Metabolismo
Os inibidores do metabolismo são compostos que interferem nas vias metabólicas, alterando a produção e utilização de energia dentro das células. Esses inibidores são usados para estudar a regulação do metabolismo, o papel das vias metabólicas em doenças como o câncer e o diabetes, e para desenvolver novas estratégias terapêuticas. Os inibidores do metabolismo podem direcionar várias enzimas e processos envolvidos na glicólise, na oxidação de ácidos graxos e em outras funções metabólicas. Na CymitQuimica, oferecemos uma ampla gama de inibidores do metabolismo de alta qualidade para apoiar sua pesquisa em bioquímica, distúrbios metabólicos e desenvolvimento de medicamentos.
Subcategorias de "Metabolismo"
- AhR(41 produtos)
- Aminopeptidase(67 produtos)
- CETP(18 produtos)
- Anidrase carbónica(177 produtos)
- Caseína quinase(130 produtos)
- DHFR(32 produtos)
- Descarboxilase(4 produtos)
- Desidrogenase(267 produtos)
- FAAH(63 produtos)
- FXR(58 produtos)
- Factor Xa(80 produtos)
- Sintase de Ácidos graxos(32 produtos)
- Ferroptose(215 produtos)
- GR(3 produtos)
- GSNOR(3 produtos)
- Glucoquinase(53 produtos)
- HIF/HIF Prolil-Hidroxilase(142 produtos)
- HMG-CoA Reductase(32 produtos)
- Hidroxilase(30 produtos)
- IDO(82 produtos)
- LDL(8 produtos)
- Lipase(96 produtos)
- Lipídio(59 produtos)
- Lipoxigenase(124 produtos)
- MAO(87 produtos)
- MPO(2 produtos)
- NAMPT(36 produtos)
- P450(6 produtos)
- PAI-1(25 produtos)
- PDE(166 produtos)
- PED(1 produtos)
- PKM(15 produtos)
- PPAR(164 produtos)
- Fosfolipase(82 produtos)
- ROR(42 produtos)
- Receptor de Retinóide(29 produtos)
- SGK(11 produtos)
- Tiorredoxina(12 produtos)
- Transferase(30 produtos)
- Tansportador(42 produtos)
- UGT(4 produtos)
- Inibidores de Xantina Oxidase (XO)(9 produtos)
Exibir 34 mais subcategorias
Foram encontrados 8595 produtos de "Metabolismo"
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PD0176078
CAS:<p>PD0176078 () is a newly blocker of N-type Calcium channel.</p>Fórmula:C23H30F2N2OPureza:99.72%Cor e Forma:SolidPeso molecular:388.49Fenleuton
CAS:<p>Fenleuton is a 5-lipoxygenase inhibitor.</p>Fórmula:C17H15FN2O3Pureza:98%Cor e Forma:SolidPeso molecular:314.31BN-82685
CAS:<p>BN-82685, a quinone-based CDC25 inhibitor, shows in vitro and in vivo efficacy, suggesting potential as an anticancer therapy.</p>Fórmula:C12H15N3O2SPureza:98%Cor e Forma:SolidPeso molecular:265.33Enpp-1-IN-8
CAS:<p>Enpp-1-IN-8: potent inhibitor of enpp-1, an enzyme breaking down various nucleotide bonds; potential in cancer/infectious disease research.</p>Fórmula:C19H26N6O4SCor e Forma:SolidPeso molecular:434.51MDK-4823
CAS:<p>MDK-4823 (LMPTP inhibitor1) blocks LMPTP, fighting insulin resistance and diabetes in obesity.</p>Fórmula:C28H36N4OCor e Forma:SolidPeso molecular:444.61ATX inhibitor 14
CAS:<p>ATX inhibitor 14, an indole carbamate, potently blocks self-adhesive proteins (IC50: 0.41 nM), aiding fibrosis research.</p>Fórmula:C26H26Cl2N4O3SCor e Forma:SolidPeso molecular:545.48L-(-)-threo-3-Hydroxyaspartic acid
CAS:<p>L-(-)-threo-3-Hydroxyaspartic acid is an EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor.</p>Fórmula:C4H7NO5Pureza:98%Cor e Forma:SolidPeso molecular:149.1Risotilide
CAS:<p>Risotilide is a voltage-dependent potassium channel inhibitor. It can prolong cardiac action potentials and refractory periods.</p>Fórmula:C15H27N3O4S2Pureza:98%Cor e Forma:SolidPeso molecular:377.52Sp-Cyclic AMPS (sodium salt)
CAS:<p>Sp-cAMPS Na salt activates PKA I/II and competitively inhibits PDE3A (Ki: 47.6 μM), also binds PDE10 GAF (EC50: 40 μM).</p>Fórmula:C10H12N5NaO5PSCor e Forma:SolidPeso molecular:367.25NC1153
CAS:<p>NC1153 blocks IL-2/JAK3/STAT5a/b, aids allograft survival, reduces toxicities.</p>Fórmula:C18H38Cl2N2OPureza:98%Cor e Forma:SolidPeso molecular:369.42MAO-B Inhibitor 58
CAS:<p>MAO-B inhibitor 58 is an effective, selective, and reversible inhibitor of monoamine oxidase B.</p>Fórmula:C14H9Cl2N3Cor e Forma:SolidPeso molecular:290.15Agn 190727
CAS:<p>Agn 190727 is a retonoic acid receptor that can induce retinoid-induced hypertriglyceridemia.</p>Fórmula:C20H22O2Cor e Forma:SolidPeso molecular:294.39α-Glycosidase-IN-1
CAS:<p>α-Glycosidase-IN-1 (compound MZ7) is a potent inhibitor of α-GLY (α-glycosidase) (IC50: 44.72 nM, Ki: 44.74 nM).</p>Fórmula:C21H19N9O6S2Cor e Forma:SolidPeso molecular:557.56Y-29794 oxalate
CAS:<p>Inhibitor of prolyl endopeptidase</p>Fórmula:C25H36N2O5S2Pureza:98%Cor e Forma:SolidPeso molecular:508.69Muristerone A
CAS:<p>Muristerone A is a phytoecdysteroid analog of ecdysone and a potent ecdysteroid receptor agonist with a K d of 1 nM [1].</p>Fórmula:C27H44O8Cor e Forma:SolidPeso molecular:496.63Glucosylceramide synthase-IN-1
CAS:<p>Potent oral GCS inhibitor T-036, crosses BBB, targets human (IC50: 31 nM) and mouse GCS (IC50: 51 nM), for Gaucher disease research.</p>Fórmula:C24H20F4N2O3Cor e Forma:SolidPeso molecular:460.42Mesopram
CAS:<p>PDE4 inhibitor, orally active</p>Fórmula:C14H19NO4Pureza:98%Cor e Forma:SolidPeso molecular:265.3LEO-29102
CAS:<p>LEO-29102: Potent, selective PDE4 inhibitor, promising for treating skin diseases, phase 2 efficacy in atopic dermatitis.</p>Fórmula:C20H22Cl2N2O5Cor e Forma:SolidPeso molecular:441.31Lp-PLA2-IN-11
CAS:<p>Lp-PLA2-IN-11, a potent Lp-PLA2 inhibitor, may be explored for atherosclerosis and Alzheimer's (WO2014114249A1, E145).</p>Fórmula:C22H20F4N4O3Cor e Forma:SolidPeso molecular:464.41Ro 41-0960
CAS:<p>Ro 41-0960 is used as a reversible and orally-active COMT-inhibitor.</p>Fórmula:C13H8FNO5Pureza:98%Cor e Forma:SolidPeso molecular:277.2TMCB
CAS:<p>CK2 and ERK8 inhibitor</p>Fórmula:C11H9Br4N3O2Pureza:98%Cor e Forma:SolidPeso molecular:534.82YM758 Phosphate
CAS:<p>YM758 Phosphate, a current channel inhibitor, selectively lowers a heart beat and decreases oxygen consumption of heart muscle.</p>Fórmula:C26H35FN3O8PPureza:98%Cor e Forma:SolidPeso molecular:567.54BMS 740808
CAS:<p>BMS-740808 is a highly effective and selective factor X inhibitor.</p>Fórmula:C31H27F3N6O3Cor e Forma:SolidPeso molecular:588.58NCX 1000
CAS:<p>NCX 1000 is a liver-specific NO donor compound,NCX 1000 derived from ursodeoxycholic acid (UDCA).</p>Fórmula:C38H55NO10Pureza:98%Cor e Forma:SolidPeso molecular:685.84MAGL-IN-1
CAS:<p>MAGL-IN-1 is a selective and potent monoacylglycerol lipase (MAGL) inhibitor with an IC50 of 80 nM.</p>Fórmula:C22H24FNO3Pureza:98%Cor e Forma:SolidPeso molecular:369.43YZ9
CAS:<p>Y29 is a potent PFKFB3 inhibitor with an IC50 of 0.183 µM, and acts as a competitive inhibitor against Fru-6-P with a Ki of 0.094 µM[1].</p>Fórmula:C12H10O5Pureza:99.59%Cor e Forma:SolidPeso molecular:234.2YM-75466
CAS:<p>YM-75466 is a factor Xa inhibitor reducing TAT in plasma dose-dependently without prolonging coagulation.</p>Fórmula:C28H35N5O8S2Cor e Forma:SolidPeso molecular:633.74ALRT 1550
CAS:<p>ALRT 1550, a retinoic acid agent (RAR) agonist, is used potentially for the treatment of cervical carcinoma.</p>Fórmula:C23H32O2Cor e Forma:SolidPeso molecular:340.5GNE-3500
CAS:<p>GNE-3500: potent, selective RORc inverse agonist; orally bioavailable; promising for treating inflammatory diseases.</p>Fórmula:C24H30FN3O3SCor e Forma:SolidPeso molecular:459.58hCAIX-IN-7
CAS:<p>hCAIX-IN-7 (6c) selectively inhibits tumor-related isoform hCAIX (KI: 410.6 nM) and weakly affects hCAI/II (KI: >10000 nM).</p>Fórmula:C18H12FNO3Cor e Forma:SolidPeso molecular:309.29CG-707
CAS:<p>CG-707 is an inhibitor of PRL-3 that acts by blocking the migration and invasion of metastatic cancer cells.</p>Fórmula:C20H17NO3S2Pureza:98%Cor e Forma:SolidPeso molecular:383.48DMPAC-Chol
CAS:<p>DMPAC-Chol, a cationic cholesterol, aids gene transfection, DNA protection, binds DNA, and lowers HepG2 viability at 37.5 μg/ml.</p>Fórmula:C33H58N2O2Cor e Forma:SolidPeso molecular:514.83Glyoxalase I inhibitor 2
CAS:<p>Glyoxalase I inhibitor 2 (compound 26) blocks GLO1 effectively (IC50: 0.5 μM), promising for depression and anxiety research.</p>Fórmula:C24H23N3O4SCor e Forma:SolidPeso molecular:449.52BI 689648
CAS:<p>BI 689648 is a highly selective inhibitor of aldosterone synthase(CYP11B1 and CYP11B2 with IC50s of 310 and 2.1 nM, respectively).</p>Fórmula:C16H18N4O2Cor e Forma:SolidPeso molecular:298.34Fluindione
CAS:<p>Fluindione is a hematologic drug.</p>Fórmula:C15H9FO2Cor e Forma:SolidPeso molecular:240.23SWE101
CAS:<p>SWE101 is a potent human and rat soluble epoxide hydrolase (sEH)-P inhibitor(IC50s of 4 μM and 2.8 μM, respectively).</p>Fórmula:C19H15Cl2NO3Pureza:98%Cor e Forma:SolidPeso molecular:376.23URB532
CAS:<p>URB532 is an irreversible fatty acid amide hydrolase (FAAH) inhibitor.</p>Fórmula:C18H21NO3Pureza:98%Cor e Forma:SolidPeso molecular:299.364,6-O-Ethylidene-α-D-glucose
CAS:<p>4,6-O-Ethylidene-α-D-glucose (Ethylidene-glucose), a derivative of glucose, serves as a competitive inhibitor for the exofacial binding site of glucose</p>Fórmula:C8H14O6Cor e Forma:SolidPeso molecular:206.19Cyt-PTPε Inhibitor-1
CAS:<p>Cyt-PTPε Inhibitor-1 (A Inhibitor-1) is an inhibitor of cytosolic protein tyrosine phosphatase ε.</p>Fórmula:C19H20N4O2SPureza:99.55% - 99.82%Cor e Forma:SolidPeso molecular:368.45AChE/hCA I/II-IN-1
CAS:<p>Compound 6: Potent inhibitor for AChE, Hca I & II with IC50s of 22.21, 60.79, 66.64 nM, useful in glaucoma, Alzheimer's, diabetes research.</p>Fórmula:C15H13N3SCor e Forma:SolidPeso molecular:267.35sEH inhibitor-6
CAS:<p>sEH inhibitor-6 (Compound 3g) is a highly potent soluble epoxide hydrolase (sEH) inhibitor, exhibiting an IC 50 value of 0.5 nM [1].</p>Fórmula:C21H14ClN3O2Cor e Forma:SolidPeso molecular:375.81OHM1
CAS:<p>OHM1, an analog of HIF1α CTAD, effectively inhibits the interaction between HIF1α CTAD and p300/CBP by targeting the CH1 domain with a binding affinity of 0.53</p>Fórmula:C24H42N6O5Cor e Forma:SolidPeso molecular:494.63CAY10762
CAS:<p>CAY10762, a MAGL inhibitor (IC50=34.1 nM), curbs H2O2-induced LDH in Neuro2a cells and boosts 2-AG in mouse brains at 10 mg/kg.</p>Fórmula:C15H13NOSCor e Forma:SolidPeso molecular:255.33EDP-305
CAS:<p>EDP-305, an oral FXR agonist, has EC50s of 34 nM/8 nM in CHO/HEK cells, aids in PBC and NASH research with antifibrotic properties.</p>Fórmula:C36H58N2O5SCor e Forma:SolidPeso molecular:630.92Anserinone B
CAS:<p>Anserinone B: Antifungal, antibacterial; inhibits S.fimicola (50%), A. furfuraceus (37%); cytotoxic to human tumor cells (GI50=4.4 µg/mL).</p>Fórmula:C11H14O4Cor e Forma:SolidPeso molecular:210.23JBP485
CAS:<p>JBP485 is an inhibitor of renal transporters OAT1 and OAT3. JBP485 is an antihepatitis agent as a substrate for intestinal PEPT1.</p>Fórmula:C8H12N2O4Cor e Forma:SolidPeso molecular:200.19Deltasonamide 2 (TFA)
CAS:<p>Deltasonamide 2 TFA is competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM.</p>Fórmula:C32H40ClF3N6O6S2Pureza:98%Cor e Forma:SolidPeso molecular:761.28ACAT-IN-1 cis isomer
CAS:<p>ACAT-IN-1 cis isomer is a potent ACAT inhibitor (IC50: 100 nM) for the study of immune system-related diseases.</p>Fórmula:C29H25NO2Pureza:>99.99%Cor e Forma:SolidPeso molecular:419.51N-Methylmoranoline
CAS:<p>N-Methylmoranoline is an inhibitor of α-glucosidase.</p>Fórmula:C7H15NO4Pureza:98%Cor e Forma:SolidPeso molecular:177.2GNF7686
CAS:<p>GNF7686 is a novel Trypanosoma cruzi inhibitor.</p>Fórmula:C15H13N3OPureza:98%Cor e Forma:SolidPeso molecular:251.28Pulixin
CAS:<p>Pulixin blocks FREP1 from P. falciparum, hinders parasite spread (EC50: 11µM), and stops its growth (EC50: 47nM).</p>Fórmula:C14H11NO4Cor e Forma:SolidPeso molecular:257.24Nampt-IN-9
CAS:<p>Nampt-IN-9 (Compound 8) is a potent inhibitor of NAMPT with anticancer properties.Nampt-IN-9 can be used to study ductal adenocarcinoma of the pancreas.</p>Fórmula:C26H33N3O4Cor e Forma:SolidPeso molecular:451.56(Rac)-RK-682
CAS:<p>(Rac)-RK-682 racemate; inhibits PTP-1B, LMW-PTP, CDC-25B with IC50s: 8.6, 12.4, 0.7 µM respectively.</p>Fórmula:C21H36O5Cor e Forma:SolidPeso molecular:368.51Ro-15-2041
CAS:<p>Ro 15-2041 is a selective inhibitor of platelet phosphodiesterase, with antithrombotic properties.</p>Fórmula:C12H12BrN3OPureza:98%Cor e Forma:SolidPeso molecular:294.15LTV-1
CAS:<p>LTV-1 has the potential for autoimmunity treatment. LTV-1 is a potent lymphoid tyrosine phosphatase (LYP) inhibitor in T cells with an IC50 of 508 nM.</p>Fórmula:C26H20N2O5SCor e Forma:SolidPeso molecular:472.51PF-04279405
CAS:<p>PF-04279405 is a potent and selective glucokinase activator.</p>Fórmula:C25H25FN4O4Cor e Forma:SolidPeso molecular:464.49JCP-170
CAS:<p>JCP-170 is an ABHD6 inhibitor.</p>Fórmula:C24H18ClNO4Pureza:98%Cor e Forma:SolidPeso molecular:419.86ML299
CAS:<p>ML299 (VU0463568) is a dual PLD1/2 inhibitor (PLD1 and PLD2, IC50 of 6 nM, 20 nM, respectively).</p>Fórmula:C23H26BrFN4O2Pureza:98%Cor e Forma:SolidPeso molecular:489.38Aminopeptidase-IN-1
CAS:<p>Aminopeptidase-IN-1: potent IRAP blocker, Ki 7.7 μM, useful for cognitive/memory disorder research.</p>Fórmula:C18H16N2O6Pureza:98.37%Cor e Forma:SolidPeso molecular:356.33Enpp-1-IN-17
CAS:<p>Enpp-1-IN-17 (example 274) is a potent inhibitor of ENPP1, exhibiting inhibition constants (Ki values) of 100 nM-1 μM for cGAMP hydrolysis and >1 μM for ATP</p>Fórmula:C18H24N4O2Cor e Forma:SolidPeso molecular:328.41IMB-XMA0038
CAS:<p>IMB-XMA0038 is a Mycobacterium tuberculosis aspartate semialdehyde dehydrogenase inhibitor with antimicrobial activity for use in tuberculosis research.</p>Fórmula:C11H10N4O6Pureza:98.94% - 99.96%Cor e Forma:SolidPeso molecular:294.22THR-0921
CAS:<p>THR-0921 (CLX-0921) is a peroxisome proliferator-activated receptor (PPAR) agonist that can be used to study cardiovascular and metabolic diseases.</p>Fórmula:C28H25NO7SPureza:100% - 99.83%Cor e Forma:SolidPeso molecular:519.57Dopropidil
CAS:<p>Dopropidil: anti-angina calcium regulator with anti-ischemic properties in animal models.</p>Fórmula:C20H35NO2Pureza:98%Cor e Forma:SolidPeso molecular:321.5FCE 28654
CAS:<p>FCE 28654 is a water-soluble acyl-CoA inhibitor.</p>Fórmula:C25H35N2O7PCor e Forma:SolidPeso molecular:506.53Pimobendan hydrochloride
CAS:<p>Pimobendan hydrochloride is a selective inhibitor of PDE3 (IC50: 0.32 μM).</p>Fórmula:C19H19ClN4O2Pureza:98%Cor e Forma:SolidPeso molecular:370.83Piritrexim
CAS:<p>Piritrexim (BW 301U) is an orally available fat-soluble dihydrofolate reductase inhibitor with pulmonary toxicity used in the study of uroepithelial carcinoma</p>Fórmula:C17H19N5O2Pureza:98.50% - >99.99%Cor e Forma:SolidPeso molecular:325.37GSK360A
CAS:<p>GSK360A is a novel prolyl hydroxylase (PHD) domain-containing enzyme inhibitor.</p>Fórmula:C17H17FN2O5Pureza:98%Cor e Forma:SolidPeso molecular:348.33Acetyl-CoA Carboxylase-IN-1
CAS:<p>Acetyl-CoA Carboxylase-IN-1 (ACC-IN-1) is a potent acetyl-CoA carboxylase (ACC) inhibitor with antibacterial activity, used in metabolic disease research.</p>Fórmula:C13H9Br2N5Pureza:98.73%Cor e Forma:SolidPeso molecular:395.05Hoquizil hydrochloride
CAS:<p>Hoquizil hydrochloride is a new bronchodilator with oral activity.</p>Fórmula:C19H27ClN4O5Pureza:98%Cor e Forma:SolidPeso molecular:426.89SCH-351591
CAS:<p>SCH-351591 is an orally active inhibitor of phosphodiesterase 4.</p>Fórmula:C17H10Cl2F3N3O3Pureza:98%Cor e Forma:SolidPeso molecular:432.18PDE7-IN-2
CAS:<p>PDE7-IN-2 is an inhibitor of phosphodiesterase 7 (IC50 = 2.1 µM) and can be used in Parkinson's disease studies.</p>Fórmula:C14H11ClN2O3SPureza:98%Cor e Forma:SolidPeso molecular:322.77IDO inhibitor 1
CAS:<p>IDO inhibitor 1 is an potent inhibitor of indoleamine-2,3 dioxygenase (IDO) ( IC50 <100 nM).with potential immunomodulating and antineoplastic activities.</p>Fórmula:C11H13BrFN7O4SPureza:99.805%Cor e Forma:SolidPeso molecular:438.23Emiglitate
CAS:<p>Emiglitate is a selective and competitive α-glucoside hydrolase inhibitor.</p>Fórmula:C17H25NO7Pureza:98%Cor e Forma:SolidPeso molecular:355.38Carbonic anhydrase inhibitor 14
CAS:<p>CA inhibitor 14 blocks hCA I/II/IX/XII (K i of 1203/99.7/9.4/27.7 nM) and CDK2 (IC50: 20.3 μM), showing antitumor effects.</p>Fórmula:C18H17N7O2SCor e Forma:SolidPeso molecular:395.44hACC2-IN-1
CAS:<p>hACC2-IN-1 is a potent inhibitor of acetyl coenzyme A carboxylase 2 (ACC2) with an IC50 value of 2.5 μM for hACC2. hACC2-IN-1 has potential for obesity studies.</p>Fórmula:C23H32N2O4SCor e Forma:SolidPeso molecular:432.58TDP1 Inhibitor-2
CAS:<p>TDP1 Inhibitor-2 strongly blocks TDP1 (IC50: 99 nM) & treats SCAN1 (IC50: 3.5 μM).</p>Fórmula:C25H14Cl2O5Cor e Forma:SolidPeso molecular:465.28CDP 840 hydrochloride
CAS:<p>CDP-840 (GR259653X), a potent oral PDE IV inhibitor, curbs early and late phase bronchoconstriction in squirrel monkeys.</p>Fórmula:C25H27NO2Cor e Forma:SolidPeso molecular:373.49ZM223
CAS:<p>ZM223 is an inhibitor of NEDD8 activating enzyme (NAE).</p>Fórmula:C23H17F3N4O2S2Pureza:99.73%Cor e Forma:SolidPeso molecular:502.53ML350
CAS:<p>ML350 (CYM-50202) is a potent KOR antagonist (IC50: 12.6 nM), selective over DOR/MOR, with high solubility and CNS penetration, lacking long-term effects.</p>Fórmula:C18H26BrN3O3Pureza:98%Cor e Forma:SolidPeso molecular:412.32L-693612
CAS:<p>L-693612 is an inhibitor of carbonic anhydrase.</p>Fórmula:C14H24N2O5S3Pureza:98%Cor e Forma:SolidPeso molecular:396.55trans-Ned 19
CAS:<p>trans-Ned 19 blocks NAADP and TPC, hindering calcium signaling and aorta relaxation at low histamine levels.</p>Fórmula:C30H31FN4O3Pureza:98%Cor e Forma:SolidPeso molecular:514.59RA 642
CAS:<p>RA 642 is used as a PDE-inhibitor.</p>Fórmula:C24H44N8O4Pureza:98%Cor e Forma:SolidPeso molecular:508.66RO6806051
CAS:<p>RO6806051 (compound 12) is a potent dual inhibitor of fatty acid binding proteins 4 and 5 (FABP4 and FABP5), exhibiting excellent selectivity and absorption, distribution, metabolism, and excretion (eADME) properties.</p>Fórmula:C21H19ClN6Cor e Forma:SolidPeso molecular:390.87NSC-79887
CAS:<p>NSC-79887 is a nucleoside hydrolase (NH) inhibitor.</p>Fórmula:C14H16ClNO4Pureza:98%Cor e Forma:SolidPeso molecular:297.73CL385319 HCl
CAS:<p>"CL385319: Inhibits H5N1 flu virus, blocks entry, low cytotoxicity, IC50=27.03μM in MDCK cells, ineffective on VSV-G pseudotypes."</p>Fórmula:C15H19ClF4N2OPureza:98%Cor e Forma:SolidPeso molecular:354.77hCAXII-IN-4
CAS:<p>hCAXII-IN-4 is a selective and potent CA XII inhibitor with a Ki value of 6.4 nM for human CA XII.</p>Fórmula:C22H27N5O6SCor e Forma:SolidPeso molecular:489.54Glucocerebrosidase-IN-1
CAS:<p>Glucocerebrosidase-IN-1 inhibits GCase with IC50 of 29.3 μM, Ki 18.5 μM, useful for Gaucher's and Parkinson's research.</p>Fórmula:C13H27NO3Cor e Forma:SolidPeso molecular:245.36GA11
CAS:<p>GA11is an inhibitor of ALDH1. It also displays anti-GBM effects in vitro and in vivo.</p>Fórmula:C19H14N2Pureza:98%Cor e Forma:SolidPeso molecular:270.33Chlorambucyl-proline
CAS:<p>Chlorambucyl-proline is a chlorambucil derivative of L-proline. It is an inhibitor of bovine lung angiotensin I-converting enzyme.</p>Fórmula:C19H26Cl2N2O3Pureza:98%Cor e Forma:SolidPeso molecular:401.3311β-HSD1-IN-6
CAS:<p>11β-HSD1-IN-6 is a potent inhibitor of 11β hydroxysteroid dehydrogenase enzymes (11β-HSDs).</p>Fórmula:C21H19ClN4OCor e Forma:SolidPeso molecular:378.8614(S)-HDHA
CAS:<p>DHA is an ω-3 important for development and therapy for inflammation and cancer; its derivative, 14(S)-HDHA, aids in reducing inflammation.</p>Fórmula:C22H32O3Cor e Forma:SolidPeso molecular:344.49Z-321
CAS:<p>Z-321 is an inhibitor of prolyl endopeptidase.</p>Fórmula:C19H24N2O2SPureza:98%Cor e Forma:SolidPeso molecular:344.47FABP4/5-IN-5
CAS:<p>FABP4/5-IN-5 (compound D9) serves as a potent inhibitor of both FABP 4 and FABP 5, demonstrating IC50 values of 4.68 μM and 10.72 μM, respectively. It is notably effective in addressing metabolic disorders such as diabetes mellitus [1].</p>Fórmula:C23H14ClF2NO4SCor e Forma:SolidPeso molecular:473.88Maxacalcitol
CAS:<p>Maxacalcitol (22-Oxacalcitriol) is a ligand of VDR-like receptors and a non-serum calcium vitamin D3 analogue.</p>Fórmula:C26H42O4Pureza:≥98%Cor e Forma:SolidPeso molecular:418.61DU717
CAS:<p>DU717 is an antihypertensive agent.</p>Fórmula:C12H15ClN4O2SPureza:99.64%Cor e Forma:SolidPeso molecular:314.79IACS-8968 R-enantiomer
CAS:<p>IACS-8968 R-enantiomer is the R-enantiomer of IACS-8968. IACS-8968 is a dual IDO and TDO inhibitor (pIC50s: 6.43 for IDO and <5 for TDO).</p>Fórmula:C17H18F3N5O2Pureza:98%Cor e Forma:SolidPeso molecular:381.35CGP-28014
CAS:<p>CGP-28014 inhibits COMT, boosts renal dopamine & DOPAC excretion, lowers HVA, no effect on renal sodium.</p>Fórmula:C12H19N3OCor e Forma:SolidPeso molecular:221.3ACC1/2-IN-2
CAS:<p>PF-3: potent ACC1/2 inhibitor; IC50: 22 nM (ACC1), 48 nM (ACC2); anti-cancer research potential.</p>Fórmula:C24H25N3O3Cor e Forma:SolidPeso molecular:403.47(3S,5S)-Pitavastatin calcium
CAS:<p>(3S,5S)-Pitavastatin calcium is the 3-epimer of Pitavastatin which is a potent HMG-CoA reductase inhibitor.</p>Fórmula:C25H26CaFNO4Pureza:98%Cor e Forma:SolidPeso molecular:463.562Protizinic acid
CAS:<p>Protizinic acid is an oral NSAID with anti-inflammatory and antipyretic properties, inhibiting PLA2 at IC50 of 210μM.</p>Fórmula:C17H17NO3SCor e Forma:SolidPeso molecular:315.39FXR agonist 4
<p>FXR agonist 4: EC50 of 1.05μM, treats hyperlipidemia, steatosis, insulin resistance, inflammation in DIO mice, for NAFLD research.</p>Fórmula:C21H28ClN3OCor e Forma:SolidPeso molecular:373.92Ciraparantag TFA
CAS:<p>Ciraparantag TFA reverses anticoagulants by inhibiting thrombin and factor Xa.</p>Fórmula:C26H50F6N12O6Pureza:98%Cor e Forma:SolidPeso molecular:740.74NP603
CAS:<p>NP603 is a cell-permeable inhibitor of FGFR1, PDGFRβ, and VEGFR2 that binds to the ATP pocket. It also is a very weak EGFR inhibitor.</p>Fórmula:C26H26N2O5Pureza:98%Cor e Forma:SolidPeso molecular:446.49OMDM-3
CAS:<p>OMDM-3 is a selective and metabolically stable anandamide cellular uptake (ACU)inhibitor(Ki of 16.6 μM).</p>Fórmula:C29H43NO3Pureza:98%Cor e Forma:SolidPeso molecular:453.66HIF-1/2α-IN-2
CAS:<p>HIF-1/2α-IN-2 is a potent inhibitor of HIF-1/2α, which effectively reduces the levels of HIF-1/2α.</p>Fórmula:C16H11FN4O2SCor e Forma:SolidPeso molecular:342.35BI-135585
CAS:<p>BI-135585 is an orally active, selective and potent inhibitor of human 11β-hydroxysteroid dehydrogenase-1 (HSD1) for the study of type 2 diabetes.</p>Fórmula:C28H32N2O4Pureza:99.45% - 99.57%Cor e Forma:SolidPeso molecular:460.577β,27-dihydroxy Cholesterol
CAS:<p>7β,27-dihydroxy Cholesterol is an oxysterol and agonist of retinoic acid receptor-related orphan receptor γ (RORγ) and RORγt.</p>Fórmula:C27H46O3Cor e Forma:SolidPeso molecular:418.65ACC1/2-IN-1
CAS:<p>ACC1/2-IN-1 is a potent inhibitor of ACC1/2 and acts on ACC1 (IC50: 98.06 nM) and ACC2 (IC50: 29.43 nM). ACC1/2-IN-1 can be used in cancer research.</p>Fórmula:C34H32N4O4Cor e Forma:SolidPeso molecular:560.64α-Glucosidase-IN-10
CAS:<p>α-Glucosidase-IN-10 (compound 13) is a potent inhibitor of α-glucosidase (IC50: 92.7 μM). α-Glucosidase-IN-10 can be used to study type II diabetes.</p>Fórmula:C21H15BrN4O2SCor e Forma:SolidPeso molecular:467.34TUPS
CAS:<p>TUPS is a selective soluble epoxide hydrolase inhibitor which protects against isoprenaline-induced cardiac hypertrophy.</p>Fórmula:C14H18F3N3O4SCor e Forma:SolidPeso molecular:381.37Rev 6207
CAS:<p>Rev 6207 is a non-sulfhydryl ACE-inhibitor.</p>Fórmula:C21H31N3O5Cor e Forma:SolidPeso molecular:405.49HFI-437
CAS:<p>HFI-437 is a potent, non-peptidic, insulin-regulated aminopeptidase (IRAP) inhibitor with a K i of 20 nM and functions as a cognitive enhancer [1].</p>Fórmula:C23H20N2O5Cor e Forma:SolidPeso molecular:404.42AX 048
CAS:<p>Group IVA cPLA2 inhibitor AX 048 halts arachidonic acid release, preventing prostaglandin production, with XI(50) of 0.022 and ED50 of 1.2 mg/kg.</p>Fórmula:C22H41NO4Cor e Forma:SolidPeso molecular:383.57CAY10485
CAS:<p>CAY10485 blocks human ACAT-1 & ACAT-2 (IC50: 95 & 81 μM) and hinders oxidation of LDL by 91% at 2 μM, possibly impacting atherosclerosis development.</p>Fórmula:C27H27NO7Cor e Forma:SolidPeso molecular:477.51JMS-053
CAS:<p>JMS-053 is a phosphatase DUSP3 inhibitor that inhibits CDC25B and prevents VEGF from disrupting the microvascular endothelial barrier.</p>Fórmula:C13H8N2O2SPureza:≥98.0%Cor e Forma:SolidPeso molecular:256.28SGK1 inhibitor
CAS:<p>SGK1 inhibitor targets SGK1/2 over SGK3, blocks GSK3β phosphorylation, lowers HCC1954 cell viability with BYL719, and reduces tumor growth in mice.</p>Fórmula:C17H12Cl2N6O2SCor e Forma:SolidPeso molecular:435.29CD 1530
CAS:<p>CD 1530 is an ARγ agonist (Kd:150 nM) with potential anticancer activity for the study of oral carcinogenesis.</p>Fórmula:C27H26O3Pureza:98.13%Cor e Forma:SolidPeso molecular:398.49JTP-4819
CAS:<p>JTP-4819: potent PEP inhibitor, may treat Alzheimer's, boosts brain peptides and acetylcholine, aiding memory.</p>Fórmula:C19H25N3O4Cor e Forma:SolidPeso molecular:359.42AMG-221
CAS:<p>AMG-221: potent 11β-HSD1 inhibitor, lowers glucose & insulin, reduces obesity in mice.</p>Fórmula:C14H22N2OSPureza:98%Cor e Forma:SolidPeso molecular:266.4Boc-Glu(OBzl)-OSu
CAS:<p>Boc-Glu(OBzl)-OSu can be used for the synthesis of solid phase peptides containing benzyl glutamate residues.</p>Fórmula:C21H26N2O8Cor e Forma:SolidPeso molecular:434.44α-Amylase/α-Glucosidase-IN-2
CAS:<p>α-Amylase/α-Glucosidase-IN-2 (compound 5) exhibits strong inhibition activity towards both α-amylase and α-glucosidase enzymes, with IC 50 values of 13.02 μM</p>Fórmula:C22H16ClN5Cor e Forma:SolidPeso molecular:385.85L 645151
CAS:<p>L 645151 is an inhibitor of lipophilic CA.</p>Fórmula:C12H14N2O4S2Cor e Forma:SolidPeso molecular:314.38ENPP1 inhibitor 43
CAS:<p>ENPP1 inhibitor 43 is a novel small molecule for cancer immunotherapy.</p>Fórmula:C16H18N6O3SCor e Forma:SolidPeso molecular:374.42MY33-3 hydrochloride
CAS:<p>MY33-3 HCl: Inhibits RPTPβ/ζ (IC50~0.1μM), PTP-1B (IC50~0.7μM), curbs alcohol intake, fights neuroinflammation and memory issues.</p>Fórmula:C16H14ClF6NS2Cor e Forma:SolidPeso molecular:433.86MAGLi 432
CAS:<p>MAGLi 432: Potent MAGL inhibitor, selective and reversible. IC50: 4.2 nM (human), 3.1 nM (mouse). Useful for neurological disorder research.</p>Fórmula:C22H24BrClN2O2Cor e Forma:SolidPeso molecular:463.8SQ-24,798
CAS:<p>SQ-24,798 is an inhibitor of the thrombin-activatable fibrinolysis and carboxypeptidase N (CPN).</p>Fórmula:C7H15N3O2SPureza:98%Cor e Forma:SolidPeso molecular:205.2824(S),25-Epoxycholesterol
CAS:<p>24(S),25-Epoxycholesterol is an oxysterol agonist of the liver X receptor.</p>Fórmula:C27H44O2Cor e Forma:SolidPeso molecular:400.64IDO1-IN-15
CAS:<p>IDO1-IN-15 is an effective IDO1 inhibitor with IC50 of 127 nM. The potency of IDO1-IN-15 against IDO1 enzyme is comparable with Epacadostat in vitro.</p>Fórmula:C13H14BrFN6O3Cor e Forma:SolidPeso molecular:401.19UCM 765
CAS:<p>UCM 765 is a partial agonist of melatonin MT(2) receptor.</p>Fórmula:C17H20N2O2Pureza:98%Cor e Forma:SolidPeso molecular:284.35Diapocynin
CAS:<p>Diapocynin (Dehydrodiacetovanillone), a dimer of Apocynin, acts as an orally administered inhibitor of NADPH oxidase.</p>Fórmula:C18H18O6Cor e Forma:SolidPeso molecular:330.333,3-Dimethyl-1-butanol
CAS:<p>3,3-Dimethyl-1-butanol (DMB) inhibits TMA/TMAO and affects p65 NF-κB, TGF-β1/Smad3 signaling; potential for CVD treatment.</p>Fórmula:C6H14OCor e Forma:SolidPeso molecular:102.17α-Glucosidase-IN-21
CAS:<p>α-Glucosidase-IN-21 (Compound 2B) is a highly potent and orally bioavailable inhibitor of α-glucosidase.</p>Fórmula:C24H23NO2SCor e Forma:SolidPeso molecular:389.51Fmoc-5-aminopentanoic acid
CAS:<p>Fmoc-5-aminopentanoic acid: alkane, Fmoc-protected amine, carboxyl group, PROTAC linker, deprotects to free amine, forms amides with activators.</p>Fórmula:C20H21NO4Cor e Forma:SolidPeso molecular:339.39mEH-IN-1
CAS:<p>mEH-IN-1 (Compound 62) is a potent mEH enzyme inhibitor with an IC50 of 2.2 nM, relevant in preeclampsia, hypercholanemia, and cancer research.</p>Fórmula:C16H17F6NOSCor e Forma:SolidPeso molecular:385.37SYN20028567
CAS:<p>SYN20028567, an aromatase (CYP19) inhibitor, exhibits an IC50 value of 9.4 nM. It has potential applications in breast cancer research [1].</p>Fórmula:C20H29N3O3SCor e Forma:SolidPeso molecular:391.53Umbralisib tosylate
CAS:<p>Umbralisib tosylate, an oral PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), shows promise for CLL research.</p>Fórmula:C38H32F3N5O6SCor e Forma:SolidPeso molecular:743.75JNJ-61803534
CAS:<p>JNJ-61803534: RORγt inverse agonist, IC50=9.6 nM, oral, anti-inflammatory, reduces IL-17A in T cells.</p>Fórmula:C23H23Cl2F6N3O4SCor e Forma:SolidPeso molecular:622.41JTP 103237
CAS:<p>JTP 103237 is a potent and selective monoacyglycerol acyltransferase 2 (MOGAT2) inhibitor.</p>Fórmula:C24H29F3N6OCor e Forma:SolidPeso molecular:474.52(R)-DNMDP
CAS:<p>(R)-DNMDP is a potent and selective cancer cytotoxic agent that directly binds PDE3A and has an EC50 500-fold lower than that of (S)-DNMDP against HeLa.</p>Fórmula:C15H20N4O3Cor e Forma:SolidPeso molecular:304.34GKA-71
CAS:<p>GKA-71 is an effective glucokinase activator (GKA).</p>Fórmula:C21H23N3O6S2Cor e Forma:SolidPeso molecular:477.55Metyltetraprole
CAS:<p>Metyltetraprole: potent fungicide, effective against Zymoseptoria, low EC50 (0.002 ppm), inhibits respiratory chain.</p>Fórmula:C19H17ClN6O2Cor e Forma:SolidPeso molecular:396.83α-Glucosidase-IN-9
CAS:<p>α-Glucosidase-IN-9 (compound 7) is a highly potent α-glucosidase inhibitor with an IC50 of 55.6 μM, making it suitable for type II diabetes research [1].</p>Fórmula:C19H12N4OSCor e Forma:SolidPeso molecular:344.39RYL-552
CAS:<p>RYL-552 is a potent inhibitor of PfNDH2.</p>Fórmula:C24H17F4NO2Pureza:98%Cor e Forma:SolidPeso molecular:427.39DHODH-IN-21
CAS:<p>DHODH-IN-21, orally active DHODH blocker with 1.1 nM IC50, shows anticancer activity, potential for AML research.</p>Fórmula:C20H19ClF4N6O4Cor e Forma:SolidPeso molecular:518.85α-Glucosidase-IN-20
CAS:<p>α-Glucosidase-IN-20 (Compound 3B) is a highly effective and orally active inhibitor of α-glucosidase.</p>Fórmula:C23H21NOSCor e Forma:SolidPeso molecular:359.48(Rac)-3′-Hydroxy simvastatin
CAS:<p>(Rac)-3′-Hydroxy Simvastatin, a metabolite of Simvastatin, acts as a competitive inhibitor of HMG-CoA reductase, demonstrating a K i value of 0.2 nM.</p>Fórmula:C25H38O6Cor e Forma:SolidPeso molecular:434.57Prenyl-IN-1
CAS:<p>Prenyl-IN-1 inhibits prenylation selectively, counters oxidative stress in Parkinson's.</p>Fórmula:C28H24ClN5O2Pureza:>99.99%Cor e Forma:SolidPeso molecular:497.98Peliglitazar racemate
CAS:<p>Peliglitazar racemate(BMS 426707-01 racemate) is the racemate of Peliglitazar.Peliglitazar racemate may be used as a potential antidiabetic and anti-obesity</p>Fórmula:C30H30N2O7Pureza:97.75%Cor e Forma:SolidPeso molecular:530.57PKM2 activator 5
CAS:<p>PKM2 activator 5 is a novel and potent PKM2 activator (AC50: 0.316 µM) with potential anticancer activity for the study of cancer metabolism-related diseases.</p>Fórmula:C18H19FN2O6S2Pureza:98%Cor e Forma:SolidPeso molecular:442.48HX-600
CAS:<p>HX-600 is a synthetic agonist for the RXR-Nurr1 heterodimer complex. HX-600 prevents ischemia-induced neuronal damage.</p>Fórmula:C29H30N2O2Cor e Forma:SolidPeso molecular:438.56TA-7552
CAS:<p>TA-7552 is a potent agent of cholesterol-lowering.</p>Fórmula:C25H26O10Pureza:98%Cor e Forma:SolidPeso molecular:486.47Teludipine hydrochloride
CAS:<p>Teludipine hydrochloride is a blocker of lipophilic calcium channel.</p>Fórmula:C28H39ClN2O6Pureza:98%Cor e Forma:SolidPeso molecular:535.07SCD1-IN-1
CAS:<p>SCD1-IN-1, a potent inhibitor of SCD1 (IC50: 5.8 nM), is valuable in dermatologic research [1].</p>Fórmula:C20H20F3NO4Cor e Forma:SolidPeso molecular:395.37Xanthine oxidoreductase-IN-1
CAS:<p>Xanthine oxidoreductase-IN-1 is a xanthine oxidoreductase (XOR) inhibitor with an IC 50 value of 7.0 nM.</p>Fórmula:C18H20N4O2Cor e Forma:SolidPeso molecular:324.38Diaplasinin
CAS:<p>Diaplasinin (PAI-749) is a potent inhibitor of plasminogen activator inhibitor-1 (PAI-1) with antithrombotic activity, used in cardiovascular disease research.</p>Fórmula:C32H31N5OPureza:99.02%Cor e Forma:SolidPeso molecular:501.62BFE-37
CAS:<p>BFE-37 is a partial agonist of beta-adrenergic.</p>Fórmula:C16H23NO3Pureza:98%Cor e Forma:SolidPeso molecular:277.36Cholesteryl behenate
CAS:<p>Cholesteryl behenate is a standard in electrospray ionization tandem mass spectrometry for the analysis of cholesteryl esters and cholesterol.</p>Fórmula:C49H88O2Pureza:98%Cor e Forma:SolidPeso molecular:709.22CYP3A4-IN-3
CAS:<p>CYP3A4-IN-3, a ritonavir analogue, is a potent CYP3A4 inhibitor with an IC50 of 0.075 μM, used as an antiviral and immunosuppressant.</p>Fórmula:C34H39N3O3SCor e Forma:SolidPeso molecular:569.76ASP3662
CAS:<p>ASP3662/SPI-62: Potent, selective CNS-penetrable 11β-HSD1 inhibitor; potential neuropathic pain treatment.</p>Fórmula:C19H16ClF3N4O2Cor e Forma:SolidPeso molecular:424.8Trandolaprilate hydrate
CAS:<p>Trandolaprilate hydrate, a powerful ACE inhibitor and Trandolapril's main metabolite, is lipophilic with partial c-fos blocking.</p>Fórmula:C22H32N2O6Cor e Forma:SolidPeso molecular:420.5PMPMEase-IN L-28
CAS:<p>PMPMEase-IN L-28 is a novel inhibitor of prenylated methylated protein methylesterase.</p>Fórmula:C17H29FO2S2Pureza:98%Cor e Forma:SolidPeso molecular:348.54YCT529 free acid
CAS:<p>YCT529 free acid is a potent, selective and orally active RAR-α inhibitor .</p>Fórmula:C29H25NO3Cor e Forma:SolidPeso molecular:435.51hCAIX/XII-IN-6
<p>hCAIX/XII-IN-6: Oral carbonic anhydrase inhibitor, targets hCA I/II/IV/IX/XII, aids rheumatoid arthritis research. Ki: 6697/2950/4093/4.1/7.7 nM.</p>Fórmula:C26H23N3O6S4Cor e Forma:SolidPeso molecular:601.74Ethylene thiourea
CAS:<p>Ethylene thiourea (NCIC03372) is a pesticide used in fruit and vegetable production.</p>Fórmula:C3H6N2SPureza:≥98%Cor e Forma:Needles Prisms From Alcohol Or Amyl AlcoholPeso molecular:102.16Pteropterin
CAS:<p>Pteropterin is an antineoplastic agent.</p>Fórmula:C29H33N9O12Pureza:98%Cor e Forma:SolidPeso molecular:699.63Sp-cAMPS
CAS:<p>Rp-cAMPS TEA salt is a cAMP-dependent protein kinase (PKA) activator.</p>Fórmula:C10H12N5O5PSCor e Forma:SolidPeso molecular:345.27Alitame
CAS:<p>Alitame is a high-intensity sweetener and sugar substitute widely used in biochemical experiments and drug synthesis research.</p>Fórmula:C14H25N3O4SPureza:98%Cor e Forma:SolidPeso molecular:331.43DCYM21
CAS:<p>DCYM21: Menin-MLL inhibitor, halts leukemia cell growth with MLL changes, causing arrest and differentiation.</p>Fórmula:C26H33ClN2Pureza:98%Cor e Forma:SolidPeso molecular:409.01hCAIX-IN-10
CAS:<p>"hCAIX-IN-10 (6i) selectively inhibits carbonic anhydrase IX/XII (Ki: 61.5/586.8 nM), markers in tumor cells, affecting acid-base balance."</p>Fórmula:C28H21N3O3SCor e Forma:SolidPeso molecular:479.55SHP844
CAS:<p>SHP844: SHP2 inhibitor, IC50 18.9 µM, affects cell growth/survival by regulating tyrosine phosphorylation.</p>Fórmula:C29H24ClN5O6Cor e Forma:SolidPeso molecular:573.98RORγt inverse agonist 28
CAS:<p>RORγt inverse agonist 28 is a potent RORγt inverse agonist.</p>Fórmula:C23H18Cl2F3NO5SCor e Forma:SolidPeso molecular:548.3611β-HSD1-IN-10
CAS:<p>11β-HSD1-IN-10, a potent inhibitor of 11β-HSD1 with an IC50 value of 1.8 µM for humans, is suitable for research into obesity, hyperglycemia, and cognitive</p>Fórmula:C16H10F3NO2Cor e Forma:SolidPeso molecular:305.25TC-E 5005
CAS:<p>PDE10A inhibitor</p>Fórmula:C15H18N4OPureza:98%Cor e Forma:SolidPeso molecular:270.33Sermetacin
CAS:<p>Sermetacin is an anti-inflammatory agent.</p>Fórmula:C22H21ClN2O6Pureza:98%Cor e Forma:SolidPeso molecular:444.86PF 04671536 hydrochloride
CAS:<p>Potent PDE8B/8A inhibitor; IC50: PDE8B-1.3nM, PDE8A-1.9nM; selective over other PDEs; enhances insulin secretion; orally bioavailable.</p>Fórmula:C14H19ClN8OSCor e Forma:SolidPeso molecular:382.87TAK 21d
CAS:<p>Potent FAAH inhibitor</p>Fórmula:C19H17F2N7OPureza:98%Cor e Forma:SolidPeso molecular:397.38SR1555 HCl
CAS:<p>SR1555: A selective RORγ inverse agonist, hinders TH17 cells, key in autoimmune diseases like RA and MS.</p>Fórmula:C22H22F6N2O2Pureza:98%Cor e Forma:SolidPeso molecular:460.41LY367385
CAS:<p>LY367385 is a highly effective and selective mGluR1a antagonist.</p>Fórmula:C10H11NO4Pureza:98%Cor e Forma:SolidPeso molecular:209.2α-Glucosidase-IN-6
CAS:<p>α-Glucosidase-IN-6 is a competitive inhibitor of α-glucosidase (IC50: 5.69 μM) and exhibits potential for anti-diabetic studies.</p>Fórmula:C24H17ClF3NO3SCor e Forma:SolidPeso molecular:491.91hCAI/II-IN-1
CAS:<p>hCAI/II-IN-1 (Compound 3h) is a human carbonic anhydrase I and II (hCA I/II) inhibitor that acts on hCA I (IC50: 0.047 μM) and hCA II (IC50: 0.024 μM).</p>Fórmula:C18H29N5O3S3Cor e Forma:SolidPeso molecular:459.65LCL521
CAS:<p>LCL521 inhibits lysosomal acid sphingomyelinase (ASMase).LCL521 is an acid ceramidase (ACDase) inhibitor.</p>Fórmula:C31H52N4O7Pureza:98%Cor e Forma:SolidPeso molecular:592.77Enpp-1-IN-6
CAS:<p>Enpp-1-IN-6, a potent enpp-1 inhibitor, may aid cancer and infectious disease studies (WO2021203772A1, compound 51).</p>Fórmula:C22H28N4O5SCor e Forma:SolidPeso molecular:460.55Oxycinchophen
CAS:<p>Oxycinchophen: Quinoline-based anti-rheumatic with P-selectin inhibition, DHOD blockade, and anti-inflammatory impacts on vascular muscle.</p>Fórmula:C16H11NO3Pureza:98%Cor e Forma:SolidPeso molecular:265.26GW648495
CAS:<p>GW648495 is a PfDHODH inhibitor that shows greater than 4,000-fold selectivity for the malarial enzyme.</p>Fórmula:C16H13N5Pureza:98%Cor e Forma:SolidPeso molecular:275.31ts-SA
CAS:<p>ts-SA is a metalloenzyme carbonic anhydrase (CA) inhibitor. It is active against 7 out of 10 human CA isoforms.</p>Fórmula:C14H15N3O5S2Pureza:98%Cor e Forma:SolidPeso molecular:369.42(-)-Ketoconazole
CAS:<p>(-)-Ketoconazole is a potential mitochondrial CYP24A1 inhibitor and has antifungal activity against Aspergillus fumigatus.</p>Fórmula:C26H28Cl2N4O4Pureza:98%Cor e Forma:SolidPeso molecular:531.43CDK2-IN-11
CAS:<p>CDK2-IN-11 inhibits CDK2 (IC50: 6.4 μM) and targets hCA II, IX, XII (Ki: 23.4-56.3 nM); suited for cancer research.</p>Fórmula:C18H14ClN7O2SCor e Forma:SolidPeso molecular:427.87Sterculic acid
CAS:<p>Sterculic acid inhibits SCD1 with IC50 of 0.9μM, affecting Δ9D desaturase activity.</p>Fórmula:C19H34O2Cor e Forma:SolidPeso molecular:294.47Fexaramate
CAS:<p>Fexaramate is a potent, selective agonist of farnesoid X receptor.</p>Fórmula:C31H37NO5Cor e Forma:SolidPeso molecular:503.63(Rac)-Etavopivat
CAS:<p>(Rac)-Etavopivat, an oral PKR activator, targets sickle cell disease and haemoglobinopathies.</p>Fórmula:C22H23N3O6SCor e Forma:SolidPeso molecular:457.5ARL-67156 trisodium salt hydrate
CAS:<p>ARL-67156 trisodium salt hydrate is an ecto-ATPase inhibitor that prevents metabolism of P2 purinoceptor agonists.</p>Fórmula:C15H24Br2N5O12P3Cor e Forma:SolidPeso molecular:719.11Seviteronel R enantiomer
CAS:<p>Seviteronel R enantiomer (VT-464 R enantiomer) is a Seviteronel isomer produced during the manufacturing process.</p>Fórmula:C18H17F4N3O3Pureza:97.97% - >99.99%Cor e Forma:SolidPeso molecular:399.34BVT-116429
CAS:<p>BVT-116429 is an inhibitor of 11β-HSD1.</p>Fórmula:C13H12F4N2OSPureza:98%Cor e Forma:SolidPeso molecular:320.31ZSET-845
CAS:<p>ZSET-845 is an enhancer of cognitive which enhances choline acetyltransferase activity in the hippocampus in the rat.</p>Fórmula:C21H18N2OPureza:98%Cor e Forma:SolidPeso molecular:314.38Langkamide
CAS:<p>Langkamide is a HIF-2 inhibitor with EC₅₀ values of 14.0 uM.</p>Fórmula:C16H17NO5Pureza:98%Cor e Forma:SolidPeso molecular:303.31HCAIX-IN-2
CAS:<p>HCAIX-IN-2 (compound 9d) is a selective inhibitor of carbonic anhydrase and acts on hCA IX (Ki: 24.6 nM) and hCA XII (Ki: 45.3 nM).</p>Fórmula:C19H16N8O4SCor e Forma:SolidPeso molecular:452.45(R)-Nepicastat HCl
CAS:<p>(R)-Nepicastat HCl (RS-25560-198 HCl), R-enantiomer, inhibits bovine/human dopamine-β-hydroxylase (IC50: 25.1/18.3 nM); not affecting other enzymes/receptors.</p>Fórmula:C14H15F2N3S·HClPureza:98%Cor e Forma:SolidPeso molecular:331.81Enazadrem
CAS:<p>Enazadrem is a 5-lipoxygenase inhibitor with antiinflammatory activities.</p>Fórmula:C18H25N3OPureza:98%Cor e Forma:SolidPeso molecular:299.41Aldophosphamide
CAS:<p>Aldophosphamide possesses apoptotic antitumor activity.</p>Fórmula:C7H15Cl2N2O3PPureza:98%Cor e Forma:SolidPeso molecular:277.09Acarbose sulfate
CAS:<p>Acarbose sulfate is an anti-diabetic drug and is an inhibitor of alpha-glucosidase.</p>Fórmula:C25H45NO22SPureza:98%Cor e Forma:SolidPeso molecular:743.68
