GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
Found 336 products of "GABA Receptor"
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Pentetrazol
CAS:<p>Pentylenetetrazol is a GABA(A) receptor antagonist, that displays activity as a central nervous system and respiratory stimulant.</p>Formula:C6H10N4Purity:99.7% - >99.99%Color and Shape:Bitter Taste Aqueous Solutions Neutral To Litmus (Ntp 1992)Molecular weight:138.17Broflanilide
CAS:<p>Broflanilide metabolite desmethyl-broflanilide blocks GABA receptor in dieldrin-resistant insects, inhibiting S. litura at IC50 1.3 nM.</p>Formula:C25H14BrF11N2O2Purity:99.82%Color and Shape:SolidMolecular weight:663.29Phenelzine sulfate
CAS:<p>Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.</p>Formula:C8H14N2O4SPurity:98.38% - 99.83%Color and Shape:SolidMolecular weight:234.27Chlormezanone
CAS:<p>Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.</p>Formula:C11H12ClNO3SPurity:99.89% - >99.99%Color and Shape:Crystals SolidMolecular weight:273.74Emamectin Benzoate
CAS:<p>Emamectin Benzoate (MK-244), by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropods</p>Formula:C56H81NO15Purity:98.68%Color and Shape:SolidMolecular weight:1008.256NEO 376
CAS:<p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>Formula:C20H24ClN3OPurity:99.56%Color and Shape:SolidMolecular weight:357.88Bemegride
CAS:<p>Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.</p>Formula:C8H13NO2Purity:99.89%Color and Shape:Physical Description White Crystalline Solid Sublimes At 212°F And 200 Mm Pressure (Ntp 1992)Molecular weight:155.19Fluxametamide
CAS:<p>Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).</p>Formula:C20H16Cl2F3N3O3Purity:99.49%Color and Shape:SolidMolecular weight:474.26Baclofen
CAS:<p>Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.</p>Formula:C10H12ClNO2Purity:98% - >99.99%Color and Shape:1992)Molecular weight:213.66L-Cycloserine
CAS:<p>L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.</p>Formula:C3H6N2O2Purity:99.45% - 99.92%Color and Shape:Crystals White PowderMolecular weight:102.09GET73
CAS:<p>GET73 (Gamma hydroxybutyric acid analogue) is an negative allosteric modulator of mGluR5.</p>Formula:C13H16F3NO2Purity:99.54%Color and Shape:SolidMolecular weight:275.27FG 7142
CAS:<p>FG 7142 (LSU-65), a benzodiazepine inverse agonist, targets α1 subunit GABAA receptors (EC50=137 nM, Ki=91 nM) and upregulates β-adrenoceptors.</p>Formula:C13H11N3OPurity:98.75%Color and Shape:SolidMolecular weight:225.25Afoxolaner
CAS:<p>Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs.</p>Formula:C26H17ClF9N3O3Purity:99.1% - 99.38%Color and Shape:SolidMolecular weight:625.87Nefiracetam
CAS:<p>Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.</p>Formula:C14H18N2O2Purity:97.37%Color and Shape:White To Off-White Crystalline PowderMolecular weight:246.3Isoguvacine hydrochloride
CAS:<p>Isoguvacine hydrochloride (1,2,3,6-tetrahydro-4-pyridinecarboxylic acid hydrochloride) is a GABA receptor agonist.</p>Formula:C6H10ClNO2Purity:99.59%Color and Shape:SolidMolecular weight:163.6Nikethamide
CAS:<p>Nikethamide is a stimulant which mainly influences the respiratory cycle. Widely known by its former sales name of Coramine, it was used in the mid-twentieth century as a medical countermeasure against tranquilizer overtreatments, before the advent of end</p>Formula:C10H14N2OPurity:99.42%Color and Shape:Followed By A Faint Sensation Of The Warmth (Ntp 1992)Molecular weight:178.23Vigabatrin
CAS:<p>Vigabatrin (Sabril), an analogue of gamma-aminobutyric acid, is an irreversible inhibitor of 4-aminobutyrate Transaminase responsible for the catabolism of γ-</p>Formula:C6H11NO2Purity:99.47% - 99.88%Color and Shape:SolidMolecular weight:129.16Topiramate
CAS:<p>Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.</p>Formula:C12H21NO8SPurity:99.79% - 99.92%Color and Shape:White To Off-White Crystalline PowderMolecular weight:339.363,4,5-Trimethoxycinnamic acid
CAS:<p>3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at the</p>Formula:C12H14O5Purity:98.91%Color and Shape:SolidMolecular weight:238.24Clomethiazole
CAS:<p>Clomethiazole (Distraneurin) is an orally active GABAA agonist and it is an anticonvulsant agent. It has potential for treating convulsive status epilepticus.</p>Formula:C6H8ClNSPurity:99.06%Color and Shape:SolidMolecular weight:161.65γ-Aminobutyric acid
CAS:<p>γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.</p>Formula:C4H9NO2Purity:99.95%Color and Shape:White Or Almost White(According To Quality Test Specification It Can Be White Or Almost White ) Solid PowderMolecular weight:103.12Flumazenil
CAS:<p>Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervous</p>Formula:C15H14FN3O3Purity:99.72% - 99.98%Color and Shape:Less Crystals Colourless CrystalsMolecular weight:303.29Etifoxine hydrochloride
CAS:<p>Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug.</p>Formula:C17H18Cl2N2OPurity:99.36%Color and Shape:SolidMolecular weight:337.24Domperidone EP Impurity A
CAS:<p>Domperidone EP Impurity A is used as pharmaceutical intermediates.</p>Formula:C12H14ClN3OPurity:99.97%Color and Shape:SolidMolecular weight:251.71Oxiracetam
CAS:<p>Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.</p>Formula:C6H10N2O3Purity:99.67%Color and Shape:White Crystalline PowderMolecular weight:158.16Phenibut
CAS:<p>Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).</p>Formula:C10H13NO2Purity:99.55%Color and Shape:SolidMolecular weight:179.22Lotilaner
CAS:<p>Lotilaner is a parasiticide.</p>Formula:C20H14Cl3F6N3O3SPurity:99.56%Color and Shape:SolidMolecular weight:596.76GABAA receptor agent 1
CAS:<p>GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.</p>Formula:C13H8ClN3O2Purity:99.31%Color and Shape:SolidMolecular weight:273.67Pivagabine
CAS:<p>Pivagabine (CXB-722), a 4-aminobutyric acid derivative, modulates GABA, CRF, and crosses the rat blood-brain barrier.</p>Formula:C9H17NO3Purity:99.87%Color and Shape:SolidMolecular weight:187.24LAU159
CAS:<p>LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).</p>Formula:C17H12ClN3O2Purity:98.7% - 99.38%Color and Shape:SolidMolecular weight:325.75Emamectin B1a
CAS:<p>Emamectin B1a can be used in relevant research in the life sciences. Its product number is T37663 and CAS number is 121124-29-6.</p>Formula:C49H75NO13Color and Shape:SolidMolecular weight:886.133Rilmazolam
CAS:<p>Rilmazolam is a triazolobenzodiazepine compound and serves as the active metabolite of Rilmazafone.</p>Formula:C19H15Cl2N5OColor and Shape:SolidMolecular weight:400.26Inaperisone
CAS:<p>Inaperisone: a novel muscle relaxant that indirectly inhibits voiding reflex via brainstem GABAB receptors.</p>Formula:C16H23NOPurity:99.48%Color and Shape:SolidMolecular weight:245.36Imagabalin
CAS:<p>Imagabalin is an active compound used in the study of neurological diseases.</p>Formula:C9H19NO2Color and Shape:SolidMolecular weight:173.253-Aminopropylphosphinic acid
CAS:<p>3-Aminopropylphosphinic acid (3-APPA) is a phosphonic analog of gamma-aminobutyric acid (GABA).</p>Formula:C3H10NO2PColor and Shape:SolidMolecular weight:123.092FGIN-1-43
CAS:<p>FGIN-1-43 is a potent and specific ligand for the mitochondrial DBI receptor.</p>Formula:C28H36Cl2N2OPurity:99.57%Color and Shape:SolidMolecular weight:487.5(Iso)-Atagabalin HCl
CAS:<p>(Iso)-Atagabalin HCl(isomer-Atagabalin HCl) is an alpha -2- delta ligand that can be used to treat non-restorative sleep.</p>Formula:C10H20ClNO2Purity:99.26% - >99.99%Color and Shape:SoildMolecular weight:221.72LU-32-176B
CAS:<p>LU32-176B is a bioactive chemical.</p>Formula:C23H24F2N2O2Color and Shape:SolidMolecular weight:398.45α-Casozepine
CAS:<p>α-Casozepine,Bioactive peptide from milk α-S1 casein. Binds GABA receptors. Anti-anxiety effects.</p>Formula:C60H94N14O16Color and Shape:SolidMolecular weight:1267.47Cinazepam
CAS:<p>Cinazepam is a GABAA receptor partial agonist and a benzodiazepine derivative with anxiolytic and sedative properties. Cinazepam can be utilized in research related to sleep disorders.</p>Formula:C19H14BrClN2O5Color and Shape:SolidMolecular weight:465.68Anticonvulsant agent 9
<p>Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.</p>Formula:C22H24N4O2Color and Shape:SolidMolecular weight:376.45Pyrazolam
CAS:<p>Pyrazolam is a psychoactive benzodiazepine compound serving as a central nervous system depressant. [Pyrazolam] can lead to psychomotor impairment.</p>Formula:C16H12BrN5Color and Shape:SolidMolecular weight:354.2GABAA receptor modulator-4
<p>GABAA receptor modulator-4 (Compound 4) acts as a negative allosteric modulator of the GABAA receptor. It inhibits the peak and steady-state currents mediated by the α1β3γ2 GABAA receptors, with an IC50 of 10 μM for both.</p>Formula:C15H17BrO4SColor and Shape:SolidMolecular weight:373.26TET-13
<p>TET-13 is a positive allosteric modulator of the GABAA receptor with an EC50 of 5.65 μM, which is more potent than Etomidate (EC50: 9.29 μM). It exhibits strong anesthetic effects in both mice and rats, with an ED50 of 0.48 mg/kg in mice and 0.69 mg/kg in rats.</p>Formula:C15H16N2O3SColor and Shape:SolidMolecular weight:304.36Anticonvulsant agent 8
<p>Anticonvulsant agent 8 (compound D4) is a chemical used in treating epilepsy by inhibiting GABAA currents. In mouse models, its ED50 values are 2.23 mg/kg for the maximal electroshock (MES) test and 24.60 mg/kg for the pentylenetetrazol (PTZ) test.</p>Formula:C15H11N5OColor and Shape:SolidMolecular weight:277.28GABAA receptor modulator-3
<p>GABAA receptor modulator-3 (compound 3b) is a positive allosteric modulator (PAM). It inhibits the peak current and steady-state current of α1β3γ2 GABAAR with IC50 values of 671 μM and 64 μM, respectively.</p>Formula:C18H22O2Color and Shape:SolidMolecular weight:270.37α5-GABAA receptor modulator 1
<p>α5-GABAA receptor modulator 1 (Compound A-4) is a selective silent allosteric modulator (SAM) targeting the α5 subunit of GABAA receptors, useful for research into central nervous system (CNS) disorders.</p>Formula:C21H20FN3O4Color and Shape:SolidMolecular weight:397.4Guvacine hydrobromide
CAS:<p>Guvacine hydrobromide, an alkaloid derived from the Areca catechu nut, serves as a potent inhibitor of GABA (GABA uptakp) uptake.</p>Formula:C6H10BrNO2Purity:98%Color and Shape:SolidMolecular weight:208.05Riluzole-13C,15N2
CAS:<p>Riluzole-13C,15N2 (PK 26124-13C,15N2) is a 13C and 15N labeled form of Riluzole, a glutamate antagonist with anticonvulsant activity, inhibiting GABA uptake.</p>Formula:CC7H5F3OS15N2Color and Shape:SolidMolecular weight:237.18Brexanolone caprilcerbate
CAS:<p>Brexanolone caprilcerbate is an effective positive allosteric modulator of the GABAA receptor.</p>Formula:C48H78O12Color and Shape:SolidMolecular weight:847.13GABA-A Receptor Ligand-1
<p>GABA-A Receptor Ligand-1 (Compound 4) is a ligand for the GABA-A receptor with a pKi of 7.27. It alleviates mitochondrial dysfunction, promotes neurite outgrowth and neuronal regeneration, and demonstrates neuroprotective effects in a rat ischemic stroke model.</p>Formula:C20H20FN3OColor and Shape:SolidMolecular weight:337.391RuBi-GABA
CAS:<p>Ruthenium-bipyridine-triphenylphosphine caged GABA</p>Formula:C42H39F6N5O2P2RuPurity:98%Color and Shape:SolidMolecular weight:922.8AHN-683
CAS:<p>AHN-683 is a fluorescent ligand. It was used for peripheral-type benzodiazepine receptors.</p>Formula:C42H32FN3O7Purity:98%Color and Shape:SolidMolecular weight:709.72Withasomniferolide B
CAS:<p>Withasomniferolide B, a withanolide from Withania somnifera root, activates GABAA receptors.</p>Formula:C28H36O4Color and Shape:SolidMolecular weight:436.58Antidepressant agent 4
<p>Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.</p>Formula:C19H38ClN5O2SColor and Shape:SolidMolecular weight:436.06Anisatin
<p>Anisatin is a useful organic compound for research related to life sciences and the catalog number is T124719.</p>Formula:C15H20O8Color and Shape:SolidMolecular weight:328.317Nitrazolam
CAS:<p>Nitrazolam is a benzodiazepine compound that may exhibit central nervous system depressant properties similar to traditional benzodiazepine drugs by acting on the GABA receptors (GABA receptor). These effects include sedation, hypnosis, anxiolytic, and anticonvulsant activities.</p>Formula:C17H13N5O2Color and Shape:SolidMolecular weight:319.323-Hydroxy desalkylflurazepam
CAS:<p>3-Hydroxy desalkylflurazepam is a benzodiazepine compound with potential sedative and anxiolytic effects.</p>Formula:C15H10ClFN2O2Color and Shape:SolidMolecular weight:304.7(1S,3R)-3-Aminocyclopentane carboxylic acid
CAS:<p>(1S,3R)-3-Aminocyclopentane carboxylic acid exhibits activity on GABAA receptors.</p>Formula:C6H11NO2Color and Shape:SolidMolecular weight:129.16Lesogaberan napadisylate
CAS:<p>Lesogaberan (AZD-3355) is a selective GABAB agonist with EC50 of 8.6 nM, Ki of 5.1 nM in rats, and acts peripherally on the esophageal sphincter.</p>Formula:C13H17FNO5PSColor and Shape:SolidMolecular weight:349.31epi-Aszonalenin A
CAS:<p>epi-Aszonalenin A: a psychoactive benzodiazepine from Aspergillus novofumigatus.</p>Formula:C25H25N3O3Color and Shape:SolidMolecular weight:415.48DAA-1106
CAS:<p>DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective agonist at the peripheral benzodiazepine receptor.</p>Formula:C23H22FNO4Purity:99.54%Color and Shape:SolidMolecular weight:395.426,7-dimethylisatin
CAS:<p>6,7-Dimethylisatin (6,7-dimethyl-1H-indole-2,3-dione) inhibits hGAT3 with IC50 of 108 μM. 6,7-Dimethylisatin also inhibits hBGT1, hGAT2.</p>Formula:C10H9NO2Purity:98.98%Color and Shape:SolidMolecular weight:175.18Azocarnil
<p>Azocarnil is a GABAergic agonist-enhancer used in neurological system research.</p>Color and Shape:Odour SolidEndosulfan I
CAS:<p>Endosulfan I is one of the two major stereoisomers of the broad-spectrum insecticide Endosulfan inhibi the GABA/benzodiazepine/picrotoxin complex</p>Formula:C9H6Cl6O3SPurity:99.86%Color and Shape:SolidMolecular weight:406.93MIDD0301
CAS:<p>MIDD0301 is a potent positive allosteric α5β3γ selective GABAA receptor (GABAAR) ligand with EC50 of 17 nM.</p>Formula:C19H13BrFN3O2Purity:98%Color and Shape:SolidMolecular weight:414.23Desalkylgidazepam
CAS:<p>Desalkylgidazepam, a benzodiazepine compound, is a metabolite of gidazepam. It is capable of activating both GABA A-type receptors and the translocator protein (TSPO).</p>Formula:C15H11BrN2OColor and Shape:SolidMolecular weight:315.17Neurotransmitter Receptor Compound Library
<p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>Color and Shape:Odour SolidNipecotic acid
CAS:<p>Compound PDK0243, with CAS No. 498-95-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0243 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Formula:C6H11NO2Color and Shape:Off-White To Pale Yellow-Beige PowderMolecular weight:129.16CGP 35348
CAS:<p>CGP 35348 是 GABAB 受体的选择性拮抗剂 (EC50 = 34 μM)。 CGP 35348 可用于研究白化新生小鼠脑损伤后的神经肌肉协调和空间学习。</p>Formula:C8H20NO4PPurity:≥98%Color and Shape:SolidMolecular weight:225.22Furosemide
CAS:<p>Furosemide is a potent NKCC2 (Na-K-2Cl symporter) inhibitor, used for edema and chronic renal insufficiency.</p>Formula:C12H11ClN2O5SPurity:99.32% - 99.89%Color and Shape:Crystals From Aqueous Ethanol Tasteless (Ntp 1992)Molecular weight:330.744Ion Channel Targeted Library
<p>A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;</p>Color and Shape:Odour Solid12,14-Dichlorodehydroabietic acid
CAS:<p>12,14-Dichlorodehydroabietic acid activates BK channels, blocks GABA A receptors, and increases calcium and neurotransmitter release.</p>Formula:C20H26Cl2O2Color and Shape:SolidMolecular weight:369.33Flufiprole
CAS:<p>Flufiprole is used as a phenylpyrazole pesticide. It has enantioselective metabolism in human and rat liver microsomes.</p>Formula:C16H10Cl2F6N4OSColor and Shape:SolidMolecular weight:491.24Fipronil sulfone
CAS:<p>Fipronil sulfone is an insecticide fipronil. Its metabolite fipronil sulphone is an inhibitor of rat ɑ1β2γ2L GABA(A) receptor.</p>Formula:C12H4Cl2F6N4O2SPurity:98%Color and Shape:SolidMolecular weight:453.14Chrodrimanin B
CAS:<p>Chrodrimanin B is a useful organic compound for research related to life sciences. The catalog number is T126052 and the CAS number is 132196-54-4.</p>Formula:C27H32O8Color and Shape:SolidMolecular weight:484.545Furosemide sodium
CAS:<p>Furosemide sodium: potent NKCC inhibitor, loop diuretic, treats heart failure, hypertension, edema, selective GABAA antagonist.</p>Formula:C12H10ClN2NaO5SPurity:99.52% - >99.99%Color and Shape:SolidMolecular weight:352.73Antidepressant agent 3
<p>Agent 3: orally active, antidepressant, anxiolytic, boosts performance and cognition.</p>Formula:C17H30ClN5O2SColor and Shape:SolidMolecular weight:403.97GABA receptor Antagonist 1
<p>GABA receptor Antagonist 1 (compound 7w) effectively inhibits the Px RDL1 GABAR at an IC50 of 7.08 nmol/L and demonstrates insecticidal efficacy against P.</p>Purity:98%Color and Shape:Odour SolidAtagabalin
CAS:<p>Atagabalin (PD 0200390), a gabamimetic for insomnia treatment and related to gabapentin, was halted due to poor trial outcomes.</p>Formula:C10H19NO2Color and Shape:SolidMolecular weight:185.263-Aminopropylphosphonic Acid
CAS:<p>3-aminopropylphosphonic acid (3-APPA) is a phosphonic analog of GABA that acts as a partial agonist of GABAB receptors (IC50 = 1.5 μM in a radioligand binding</p>Formula:C3H10NO3PPurity:99.84%Color and Shape:Light Yellow LiquidMolecular weight:139.09Etifoxine
CAS:<p>Etifoxine targets β2/β3 GABAA receptors, is anxiolytic in humans/rodents, boosts GABAA, binds TSPO, aids axon regeneration, no sedative effects.</p>Formula:C17H17ClN2OPurity:98%Color and Shape:SolidMolecular weight:300.78L-655708
CAS:<p>L-655708 is a selective and highly potent GABAA receptor reverse agonist with a Ki value of 0.45 nM.</p>Formula:C18H19N3O4Purity:98.41%Color and Shape:PowderMolecular weight:341.36Padsevonil
CAS:<p>Padsevonil (UCB-0942) is a potential GABA A receptor orthosteric modulator with antiepileptic activity for the treatment of epilepsy.</p>Formula:C14H14ClF5N4O2SPurity:99.63%Color and Shape:SolidMolecular weight:432.80MRK-016
CAS:<p>MRK-016 is a selective GABAA α5 receptor inverse agonist/ negative allosteric modulator, orally available and penetrating the BBB. MRK-016 is antidepressant.</p>Formula:C17H20N8O2Purity:99.76%Color and Shape:SolidMolecular weight:368.39TACA
CAS:<p>GABAA agonist</p>Formula:C4H7NO2Purity:98%Color and Shape:White SolidMolecular weight:101.1CGP 36742
CAS:<p>CGP 36742 blocks GABAB receptor, crosses blood-brain barrier, aids depression treatment (IC50: 32 μM).</p>Formula:C7H18NO2PColor and Shape:SolidMolecular weight:179.2Vigabatrin Hydrochloride
CAS:<p>Vigabatrin Hydrochloride (γ-Vinyl-GABA hydrochloride) is a structural analog of the GABA, irreversibly inhibiting the catabolism of GABA by GABA transaminase.</p>Formula:C6H11NO2·HClPurity:98%Color and Shape:SolidMolecular weight:165.62Furosemide-d5
CAS:<p>Furosemide-d5 is a deuterium marker for Furosemide and used in isotope tracer experiments. orally active inhibitor of Na+/K+/2Cl- (NKCC) diuretic reagent.</p>Formula:C12H11ClN2O5SColor and Shape:SolidMolecular weight:335.78(-)-α-Pinene
CAS:<p>(-)-α-Pinene ((1S)-(-)-Alpha-Pinene) enhances the quantity of NREMS without affecting the intensity of NREMS by prolonging GABAergic synaptic transmission,</p>Formula:C10H16Purity:98.02% - 98.60%Color and Shape:Colourless LiquidMolecular weight:136.23Valnoctamide
CAS:<p>Valnoctamide (Valmethamide) has antiepileptic and anticonvulsant activity and may be used in the study of neurological disorders.</p>Formula:C8H17NOPurity:98%Color and Shape:SolidMolecular weight:143.23Dipropofol
CAS:<p>Dipropofol (4,4-Bis(2,6-di-isopropylphenol)) is a small molecule GABAA receptor agonist that can be used to study epilepsy.</p>Formula:C24H34O2Purity:99.51%Color and Shape:SolidMolecular weight:354.53Propanidid
CAS:<p>Propanidid (Sombrevin) is a gamma-aminobutyric acid type A receptor (GABAA) agonist and an intravenous anesthetic that lowers arterial blood pressure.</p>Formula:C18H27NO5Purity:99.64%Color and Shape:SolidMolecular weight:337.41p-Hydroxybenzaldehyde
CAS:<p>1.</p>Formula:C7H6O2Purity:99.05% - 99.86%Color and Shape:SolidMolecular weight:122.12(R)-baclofen
CAS:<p>(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.</p>Formula:C10H12ClNO2Purity:97.20% - 98.94%Color and Shape:SolidMolecular weight:213.66Ocinaplon
CAS:<p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>Formula:C17H11N5OPurity:99.81%Color and Shape:SolidMolecular weight:301.3Cyclothiazide
CAS:<p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>Formula:C14H16ClN3O4S2Purity:98.23% - 99.49%Color and Shape:Crystals From Dilute Alcohol SolidMolecular weight:389.88Arecaidine hydrochloride
CAS:<p>Arecaidine hydrochloride may have carcinogenesis.</p>Formula:C7H12ClNO2Purity:99.69% - ≥95%Color and Shape:SolidMolecular weight:177.63U93631
CAS:<p>GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.</p>Formula:C17H21N3O2Purity:99.65% - 99.76%Color and Shape:SolidMolecular weight:299.37Pipequaline hydrochloride
CAS:<p>Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.</p>Formula:C22H25ClN2Purity:99.46%Color and Shape:SolidMolecular weight:352.9Fluralaner
CAS:<p>Fluralaner (A1443) is an isoxazoline ectoparasiticide.</p>Formula:C22H17Cl2F6N3O3Purity:99.72% - 99.90%Color and Shape:Solid PowderMolecular weight:556.29L-DABA
CAS:<p>L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).</p>Formula:C4H10N2O2Purity:99.32%Color and Shape:SolidMolecular weight:118.13ONO-8590580
CAS:<p>ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.</p>Formula:C21H21FN6Purity:99.43%Color and Shape:SolidMolecular weight:376.43Kavain
CAS:<p>Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation of</p>Formula:C14H14O3Purity:99.93% - ≥95%Color and Shape:SolidMolecular weight:230.26Isoflurane
CAS:<p>Isoflurane (Forane) is a stable, non-explosive inhalation anesthetic that has been reported to induce caspase-3 activation.</p>Formula:C3H2ClF5OPurity:98%Color and Shape:Clear Colorless Liquid LiquidMolecular weight:184.49Ginsenoside Rc
CAS:<p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>Formula:C53H90O22Purity:98.83% - 99.56%Color and Shape:White PowderMolecular weight:1079.272'-O-Methylisoliquiritigenin
CAS:<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Formula:C16H14O4Purity:98.75%Color and Shape:SolidMolecular weight:270.28NS11394
CAS:<p>NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(</p>Formula:C23H19N3OPurity:99.44% - 99.86%Color and Shape:SolidMolecular weight:353.42Afloqualone
CAS:<p>Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.</p>Formula:C16H14FN3OPurity:99.72%Color and Shape:SolidMolecular weight:283.3Songorine
CAS:<p>Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.</p>Formula:C22H31NO3Purity:98% - 99.92%Color and Shape:SolidMolecular weight:357.49Pikamilone
CAS:<p>Pikamilone (Picamilon) is an intelligent medicine.</p>Formula:C10H12N2O3Purity:99.38%Color and Shape:White Crystalline PowderMolecular weight:208.21AZD-6280
CAS:<p>AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.</p>Formula:C20H22N4O3Purity:98.99%Color and Shape:SolidMolecular weight:366.41(-)-Securinine
CAS:<p>(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.</p>Formula:C13H15NO2Purity:99.58% - 99.87%Color and Shape:SolidMolecular weight:217.26Thiocolchicoside
CAS:<p>Thiocolchicoside, a muscle relaxant, has anti-inflammatory and analgesic properties; not for seizure-prone people.</p>Formula:C27H33NO10SPurity:99.11% - 99.39%Color and Shape:SolidMolecular weight:563.62Loreclezole
CAS:<p>Loreclezole is a selective GABAA receptor modulator and acts as a positive allosteric modulator of β2 or β3-subunit-containing receptors.</p>Formula:C10H6Cl3N3Purity:99.78%Color and Shape:SolidMolecular weight:274.53Bicuculline
CAS:<p>Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.</p>Formula:C20H17NO6Purity:98% - 99.99%Color and Shape:Light Yellow PowderMolecular weight:367.35Baclofen hydrochloride
CAS:<p>Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.</p>Formula:C10H13Cl2NO2Purity:99.55%Color and Shape:SolidMolecular weight:250.122γ-Acetylenic GABA
CAS:<p>γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.</p>Formula:C6H9NO2Color and Shape:SolidMolecular weight:127.143Tiagabine hydrochloride
CAS:<p>Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.</p>Formula:C20H25NO2S2·HClPurity:99.09% - 99.77%Color and Shape:White To Off-White SolidMolecular weight:412.01Dihydroergotoxine mesylate
CAS:<p>Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.</p>Formula:C20H29N3O5SPurity:99.39% - ≥95%Color and Shape:SolidMolecular weight:423.536-Methylflavone
CAS:<p>6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.</p>Formula:C16H12O2Purity:99.69%Color and Shape:SolidMolecular weight:236.27Basmisanil
CAS:<p>Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for the</p>Formula:C21H20FN3O5SPurity:99.21% - 99.42%Color and Shape:SolidMolecular weight:445.46Gabazine free base
CAS:<p>Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.</p>Formula:C15H17N3O3Color and Shape:SolidMolecular weight:287.31rac-BHFF
CAS:<p>rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.</p>Formula:C17H21F3O3Purity:99.69% - >99.99%Color and Shape:SolidMolecular weight:330.34Acamprosate calcium
CAS:<p>Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.</p>Formula:C10H20CaN2O8S2Purity:98% - 99.93%Color and Shape:White Odorless Or Nearly Odorless PowderMolecular weight:400.486-Aminonicotinic acid
CAS:<p>6-Aminonicotinic acid is a natural product.</p>Formula:C6H6N2O2Purity:99.94%Color and Shape:SoildMolecular weight:138.1238DL-Menthol
CAS:<p>DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.</p>Formula:C10H20OPurity:99.74%Color and Shape:White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Molecular weight:156.27Lorediplon
CAS:<p>Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.</p>Formula:C20H15FN4O2SPurity:99.12% - 99.19%Color and Shape:SolidMolecular weight:394.42Suritozole
CAS:<p>Suritozole (MDL-26479) is a negative modulator at the gamma-aminobutyric acidA (GABAA) receptor</p>Formula:C10H10FN3SPurity:99.25%Color and Shape:SolidMolecular weight:223.27CL 218872
CAS:<p>CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.</p>Formula:C13H9F3N4Purity:99.92%Color and Shape:SolidMolecular weight:278.23Imidazenil
CAS:<p>Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.</p>Formula:C18H12BrFN4OPurity:98.4%Color and Shape:SolidMolecular weight:399.22(E)-3,4,5-Trimethoxycinnamic acid
CAS:<p>(E)-3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) is a natural product from the roots and rhizomes of Notopterygium incisum.</p>Formula:C12H14O5Purity:99.83%Color and Shape:SolidMolecular weight:238.24CGP52432
CAS:<p>CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).</p>Formula:C15H24Cl2NO4PPurity:98.75%Color and Shape:SolidMolecular weight:384.244-Acetamidobutanoic acid
CAS:<p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>Formula:C6H11NO3Purity:98.51%Color and Shape:SolidMolecular weight:145.16Cholesterol myristate
CAS:<p>Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.</p>Formula:C41H72O2Purity:99.65%Color and Shape:SolidMolecular weight:597.01Guvacine hydrochloride
CAS:<p>Guvacine hydrochloride is an inhibits of GABA uptake (IC50 : 10 μM)</p>Formula:C6H10ClNO2Purity:98.42%Color and Shape:SolidMolecular weight:163.602α-Thujone
CAS:<p>α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.</p>Formula:C10H16OPurity:97.02% - 98.41%Color and Shape:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Molecular weight:152.23(2S)-6-Prenylnaringenin
CAS:<p>(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.</p>Formula:C20H20O5Purity:99.47%Color and Shape:SolidMolecular weight:340.37Piperazine citrate
CAS:<p>Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.</p>Formula:C24H46N6O14Purity:99.8%Color and Shape:Crystals IndicationMolecular weight:642.65(+)-Kavain
CAS:<p>(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.</p>Formula:C14H14O3Purity:97% - ≥95%Color and Shape:White Fine PowderMolecular weight:230.26α-Asarone
CAS:<p>alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.</p>Formula:C12H16O3Purity:99.64% - 99.64%Color and Shape:Monoclinic Needles From Water Monoclinic Needles From WaterMolecular weight:208.25SSD114 HCl
CAS:<p>SSD114 is a novel GABAB receptor positive allosteric modulator.</p>Formula:C18H21ClF3N3OPurity:99.03% - 99.95%Color and Shape:SolidMolecular weight:387.83Loreclezole hydrochloride
CAS:<p>Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.</p>Formula:C10H7Cl4N3Color and Shape:SolidMolecular weight:310.99Temgicoluril
CAS:<p>Temgicoluril (mebikar) acts on GABA Receptor.</p>Formula:C8H14N4O2Purity:99.8%Color and Shape:SolidMolecular weight:198.22Phenibut (hydrochloride)
CAS:<p>Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.</p>Formula:C10H14ClNO2Purity:99.93%Color and Shape:White Crystalline PowderMolecular weight:215.68Saclofen
CAS:<p>Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.</p>Formula:C9H12ClNO3SPurity:99.17%Color and Shape:White Crystalline SolidMolecular weight:249.71AZD7325
CAS:<p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>Formula:C19H19FN4O2Purity:99.83%Color and Shape:SolidMolecular weight:354.38Tiagabine hydrochloride hydrate
CAS:<p>Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.</p>Formula:C20H28ClNO3S2Color and Shape:SolidMolecular weight:430.022'MeO6MF
CAS:<p>2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functional</p>Formula:C17H14O3Purity:99.28% - 99.63%Color and Shape:SolidMolecular weight:266.29Jujuboside A
CAS:<p>Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.</p>Formula:C58H94O26Purity:98% - >99.99%Color and Shape:SolidMolecular weight:1207.35Miltirone
CAS:<p>Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.</p>Formula:C19H22O2Purity:99.22% - 99.66%Color and Shape:SolidMolecular weight:282.38SKF89976A hydrochloride
CAS:<p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>Formula:C22H26ClNO2Purity:98.02%Color and Shape:SolidMolecular weight:371.9Piperazine
CAS:<p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>Formula:C4H10N2Color and Shape:SolidMolecular weight:86.14Ginkgolide A
CAS:<p>Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.</p>Formula:C20H24O9Purity:98.76% - 99.81%Color and Shape:White PowderMolecular weight:408.4Imepitoin
CAS:<p>Imepitoin (AWD 131-138), a new low-affinity partial benzodiazepine receptor agonist, shows potent anticonvulsant and anxiolytic properties in rodent models.</p>Formula:C13H14ClN3O2Purity:99.82%Color and Shape:SolidMolecular weight:279.72Isonipecotic acid
CAS:<p>Isonipecotic acid (4-Piperidinecarboxylic acid) is a heterocyclic compound. Isonipecotic acid mainly characterized as a GABAA receptor partial agonist.</p>Formula:C6H11NO2Purity:99.82%Color and Shape:White To Faint Pink-Beige PowderMolecular weight:129.16Gabazine
CAS:<p>Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)</p>Formula:C15H18BrN3O3Purity:98.51% - 99.24%Color and Shape:SolidMolecular weight:368.23Tiagabine
CAS:<p>Tiagabine (NO050328) is an Anti-epileptic Agent.</p>Formula:C20H25NO2S2Purity:99.25%Color and Shape:White To Off-White Crystalline SolidMolecular weight:375.55Acetoxyvalerensre
CAS:<p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>Formula:C17H24O4Purity:98.22%Color and Shape:SolidMolecular weight:292.37Amentoflavone
CAS:<p>Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.</p>Formula:C30H18O10Purity:98.21% - 99.22%Color and Shape:Odourless Whitish SolidMolecular weight:538.46Aminooxyacetic acid hemihydrochloride
CAS:<p>Aminooxyacetic acid hemihydrochloride (Carboxymethoxylamine Hemihydrochloride) is a malate-aspartate shuttle (MAS) inhibitor which also inhibits the GABA</p>Formula:C2H5NO3·5HClPurity:98.03%Color and Shape:Light Beige Crystalline PowderMolecular weight:109.36-(4-Methoxyphenyl)-3-pyridazinamine
CAS:<p>6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist</p>Formula:C11H11N3OPurity:99.03%Color and Shape:SolidMolecular weight:201.22Fipronil
CAS:<p>Fipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.</p>Formula:C12H4Cl2F6N4OSPurity:97.21%Color and Shape:Solid PowderMolecular weight:437.15Darigabat
CAS:<p>Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.</p>Formula:C22H21FN4O3SPurity:98.42% - 99.29%Color and Shape:SolidMolecular weight:440.49Riluzole
CAS:<p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>Formula:C8H5F3N2OSPurity:99.71% - 99.88%Color and Shape:PowderMolecular weight:234.2CGP 36216 hydrochloride
CAS:<p>CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).</p>Formula:C5H14NO2PPurity:98%Color and Shape:SolidMolecular weight:151.14β-CCB
CAS:<p>benzodiazepine receptor ligand</p>Formula:C16H16N2O2Purity:98%Color and Shape:SolidMolecular weight:268.31NO 711
CAS:<p>NO 711（NNC-711 free acid） is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.</p>Formula:C21H22N2O3Purity:99.70%Color and Shape:SolidMolecular weight:350.41(±)-Homoproline Hydrochloride
CAS:<p>(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can Trust</p>Formula:C6H12ClNO2Purity:99.69%Color and Shape:SolidMolecular weight:165.62CP-457920
CAS:<p>CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.</p>Formula:C18H17N3O3Purity:99.06% - 99.74%Color and Shape:SolidMolecular weight:323.35Ro 41-3290
CAS:<p>Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is an agonist of nonbenzodiazepine partial at the benzodiazepine receptor.</p>Formula:C24H21ClN2O3Purity:98%Color and Shape:SolidMolecular weight:420.89PF-0713
CAS:<p>PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.</p>Formula:C14H22OPurity:98%Color and Shape:SolidMolecular weight:206.32HZ166
CAS:<p>HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.</p>Formula:C21H16N4O2Purity:98%Color and Shape:SolidMolecular weight:356.38Pregabalin arenacarbil
CAS:<p>Pregabalin arenacarbil is a gabamimetic.</p>Formula:C15H27NO6Color and Shape:SolidMolecular weight:317.38NCS-382
CAS:<p>γ-Hydroxybutyric acid antagonist</p>Formula:C13H14O3Purity:98%Color and Shape:SolidMolecular weight:218.25Ro 19-4603
CAS:<p>Benzodiazepine inverse agonist</p>Formula:C15H17N3O3SPurity:98%Color and Shape:SolidMolecular weight:319.38GABAA receptor agent 4
CAS:<p>Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.</p>Formula:C17H24N2OColor and Shape:SolidMolecular weight:272.39mGAT3/4-IN-1
CAS:<p>mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.</p>Formula:C26H31ClN2O2S2Color and Shape:SolidMolecular weight:503.12CGP11952
CAS:<p>CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.</p>Formula:C21H21Cl2N5O2Purity:98%Color and Shape:SolidMolecular weight:446.3317-PA
CAS:<p>17-PA is a GABAA receptor antagonist.</p>Formula:C25H34OPurity:98%Color and Shape:SolidMolecular weight:350.54MK-0343
CAS:<p>MK0343 is an orally bioavailable GABAA receptor subtype-selective partial agonist and is a non-sedating anxiolytic.</p>Formula:C19H17F2N7OPurity:98%Color and Shape:SolidMolecular weight:397.38DS2
CAS:<p>Positive allosteric modulator of δ-subunit containing GABAA receptors</p>Formula:C18H12ClN3OSPurity:98%Color and Shape:SolidMolecular weight:353.83CGS8216
CAS:<p>CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.</p>Formula:C16H11N3OPurity:98.53%Color and Shape:SolidMolecular weight:261.28BHF-177
CAS:<p>BHF-177 is a positive allosteric modulator of the GABAB receptor. BHF-177 reduces self-administration of nicotine in animal studies.</p>Formula:C19H20F3N3Color and Shape:SolidMolecular weight:347.38SKF 97541
CAS:<p>GABAB agonist</p>Formula:C4H12NO2PPurity:98%Color and Shape:SolidMolecular weight:137.12CGP 7930
CAS:<p>Positive allosteric modulator of GABAB receptors</p>Formula:C19H32O2Purity:98%Color and Shape:SolidMolecular weight:292.46TPA-023B
CAS:<p>TPA-023B: oral GABAA α2/α3 agonist (Kis: 0.73/2 nM), α1 antagonist (Ki: 1.8 nM), non-sedating anxiolytic.</p>Formula:C21H15F2N5OPurity:98%Color and Shape:SolidMolecular weight:391.37U-101017
CAS:<p>U-101017 is a partial benzodiazepine receptor and GABAA receptor agonist.</p>Formula:C23H27ClN4O3Purity:98%Color and Shape:SolidMolecular weight:442.94Org 20599
CAS:<p>GABAA receptor agonist</p>Formula:C25H40ClNO3Purity:98%Color and Shape:SolidMolecular weight:438.04SX-3228
CAS:<p>SX-3228 is a selective agonist of benzodiazepine1 (BZ1) receptor(IC50 of 17 nM).</p>Formula:C18H18N4O3Purity:98%Color and Shape:SolidMolecular weight:338.36CGS 20625
CAS:<p>partial agonist for the benzodiazepine binding site of the GABAA receptor</p>Formula:C18H19N3O2Purity:99.61%Color and Shape:SolidMolecular weight:309.362-Hydroxysaclofen
CAS:<p>2-Hydroxysaclofen is a GABAB receptor antagonist.</p>Formula:C9H12ClNO4SPurity:98%Color and Shape:White SolidMolecular weight:265.71Ro15-4513
CAS:<p>Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.</p>Formula:C15H14N6O3Purity:98%Color and Shape:SolidMolecular weight:326.313-Methyl-GABA
CAS:<p>3-Methyl-GABA activates GABA aminotransferase, fits GABAaR, stimulates GAD, and acts as an anticonvulsant.</p>Formula:C20H30N2O10S2Purity:98%Color and Shape:SolidMolecular weight:522.59DS1
CAS:<p>DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.</p>Formula:C18H10Br2ClN3OSColor and Shape:SolidMolecular weight:511.62Cyprodenate
CAS:<p>Cyprodenate (Actebral) is a potent orally active brain-activating agent with appetite-suppressing properties, useful in studying metabolic.</p>Formula:C13H25NO2Color and Shape:SolidMolecular weight:227.34Y 23684
CAS:<p>Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.</p>Formula:C18H13ClN2O2SPurity:98%Color and Shape:SolidMolecular weight:356.83U-7524
CAS:<p>U-7524 (AOAA), an inhibitor of GABA-T and other PLP-dependent enzymes, disrupts the Schiff base linkage, forming oxime complexes.</p>Formula:C2H5NO3Color and Shape:SolidMolecular weight:91.07Ethyl dirazepate
CAS:<p>Ethyl dirazepate has anxiolytic and hypnotic and possibly other characteristic benzodiazepine properties,is a drug which is a benzodiazepine derivative.</p>Formula:C18H14Cl2N2O3Purity:98%Color and Shape:SolidMolecular weight:377.22Arbaclofen placarbil
CAS:<p>Arbaclofen placarbil is a GABA(B) receptor agonist with better ADMET than R-baclofen, reducing postprandial reflux in GERD.</p>Formula:C19H26ClNO6Color and Shape:SolidMolecular weight:399.87
