Metabolismo
Os inibidores do metabolismo são compostos que interferem nas vias metabólicas, alterando a produção e utilização de energia dentro das células. Esses inibidores são usados para estudar a regulação do metabolismo, o papel das vias metabólicas em doenças como o câncer e o diabetes, e para desenvolver novas estratégias terapêuticas. Os inibidores do metabolismo podem direcionar várias enzimas e processos envolvidos na glicólise, na oxidação de ácidos graxos e em outras funções metabólicas. Na CymitQuimica, oferecemos uma ampla gama de inibidores do metabolismo de alta qualidade para apoiar sua pesquisa em bioquímica, distúrbios metabólicos e desenvolvimento de medicamentos.
Subcategorias de "Metabolismo"
- AhR(41 produtos)
- Aminopeptidase(67 produtos)
- CETP(18 produtos)
- Anidrase carbónica(177 produtos)
- Caseína quinase(130 produtos)
- DHFR(32 produtos)
- Descarboxilase(4 produtos)
- Desidrogenase(267 produtos)
- FAAH(63 produtos)
- FXR(58 produtos)
- Factor Xa(80 produtos)
- Sintase de Ácidos graxos(32 produtos)
- Ferroptose(215 produtos)
- GR(3 produtos)
- GSNOR(3 produtos)
- Glucoquinase(53 produtos)
- HIF/HIF Prolil-Hidroxilase(142 produtos)
- HMG-CoA Reductase(32 produtos)
- Hidroxilase(30 produtos)
- IDO(82 produtos)
- LDL(8 produtos)
- Lipase(96 produtos)
- Lipídio(59 produtos)
- Lipoxigenase(124 produtos)
- MAO(87 produtos)
- MPO(2 produtos)
- NAMPT(36 produtos)
- P450(6 produtos)
- PAI-1(25 produtos)
- PDE(166 produtos)
- PED(1 produtos)
- PKM(15 produtos)
- PPAR(164 produtos)
- Fosfolipase(82 produtos)
- ROR(42 produtos)
- Receptor de Retinóide(29 produtos)
- SGK(11 produtos)
- Tiorredoxina(12 produtos)
- Transferase(30 produtos)
- Tansportador(42 produtos)
- UGT(4 produtos)
- Inibidores de Xantina Oxidase (XO)(9 produtos)
Exibir 34 mais subcategorias
Foram encontrados 8595 produtos de "Metabolismo"
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NF-1819
CAS:<p>NF-1819: strong, selective MGL inhibitor; eases MS symptoms; analgesic; penetrates brain with high permeability.</p>Fórmula:C24H22FN5O4Pureza:99.55%Cor e Forma:SolidPeso molecular:463.46AZD8329
CAS:<p>AZD8329 is an 11β-HSD1 inhibitor that inhibits 11β-HSD2, 17β-HSD1, 17β-HSD3, and can be used to study allergic reactions in humans.</p>Fórmula:C25H31N3O3Pureza:99.31%Cor e Forma:SolidPeso molecular:421.53Albaconazole
CAS:<p>Albaconazole, a small fungal CYP51A1 inhibitor, treats fungal infections and some musculoskeletal disorders.</p>Fórmula:C20H16ClF2N5O2Pureza:99.27%Cor e Forma:SolidPeso molecular:431.82LCL521 dihydrochloride
CAS:<p>LCL521 dihydrochloride is a dual inhibitor of ACDase and ASMase, modulating sphingolipid metabolism with potential in cancer and metabolic research.</p>Fórmula:C31H54Cl2N4O7Pureza:98%Cor e Forma:SolidPeso molecular:665.69DHODH-IN-17
CAS:<p>DHODH-IN-17 is a human DHODH inhibitor with an IC50 of 0.40 μM.</p>Fórmula:C12H9ClN2O2Pureza:99.41% - 99.52%Cor e Forma:SolidPeso molecular:248.672-Hydroxy atorvastatin calcium salt
CAS:<p>2-Hydroxy atorvastatin calcium salt is a hydroxy metabolite of Atorvastatin calcium salt which is a potent HMG-CoA reductase inhibitor (IC50 = 8 nM).</p>Fórmula:C33H34FN2O60·5CaPureza:97.06%Cor e Forma:SolidPeso molecular:593.68LGE-899
CAS:<p>LGE-899 (Sonidegib metabolite M48) is a main metabolite of Sonidegib which is an inhibitor of the hedgehog pathway.</p>Fórmula:C15H11F3O3Pureza:99.93%Cor e Forma:SolidPeso molecular:296.24Ocaphane Hydrochloride
CAS:<p>Ocaphane Hydrochloride is a strong antitumor agent used on a number of animal tumors.</p>Fórmula:C14H22Cl4N2O2Pureza:98%Cor e Forma:SolidPeso molecular:392.14Roflurane
CAS:<p>Roflurane is a halocarbon drug. It has been investigated as an inhalational anesthetic.</p>Fórmula:C3H4BrF3OPureza:98%Cor e Forma:SolidPeso molecular:192.96Hexazinone
CAS:<p>Hexazinone: a triazine herbicide blocks photosynthesis by binding to D-1 protein in photosystem II.</p>Fórmula:C12H20N4O2Pureza:99.99%Cor e Forma:SolidPeso molecular:252.31PDE10-IN-5
CAS:<p>PDE10-IN-5 is a phosphodiesterase 10 (PDE 10) inhibitor that can be used to study certain central nervous system disorders.</p>Fórmula:C26H19F3N4OCor e Forma:SolidPeso molecular:460.45JCP-170
CAS:<p>JCP-170 is an ABHD6 inhibitor.</p>Fórmula:C24H18ClNO4Pureza:98%Cor e Forma:SolidPeso molecular:419.86TM-1
CAS:<p>TM-1: PDHK inhibitor, IC50 - PDHK1: 2.97μM, PDHK2: 5.2μM, prevents PDHC phosphorylation, inhibits cancer cell growth.</p>Fórmula:C26H32N2O6Cor e Forma:SolidPeso molecular:468.54Adenosine 5'-phosphosulfate (sodium salt)
CAS:<p>Adenosine 5'-phosphosulfate (sodium salt) (APS) is a key intermediate in sulphur metabolism and a substrate for adenosine 5'-phosphosulfate kinase (APSK).</p>Fórmula:C10H12N5Na2O10PSCor e Forma:SolidPeso molecular:471.24PDE2/PDE10-IN-1
CAS:<p>PDE2/PDE10-IN-1 is a inhibitor of phosphodiesterase 2 (PDE2) and PDE10(IC50s of 29 and 480 nM, respectively).</p>Fórmula:C15H10ClN5Pureza:98%Cor e Forma:SolidPeso molecular:295.73Quazodine
CAS:<p>Quazodine is a phosphodiesterase inhibitor.</p>Fórmula:C12H14N2O2Cor e Forma:SolidPeso molecular:218.25CAY10762
CAS:<p>CAY10762, a MAGL inhibitor (IC50=34.1 nM), curbs H2O2-induced LDH in Neuro2a cells and boosts 2-AG in mouse brains at 10 mg/kg.</p>Fórmula:C15H13NOSCor e Forma:SolidPeso molecular:255.33hCAII-IN-1
CAS:<p>hCAII-IN-1 (7f) inhibits CA II/IX with Kis 1.2 nM/113.6 nM, potential for cancer treatment.</p>Fórmula:C21H21BrN6O4SCor e Forma:SolidPeso molecular:533.4Kurasoin B
CAS:<p>Kurasoin B is an inhibitor of protein farnesyltransferase.</p>Fórmula:C18H17NO2Cor e Forma:SolidPeso molecular:279.33CAY10486
CAS:<p>CAY10486 blocks ACAT-1/2, which form cholesterol esters, potentially reducing atherosclerosis; inhibits LDL oxidation. IC50 ~60μM; 28% effect at 3μM.</p>Fórmula:C19H19NO4Cor e Forma:SolidPeso molecular:325.36Valibose
CAS:<p>Valibose, α-glucosidase inhibitor, improves glucose/lipid metabolism, lowers serum BUN/NAG, reduces kidney weight index.</p>Fórmula:C10H21NO6Cor e Forma:SolidPeso molecular:251.28(R)-Irsenontrine
CAS:<p>(R)-Irsenontrine (R-E2027), R-enantiomer, is a potent PDE9 inhibitor, IC50 = 0.041 μM, for neurological disease research.</p>Fórmula:C22H22N4O3Cor e Forma:SolidPeso molecular:390.44hCAI/II-IN-3
CAS:<p>"hCAI/II-IN-3 (compound 5b) is a potent dual hCA I/II inhibitor with Ki: 51.25nM (I), 13.15nM (II), helps treat AMS."</p>Fórmula:C16H18N4O4S2Cor e Forma:SolidPeso molecular:394.47hCAXII-IN-2
CAS:<p>hCAXII-IN-2 is a potent inhibitor of hCA XII (Ki: 84.2 nM) and hCA IX (Ki: 268.5 nM), with low activity on hCA I/II.</p>Fórmula:C21H18ClN3O4Cor e Forma:SolidPeso molecular:411.84Teglicar
CAS:<p>Teglicar is a selective and reversible liver isoform of carnitine palmitoyl-transferase 1 (L-CPT1) inhibitor.</p>Fórmula:C22H45N3O3Pureza:98%Cor e Forma:SolidPeso molecular:399.61M77976
CAS:<p>M77976 inhibits PDK4 with an IC50 of 648 μM, targeting obesity and diabetes research.</p>Fórmula:C17H16N2O3Pureza:99.43%Cor e Forma:SolidPeso molecular:296.32α-Glucosidase-IN-16
CAS:<p>α-Glucosidase-IN-16 is a highly effective and orally bioavailable inhibitor of α-glucosidase, displaying a remarkable IC50 value of 3.28 μM.</p>Fórmula:C22H18FNSCor e Forma:SolidPeso molecular:347.45ALDH3A1-IN-2
CAS:<p>ALDH3A1-IN-2 is a potent inhibitor targeting ALDH3A1 (IC50=1.29µM), potentially useful in cancer research.</p>Fórmula:C11H14N2O3Cor e Forma:SolidPeso molecular:222.24GNF7686
CAS:<p>GNF7686 is a novel Trypanosoma cruzi inhibitor.</p>Fórmula:C15H13N3OPureza:98%Cor e Forma:SolidPeso molecular:251.28SAR127303
CAS:<p>SAR127303 is an effective covalent inhibitor of MAGL. SAR127303 behaves as a selective and competitive inhibitor of mouse and human MAGL.</p>Fórmula:C16H17ClF6N2O4SPureza:98%Cor e Forma:SolidPeso molecular:482.83Sp-cAMPS
CAS:<p>Rp-cAMPS TEA salt is a cAMP-dependent protein kinase (PKA) activator.</p>Fórmula:C10H12N5O5PSCor e Forma:SolidPeso molecular:345.27Pparδ agonist 2
CAS:<p>Pparδ agonist 2 is an agonist of PPARδ.</p>Fórmula:C20H18F3N3O3SPureza:98%Cor e Forma:SolidPeso molecular:437.44hCAIX-IN-10
CAS:<p>"hCAIX-IN-10 (6i) selectively inhibits carbonic anhydrase IX/XII (Ki: 61.5/586.8 nM), markers in tumor cells, affecting acid-base balance."</p>Fórmula:C28H21N3O3SCor e Forma:SolidPeso molecular:479.55Emiglitate
CAS:<p>Emiglitate is a selective and competitive α-glucoside hydrolase inhibitor.</p>Fórmula:C17H25NO7Pureza:98%Cor e Forma:SolidPeso molecular:355.38BNS
CAS:<p>BNS is a potent, prolyl-hydroxylase 2 (PHD2)-selective inhibitor.</p>Fórmula:C18H16N2O6S2Pureza:98%Cor e Forma:SolidPeso molecular:420.46SHP844
CAS:<p>SHP844: SHP2 inhibitor, IC50 18.9 µM, affects cell growth/survival by regulating tyrosine phosphorylation.</p>Fórmula:C29H24ClN5O6Cor e Forma:SolidPeso molecular:573.98RORγt inverse agonist 28
CAS:<p>RORγt inverse agonist 28 is a potent RORγt inverse agonist.</p>Fórmula:C23H18Cl2F3NO5SCor e Forma:SolidPeso molecular:548.3611β-HSD1-IN-10
CAS:<p>11β-HSD1-IN-10, a potent inhibitor of 11β-HSD1 with an IC50 value of 1.8 µM for humans, is suitable for research into obesity, hyperglycemia, and cognitive</p>Fórmula:C16H10F3NO2Cor e Forma:SolidPeso molecular:305.25VEC6
CAS:<p>VEC6 is a VEZF1–DNA interaction inhibitor that recapitulates RhoB loss in ischaemic retinopathy.</p>Fórmula:C14H20N4Pureza:98%Cor e Forma:SolidPeso molecular:244.34NSC117079
CAS:<p>NSC117079 is a novel PHLPP1/2 (Pleckstrin homology domain and leucine rich repeat protein phosphatase) inhibitor that activates neuronal AKT .</p>Fórmula:C20H15N3O7S2Pureza:98.11%Cor e Forma:SolidPeso molecular:473.48ML202
CAS:<p>ML202 activates human pyruvate kinase M2, affecting PEP cooperativity with minimal impact on ADP binding.</p>Fórmula:C18H17N3O3S2Cor e Forma:SolidPeso molecular:387.48GNE-3500
CAS:<p>GNE-3500: potent, selective RORc inverse agonist; orally bioavailable; promising for treating inflammatory diseases.</p>Fórmula:C24H30FN3O3SCor e Forma:SolidPeso molecular:459.58BCM-599
CAS:<p>BCM-599 is a HBV capsid assembly inhibitor. BCM-599 showed IC50 of 0.88 μM and CC50 of 144 μM in HepG2.2.15 cells.</p>Fórmula:C14H10Cl2FN3O2Cor e Forma:SolidPeso molecular:342.15Hoquizil hydrochloride
CAS:<p>Hoquizil hydrochloride is a new bronchodilator with oral activity.</p>Fórmula:C19H27ClN4O5Pureza:98%Cor e Forma:SolidPeso molecular:426.89YM-75466
CAS:<p>YM-75466 is a factor Xa inhibitor reducing TAT in plasma dose-dependently without prolonging coagulation.</p>Fórmula:C28H35N5O8S2Cor e Forma:SolidPeso molecular:633.74IDO-IN-12
CAS:<p>IDO-IN-12 is an inhibitor of indoleamine 2,3-dioxygenase (IDO).</p>Fórmula:C13H11BrFN5O3SPureza:99.727%Cor e Forma:SolidPeso molecular:416.23Afegostat
CAS:<p>Afegostat is a pharmacological chaperone that specifically and reversibly binds acid-β-glucosidase (GCase) in the endoplasmic reticulum with high affinity.</p>Fórmula:C6H13NO3Pureza:98%Cor e Forma:Yellow Low-Melting SolidPeso molecular:147.17PF 04671536 hydrochloride
CAS:<p>Potent PDE8B/8A inhibitor; IC50: PDE8B-1.3nM, PDE8A-1.9nM; selective over other PDEs; enhances insulin secretion; orally bioavailable.</p>Fórmula:C14H19ClN8OSCor e Forma:SolidPeso molecular:382.87TAK 21d
CAS:<p>Potent FAAH inhibitor</p>Fórmula:C19H17F2N7OPureza:98%Cor e Forma:SolidPeso molecular:397.38DSHN
CAS:<p>DSHN activates SHP, boosting its mRNA and protecting it from ubiquitination and degradation.</p>Fórmula:C15H17NO5SPureza:98%Cor e Forma:SolidPeso molecular:323.36JNJ-DGAT1-A
CAS:<p>JNJ-DGAT1-A is a DGAT1-selective inhibitor.</p>Fórmula:C31H35Cl2N5O3Cor e Forma:SolidPeso molecular:596.55TRC210258
CAS:<p>TRC210258 is a TGR5 agonist that acts by decreasing glycemic and dyslipidemic cardiovascular risk in animal models of diabesity.</p>Fórmula:C20H14ClFN4O2Pureza:98%Cor e Forma:SolidPeso molecular:396.8Statine
CAS:<p>Statine is a protease inhibitor that is active against pepsin and other acid proteases.</p>Fórmula:C8H17NO3Pureza:98%Cor e Forma:SolidPeso molecular:175.23Trandolaprilat
CAS:<p>Trandolaprilat is an inhibitor of non-sulfhydryl angiotensin-converting enzyme.</p>Fórmula:C22H30N2O5Cor e Forma:Pale Yellow SolidPeso molecular:402.48Mixanpril
CAS:<p>Mixanpril is an RB 105 lipophilic prodrug.</p>Fórmula:C21H23NO4SPureza:98%Cor e Forma:SolidPeso molecular:385.48Loxoprofenol-SRS
CAS:<p>Loxoprofenol-SRS, a potent metabolite of Loxoprofen, is an IV NSAID with enhanced anti-inflammatory and pain relief properties.</p>Fórmula:C15H20O3Cor e Forma:SolidPeso molecular:248.32α-Glucosidase-IN-20
CAS:<p>α-Glucosidase-IN-20 (Compound 3B) is a highly effective and orally active inhibitor of α-glucosidase.</p>Fórmula:C23H21NOSCor e Forma:SolidPeso molecular:359.48TPN729
CAS:<p>TPN729, a PDE5 inhibitor, has an IC50 of 2.28 nM, used to research erectile dysfunction.</p>Fórmula:C25H36N6O4SCor e Forma:SolidPeso molecular:516.66KT185
CAS:<p>KT185 is an orally-bioavailable and brain-penetrant ABHD6 inhibitor (IC50: 0.21 nM in Neuro2A cells).</p>Fórmula:C32H33N5O2Pureza:98%Cor e Forma:SolidPeso molecular:519.64(R)-MLN-4760
CAS:<p>(R)-MLN-4760, the R-enantiomer of MLN-4760, functions as an ACE2 inhibitor and exhibits a half maximal inhibitory concentration (IC50) of 8.4 μM, identifying it</p>Fórmula:C19H23Cl2N3O4Cor e Forma:SolidPeso molecular:428.31Tibenelast sodium
CAS:Tibenelast sodium is an inhibitor of phosphodiesterase.Fórmula:C13H14NaO4SPureza:98%Cor e Forma:SolidPeso molecular:289.3BRD6897
CAS:<p>BRD6897 is a mitochondrial content inducer that increases the cellular content of mitochondria.</p>Fórmula:C25H21N3O2S2Pureza:97.74%Cor e Forma:SolidPeso molecular:459.5814-dehydro Zymostenol
CAS:<p>14-dehydro Zymostenol, a cholesterol precursor, boosts MBP+ oligodendrocytes from precursors at 5.8-17 μM.</p>Fórmula:C27H44OCor e Forma:SolidPeso molecular:384.64Deltasonamide 2 (TFA)
CAS:<p>Deltasonamide 2 TFA is competitive, high affinity PDEδ inhibitor with a Kd of ~385 pM.</p>Fórmula:C32H40ClF3N6O6S2Pureza:98%Cor e Forma:SolidPeso molecular:761.28ACAT-IN-1 cis isomer
CAS:<p>ACAT-IN-1 cis isomer is a potent ACAT inhibitor (IC50: 100 nM) for the study of immune system-related diseases.</p>Fórmula:C29H25NO2Pureza:>99.99%Cor e Forma:SolidPeso molecular:419.51Peliglitazar racemate
CAS:<p>Peliglitazar racemate(BMS 426707-01 racemate) is the racemate of Peliglitazar.Peliglitazar racemate may be used as a potential antidiabetic and anti-obesity</p>Fórmula:C30H30N2O7Pureza:97.75%Cor e Forma:SolidPeso molecular:530.57Imazodan
CAS:<p>Imazodan is a compound with positive inotropic activity and is a type III phosphodiesterase inhibitor that can be used to study heart failure.</p>Fórmula:C13H12N4OPureza:98% - 98.31%Cor e Forma:SolidPeso molecular:240.26sEH inhibitor-14
CAS:<p>sEH inhibitor-14, a benzoxazolone-5-urea analogue, acts as an efficient soluble Epoxide Hydrolase (sEH) inhibitor, demonstrating significant activity with an</p>Fórmula:C16H12F3N3O4Cor e Forma:SoildPeso molecular:367.28PKM2 activator 5
CAS:<p>PKM2 activator 5 is a novel and potent PKM2 activator (AC50: 0.316 µM) with potential anticancer activity for the study of cancer metabolism-related diseases.</p>Fórmula:C18H19FN2O6S2Pureza:98%Cor e Forma:SolidPeso molecular:442.48Andolast
CAS:<p>Andolast (CR-2039) is an anti-allergic for asthma and COPD, inhibiting IgE synthesis and improving airflow.</p>Fórmula:C15H11N9OCor e Forma:SolidPeso molecular:333.31Pulixin
CAS:<p>Pulixin blocks FREP1 from P. falciparum, hinders parasite spread (EC50: 11µM), and stops its growth (EC50: 47nM).</p>Fórmula:C14H11NO4Cor e Forma:SolidPeso molecular:257.24SHP2 inhibitor LY6
CAS:<p>SHP2 inhibitor LY6 (LY6) is a potent and selective SHP2 inhibitor (IC50: 9.8 μM) that blocks SHP2-mediated cell signaling and proliferation.</p>Fórmula:C30H27Cl2N3O4Cor e Forma:SolidPeso molecular:564.46Sch 34826
CAS:<p>Sch 34826 is a potent, selective neutral endopeptidase inhibitor.</p>Fórmula:C27H34N2O7Pureza:98%Cor e Forma:SolidPeso molecular:498.57BMS-351
CAS:<p>BMS-351: potent, selective CYP17A1 inhibitor, promising for prostate cancer, minimal side effects.</p>Fórmula:C15H12F3N3Cor e Forma:SolidPeso molecular:291.27NPD-1335
CAS:<p>NPD1335: potent TbrPDEB1 inhibitor, submicromolar efficacy, low toxicity, raises cAMP, disrupts cell cycle, kills T. brucei.</p>Fórmula:C28H29N3O3Pureza:98%Cor e Forma:SolidPeso molecular:455.55CYP3A4-IN-3
CAS:<p>CYP3A4-IN-3, a ritonavir analogue, is a potent CYP3A4 inhibitor with an IC50 of 0.075 μM, used as an antiviral and immunosuppressant.</p>Fórmula:C34H39N3O3SCor e Forma:SolidPeso molecular:569.76Glyoxalase I inhibitor 2
CAS:<p>Glyoxalase I inhibitor 2 (compound 26) blocks GLO1 effectively (IC50: 0.5 μM), promising for depression and anxiety research.</p>Fórmula:C24H23N3O4SCor e Forma:SolidPeso molecular:449.52HSL-IN-1
CAS:<p>HSL-IN-1 is an HSL inhibitor that significantly reduces the reactive metabolite load and reduces the release of free fatty acids from stored fat.</p>Fórmula:C19H13BClF3N2O4Pureza:>99.99%Cor e Forma:SolidPeso molecular:436.58ATX inhibitor 8
CAS:<p>ATX inhibitor 8 is an inhibitor of the autocrine motor factor Autotaxin (ATX).</p>Fórmula:C28H26N10OCor e Forma:SolidPeso molecular:518.57D-threo-PPMP hydrochloride
CAS:<p>D-threo-PPMP inhibits GlyCer synthetase; active enantiomer; reduces MDCK cell growth by 70% at 20 μM.</p>Fórmula:C29H51ClN2O3Cor e Forma:SolidPeso molecular:511.19TTA-A8
CAS:<p>TTA-A8 is an antagonist of T-type calcium channel.</p>Fórmula:C22H21F3N4O2Pureza:99.22%Cor e Forma:SolidPeso molecular:430.42NBD-125
CAS:<p>NBD-125 (B-12) is a berberine analogue. NBD-125 is an RXRα activator. The IC50 value of NBD-125 in KM12C cell is 31.10 μM [1].</p>Fórmula:C19H18ClNO2Cor e Forma:SolidPeso molecular:327.81CL67
CAS:<p>CL67 is a hypoxia-inducible factor pathway inhibitor. It acts by binding to a G-quadruplex higher-order structure in the HIF promoter sequence in vitro.</p>Fórmula:C38H42N10O2Cor e Forma:SolidPeso molecular:670.81hCAIX-IN-8
CAS:<p>hCAIX-IN-8, a selective hCAIX inhibitor, IC50: 0.024 μM. Also affects CAII, CAVA (IC50s: 1.99, 1.10 μM), limits cell migration, and induces apoptosis.</p>Fórmula:C19H16N4O6Cor e Forma:SolidPeso molecular:396.355β-Dutasteride
CAS:<p>5β-Dutasteride is the S configuration of Dutasteride. It is a potent inhibitor of both 5 alpha-reductase isozymes.</p>Fórmula:C27H30F6N2O2Pureza:98%Cor e Forma:SolidPeso molecular:528.53Otamixaban
CAS:<p>Otamixaban (FXV673) is a selective and highly effective Xa inhibitor that inhibits the generation of thrombin and can be used to study acute coronary syndrome.</p>Fórmula:C25H26N4O4Pureza:98.08%Cor e Forma:SolidPeso molecular:446.5PDE4-IN-11
CAS:<p>PDE4-IN-11: Potent PDE4 inhibitor with strong bronchodilatory and anti-inflammatory effects for airway disease research.</p>Fórmula:C21H19FN2O2Cor e Forma:SolidPeso molecular:350.39RV01
CAS:<p>RV01, a resveratrol-like quinoline, inhibits DNA damage, ALDH2 expression, and has antioxidant and anti-inflammatory properties.</p>Fórmula:C17H13NO2Pureza:99.93%Cor e Forma:SolidPeso molecular:263.29MY33-3 hydrochloride
CAS:<p>MY33-3 HCl: Inhibits RPTPβ/ζ (IC50~0.1μM), PTP-1B (IC50~0.7μM), curbs alcohol intake, fights neuroinflammation and memory issues.</p>Fórmula:C16H14ClF6NS2Cor e Forma:SolidPeso molecular:433.86hCAIX-IN-14
CAS:<p>hCAIX-IN-14 is a potent inhibitor of human CA IX with a K i value of 134.8 nM .</p>Fórmula:C11H17ClN6O2SCor e Forma:SolidPeso molecular:332.81hCAI/II-IN-2
CAS:<p>hCAI/II-IN-2 (2b) inhibits hCA I/II (Ki: 40.97 nM, 15.15 nM) and IX (61.88 nM), fights AMS with anti-hypoxic effects, but has low cellular activity.</p>Fórmula:C12H12N4O5S2Cor e Forma:SolidPeso molecular:356.38PKM2 activator 4
CAS:<p>PKM2 Activator 4, a chemical compound, functions as an activator of PKM2 with an activation concentration (AC 50) ranging from 1 to 10 μM.</p>Fórmula:C16H16N2O4SCor e Forma:SolidPeso molecular:332.37LCL521
CAS:<p>LCL521 inhibits lysosomal acid sphingomyelinase (ASMase).LCL521 is an acid ceramidase (ACDase) inhibitor.</p>Fórmula:C31H52N4O7Pureza:98%Cor e Forma:SolidPeso molecular:592.77BN-82685
CAS:<p>BN-82685, a quinone-based CDC25 inhibitor, shows in vitro and in vivo efficacy, suggesting potential as an anticancer therapy.</p>Fórmula:C12H15N3O2SPureza:98%Cor e Forma:SolidPeso molecular:265.33SCH-351591
CAS:<p>SCH-351591 is an orally active inhibitor of phosphodiesterase 4.</p>Fórmula:C17H10Cl2F3N3O3Pureza:98%Cor e Forma:SolidPeso molecular:432.18Seviteronel R enantiomer
CAS:<p>Seviteronel R enantiomer (VT-464 R enantiomer) is a Seviteronel isomer produced during the manufacturing process.</p>Fórmula:C18H17F4N3O3Pureza:97.97% - >99.99%Cor e Forma:SolidPeso molecular:399.34JZP-MA-13
<p>JZP-MA-13: selective α/β-hydrolase domain 6 inhibitor, IC 50 392 nM, doesn't inhibit MAGL/ABHD12/FAAH, used in PET imaging.</p>Fórmula:C14H15FN4O3SCor e Forma:SolidPeso molecular:338.36GSK2945
CAS:<p>GSK2945, a specific Rev-erbα antagonist, boosts CYP7A1 and cholesterol metabolism. EC50: 21.5 μM (mouse), 20.8 μM (human).</p>Fórmula:C20H18Cl2N2O2SPureza:98%Cor e Forma:SolidPeso molecular:421.34Seviteronel
CAS:<p>Seviteronel (VT-464) is a novel CYP17 cleavage enzyme inhibitor and androgen receptor antagonist for the study of breast and prostate cancer.</p>Fórmula:C18H17F4N3O3Pureza:99.67% - 99.98%Cor e Forma:SolidPeso molecular:399.34FABP-IN-2
CAS:<p>FABP-IN-2, a novel ligand for FABP3, demonstrates inhibition of both FABP3 and FABP4 with IC50 values of 1.16 μM and 4.27 μM, respectively.</p>Fórmula:C25H21ClN2O3Cor e Forma:SolidPeso molecular:432.9ARL-67156 trisodium salt hydrate
CAS:<p>ARL-67156 trisodium salt hydrate is an ecto-ATPase inhibitor that prevents metabolism of P2 purinoceptor agonists.</p>Fórmula:C15H24Br2N5O12P3Cor e Forma:SolidPeso molecular:719.11Cholesteryl behenate
CAS:<p>Cholesteryl behenate is a standard in electrospray ionization tandem mass spectrometry for the analysis of cholesteryl esters and cholesterol.</p>Fórmula:C49H88O2Pureza:98%Cor e Forma:SolidPeso molecular:709.22A-908292
CAS:<p>A-908292: potent ACC2 inhibitor with 38 nM IC50, useful for studying fatty acid metabolism.</p>Fórmula:C18H20N2O4SCor e Forma:SolidPeso molecular:360.43CDP 840 hydrochloride
CAS:<p>CDP-840 (GR259653X), a potent oral PDE IV inhibitor, curbs early and late phase bronchoconstriction in squirrel monkeys.</p>Fórmula:C25H27NO2Cor e Forma:SolidPeso molecular:373.49Arasertaconazole
CAS:<p>Arasertaconazole, a sterol-14-alpha demethylation inhibitor, is used potentially for the treatment of vulvovaginal candcanidiasis.</p>Fórmula:C20H15Cl3N2OSCor e Forma:SolidPeso molecular:437.77IDO1-IN-2
CAS:<p>IDO1-IN-2 is a potent and selective IDO1 inhibitor with IC50s of 81 nM, 59 nM (mouse), and 28 nM (rat), respectively. It has anti-cancer activity.</p>Fórmula:C15H17FN6O4Pureza:98%Cor e Forma:SolidPeso molecular:364.33TDP1 Inhibitor-2
CAS:<p>TDP1 Inhibitor-2 strongly blocks TDP1 (IC50: 99 nM) & treats SCAN1 (IC50: 3.5 μM).</p>Fórmula:C25H14Cl2O5Cor e Forma:SolidPeso molecular:465.28Spirapril
CAS:<p>Spiropril is an ACE inhibitor antihypertensive drug, which belongs to the bicarboxyl group of ACE inhibitors and is used in the treatment of hypertension.</p>Fórmula:C22H30N2O5S2Cor e Forma:SolidPeso molecular:466.6111β-HSD1-IN-9
CAS:<p>11β-HSD1-IN-9 is a potent inhibitor of 11β-HSD1, displaying IC50 values of 0.48 µM for human and 1.3 µM for murine variants, respectively.</p>Fórmula:C13H9F3N2OCor e Forma:SolidPeso molecular:266.22CL 242817
CAS:<p>CL 242817 is an inhibitor of angiotensin converting enzyme (ACE).</p>Fórmula:C18H21NO5SCor e Forma:SolidPeso molecular:363.43LY 113174
CAS:<p>LY 113174, a novel nonsteroidal aromatase inhibitor, may prove useful in the treatment of estrogen-dependent diseases.</p>Fórmula:C17H10Cl2N2Cor e Forma:SolidPeso molecular:313.18LY 56110
CAS:<p>LY 56110 is a novel nonsteroidal aromatase inhibitor.</p>Fórmula:C17H12Cl2N2Pureza:98%Cor e Forma:SolidPeso molecular:315.2PF-06424439
CAS:<p>PF-06424439 is an oral and selective inhibitor of imidazopyridine diacylglycerol acyltransferase 2 (DGAT2) (IC50 of 14 nM).</p>Fórmula:C22H26ClN7OPureza:98%Cor e Forma:SolidPeso molecular:439.94Cefetrizole
CAS:<p>Ceftezole is an α-Glucosidase inhibitor (IC50: 2.1 μM; Ki: 0.578 μM).</p>Fórmula:C16H15N5O4S3Pureza:98%Cor e Forma:SolidPeso molecular:437.52(Rac)-Etavopivat
CAS:<p>(Rac)-Etavopivat, an oral PKR activator, targets sickle cell disease and haemoglobinopathies.</p>Fórmula:C22H23N3O6SCor e Forma:SolidPeso molecular:457.5BRD9500
CAS:<p>BRD9500 is an oral PDE3 inhibitor, IC50: 10 nM (PDE3A), 27 nM (PDE3B); effective in SK-MEL-3 cancer model.</p>Fórmula:C15H18FN3O2Cor e Forma:SolidPeso molecular:291.32Acetyltrialanine
CAS:<p>Acetyltrialanine is a dipeptide compound that binds at two sites on the Tb+3-pancreatic elastase complex and can be used as a nitrogen source.</p>Fórmula:C11H19N3O5Pureza:99.53%Cor e Forma:White PowderPeso molecular:273.29MDPD
CAS:<p>MDPD boosts AtFAAH, the enzyme degrading NAEs in Arabidopsis, reducing NAE 12:0's growth inhibition.</p>Fórmula:C21H19N3O3Cor e Forma:SolidPeso molecular:361.39TFB-TBOA
CAS:<p>glial glutamate transporter EAAT1 and EAAT2 inhibitor</p>Fórmula:C19H17F3N2O6Pureza:98%Cor e Forma:SolidPeso molecular:426.34Carbonic anhydrase inhibitor 14
CAS:<p>CA inhibitor 14 blocks hCA I/II/IX/XII (K i of 1203/99.7/9.4/27.7 nM) and CDK2 (IC50: 20.3 μM), showing antitumor effects.</p>Fórmula:C18H17N7O2SCor e Forma:SolidPeso molecular:395.44Enpp-1-IN-6
CAS:<p>Enpp-1-IN-6, a potent enpp-1 inhibitor, may aid cancer and infectious disease studies (WO2021203772A1, compound 51).</p>Fórmula:C22H28N4O5SCor e Forma:SolidPeso molecular:460.5511β-HSD1-IN-6
CAS:<p>11β-HSD1-IN-6 is a potent inhibitor of 11β hydroxysteroid dehydrogenase enzymes (11β-HSDs).</p>Fórmula:C21H19ClN4OCor e Forma:SolidPeso molecular:378.86Aminopeptidase-IN-1
CAS:<p>Aminopeptidase-IN-1: potent IRAP blocker, Ki 7.7 μM, useful for cognitive/memory disorder research.</p>Fórmula:C18H16N2O6Pureza:98.37%Cor e Forma:SolidPeso molecular:356.33GS 389
CAS:<p>GS 389, a tetrahydroisoquinoline, relaxes blood vessels by inhibiting brain PDE and raising aorta cGMP.</p>Fórmula:C19H23NO3Pureza:98%Cor e Forma:SolidPeso molecular:313.39Acarbose sulfate
CAS:<p>Acarbose sulfate is an anti-diabetic drug and is an inhibitor of alpha-glucosidase.</p>Fórmula:C25H45NO22SPureza:98%Cor e Forma:SolidPeso molecular:743.68TK-642
CAS:<p>TK-642 is a potent and selective SHP2 inhibitor with oral activity, based on pyrazole and pyrazine structures (IC50 = 2.7 nmol/L). It effectively inhibits the proliferation of esophageal carcinoma cells and induces apoptosis, making it useful for studying esophageal cancer.</p>Fórmula:C17H20ClN7SCor e Forma:SolidPeso molecular:389.91Anti-hyperglycemic agent-1
CAS:<p>Anti-hyperglycemic agent 1 is a potent inhibitor of alpha-glucosidase (IC50: 0.53 μM). anti-Hyperglycemic agent 1 can be used to study diabetes.</p>Fórmula:C20H15BrN2O3Cor e Forma:SolidPeso molecular:411.25Anticancer agent 70
CAS:<p>Compound 21 is a powerful anticancer agent with cytotoxicity against various cancers, causing cell cycle arrest and affecting p53/p21 levels and mitochondria.</p>Fórmula:C13H9Cl2N3O2SCor e Forma:SolidPeso molecular:342.2LAZABEMIDE
CAS:<p>Lazabemide (Ro 19-6327) is selective, reversible monoamine oxidase B (MAO-B) inhibitor (IC50 values are 0.03 and > 100 μM for MAO-B and MAO-A respectively).</p>Fórmula:C8H10ClN3OPureza:98%Cor e Forma:SolidPeso molecular:199.64Gcase activator 3
CAS:<p>Gcase activator 3 is a glucocerebrosidase (GCase) activator that enhances GBA1 mutant fibroblast lysosomal GCase activity.</p>Fórmula:C23H20N4O2Pureza:99.08%Cor e Forma:SolidPeso molecular:384.43Phosphodiesterase-IN-1
CAS:<p>Phosphodiesterase-IN-1 (Compound 7), a phosphodiesterase (PDE) inhibitor, exhibits anti-Plasmodium and antiproliferative activities. It effectively inhibits P. falciparum (strain 3D7) with an IC 50 value of 0.64 μM [1].</p>Fórmula:C15H15FN4OCor e Forma:SolidPeso molecular:286.3HM-50316
CAS:<p>HM-50316 is a High affinity FABP4 inhibitor (Ki < 1 nM).</p>Fórmula:C29H23ClN2O3SPureza:98%Cor e Forma:SolidPeso molecular:515.02MMPX
CAS:<p>calmodulin-sensitive cyclic GMP phosphodiesterase inhibitor</p>Fórmula:C12H18N4O3Pureza:98%Cor e Forma:SolidPeso molecular:266.3hCAIX/XII-IN-4
CAS:<p>hCAIX/XII-IN-4 inhibits CAIX/XII with Ki: 4.5 nM (CAXII), 23.6 nM (CAIX), and >10000 nM (CAI/CAII).</p>Fórmula:C20H16N2O5Cor e Forma:SolidPeso molecular:364.35Zidovudine glucuronide
CAS:<p>Zidovudine glucuronide: an NRTI antiretroviral for HIV/AIDS treatment; blocks HIV reverse transcriptase, stops viral DNA formation.</p>Fórmula:C16H21N5O10Cor e Forma:SolidPeso molecular:443.37AX 048
CAS:<p>Group IVA cPLA2 inhibitor AX 048 halts arachidonic acid release, preventing prostaglandin production, with XI(50) of 0.022 and ED50 of 1.2 mg/kg.</p>Fórmula:C22H41NO4Cor e Forma:SolidPeso molecular:383.57MEDS433
CAS:<p>MEDS433 inhibits dihydroorotate dehydrogenase (IC50 1.2 nM) and blocks replication of hCoV-OC43, hCoV-229E, SARS-CoV-2 at nanomolar levels.</p>Fórmula:C20H11F4N3O2Cor e Forma:SolidPeso molecular:401.31YM 26734
CAS:<p>Competitive inhibitor of secretory phospholipase A2 (sPLA2)</p>Fórmula:C45H62O8Pureza:98%Cor e Forma:SolidPeso molecular:730.97SCD1 Inhibitor
CAS:<p>SCD1 Inhibitor is a novel stearoyl-CoA desaturase1 (SCD1) inhibitor.</p>Fórmula:C21H20F3N3O3Cor e Forma:SolidPeso molecular:419.4Tritoqualine
CAS:<p>Tritoqualine is used as an inhibitor of histidine decarboxylase.</p>Fórmula:C26H32N2O8Pureza:98%Cor e Forma:SolidPeso molecular:500.54SQ-24,798
CAS:<p>SQ-24,798 is an inhibitor of the thrombin-activatable fibrinolysis and carboxypeptidase N (CPN).</p>Fórmula:C7H15N3O2SPureza:98%Cor e Forma:SolidPeso molecular:205.28SCH-51866
CAS:<p>SCH-51866 is a PDE1 and PDE5 phosphodiesterase inhibitor with IC50 value of 0.070 μM and IC50 0.060 μM respectively.</p>Fórmula:C19H18F3N5OPureza:98%Cor e Forma:SolidPeso molecular:389.37Ciraparantag
CAS:<p>Ciraparantag inhibits thrombin, factor Xa, and reverses various anticoagulants.</p>Fórmula:C22H48N12O2Pureza:98%Cor e Forma:SolidPeso molecular:512.7Y-29794 oxalate
CAS:<p>Inhibitor of prolyl endopeptidase</p>Fórmula:C25H36N2O5S2Pureza:98%Cor e Forma:SolidPeso molecular:508.69UK-414,495
CAS:<p>UK-414,495 is a potent, selective inhibitor of the neutral endopeptidase, the enzyme normally serves to break down the neuropeptide VIP.</p>Fórmula:C16H25N3O3SCor e Forma:SolidPeso molecular:339.45FABP4/5-IN-5
CAS:<p>FABP4/5-IN-5 (compound D9) serves as a potent inhibitor of both FABP 4 and FABP 5, demonstrating IC50 values of 4.68 μM and 10.72 μM, respectively. It is notably effective in addressing metabolic disorders such as diabetes mellitus [1].</p>Fórmula:C23H14ClF2NO4SCor e Forma:SolidPeso molecular:473.88JNJ-61803534
CAS:<p>JNJ-61803534: RORγt inverse agonist, IC50=9.6 nM, oral, anti-inflammatory, reduces IL-17A in T cells.</p>Fórmula:C23H23Cl2F6N3O4SCor e Forma:SolidPeso molecular:622.41BML-111
CAS:<p>inhibits leukotriene B4 (LTB4)-induced polymorphonuclear neutrophils (PMN) chemotaxis</p>Fórmula:C8H16O5Cor e Forma:SolidPeso molecular:192.21RO6806051
CAS:<p>RO6806051 (compound 12) is a potent dual inhibitor of fatty acid binding proteins 4 and 5 (FABP4 and FABP5), exhibiting excellent selectivity and absorption, distribution, metabolism, and excretion (eADME) properties.</p>Fórmula:C21H19ClN6Cor e Forma:SolidPeso molecular:390.87Benproperine
CAS:<p>Benproperine is a bioactive molecule with antineoplastic properties.</p>Fórmula:C21H27NOPureza:98%Cor e Forma:SolidPeso molecular:309.45Methazolamide-d6
CAS:<p>Methazolamide-d6 is a GC/LC-MS standard for measuring methazolamide, a glaucoma drug that lowers eye pressure and fluid, reduces seizures, and combats ROS.</p>Fórmula:C5H2D6N4O3S2Cor e Forma:SolidPeso molecular:242.31mIDH1-IN-1
CAS:<p>mIDH1-IN-1 is a selective mIDH1 inhibitor (IC50: 961.5 nM), blocks 2-HG production, and hinders IDH1 mutant cell growth (IC50: 41.8 nM).</p>Fórmula:C25H27N3O5Cor e Forma:SolidPeso molecular:449.5Umbralisib tosylate
CAS:<p>Umbralisib tosylate, an oral PI3Kδ/CK1ε inhibitor (EC50: 22.2 nM/6.0 μM), shows promise for CLL research.</p>Fórmula:C38H32F3N5O6SCor e Forma:SolidPeso molecular:743.75CS-722 Free base
CAS:<p>CS-722 Free base: synthetic muscle relaxant; inhibits spinal reflex and sodium/calcium currents affecting synaptic activity.</p>Fórmula:C16H19ClN2O4Pureza:99.52%Cor e Forma:SolidPeso molecular:338.79CG-707
CAS:<p>CG-707 is an inhibitor of PRL-3 that acts by blocking the migration and invasion of metastatic cancer cells.</p>Fórmula:C20H17NO3S2Pureza:98%Cor e Forma:SolidPeso molecular:383.48Imidazoleacetic acid
CAS:<p>Imidazoleacetic acid, an endogenous ligand, stimulates imidazole receptors.</p>Fórmula:C5H6N2O2Pureza:98%Cor e Forma:SolidPeso molecular:126.11Sp-Cyclic AMPS (sodium salt)
CAS:<p>Sp-cAMPS Na salt activates PKA I/II and competitively inhibits PDE3A (Ki: 47.6 μM), also binds PDE10 GAF (EC50: 40 μM).</p>Fórmula:C10H12N5NaO5PSCor e Forma:SolidPeso molecular:367.25LAS-31180
CAS:<p>LAS-31180 is a phosphodiesterase 3 inhibitor. It also has positive inotropic and vasodilator properties.</p>Fórmula:C11H12N2O3SPureza:98%Cor e Forma:SolidPeso molecular:252.29GKA-22
CAS:<p>GKA-22 is a human glucokinase allosteric activator in the absence of glucose.</p>Fórmula:C22H22N2O5SPureza:98%Cor e Forma:SolidPeso molecular:426.49Glucocerebrosidase-IN-1
CAS:<p>Glucocerebrosidase-IN-1 inhibits GCase with IC50 of 29.3 μM, Ki 18.5 μM, useful for Gaucher's and Parkinson's research.</p>Fórmula:C13H27NO3Cor e Forma:SolidPeso molecular:245.36SHP2-IN-13
CAS:<p>SHP2-IN-13 is an orally active, highly selective allosteric inhibitor targeting the SHP2 “tunnel site,” exhibiting an IC50 of 83.0 nM.</p>Fórmula:C16H21N7OCor e Forma:SolidPeso molecular:327.38Win-62005
CAS:<p>Win-62005 is an inhibitor of cyclic AMP phosphodiesterase III (PDE III)(Kis: 25 and 26 nM for rat heart and canine aorta).</p>Fórmula:C12H10N4OPureza:98%Cor e Forma:SolidPeso molecular:226.23ML218
CAS:<p>ML218 is an inhibitor of T-type Ca2+ channels (Cav3.1, Cav3.2, Cav3.3).ML218 inhibits the synaptic activity of subthalamic nucleus (STN) neurons.</p>Fórmula:C19H26Cl2N2OPureza:99.2% - 99.45%Cor e Forma:SolidPeso molecular:369.33TM6008
CAS:<p>TM6008 is an inhibitor of prolyl hydroxylase that protects against cell death after hypoxia.</p>Fórmula:C21H17N5O3Pureza:98%Cor e Forma:SolidPeso molecular:387.39DMPAC-Chol
CAS:<p>DMPAC-Chol, a cationic cholesterol, aids gene transfection, DNA protection, binds DNA, and lowers HepG2 viability at 37.5 μg/ml.</p>Fórmula:C33H58N2O2Cor e Forma:SolidPeso molecular:514.83FR-221647
CAS:<p>FR-221647: non-nucleoside adenosine deaminase blocker, moderate efficacy, better pharmacokinetics than EHNA/Pentostatin.</p>Fórmula:C14H17N3O2Cor e Forma:SolidPeso molecular:259.3LP-533401
CAS:<p>LP-533401 is an inhibitor of Tryptophan hydroxylase 1. It is used for regulates serotonin production in the gut.</p>Fórmula:C27H22F4N4O3Pureza:98%Cor e Forma:SolidPeso molecular:526.48Enpp-1-IN-5
CAS:<p>Enpp-1-IN-5 is a potent enpp-1 inhibitor with potential in cancer and infectious disease research.</p>Fórmula:C17H26N6O4SCor e Forma:SolidPeso molecular:410.49MitoTEMPO hydrate
CAS:<p>MitoTEMPO, a mitochondria-targeted antioxidant, scavenges superoxide and alkyl radicals supporting potential therapy for mitochondrial dysfunction.</p>Fórmula:C29H35N2O2P·Cl·H2OCor e Forma:SolidPeso molecular:528.04CAY10761
CAS:<p>CAY10761 inhibits ENPP1 (IC50: 467 μM human, 429 μM snake), mushroom tyrosinase (Ki: 1.9 μM), and urease from different sources (IC50: 0.093-<0.125 mM).</p>Fórmula:C7H8N4O2S2Cor e Forma:SolidPeso molecular:244.29ML-262
CAS:<p>ML-262 is an effective inhibitor of hepatic lipid droplet formation and is used in studies of non-alcoholic fatty liver disease.</p>Fórmula:C27H32N2O4SCor e Forma:SolidPeso molecular:480.62PKM2 activator 3
CAS:<p>PKM2 activator 3, with 90 nM AC50, enhances PKM2. It has good Caco-2 permeability, stable, and aids cancer research.</p>Fórmula:C15H11ClF2N2O3SCor e Forma:SolidPeso molecular:372.7711β-HSD1-IN-12
CAS:<p>11β-HSD1-IN-12 is an 11β-HSD1 inhibitor.11β-HSD1-IN-12 is implicated in the conversion of glucocorticoids in vivo and can be used to study metabolic syndrome</p>Fórmula:C19H27ClN2O3SPureza:99.68%Cor e Forma:SolidPeso molecular:398.95Gemcabene
CAS:<p>Gemcabene (PD-72953) lowers LDL and triglycerides, boosts HDL, and reduces inflammation by decreasing C-reactive protein.</p>Fórmula:C16H30O5Pureza:≥98%Cor e Forma:SolidPeso molecular:302.41Z-321
CAS:<p>Z-321 is an inhibitor of prolyl endopeptidase.</p>Fórmula:C19H24N2O2SPureza:98%Cor e Forma:SolidPeso molecular:344.47IDO1-IN-17
CAS:<p>IDO1-IN-17 (I-4) is an IDO1 inhibitor, with an IC 50 of 0.44 μM in hela cells .</p>Fórmula:C28H32BrClFN5O2Cor e Forma:SolidPeso molecular:604.94Endothall
CAS:<p>Endothall is an effective protein phosphatase 2A (PP2A) inhibitor, exerting inhibitory effects on both PP2A and PP1, with IC50 values of 90 nM and 5 µM,</p>Fórmula:C8H10O5Pureza:98.92% - ≥98%Cor e Forma:Cyrstalline White Solid The Monohydrate Is In The Form Of Colorless Crystals Non Corrosive Used As A Selective HerbicidePeso molecular:186.16DU717
CAS:<p>DU717 is an antihypertensive agent.</p>Fórmula:C12H15ClN4O2SPureza:99.64%Cor e Forma:SolidPeso molecular:314.79Enazadrem
CAS:<p>Enazadrem is a 5-lipoxygenase inhibitor with antiinflammatory activities.</p>Fórmula:C18H25N3OPureza:98%Cor e Forma:SolidPeso molecular:299.41α-Glycosidase-IN-1
CAS:<p>α-Glycosidase-IN-1 (compound MZ7) is a potent inhibitor of α-GLY (α-glycosidase) (IC50: 44.72 nM, Ki: 44.74 nM).</p>Fórmula:C21H19N9O6S2Cor e Forma:SolidPeso molecular:557.56Hydroxythiohomosildenafil
CAS:<p>Hydroxythiohomosildenafil, an analogue of sildenafil, is a phosphodiesterase-5 (PDE-5) inhibitor.</p>Fórmula:C23H32N6O4S2Pureza:99.45%Cor e Forma:SolidPeso molecular:520.67Tenuazonic acid
CAS:<p>Tenuazonic acid, a nonhost-selective mycotoxin from Alternaria alternate, inhibits PSII by blocking electron transport at D1 protein.</p>Fórmula:C10H15NO3Pureza:98%Cor e Forma:SolidPeso molecular:197.23Agn 190727
CAS:<p>Agn 190727 is a retonoic acid receptor that can induce retinoid-induced hypertriglyceridemia.</p>Fórmula:C20H22O2Cor e Forma:SolidPeso molecular:294.39CGP-28014
CAS:<p>CGP-28014 inhibits COMT, boosts renal dopamine & DOPAC excretion, lowers HVA, no effect on renal sodium.</p>Fórmula:C12H19N3OCor e Forma:SolidPeso molecular:221.3RWJ 63556
CAS:<p>RWJ 63556 is an orally active inhibitor of COX-2 selective/5-lipoxygenase, shows anti-inflammatory activities.</p>Fórmula:C11H10FNO3S2Pureza:99.92%Cor e Forma:SolidPeso molecular:287.33MDK-4683
CAS:<p>MDK-4683, also known as CA IX/XII Inhibitor, is a hCA IX and hCA XII inhibitor.</p>Fórmula:C13H12N4O5SPureza:98%Cor e Forma:SolidPeso molecular:336.32HFI-437
CAS:<p>HFI-437 is a potent, non-peptidic, insulin-regulated aminopeptidase (IRAP) inhibitor with a K i of 20 nM and functions as a cognitive enhancer [1].</p>Fórmula:C23H20N2O5Cor e Forma:SolidPeso molecular:404.42MitoPBN
CAS:<p>MitoPBN: mitochondria-targeted antioxidant, inhibits UCP1-3 at 250 nM, traps hydroxyl & carbon radicals, prevents lipid peroxidation.</p>Fórmula:C33H37BrNO2PCor e Forma:SolidPeso molecular:590.542Ciraparantag TFA
CAS:<p>Ciraparantag TFA reverses anticoagulants by inhibiting thrombin and factor Xa.</p>Fórmula:C26H50F6N12O6Pureza:98%Cor e Forma:SolidPeso molecular:740.74NP603
CAS:<p>NP603 is a cell-permeable inhibitor of FGFR1, PDGFRβ, and VEGFR2 that binds to the ATP pocket. It also is a very weak EGFR inhibitor.</p>Fórmula:C26H26N2O5Pureza:98%Cor e Forma:SolidPeso molecular:446.49FKGK11
CAS:<p>FKGK11 is a potent inhibitor of GVIA iPLA2.</p>Fórmula:C13H13F5OPureza:98%Cor e Forma:SolidPeso molecular:280.23Carbonic anhydrase inhibitor 13
CAS:<p>Carbonic anhydrase inhibitor 13 (compound 7) is a potent inhibitor of carbonic anhydrase (CA).</p>Fórmula:C17H15N5O3S2Cor e Forma:SolidPeso molecular:401.46Amastatin
CAS:<p>Amastatin is a non-toxic inhibitor of aminopeptidase A and leucine aminopeptidase, and its Ki for aminopeptidase A is 1 μM .</p>Fórmula:C21H38N4O8Pureza:98%Cor e Forma:SolidPeso molecular:474.559(S)-HpODE
CAS:<p>9(S)-HpODE is produced by the action of arachidonate 5-LO on linoleic acid. It can be further metabolized by potato hydroperoxide dehydratase to colneleic acid.</p>Fórmula:C18H32O4Cor e Forma:SolidPeso molecular:312.44Tebuconazole-d9
CAS:<p>Tebuconazole-d9 is a GC/LC-MS standard for quantifying the triazole fungicide tebuconazole, affecting seed/foliar fungi and androgen receptors.</p>Fórmula:C16H13ClD9N3OCor e Forma:SolidPeso molecular:316.87hCAIX-IN-6
CAS:<p>6B and 14g inhibit tumor-associated HCA IX with low nanomolar potency; 6K targets HCA XII. All are potential cancer drug leads.</p>Fórmula:C18H12N2O4SCor e Forma:SolidPeso molecular:352.36Arcapillin
CAS:<p>Arcapillin, an anticancer agent, induces apoptosis mediated at least in part by the ERS pathway and inhibits hepatoma tumor growth.</p>Fórmula:C18H16O8Cor e Forma:SolidPeso molecular:360.31α-Glucosidase-IN-9
CAS:<p>α-Glucosidase-IN-9 (compound 7) is a highly potent α-glucosidase inhibitor with an IC50 of 55.6 μM, making it suitable for type II diabetes research [1].</p>Fórmula:C19H12N4OSCor e Forma:SolidPeso molecular:344.39DNJNAc
CAS:<p>DNJNAc (2-Acetamido-1,2-dideoxynojirimycin) is a potent β-hexosaminidase inhibitor, reducing cartilage matrix degradation, relevant in glycoconjugate studies.</p>Fórmula:C8H16N2O4Pureza:98.65% - 99.37%Cor e Forma:SolidPeso molecular:204.22Eggmanone
CAS:<p>EGM1: potent PDE4D3 inhibitor, IC50=72 nM, 40-50x selectivity over other PDEs, activates PKA, blocks Hh.</p>Fórmula:C20H20N2O2S3Cor e Forma:SolidPeso molecular:416.58
