Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(92 products)
- Adiponectin receptor(5 products)
- CFTR(66 products)
- CGRP Receptor(55 products)
- Calcium Channel(578 products)
- Chloride channel(53 products)
- GABA Receptor(367 products)
- Monoamine Transporter(30 products)
- Monocarboxylate transporter(18 products)
- NKCC(2 products)
- NPC1L1(1 products)
- Na-K-Cl cotransporter(9 products)
- OAT(31 products)
- OCT(7 products)
- P-gp(56 products)
- Potassium Channel(318 products)
- Proton pump(42 products)
- SGLT(32 products)
- Sodium Channel(273 products)
- TRP/TRPV Channel(97 products)
Show 13 more subcategories
Found 2691 products for "Membrane Transporter/Ion Channel".
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1-EBIO
CAS:1-EBIO (1-EBIO) is a calium channel agonist.Formula:C9H10N2OPurity:98.75% - 99.96%Color and Shape:SolidMolecular weight:162.19Baclofen
CAS:Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.Formula:C10H12ClNO2Purity:98% - 99.94%Color and Shape:White SolidMolecular weight:213.66γ-DGG acetate(6729-55-1 free base)
CAS:gamma-DGG acetate(6729-55-1 free base) (γ-D-Glutamylglycine) is a competitive blocker of AMPA receptor.Formula:C9H16N2O7Purity:99.92%Color and Shape:SolidMolecular weight:264.23Econazole
CAS:Econazole ((±)-Econazol) is an imidazole derivative that is commonly used as a topical antifungal agent.Formula:C18H15Cl3N2OPurity:98.11% - 99.97%Color and Shape:SolidMolecular weight:381.68Bupivacaine hydrochloride
CAS:Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.Formula:C18H28N2O·HClPurity:99.89% - 99.9%Color and Shape:White SolidMolecular weight:324.89NS13001
CAS:NS13001, an oral SK channel modulator, shows promise for SCA2 therapy; EC50: 1.8 µM (SK2), 0.14 µM (SK3).Formula:C17H16ClN7Purity:99.55%Color and Shape:White SolidMolecular weight:353.81MRZ 2-514
CAS:MRZ 2-514 (8-bromo-4,5-dihydroxypyridazino[4,5-b]quinolin-1-one) is a strychnine-insensitive modulatory site of the NMDA receptor (glycineB)antagonist with KiFormula:C11H6BrN3O3Purity:98.45%Color and Shape:SolidMolecular weight:308.09Ref: TM-T12110
1mg92.00€5mg192.00€1mL*10mM (DMSO)212.00€10mg313.00€25mg620.00€50mg1,044.00€100mg1,404.00€Indapamide
CAS:Indapamide (Noranat) is a non-thiazide sulphonamide diuretic compound, generally used in the treatment of hypertension, as well as decompensated cardiac failure.Formula:C16H16ClN3O3SPurity:98.97% - 99.83%Color and Shape:SolidMolecular weight:365.83Lotilaner
CAS:Lotilaner is a parasiticide.Formula:C20H14Cl3F6N3O3SPurity:99.56%Color and Shape:SolidMolecular weight:596.76Ref: TM-T15775
1mg42.00€2mg55.00€5mg89.00€1mL*10mM (DMSO)105.00€10mg137.00€25mg318.00€50mg522.00€100mg835.00€200mg1,125.00€CGP37157
CAS:CGP37157 (7-Chloro-5-(2-chlorophenyl)-1,5-dihydro-4,1-benzothiazepine-2(3H)-one) is a Na+/Ca2+ exchanger inhibitor, inhibits Na+-induced Ca2+ release fromFormula:C15H11Cl2NOSPurity:99.92%Color and Shape:SolidMolecular weight:324.22Endovion
CAS:Endovion (NS3728) is a pharmacological anion channel and an Anoctamin-1 (ANO 1) channel inhibitor. Endovion is also the specific VRAC/VSOAC blocker.Formula:C16H9BrF6N6OPurity:98.51%Color and Shape:SolidMolecular weight:495.18Norverapamil hydrochloride
CAS:Norverapamil HCl, a Verapamil metabolite, blocks L-type calcium channels and inhibits P-gp function.Formula:C26H37ClN2O4Purity:99.47%Color and Shape:SolidMolecular weight:477.04Ref: TM-T16339
1mg34.00€5mg105.00€1mL*10mM (DMSO)110.00€10mg177.00€25mg299.00€50mg447.00€100mg602.00€200mg842.00€Vocacapsaicin hydrochloride
CAS:Vocacapsaicin hydrochloride (CA-008 hydrochloride) is a non-opioid TRPV1 agonist, a raw material for capsaicin, and is used for pain relief.Formula:C26H42ClN3O4Purity:99.66% - 99.80%Color and Shape:SolidMolecular weight:496.08DSP-2230
CAS:DSP-2230 is a selective blocker of Nav1.7/Nav1.8.Formula:C20H20F3N5O2Purity:97.14%Color and Shape:SolidMolecular weight:419.4Ref: TM-T15174
1mg34.00€5mg66.00€1mL*10mM (DMSO)73.00€10mg99.00€25mg205.00€50mg334.00€100mg537.00€200mg762.00€Otilonium bromide
CAS:Otilonium bromide (SP63) , an antimuscarinic, is utilized as a spasmolytic agent.Formula:C29H43BrN2O4Purity:99.78% - 99.88%Color and Shape:SolidMolecular weight:563.57Bemegride
CAS:Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.Formula:C8H13NO2Purity:99.89%Color and Shape:SolidMolecular weight:155.19Gabapentin
CAS:Gabapentin (Neurontin) is an Anti-epileptic Agent.Formula:C9H17NO2Purity:99.55% - 99.91%Color and Shape:White SolidMolecular weight:171.24CRAC intermediate 2
CAS:CRAC intermediate 2 is a intermediate compound for CRAC inhibitor synthesis.Formula:C11H7F6N3Purity:99.69%Color and Shape:SolidMolecular weight:295.18IK1 inhibitor PA-6
CAS:IK1 inhibitor PA-6 (PA-6) is a selective and potent inhibitor of IK1 (KIR2.x ion-channel-carried inward rectifier current)(IC50 of 12-15 nM for human and mouseFormula:C31H32N4O2Purity:98.9%Color and Shape:SolidMolecular weight:492.61Z433927330
CAS:Z433927330 is a potent and selective Aquaporin-7 (AQP7) inhibitor(IC50s of 0.2).Formula:C20H20N4O3Purity:99.64%Color and Shape:SolidMolecular weight:364.4VU6036720
VU6036720 is a potent and selective inhibitor of the isomeric Kir4.1/5.1.VU6036720 inhibits Kir4.1/5.1 activity by decreasing the channel open-circuitFormula:C20H22ClFN4O2SPurity:98.1%Color and Shape:SolidMolecular weight:436.93Cromolyn sodium
CAS:Cromolyn sodium (FPL-670) is a chromone complex that acts by inhibiting the release of chemical mediators from sensitized mast cells.Formula:C23H14Na2O11Purity:99.4% - 99.95%Color and Shape:White SolidMolecular weight:512.33Tolazamide
CAS:Tolazamide (U-17835) is a sulphonylurea hypoglycemic agent with actions and uses similar to those of CHLORPROPAMIDE.Formula:C14H21N3O3SPurity:98% - >99.99%Color and Shape:SolidMolecular weight:311.40Ref: TM-T1333
2mg34.00€5mg50.00€1mL*10mM (DMSO)58.00€10mg66.00€25mg92.00€50mg118.00€100mg152.00€200mg219.00€Mephenesin
CAS:Mephenesin (Cresoxydiol) is a centrally acting muscle relaxant with a short duration of action.Formula:C10H14O3Purity:99.49% - 99.87%Color and Shape:SolidMolecular weight:182.22Cav 2.2 blocker 1
CAS:Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.Formula:C25H29ClN2O2Purity:99.44%Color and Shape:SolidMolecular weight:424.96Ref: TM-T10690
1mg48.00€5mg105.00€1mL*10mM (DMSO)111.00€10mg173.00€25mg323.00€50mg494.00€100mg740.00€200mg973.00€Boc-LRR-AMC TFA
Boc-LRR-AMC TFA is a fluorogenic protease substrate for detecting trypsin-like activity in the 26S proteasome or 20S proteasome core.Formula:C35H53F3N10O9Purity:97.70%Color and Shape:SolidMolecular weight:814.85VU0134992 hydrochloride
CAS:VU0134992 hydrochloride is the first subtype-preferring, orally active and selective blocker of Kir4.1 potassium channel pore(IC50 : 0.97 μM).Formula:C20H32BrClN2O2Purity:>99.99%Color and Shape:SolidMolecular weight:447.84AZD9056 hydrochloride
CAS:AZD9056 hydrochloride is a P2X7 inhibitor，Which plays a significant role in pain-causing diseases and inflammation.Formula:C24H36Cl2N2O2Purity:99.68%Color and Shape:SolidMolecular weight:455.46Nilvadipine
CAS:Nilvadipine (FK235), a calcium channel blocker (CCB), is utilized for treatment of hypertension.Formula:C19H19N3O6Purity:99.86% - 99.93%Color and Shape:SolidMolecular weight:385.37Flumazenil
CAS:Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervousFormula:C15H14FN3O3Purity:99.72% - 99.98%Color and Shape:White SolidMolecular weight:303.29Clevidipine
CAS:Clevidipine (Clevidipine butyrate) is a dihydropyridine L-type calcium channel blocker that is selective for vascular smooth muscle and is indicated for bloodFormula:C21H23Cl2NO6Purity:99.40%Color and Shape:PowderMolecular weight:456.32Devapamil
CAS:Devapamil (Devapamilo) is a phenylalkylamine that blocks L-type calcium currents from the inner side of membrane cells in a use-dependent manner.Formula:C26H36N2O3Purity:99.63%Color and Shape:SolidMolecular weight:424.58Ethaverine hydrochloride
CAS:Ethaverine hydrochloride is a homologue of papaverine and is used as a vasodilator and antispasmodic.Cost-effective and quality-assured.Formula:C24H30ClNO4Purity:99.66% - 99.73%Color and Shape:SolidMolecular weight:431.96Synta66
CAS:Synta66 is a store-operated calcium entry channel Orai inhibitor, and used for the research of neurological disease.Formula:C20H17FN2O3Purity:99.57% - 99.84%Color and Shape:SolidMolecular weight:352.36Ref: TM-T13047
2mg34.00€5mg50.00€1mL*10mM (DMSO)55.00€10mg80.00€25mg147.00€50mg227.00€100mg339.00€200mg482.00€A 438079
CAS:A 438079 is a potent, and selective antagonist of P2X7 receptor (pIC50: 6.9).Formula:C13H9Cl2N5Purity:99.70% - 99.82%Color and Shape:SolidMolecular weight:306.15Praziquantel
CAS:Praziquantel (Droncit) is an anthelmintic that paralyzes worms by increasing calcium in muscle cells, causing tegument damage and immune response.Formula:C19H24N2O2Purity:99.67% - 99.69%Color and Shape:SolidMolecular weight:312.41Pramocaine hydrochloride
CAS:Pramocaine hydrochloride (Pramoxine HCl), a topical anesthetic, is served as an antipruritic.Formula:C17H27NO3·HClPurity:99.15% - 99.61%Color and Shape:SolidMolecular weight:329.86Tetracaine hydrochloride
CAS:Tetracaine HCl (Pontocaine), a potent local anesthetic and antipruritic, is used in eye care and for surface/spinal anesthesia.Formula:C15H25ClN2O2Purity:99.72% - 99.94%Color and Shape:White SolidMolecular weight:300.82Vigabatrin
CAS:Vigabatrin (Sabril), an analogue of gamma-aminobutyric acid, is an irreversible inhibitor of 4-aminobutyrate Transaminase responsible for the catabolism of γ-Formula:C6H11NO2Purity:99.47% - 99.88%Color and Shape:SolidMolecular weight:129.16Acetohexamide
CAS:Acetohexamide (Acetohexamid) is an intermediate-acting, first-generation sulfonylurea with hypoglycemic activity.Formula:C15H20N2O4SPurity:99.01% - 99.19%Color and Shape:White SolidMolecular weight:324.40Phenibut
CAS:Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).Formula:C10H13NO2Purity:99.55%Color and Shape:White SolidMolecular weight:179.22ML418
CAS:ML418 is a potent, selective and CNS penetrating Kir7.1 potassium channel blocker (IC50 = 310 nM), and also potently inhibits Kir6.2/SUR1.Formula:C19H24ClN3O3Purity:99.3%Color and Shape:SolidMolecular weight:377.87Ref: TM-T16110
1mg37.00€5mg79.00€1mL*10mM (DMSO)84.00€10mg111.00€25mg178.00€50mg288.00€100mg414.00€200mg583.00€4-Aminopyridine
CAS:4-Aminopyridine (Dalfampridine) is a nonselective potassium (K+) channel blocker that binds to the cytoplasmic side of the cell membrane.Formula:C5H6N2Purity:91.61%Color and Shape:SolidMolecular weight:94.11BuChE-IN-9
BuChE-IN-9 (compound 22a), an eqBuChE (equine serum-derived butyrylcholinesterase) inhibitor, exhibits potent activity with an IC50 of 173 nM.Formula:C28H34N4O2Color and Shape:SolidMolecular weight:458.6Dofetilide N-oxide
CAS:Dofetilide N-oxide (UK-116856) is a metabolite of dofetilide. Dofetilide can block potassium channels and is a tertiary antiarrhythmic drug.Formula:C19H27N3O6S2Purity:98%Color and Shape:SolidMolecular weight:457.56Prilocaine acetate
Prilocaine acetate, an amino amide compound, functions as a Na/K-ATPase inhibitor, exhibiting neurotoxic effects [1] [2].Formula:C15H24N2O3Color and Shape:SolidMolecular weight:280.36Anticonvulsant agent 8
Anticonvulsant agent 8 (compound D4) is a chemical used in treating epilepsy by inhibiting GABAA currents. In mouse models, its ED50 values are 2.23 mg/kg for the maximal electroshock (MES) test and 24.60 mg/kg for the pentylenetetrazol (PTZ) test.Formula:C15H11N5OColor and Shape:SolidMolecular weight:277.28UCL 1684 dibromide
CAS:apamin-sensitive Ca2+-activated K+ channel (KCa2.1) blockerFormula:C34H30Br2N4Purity:98%Color and Shape:SolidMolecular weight:654.45Tariquidar dimesylate
CAS:Tariquidar, a non-competitive P-glycoprotein inhibitor, may help combat cancer drug resistance.Formula:C80H94N8O25S4Purity:98%Color and Shape:SolidMolecular weight:1695.9PptT-IN-4
PptT-IN-4 (Compound 3a) is a PptT inhibitor exhibiting an IC50 of 0.71 μM.Formula:C17H23N3Purity:98%Color and Shape:SolidMolecular weight:269.38
