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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2277 products of "Membrane Transporter/Ion Channel"

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  • Phenibut
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    Phenibut

    CAS:
    <p>Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).</p>
    Formula:C10H13NO2
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:179.22

    Ref: TM-T2990

  • γ-DGG acetate(6729-55-1 free base)
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    γ-DGG acetate(6729-55-1 free base)

    CAS:
    <p>gamma-DGG acetate(6729-55-1 free base) (γ-D-Glutamylglycine) is a competitive blocker of AMPA receptor.</p>
    Formula:C9H16N2O7
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:264.23

    Ref: TM-T15369L

  • GET73
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    GET73

    CAS:
    <p>GET73 (Gamma hydroxybutyric acid analogue) is an negative allosteric modulator of mGluR5.</p>
    Formula:C13H16F3NO2
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:275.27

    Ref: TM-T11393

  • Etimizol
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    Etimizol

    CAS:
    <p>Etimizol improves memory by aiding the consolidation stage, effective against amnesia from hypoxia or brain injury.</p>
    Formula:C9H14N4O2
    Purity:99%
    Color and Shape:Solid
    Molecular weight:210.23

    Ref: TM-T11244

  • Oxybuprocaine hydrochloride
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    Oxybuprocaine hydrochloride

    CAS:
    <p>Oxybuprocaine hydrochloride (Oxybuprocaine HCl), a local anesthetic, is used especially in otolaryngology and ophthalmology.</p>
    Formula:C17H29ClN2O3
    Purity:>99.99%
    Color and Shape:White Crystalline Powder
    Molecular weight:344.88

    Ref: TM-T0378

  • DCPIB
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    DCPIB

    CAS:
    <p>DCPIB, a known specific and potent inhibitor of volume-regulated anion channels (VRAC),DCPIB displayed superior selectivity toward TRESK with an IC50 of 0.14 μM</p>
    Formula:C22H28Cl2O4
    Purity:99.79% - 99.87%
    Color and Shape:Solid
    Molecular weight:427.36

    Ref: TM-T10979

  • Doxapram hydrochloride hydrate
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    Doxapram hydrochloride hydrate

    CAS:
    <p>Doxapram hydrochloride hydrate (Doxapram HCl) inhibits TASK-1, TASK-3, TASK-1/TASK-3 heterodimeric channel function with EC50 of 0.41, 37, 9 μM, respectively.</p>
    Formula:C24H33ClN2O3C24H30N2O2·ClH·H2O
    Purity:99.64% - >99.99%
    Color and Shape:Solid
    Molecular weight:432.99

    Ref: TM-T0038

  • Glimepiride
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    Glimepiride

    CAS:
    <p>Glimepiride (HOE-490) is a long-acting, third-generation sulfonylurea with hypoglycemic activity.</p>
    Formula:C24H34N4O5S
    Purity:97.84% - 98.87%
    Color and Shape:White Cyrstalline Solid
    Molecular weight:490.62

    Ref: TM-T0127

  • Disopyramide
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    Disopyramide

    CAS:
    <p>Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.</p>
    Formula:C21H29N3O
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:339.47

    Ref: TM-T1320

  • 3,4,5-Trimethoxycinnamic acid
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    3,4,5-Trimethoxycinnamic acid

    CAS:
    <p>3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at the</p>
    Formula:C12H14O5
    Purity:98.91%
    Color and Shape:Solid
    Molecular weight:238.24

    Ref: TM-T2983

  • Butamben
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    Butamben

    CAS:
    <p>Butamben (Butyl 4-aminobenzoate) is a long-duration local anesthetic used for the treatment of chronic pain.</p>
    Formula:C11H15NO2
    Purity:99.43%
    Color and Shape:Crystals From Alc Physical Description Yellow Powder Insoluble In Water (Ntp 1992)
    Molecular weight:193.24

    Ref: TM-T0916

  • Penicillin G sodium salt
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    Penicillin G sodium salt

    CAS:
    <p>Penicillin G sodium(Benzylpenicillin sodium) salt is a penicillin derivative commonly used in the form of its sodium or potassium salts in the treatment of a</p>
    Formula:C16H17N2NaO4S
    Purity:98.11%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:356.37

    Ref: TM-T0958

  • 5,5-Dimethyloxazolidine-2,4-dione
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    5,5-Dimethyloxazolidine-2,4-dione

    CAS:
    <p>5,5-Dimethyloxazolidine-2,4-dione (Dimethadione) is an anticonvulsant that is the active metabolite of TRIMETHADIONE.</p>
    Formula:C5H7NO3
    Purity:99.12%
    Color and Shape:Drypowder Pelletslargecrystals
    Molecular weight:129.11

    Ref: TM-T1234

  • Leptomycin A
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    Leptomycin A

    CAS:
    <p>Leptomycin A from Streptomyces inhibits CRM1, reducing HIV-1 replication, less potent than Leptomycin B, blocks protein nuclear export.</p>
    Formula:C32H46O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:526.7

    Ref: TM-T11837

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    EVT-401

    <p>EVT-401 (P2X7 receptor antagonist-1), a purinergic P2X7 receptor antagonist, demonstrates efficacy in combating neuroinflammation [1].</p>
    Formula:C22H20F4N2O3
    Color and Shape:Solid
    Molecular weight:436.4

    Ref: TM-T74409

  • Cavα2δ-IN-1
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    Cavα2δ-IN-1

    CAS:
    <p>Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a Ki</p>
    Formula:C18H27N5O
    Color and Shape:Solid
    Molecular weight:329.448

    Ref: TM-T40071

  • Nitrazolam
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    Nitrazolam

    CAS:
    <p>Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.</p>
    Formula:C17H13N5O2
    Color and Shape:Solid
    Molecular weight:319.32

    Ref: TM-T203627

  • Elgodipine
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    Elgodipine

    CAS:
    <p>Elgodipine decreases angina severity, inhibits muscle growth, and is voltage-sensitive, showing promise for angina treatment.</p>
    Formula:C29H33FN2O6
    Purity:98.95% - 99.50%
    Color and Shape:Solid
    Molecular weight:524.58

    Ref: TM-T68060

  • GS-9191 PM
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    GS-9191 PM

    <p>GS-9191 PM: novel antitumorviral bis-amide prodrug, inhibits MDR1/BCRP, has antiproliferative activity.</p>
    Formula:C11H16N6O
    Purity:99.79%
    Color and Shape:Soild
    Molecular weight:248.28

    Ref: TM-T67821

  • TRPA1 Antagonist 3
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    TRPA1 Antagonist 3

    CAS:
    <p>TRPA1 Antagonist 3 is a compound with photoswitchable properties that acts as an agonist on the TRPA1 channel, providing the ability for optical control.</p>
    Formula:C11H8ClN3
    Color and Shape:Solid
    Molecular weight:217.66

    Ref: TM-T40822

  • (1S,3R)-3-Aminocyclopentane carboxylic acid
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    (1S,3R)-3-Aminocyclopentane carboxylic acid

    CAS:
    <p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>
    Formula:C6H11NO2
    Color and Shape:Solid
    Molecular weight:129.16

    Ref: TM-T203289

  • GsMTx4
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    GsMTx4

    CAS:
    <p>GsMTx-4, mechanosensitive and stretch-activated ion channel inhibitor (CAS 1209500-46-8).</p>
    Formula:C185H273N49O45S6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4095.84

    Ref: TM-TP1670

  • BeKm-1
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    BeKm-1

    CAS:
    <p>Potent, selective hERG (KV11.1) blocker; doesn't affect 14 other K+ channels; extends QTc in rabbit heart dose-dependently.</p>
    Formula:C174H261N51O52S6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4091.65

    Ref: TM-TP2072

  • GeX-2
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    GeX-2

    CAS:
    <p>GeX-2 is a truncated analogue of αO-conotoxin. It has the ability to activate GABAB receptors and inhibit α9α10nAChR as well as CaV2.2 channels. Additionally, GeX-2 is effective in alleviating pain in a rat model of chronic constriction injury.</p>
    Formula:C103H169N43O27
    Color and Shape:Solid
    Molecular weight:2441.72

    Ref: TM-TP3132

  • α,β-Methylene-ATP dilithium
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    α,β-Methylene-ATP dilithium

    CAS:
    <p>α,β-Methylene ATP dilithium, a phosphonic analog of ATP, serves as a ligand for P2X3 and P2X7 receptors.</p>
    Formula:C11H16Li2N5O12P3
    Color and Shape:Solid
    Molecular weight:517.07

    Ref: TM-T38444

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    GpTx-1 TFA

    <p>GpTx-1 TFA is a polypeptide NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. It exhibits potent inhibitory activity on the NaV1.7 channel with an IC50 value of 10 nM, demonstrating excellent selectivity over NaV1.4 (IC50 = 0.301 μM) and NaV1.5 (IC50 = 4.20 μM) with &gt;20-fold and &gt;950-fold selectivity, respectively.</p>
    Color and Shape:Odour Solid

    Ref: TM-TP3232

  • WAY-326766
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    WAY-326766

    CAS:
    <p>WAY-326766 increases ion transport through mutant CFTR and can be used to alter the lifespan of eukaryotes.WAY-326766 can be used to treat cystic fibrosis (CF).</p>
    Formula:C21H23N3O5
    Purity:98.76%
    Color and Shape:Solid
    Molecular weight:397.42

    Ref: TM-T77604

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    AChE/Aβ-IN-1

    <p>AChE/Aβ-IN-1 (compound 32) is a potent, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 86 nM and an NMDA receptor antagonist targeting the</p>
    Formula:C20H25BrN4
    Color and Shape:Solid
    Molecular weight:401.34

    Ref: TM-T79569

  • Anisatin
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    Anisatin

    <p>Anisatin is a useful organic compound for research related to life sciences and the catalog number is T124719.</p>
    Formula:C15H20O8
    Color and Shape:Solid
    Molecular weight:328.317

    Ref: TM-T124719

  • Trans (2,3)-Dihydrotetrabenazine
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    Trans (2,3)-Dihydrotetrabenazine

    CAS:
    <p>Trans (2,3)-Dihydrotetrabenazine is a Tetrabenazine metabolite, shows inhibition activity on vesicular monoamine transporter (VMAT2).</p>
    Formula:C19H29NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:319.44

    Ref: TM-T12190

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    LRRK2-IN-15

    <p>LRRK2-IN-15 is an inhibitor of LRRK2. It exhibits an IC50 value of 5 nM in PBMC cells and 1.5 μM for BCRP. This compound is utilized in the research of Parkinson's disease.</p>
    Color and Shape:Odour Solid

    Ref: TM-T200475

  • TP-050
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    TP-050

    CAS:
    <p>TP-050: potent, selective NMDAR agonist, EC50 0.51 µM (GluN2A), 9.6 µM (GluN2D), BBB permeable, boosts hippocampal LTP.</p>
    Formula:C16H15ClF2N6O
    Color and Shape:Solid
    Molecular weight:380.78

    Ref: TM-T73491

  • Albanin A
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    Albanin A

    <p>Albanin A is a useful organic compound for research related to life sciences and the catalog number is T124310.</p>
    Formula:C20H18O6
    Color and Shape:Solid
    Molecular weight:354.358

    Ref: TM-T124310

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    Jingzhaotoxin-XII TFA

    <p>Jingzhaotoxin-XII (JzTx-XII) TFA is a specific inhibitor of the Kv4.1 channel, exhibiting an IC50 of 0.363 μM. It interacts with the channel by altering gating behavior.</p>
    Color and Shape:Odour Solid

    Ref: TM-TP2888

  • 3-Aminopropylphosphinic acid
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    3-Aminopropylphosphinic acid

    CAS:
    <p>3-Aminopropylphosphinic acid (3-APPA) is a phosphonic analog of gamma-aminobutyric acid (GABA).</p>
    Formula:C3H10NO2P
    Color and Shape:Solid
    Molecular weight:123.092

    Ref: TM-T38438

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    Huwentoxin I

    CAS:
    <p>Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.</p>
    Formula:C161H246N48O44S6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3750.36

    Ref: TM-T80185

  • LY-466195
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    LY-466195

    CAS:
    <p>LY-466195 is a competitive antagonist of GLUK5 receptor.</p>
    Formula:C16H24F2N2O4
    Color and Shape:Solid
    Molecular weight:346.37

    Ref: TM-T27958

  • Hyp9
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    Hyp9

    CAS:
    <p>Hyp9, a specific agonist for the transient receptor potential canonical 6 (TRPC6) channel, is utilized in spinal cord injury (SCI) research [1].</p>
    Formula:C18H26O5
    Color and Shape:Solid
    Molecular weight:322.40

    Ref: TM-T75550

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    AChE/Aβ-IN-2

    <p>AChE/Aβ-IN-2 (compound 33) is a powerful, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 135 nM.</p>
    Formula:C20H25ClN4
    Color and Shape:Solid
    Molecular weight:356.89

    Ref: TM-T79571

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    Chlorotoxin TFA

    <p>Chlorotoxin TFA, a scorpion venom peptide, blocks chloride channels and has anti-cancer properties.</p>
    Formula:C160H250F3N53O49S11
    Color and Shape:Solid
    Molecular weight:4109.74

    Ref: TM-T75722

  • JAMI1001A
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    JAMI1001A

    CAS:
    <p>JAMI1001A enhances AMPA receptor signaling, slows deactivation/desensitization for flip/flop isoforms.</p>
    Formula:C16H17F3N4O3S
    Color and Shape:Solid
    Molecular weight:402.39

    Ref: TM-T38392

  • SLC26A3-IN-2
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    SLC26A3-IN-2

    CAS:
    <p>Vilobelimab (CaCP-29) is a human-mouse chimeric IgG antibody targeting human complement component 5a, a C5a inhibitor that inhibits neutrophil activation.</p>
    Formula:C19H13ClN2O2S
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:368.84

    Ref: TM-T74815

  • Homocarnosine
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    Homocarnosine

    CAS:
    <p>Homocarnosine is an endogenous dipeptide in cerebral regions and cerebrospinal fluid.</p>
    Formula:C10H16N4O3
    Color and Shape:Solid
    Molecular weight:240.26

    Ref: TM-T32098

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    Idactamab

    CAS:
    <p>Idactamab (INT-001) is a monoclonal antibody to the human amino acid transport protein ASCT2.</p>
    Purity:> 95%
    Color and Shape:Liquid
    Molecular weight:146.2 kDa

    Ref: TM-T77385

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    Anticonvulsant agent 9

    <p>Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.</p>
    Formula:C22H24N4O2
    Color and Shape:Solid
    Molecular weight:376.45

    Ref: TM-T205256

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    Crofelemer

    CAS:
    <p>Crofelemer (Provir) is an orally active antidiarrheal agent. It targets the cystic fibrosis transmembrane conductance regulator (CFTR) and calcium-activated chloride channels (CACC), which are responsible for chloride and fluid secretion in the gastrointestinal tract. Crofelemer is applicable for research in diarrhea-related conditions.</p>
    Color and Shape:Solid

    Ref: TM-T205474

  • 2,4,6-Tri-tert-butylphenol
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    2,4,6-Tri-tert-butylphenol

    CAS:
    <p>2,4,6-Tri-tert-butylphenol inhibits the Ca2+ ATPase activity of human red blood cell membranes and can be used in related research in the field of life sciences.</p>
    Formula:C18H30O
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:262.43

    Ref: TM-TN9644

  • Bendroflumethiazide
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    Bendroflumethiazide

    CAS:
    <p>Bendroflumethiazide (Naturetin) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE. It has been used in the treatment of familial hyperkalemia, hypertension, edema, and urinary tract disorders. (From Martindale, The Extra Pharmacopoeia, 30th ed, p810)</p>
    Formula:C15H14F3N3O4S2
    Purity:98% - >99.99%
    Color and Shape:Crystals From Dioxane Solid
    Molecular weight:421.41

    Ref: TM-T1204

  • Levamlodipine besylate Hemipentahydrate
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    Levamlodipine besylate Hemipentahydrate

    CAS:
    <p>Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.</p>
    Formula:C20H25ClN2O5·C6H6O3SH2O
    Color and Shape:Solid
    Molecular weight:1224.18

    Ref: TM-T204904

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    Analgesic/antidepressant agent-1

    <p>Analgesic/antidepressant agent-1 (Compound k1) is an orally active N-acetylamino chloro ketone derivative capable of crossing the blood-brain barrier. It exhibits high affinity for NMDA receptors and demonstrates analgesic, anti-inflammatory, and antidepressant properties, with low psychotomimetic activity.</p>
    Formula:C22H25ClN2O2
    Color and Shape:Solid
    Molecular weight:384.9

    Ref: TM-T205604