.96%
    Cor e Forma:Solid
    Peso molecular:563.94
  • CETP-IN-4

    CAS:
    <p>CETP-IN-4 is a cholesteryl ester transfer protein (CETP) inhibitor.</p>
    Fórmula:C36H28F9N3O4
    Cor e Forma:Solid
    Peso molecular:737.623
  • Tetracosanoyl-sulfatide

    CAS:
    <p>C24 3'-sulfo Galactosylceramide is a key myelin sulfatide, high in leukodystrophy patients, non-immunogenic compared to C24:1 variant.</p>
    Fórmula:C48H93NO11S
    Cor e Forma:Solid
    Peso molecular:892.32
  • Streptolysin O

    CAS:
    <p>Streptolysin O: lyses cells, cardiotoxic, used for cell permeabilization, has active and inactive states.</p>
    Pureza:98%
    Cor e Forma:Solid
  • (±)-Hexanoylcarnitine chloride

    CAS:
    <p>(±)-Hexanoylcarnitine chloride is a fatty acid metabolite that breaks down fatty acids into small compounds that can be utilized by the body.</p>
    Fórmula:C13H26ClNO4
    Pureza:99.45%
    Cor e Forma:Solid
    Peso molecular:295.8
  • (1S)-Calcitriol

    CAS:
    <p>(1S)-Calcitriol, a natural 1α,25(OH)2D3 metabolite, regulates VDR actions like keratinocyte growth inhibition.</p>
    Fórmula:C27H44O3
    Cor e Forma:Solid
    Peso molecular:416.646
  • Ruthenoleuton


    <p>Ruthenoleuton is a 5-lipoxygenase (5-LOX) inhibitor with an IC50 of 3.49 μM and a Ki of 0.80 μM. It possesses antioxidant properties and is applicable in research on inflammatory diseases.</p>
    Fórmula:C13H16N2O2Ru
    Cor e Forma:Solid
    Peso molecular:333.35
  • Ribulose, L-

    CAS:
    <p>Ribulose: key in pentose metabolism, aids L-ribose isomerase study, yeast engineering, and chiral compound research.</p>
    Fórmula:C5H10O5
    Cor e Forma:Solid
    Peso molecular:150.13
  • Bicyclic UK18

    CAS:
    <p>Bicyclic UK18 is a competitive inhibitor of human urokinase-type plasminogen activator (uPA) with a Ki value of 53 nM.</p>
    Fórmula:C77H118N26O25S3
    Cor e Forma:Solid
    Peso molecular:1904.11
  • γ-Glu-Gly TFA


    <p>γ-Glu-Gly TFA, a γ-glutamyl dipeptide, is a human lipid metabolite with a structure resembling GABA (γ-aminobutyric acid).</p>
    Cor e Forma:Liquid
  • Trimipramine N-oxide

    CAS:
    <p>Trimipramine N-oxide, a trimipramine metabolite, inhibits hNAT, hSERT, hDAT, and hOCT1/2 with IC50s 11.7-27.4 nM; for depression/anxiety research.</p>
    Fórmula:C20H26N2O
    Cor e Forma:Solid
    Peso molecular:310.43
  • α-D-Glucose-1-phosphate disodium hydrate

    CAS:
    <p>α-D-Glucose-1-phosphate disodium hydrate serves multiple roles in medical and biochemical applications, including as a precursor in the synthesis of glucuronic</p>
    Fórmula:C6H15Na2O11P
    Cor e Forma:Solid
    Peso molecular:340.13
  • DSPE-PEG3000-R6H4


    <p>DSPE-PEG3000-R6H4 is a PEG compound composed of DSPE and the pH-responsive transmembrane peptide (R6H4). R6H4 is applicable for pH-responsive anticancer drug delivery. DSPE-PEG3000-R6H4 can be utilized for drug delivery purposes.</p>
    Cor e Forma:Odour Solid
  • 4-Hydroxybenzoic acid-d4

    CAS:
    <p>4-Hydroxybenzoicacid-d4 is a deuterated form of 4-Hydroxybenzoicacid, which is a phenolic derivative of benzoic acid. It is effective in inhibiting most Gram-positive bacteria and some Gram-negative bacteria with an IC50 of 160 μg/mL.</p>
    Fórmula:C7H6O3
    Cor e Forma:Solid
    Peso molecular:142.15
  • trans-2-Hexadecenoyl-L-carnitine

    CAS:
    <p>trans-2-Hexadecenoyl-L-carnitine is an endogenous metabolite in urine[1].</p>
    Fórmula:C23H43NO4
    Cor e Forma:Solid
    Peso molecular:397.59
  • Quinaprilat hydrate

    CAS:
    <p>Quinaprilat: active form of quinapril; treats heart failure, hypertension.</p>
    Fórmula:C23H28N2O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:428.48
  • Diglycyl-histidine

    CAS:
    <p>Diglycyl-histidine is a tripeptide complexed with cupric ion designed to mimic specific Cu(II) transport site of ascorbate on albumin molecule.</p>
    Fórmula:C10H15N5O4
    Cor e Forma:Solid
    Peso molecular:269.26
  • Kyotorphin

    CAS:
    <p>Kyotorphin is a Morphine-like dipeptide.</p>
    Fórmula:C15H23N5O4
    Cor e Forma:Solid
    Peso molecular:337.38
  • Deoxyadenosine diphosphate sodium

    CAS:
    <p>Deoxyadenosine diphosphate sodium is a diphosphate nucleoside featuring deoxyadenosine as its nucleoside component. It plays a role in the synthesis and repair of DNA. Deoxyadenosine diphosphate sodium acts as an inhibitor of polynucleotide phosphorylase, thereby interfering with the polymerization of ADP and CDP.</p>
    Fórmula:C10H12N5Na3O9P2
    Cor e Forma:Solid
    Peso molecular:477.15
  • Transketolase-IN-6


    <p>Transketolase-IN-6 (Compound 6bj) serves as a lead compound for herbicides. It achieves approximately 80% root inhibition in redroot pigweed (Amaranthus retroflexus) and green foxtail (Setaria viridis). Moreover, Transketolase-IN-6 is an effective inhibitor of transketolase (TK).</p>
    Fórmula:C23H27ClN6O
    Peso molecular:438.19349
  • BVT-2733 hydrochloride

    CAS:
    <p>BVT-2733 hydrochloride is a potent, selective, and orally active non-steroidal 11β-HSD1 inhibitor. It exhibits stronger inhibition on mouse 11β-HSD1 enzyme (IC50=96 nM) compared to the human 11β-HSD1 enzyme (IC50=3341 nM). BVT-2733 hydrochloride shows potential for research in arthritis and obesity-related diseases.</p>
    Fórmula:C17H22Cl2N4O3S2
    Cor e Forma:Solid
    Peso molecular:465.42
  • MPO-IN-7


    <p>MPO-IN-7 (compound MDC) is a myeloperoxidase inhibitor with IC50 values of 41 μM for α-glucosidase, 25 μM for dipeptidyl peptidase-4, and 4.5 μM for myeloperoxidase. MPO-IN-7 exhibits antioxidant and anti-inflammatory activities in vitro.</p>
    Fórmula:C16H14N2O6
    Peso molecular:330.08519
  • Decanoyl coenzyme A

    CAS:
    <p>Decanoyl coenzyme A (Decanoyl CoA) serves as a primer for the fatty acid elongation system in Mycobacterium smegmatis [1].</p>
    Fórmula:C31H54N7O17P3S
    Cor e Forma:Solid
    Peso molecular:921.78
  • (24S)-MC 976

    CAS:
    <p>(24S)-MC 976 is a derivative of Vitamin D3.</p>
    Fórmula:C27H42O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:414.62
  • IDO1/TDO-IN-7


    <p>IDO1/TDO-IN-7 (Compound 43b), an isochinoline derivative, functions as a potent dual inhibitor of IDO1/TDO with IC50 values of 0.31 μM and 0.08 μM, respectively. Demonstrating favorable pharmacokinetics and strong antitumor efficacy in the B16-F10 tumor model, this compound also exhibits low toxicity.</p>
    Cor e Forma:Odour Solid