
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,003 products)
- Adenosine Receptor(247 products)
- Adrenergic Receptor(3,010 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(60 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(215 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(435 products)
- Endothelin Receptor(83 products)
- GNRH Receptor(82 products)
- GPCR19(33 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(190 products)
- Hedgehog/Smoothened(48 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(321 products)
- PAFR(13 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5838 products of "GPCR/G-Protein"
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Chemerin-9 (149-157) TFA
Chemerin-9 (149-157) TFA is a peptide located at positions 149-157 of chemerin-9, acting as a ChemR23/CMKLR1 agonist.Formula:C56H67F3N10O15Purity:99.77%Color and Shape:SolidMolecular weight:1177.18A71378
CAS:A71378 is a high potency, selectivity CCK-A receptors agonist.Formula:C48H62N8O13SPurity:98%Color and Shape:SolidMolecular weight:991.12PF-03382792
CAS:PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.Formula:C23H32FN3O4Purity:99.64%Color and Shape:SolidMolecular weight:433.52PY-60
CAS:<p>PY-60 can effectively activate YAP transcriptional activity against annexin A2 (ANXA2).Cost-effective and quality-assured.</p>Formula:C16H15N3O2SPurity:99.5% - 99.67%Color and Shape:SolidMolecular weight:313.37GLP-1R agonist 29
<p>GLP-1R agonist 29 (Compound 20) is a GLP-1R agonist that induces hGLP-1R-mediated cAMP stimulation with an EC50 of 0.018 nM. It exhibits favorable pharmacokinetic properties and shows good in vivo exposure, with an AUC0-∞,sc of 77688 ng·h/mL.</p>Color and Shape:Odour SolidBradykinin (1-6)
CAS:Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.Formula:C30H45N9O8Purity:98%Color and Shape:SolidMolecular weight:659.73CCR4 antagonist 3 hydrochloride
CAS:Orally active CCR4 antagonist 3 hydrochloride with potent selectivity, IC50s: 22/50 nM; has antitumor properties.Formula:C24H27Cl2N7O·xHClColor and Shape:SolidPlecanatide acetate
CAS:Plecanatide acetate: GC-C receptor agonist, EC50=190 nM (T84 cells), anti-inflammatory in murine colitis.Formula:C67H108N18O28S4Purity:98%Color and Shape:SolidMolecular weight:1741.94THX-B
CAS:THX-B, a potent non-peptidic p75 NTR antagonist, aids in researching diabetic kidney disease and neurodegenerative and inflammatory disorders.Formula:C16H24N6O4Color and Shape:SolidMolecular weight:364.4Substance P (1-9)
CAS:Substance P (1-9), a nonapeptide, slows its own inactivation and stimulates neurons.Formula:C52H77N15O12Purity:98%Color and Shape:SolidMolecular weight:1104.26Imnopitant dihydrochloride
CAS:Imnopitant dihydrochloride is a neurokinin NK1 receptor antagonist [1] .Formula:C28H30Cl2F6N4OColor and Shape:SolidMolecular weight:623.46Lys-γ3-MSH(human)
CAS:Pro-opiomelanocortin (POMC) derived peptide that stimulates lipolysisFormula:C128H193N45O39SPurity:98%Color and Shape:SolidMolecular weight:3018.25Albiglutide fragment TFA
Albiglutide fragment (GLP-1 (7-36) analog) TFA represents a biologically active segment of Albiglutide, resistant to DPP-4 degradation due to its structure as aFormula:C148H224N40O45·xC2HF3O2Color and Shape:SolidAlverine hydrochloride
CAS:<p>Alverine hydrochloride is a parasympatholytic.</p>Formula:C20H28ClNColor and Shape:SolidMolecular weight:317.9[Ala1,3,11,15]-Endothelin
CAS:Selective ETB endothelin receptor agonist (IC50 values are 0.33 and 2200 nM for displacing [125I]-ET-1 from ETB and ETA receptors respectively).Formula:C109H163N25O32SPurity:98%Color and Shape:SolidMolecular weight:2368Vicasinabin
CAS:Vicasinabin: potent CB2 agonist; researches chronic pain, atherosclerosis, bone mass, neuroinflammation.Formula:C15H22N10OColor and Shape:SolidMolecular weight:358.41PACAP (6-38), human, ovine, rat
CAS:<p>PACAP (6-38) in humans, sheep, rats: a strong inhibitor of PACAP 38, outperforms PACAP (6-27) in blocking PACAP-27-induced adenylate cyclase.</p>Formula:C182H300N56O45SPurity:98%Color and Shape:SolidMolecular weight:4024.74Hemokinin 1 (mouse)
CAS:<p>Hemokinin 1 (mouse) is a selective excitogen 1 receptor agonist with a Ki value of 0.175 nM for the human NK1 receptor and 560 nM for the human NK2 receptor.</p>Formula:C61H100N22O15SPurity:98%Color and Shape:White PowderMolecular weight:1413.65Ramelteon metabolite M-II
CAS:Ramelteon M-II binds MT1/MT2 with IC50s: 208/1470 pM; it's the main metabolite and a melatonin receptor agonist.Formula:C16H21NO3Purity:98%Color and Shape:SolidMolecular weight:275.34BIBP3226
CAS:<p>BIBP3226 is a potent and selective antagonist for the Neuropeptide Y receptor Y1 and the neuropeptide FF receptor.</p>Formula:C27H31N5O3Color and Shape:SolidMolecular weight:473.57Metaraminol
CAS:Metaraminol is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.Formula:C9H13NO2Color and Shape:SolidMolecular weight:167.2117-phenoxy trinor Prostaglandin F2α ethyl amide
CAS:Prostaglandin F2α (PGF2α), acting through the FP receptor, causes smooth muscle contraction and exhibits potent luteolytic activity.Formula:C25H37NO5Color and Shape:SolidMolecular weight:431.573Piperulin A
CAS:Piperulin A effectively inhibits platelet-activating factor receptor (PAFR) by specifically blocking its binding to isolated rabbit platelet plasma membranes,Formula:C23H28O6Color and Shape:SolidMolecular weight:400.46Bz-Dab(nbd)-awfpp-nle-NH2
CAS:Bz-Dab(nbd)-ala-trp-phe-pro-pro-nle-NH2 is a fluorescent NK2 antagonist.Formula:C56H65N13O11Color and Shape:SolidMolecular weight:1096.2Gulgafafusp alfa
CAS:Gulgafafusp alfa is a human IgG2κ monoclonal antibody that selectively binds to the glucagon-like peptide 1 receptor (GLP1R) [1].Color and Shape:Liquidd[Leu4,Lys8]-VP
CAS:Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.Formula:C47H67N11O11S2Purity:98%Color and Shape:SolidMolecular weight:1026.2Neuropeptide Y 13-36 (porcine)
CAS:Neuropeptide Y 13-36 (porcine) is a selective neuropeptide Y2 receptor agonist.Formula:C135H209N41O36Color and Shape:SolidMolecular weight:2982.408L-797,591
CAS:L-797,591 is a selective agonist of somatostatin receptor subtype 1.Formula:C38H49N5O2Color and Shape:SolidMolecular weight:607.83GB-110 hydrochloride
GB-110 HCl: potent, nonpeptidic oral PAR2 agonist; triggers Ca2+ release in HT29 cells; EC50 0.28 μM.Formula:C33H49ClN6O5Color and Shape:SolidMolecular weight:645.23Glucagon-like peptide 1 (1-37), human TFA
Human Glucagon-like peptide 1 (1-37) TFA is a potent GLP-1 receptor agonist derived from proglucagon.Formula:C188H276N51F3O61Purity:98%Color and Shape:SolidMolecular weight:4283.5Bodilisant
CAS:Bodilisant: nanomolar-affinity hH3R ligand, derived from piperidine, with BODIPY fluorophore.Formula:C27H34BF2N3OColor and Shape:SolidMolecular weight:465.4Bremelanotide
CAS:<p>Bremelanotide is a synthetic peptide analog of alpha-MSH and is an agonist at melanocortin receptors including the MC3R and MC4R.</p>Formula:C50H68N14O10Purity:98%Color and Shape:White PowderMolecular weight:1025.161a,1b-dihomo Prostaglandin E1
CAS:1a,1b-dihomo Prostaglandin E1 is a class of prostaglandin compounds.Formula:C22H38O5Color and Shape:SolidMolecular weight:382.541Neuropeptide FF
CAS:Endogenous antiopioid peptide and agonist at NPFF1 and NPFF2 receptors (Ki values are 2.82 and 0.21 nM respectively).Formula:C54H76N14O10Purity:98%Color and Shape:SolidMolecular weight:1081.27HTL22562
CAS:HTL22562 is a calcitonin gene-related peptide (CGRP) receptor antagonist for acute treatment of migraine.Formula:C40H49N11O5Color and Shape:SolidMolecular weight:763.904Secretin (33-59), rat TFA
Secretin (33-59), rat (TFA), a 27-aa peptide, stimulates the secretin receptor, increasing pancreas secretion of bicarbonate, enzymes, and K+.Formula:C131H217F3N42O44Color and Shape:SolidMolecular weight:3141.37RGS2-Galpha-q interaction-IN-1
RGS2–Galpha-q interaction-IN-1 (Compound AJ-3) is an inhibitor of the RGS2-Galpha-q interaction. It inhibits the growth of cancer cell lines that express RGS2 and has anti-cell migration properties.Formula:C30H30ClN7O3Color and Shape:SolidMolecular weight:572.06GRL093-22
<p>GRL093-22 is an effective and selective inhibitor of G protein-coupled receptor kinases (GRK), with IC50 values of 60 nM for GRK5 and 40 nM for GRK6. It shows potential for research in heart failure and multiple myeloma.</p>Formula:C33H29FN6O3Color and Shape:SolidMolecular weight:576.62Jmv 167
CAS:Jmv 167 is an antagonist of the Cholecystokinin receptor.Formula:C51H68N8O14SPurity:98%Color and Shape:SolidMolecular weight:1049.21Vatinoxan
CAS:Vatinoxan is a peripheral α2 adrenoreceptor antagonist.Formula:C20H26N4O4SPurity:98%Color and Shape:SolidMolecular weight:418.51Neurokinin B
CAS:<p>NKB, a tachykinin peptide, impacts human functions like gonadotropin-releasing hormone secretion.</p>Formula:C55H79N13O14S2Purity:98%Color and Shape:SolidMolecular weight:1210.42PACAP (1-27), human, ovine, rat
CAS:PACAP (1-27) (the N-terminal fragment of PACAP-38) is a novel neuropeptides originally isolated from bovine hypothalamus, also found in humans and rats.Formula:C142H224N40O39SPurity:98%Color and Shape:SolidMolecular weight:3147.66NI-0701
<p>NI-0701 is a humanized antibody targeting CCL5/RANTES.</p>Purity:95.4% (SDS-PAGE); 99.4% (SEC-HPLC) - 95.4% (SDS-PAGE); 99.4% (SEC-HPLC)Color and Shape:LiquidMolecular weight:145.5kDa[D-Phe12]-Bombesin
CAS:<p>Bombesin receptor antagonist</p>Formula:C74H112N22O18SPurity:98%Color and Shape:SolidMolecular weight:1629.8815(S)-15-methyl Prostaglandin E2
CAS:15(S)-15-methyl PGE2: A stable PGE2 analog; strong antiulcer with double PGE2 affinity; excels PGE1 in uterine contraction.Formula:C21H34O5Color and Shape:SolidMolecular weight:366.49Galanin (1-16), mouse, porcine, rat TFA
Galanin (1-16) agonizes hippocampal receptors; Kd 3 nM. Active on locus coeruleus neurons in mice, pigs, rats.Formula:C80H117F3N20O23Purity:98%Color and Shape:SolidMolecular weight:1783.9JNJ-10181457 (hydrochloride)
CAS:JNJ-10181457 (hydrochloride) is a non-imidazole H3 receptor antagonist that is brain-penetrating and selective, increasing NE and acetylcholine concentrationsFormula:C20H30Cl2N2OColor and Shape:SolidMolecular weight:385.3715-keto Latanoprost
CAS:Latanoprost, a PG analog for ocular pressure, metabolizes into 15-keto latanoprost, a less potent variant reducing intraocular pressure and pupil size.Formula:C26H38O5Color and Shape:SolidMolecular weight:430.58Adenosine 2',5'-diphosphate sodium
CAS:<p>Adenosine 2',5'-diphosphate sodium is a competitive P2Y1 antagonist with non-selective antagonism at recombinant and human platelet P2X1 receptors.</p>Formula:C10H15N5NaO10P2Color and Shape:SolidMolecular weight:450.192[Nle11]-Substance P
CAS:<p>'[Nle11]-Substance P is a gut and brain peptide, resisting methionine oxidation and causing excitatory neural effects.'</p>Formula:C64H100N18O13Purity:98%Color and Shape:SolidMolecular weight:1329.59CCR4 antagonist 3
CAS:Orally active CCR4 antagonist with piperidinyl-azetidine; IC50: 22 nM (calcium flux), 50 nM (CTX); antitumor effects.Formula:C24H27Cl2N7OColor and Shape:SolidMolecular weight:500.43Glucagon receptor antagonists-1
CAS:Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.Formula:C29H34FNO2Purity:98%Color and Shape:SolidMolecular weight:447.58Cetirizine D8 dihydrochloride
CAS:<p>Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.</p>Formula:C21H26Cl2N2O3Purity:98%Color and Shape:SolidMolecular weight:433.4DSP-1053
CAS:Dsp-1053 is a powerful SERT (Ki=1.02 nM) inhibitor with partial 5-HT1A receptor (Ki=5.05 nM) agonizing activity.Formula:C26H32BrNO4Purity:98%Color and Shape:SolidMolecular weight:502.44Methapyrilene hydrochloride
CAS:<p>Methapyrilene hydrochloride is a biochemical.</p>Formula:C14H20ClN3SColor and Shape:Liquid Solution) 5 5 (Ntp 1992)Molecular weight:297.85IRL-1620
CAS:<p>IRL-1620 is an effective and selective agonist of endothelin receptor type B (ETB) (Ki: 16 pM).</p>Formula:C86H117N17O27Purity:98%Color and Shape:SolidMolecular weight:1820.974Prazobind
CAS:<p>Prazobind is a prazosinoid substance that blocks insulin stimulation of IP1 (inositol phosphate) accumulation and is an effective α1 adrenoceptor blocker.</p>Formula:C23H27N5O3Color and Shape:SolidMolecular weight:421.501α-CGRP, rat
CAS:Endogenous neuropeptide, potent vasodilatorFormula:C162H262N50O52S2Purity:98%Color and Shape:SolidMolecular weight:3806.25Avorelin
CAS:Avorelin, a luteinizing hormone releasing hormone (LH-RH) agonist, is used potentially for the treatment of prostate.Formula:C65H85N17O12Purity:98%Color and Shape:SolidMolecular weight:1296.48α-Helical CRF(9-41)
CAS:Corticotropin-releasing factor receptor antagonist (Ki values are 17, 5 and 0.97 at human CRF1, rat CRF2α and mouse CRF2β receptors respectively).Formula:C166H274N46O53S2Purity:98%Color and Shape:SolidMolecular weight:3827GLP-1R Antagonist 1
CAS:<p>GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).</p>Formula:C16H11ClF6N4O2Purity:99.84%Color and Shape:SolidMolecular weight:440.73Calcitonin Gene Related Peptide (CGRP) II, rat
CAS:CGRP II is a potent vasodilator that boosts pancreatic enzyme levels by activating β-cell receptors.Formula:C163H267N51O50S2Purity:98%Color and Shape:SolidMolecular weight:3805.31ACTH (1-14)
CAS:ACTH (1-14) is a pituitary hormone fragment that controls cortisol and androgen levels.Formula:C77H109N21O20SPurity:98%Color and Shape:SolidMolecular weight:1680.88β-CGRP, human
CAS:<p>β-CGRP, human ,a 37-amino acid peptide,is the beta form of Calcitonin-gene-related peptide (β-CGRP), involved extensively in regulation of the cardiovascular</p>Formula:C162H267N51O48S3Purity:98%Color and Shape:SolidMolecular weight:3793.4117-phenyl trinor Prostaglandin F2α cyclopropyl amide
CAS:<p>17-phenyl trinor Prostaglandin F2α cyclopropyl amide (17-phenyl trinor PGF2α cyclopropyl amide) is a novel analog of 17-phenyl trinor PGF2α ethyl amide.</p>Formula:C26H37NO4Color and Shape:SolidMolecular weight:427.585(3R,5R,6S)-Atogepant
(3R,5R,6S)-Atogepant (MK-8031) is a CGRP antagonist enantiomer used in migraine research.Formula:C29H23F6N5O3Color and Shape:SolidMolecular weight:603.52Apelin-36(rat, mouse)
CAS:Endogenous APJ agonist from adipocytes; binds APJ tightly, inhibits cAMP, regulates heart function and fluid balance, blocks some HIV strains.Formula:C185H304N68O43SPurity:98%Color and Shape:SolidMolecular weight:4200.93Neuropeptide Y (human)
CAS:Neuropeptide Y (29-64), amide, human is a biologically active 36-amino acid peptide.Formula:C189H285N55O57SPurity:98%Color and Shape:SolidMolecular weight:4271.68SR-31747 free base
CAS:SR-31747: immunosuppressive anti-inflammatory agent, inhibits cell growth by blocking sterol isomerase.Formula:C23H34ClNColor and Shape:SolidMolecular weight:359.98BMS-753426
CAS:<p>BMS-753426 is a potent and orally bioavailable antagonist of CCR2 .</p>Formula:C25H33F3N6O2Color and Shape:SolidMolecular weight:506.574Spantide II
CAS:<p>Spantide II is an antagonist of tachykinin.</p>Formula:C86H104Cl2N18O13Purity:98%Color and Shape:SolidMolecular weight:1668.77Somatostatin-28 (1-14)
CAS:Somatostatin-28 (1-14) is a truncated neuropeptide from prosomatostatin cleavage.Formula:C61H105N23O21SPurity:98%Color and Shape:SolidMolecular weight:1528.71Khusimol
CAS:Khusimol is a vasopressin V1a receptors non-peptide ligand that acts by inhibiting the binding of vasopressin.Formula:C15H24OPurity:98%Color and Shape:SolidMolecular weight:220.35Nebentan
CAS:<p>Nebentan (YM598) is an oral, selective ETA antagonist; Ki: 0.697 nM (ETA), 569 nM (ETB); may slow cor pulmonale, myocardial infarction.</p>Formula:C24H21N5O5SColor and Shape:SolidMolecular weight:491.5217-phenyl trinor Prostaglandin F2α cyclopropyl methyl amide
CAS:Prostaglandin F2α (PGF2α) activates the FP receptor, promoting smooth muscle contraction and luteolysis.Formula:C27H39NO4Color and Shape:SolidMolecular weight:441.612Antisauvagine-30
CAS:<p>CRF2 receptor antagonist; Kd 1.4 nM (mCRF2β), 153.6 nM (rCRF1). Blocks sauvagine-induced cAMP in cells & stress-related responses in mice.</p>Formula:C161H274N48O46SPurity:98%Color and Shape:SolidMolecular weight:3650.29Amylin (8-37), rat
CAS:Amylin (8-37), rat, an analog of IAPP, blocks insulin's effects on muscle glucose uptake and glycogen storage.Formula:C140H227N43O43Purity:98%Color and Shape:SolidMolecular weight:3200.61(S, R)-LSN 3318839
CAS:(S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.Formula:C26H23Cl2N3O2Purity:99.57%Color and Shape:SoildMolecular weight:480.39LU AA33810
CAS:<p>LU AA33810 is a neuropeptide Y (NPY) Y5 receptor antagonist.</p>Formula:C19H25N3O2S3Purity:98%Color and Shape:SolidMolecular weight:423.62{Val1}-Exendin-3/4
{Val1}- exendin-3/4 is the first n-terminal 1-28 residue of exendin-4 peptide.Formula:NAPurity:98%Color and Shape:SolidMolecular weight:3241.7Losulazine
CAS:<p>Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.</p>Formula:C27H22F4N4O3SPurity:98.83%Color and Shape:SolidMolecular weight:558.5516-phenoxy tetranor Prostaglandin F2α methyl ester
CAS:<p>Prostaglandin F2α (PGF2α) drives luteolysis and smooth muscle contraction by activating the FP receptor.</p>Formula:C23H32O6Color and Shape:SolidMolecular weight:404.503Bertilimumab
CAS:<p>Bertilimumab (CAT 213; iCo-008), a human monoclonal antibody that targets eotaxin-1 (CCL11), shows promise in the research of allergic disorders [1].</p>Color and Shape:LiquidSC-53116
CAS:SC-53116 HCl can increase the production of serotonin in central nervous system tissues and is a psychoactive agent.Formula:C16H22ClN3O2Color and Shape:SolidMolecular weight:323.82CAY10606
CAS:<p>CAY10606 has a wide range of applications in life science related research.</p>Formula:C22H18ClNO3Color and Shape:SolidMolecular weight:379.84Cloprostenol isopropyl ester
CAS:(+)-Chloprostol is a PGF2α agonist, mimics prostaglandin F2α, induces luteal dissolution in mares without side effects or stress.Formula:C25H35ClO6Color and Shape:SolidMolecular weight:466.99(R)-CJ 11974
CAS:(R)-CJ 11974: non-peptide NK1 receptor antagonist, may relieve pain and prevent chemo-induced vomiting.Formula:C31H38N2OPurity:97.15%Color and Shape:SoildMolecular weight:454.65Preclamol hydrochloride
CAS:Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.Formula:C14H22ClNOColor and Shape:SolidMolecular weight:255.78INCB3344 R-isomer
<p>INCB3344 is a potent CCR2 antagonist. INCB3344 R-isomer is the R-isomer of INCB3344.</p>Formula:C29H34F3N3O6Purity:98%Color and Shape:SolidMolecular weight:577.59I-BOP
CAS:I-BOP is an agonist (KD=0.61 nM) at the thromboxane A2 receptor (TP).Formula:C23H29IO5Color and Shape:SolidMolecular weight:512.384Apelin-36(human)
CAS:Endogenous APJ agonist, EC50=20nM, regulates cardiovascular function, fluid balance, and feeding; blocks certain HIV strains.Formula:C184H297N69O43SPurity:98%Color and Shape:SolidMolecular weight:4195.87CAP-100
CAP-100 is a monoclonal antibody targeting CCR7. It neutralizes the ligand binding site and signaling of CCR7. This compound effectively inhibits migration, extravasation, homing, and survival in chronic lymphocytic leukemia (CLL) samples induced by CCR7. CAP-100 can mediate potent tumor cell killing through host immune mechanisms and exhibits favorable toxicity profiles in related hematopoietic cell subsets. It is involved in research on antitumor activity and diseases like chronic lymphocytic leukemia (CLL).Color and Shape:Odour LiquidNF157
CAS:<p>NF157, a selective P2Y11 antagonist with pKi 7.35, lowers MMP-3/MMP-13, aiding OA treatment; IC50s: P2Y11 463 nM, P2Y1 1811 μM, P2Y2 170 μM.</p>Formula:C49H28F2N6Na6O23S6Purity:98%Color and Shape:SolidMolecular weight:1437.1Dipentylone hydrochloride
CAS:Dipentylone hydrochloride (Bk-dmbdp HCl) is a psychoactive synthetic cathinone and sympathomimetic stimulant. Its inhibitory activity towards the dopamine transporter (IC50=0.233µM) is tenfold higher than that towards NET and SERT, inhibiting dopamine uptake and stimulating locomotor activity in mice.Formula:C14H20ClNO3Purity:99.94%Color and Shape:SolidMolecular weight:285.77AB21 HCl
AB21 HCl: σ1 receptor antagonist, Ki 13 nM; less potent at σ2 (102 nM). Reduces mechanical hypersensitivity.Formula:C23H29ClN2OPurity:99.91%Color and Shape:SolidMolecular weight:384.2CAY10580
CAS:CAY10580 is a potent and selective prostaglandin EP 4 receptor agonist ( K i =35 nM).Formula:C19H35NO4Color and Shape:SolidMolecular weight:341.49GLP-1R agonist 16
CAS:Compound 115a, a GLP-1R agonist, effectively activates the GLP-1 receptor with an EC50 of 0.15 nM [1].Formula:C50H58FN10O6PColor and Shape:SolidMolecular weight:945.03Eletriptan
CAS:<p>Eletriptan, second-generation triptans used to treat migraines, is used as an abortion drug.</p>Formula:C22H26N2O2SColor and Shape:SolidMolecular weight:382.52Hemokinin 1, human
CAS:Endogenous P-like compound, NK1 receptor agonist; IC50: NK1-1.8 nM, NK3-370 nM, NK2-480 nM; boosts B-cell growth, antiapoptotic, lowers blood pressure in vivo.Formula:C54H84N14O14SPurity:98%Color and Shape:SolidMolecular weight:1185.4Ecraprost
CAS:<p>Ecraprost is used as a prodrug of prostaglandin E1.</p>Formula:C28H48O6Color and Shape:SolidMolecular weight:480.68

