GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5838 products of "GPCR/G-Protein"

Purity (%)

100

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26Rfa, Hypothalamic Peptide, human
CAS:
- 600171-68-4
26RFa, a human neuropeptide, stimulates appetite and possibly regulates feeding and the gonadotropic axis, with ≈80% identity across human, rat, and frog.
Formula:C₁₂₇H₁₉₅N₃₇O₃₇
Purity:98%
Color and Shape:Solid
Molecular weight:2832.13
Ref: TM-TP1542
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Pemvidutide TFA
Pemvidutide (TFA), a GLP-1R/GCGR dual agonist, effectively reduces body weight, liver fat, and serum lipid levels, and is utilized in research on non-alcoholic
Formula:C₁₈₂H₂₇₅N₃₉O₅₄·xC₂HF₃O₂
Color and Shape:Solid
Molecular weight:3873.35 (free base)
Ref: TM-T78658
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AD186
AD186, a potent and selective S1R agonist, exhibits dissociation constants (Kis) of 2.7 nM for S1R and 27 nM for S2R.
Formula:C₂₂H₂₈N₂
Purity:98%
Color and Shape:Solid
Molecular weight:320.47
Ref: TM-T78915
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(+)-5-trans Cloprostenol
CAS:
- 57968-81-7
Cloprostenol, a synthetic PGF2α derivative, induces estrus and treats reproductive issues in livestock; its minor impurity, (+)-5-trans, is less effective.
Formula:C₂₂H₂₉ClO₆
Color and Shape:Solid
Molecular weight:424.92
Ref: TM-T37230
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Brain Natriuretic Peptide-45, rat
CAS:
- 123337-89-3
BNP-45 (rat) is a circulating form of rat brain natriuretic peptide isolated from rat heart with potent hypotensive and natriuretic potency.
Formula:C₂₁₃H₃₄₉N₇₁O₆₅S₃
Purity:98%
Color and Shape:Solid
Molecular weight:5040.67
Ref: TM-TP1207
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Ala5-Galanin (2-11)
CAS:
- 859843-84-8
Ala5-Galanin (2-11) is a specific agonist for the galanin receptor 2 (GAL2R) with an affinity constant (Ki) of 258 nM [1].
Formula:C₅₄H₈₁N₁₃O₁₃
Purity:98%
Color and Shape:Solid
Molecular weight:1120.3
Ref: TM-T80517
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15-keto-17-phenyl trinor Prostaglandin F2α ethyl amide
CAS:
- 1163135-96-3
Bimatoprost is the Allergan trade name for 17-phenyl trinor prostaglandin F2α ethyl amide (17-phenyl trinor PGF2α ethyl amide), an F-series PG analog which has
Formula:C₂₅H₃₅NO₄
Color and Shape:Solid
Molecular weight:413.558
Ref: TM-T35944
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Val9-Oxytocin
CAS:
- 1021701-88-1
Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor.
Formula:C₄₆H₇₂N₁₂O₁₂S₂
Purity:98%
Color and Shape:Solid
Molecular weight:1049.27
Ref: TM-T80136
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Ebiratide
CAS:
- 105250-86-0
Ebiratide is an analog of ACTH 4-9.
Formula:C₄₈H₇₃N₁₁O₁₀S
Purity:98%
Color and Shape:Solid
Molecular weight:996.23
Ref: TM-TP2379
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Stressin I TFA
Stressin I (Cyclo(31-34)[DPhe12, Nle21, 38, Glu31, Lys34]Ac-hCRF(4-41)) TFA, with a K i of 1.7 nM, is a potent and selective agonist of the CRF1 receptor.
Purity:98%
Color and Shape:Odour Solid
Ref: TM-T81081
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A3AR agonist 2
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.
Formula:C₃₄H₃₄N₆O₆
Purity:98%
Color and Shape:Solid
Molecular weight:622.67
Ref: TM-T79373
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Synephrine hemitartrate
CAS:
- 16589-24-5
Synephrine hemitartrate, an alkaloid from Citrus aurantium, is a sympathomimetic for weight loss, with α and β-adrenergic action.
Formula:C₉H₁₃NO₂C₄H₆O₆
Color and Shape:Solid
Molecular weight:242.26
Ref: TM-T75425
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Suntinorexton
CAS:
- 2274802-89-8
Suntinorexton (TAK 861) is an orexin type 2 receptor (OX2R) agonist used in the study of neurologic disorders.
Formula:C₂₃H₂₈F₂N₂O₄S
Purity:99.89%
Color and Shape:Solid
Molecular weight:466.54
Ref: TM-T39807
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Semaglutide, FITC labeled
Semaglutide (FITC-labeled Semaglutide) is a long-acting analog of human glucagon-like peptide-1, functioning as an agonist of the GLP-1 receptor. It shows potential for research related to type 2 diabetes.
Formula:C₂₀₉H₃₀₄N₄₆O₆₃S
Molecular weight:4498.17191
Ref: TM-TP3655
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(Des-Bromo)-Neuropeptide B (1-23) (human)
CAS:
- 434897-64-0
'(Des-Bromo)-Neuropeptide B (1-23) (human)' is an agonist for orphan G-protein-coupled receptors, exhibiting a K i of 1.2 nM for GPR7 (NPBW1) and 341 nM for
Formula:C₁₀₇H₁₆₂N₃₀O₃₀
Molecular weight:2348.61
Ref: TM-T83547
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Onvitrelin ucalontide
CAS:
- 1174415-90-7
Onvitrelin ucalontide is a LHRH analogue with anticancer effect; halts breast, ovarian, and prostate tumors in mice.
Formula:C₁₆₃H₂₄₃N₄₃O₃₂
Molecular weight:3316.94
Ref: TM-T76558
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Rp-UTP-α-S tetrasodium
Rp-UTP-α-S (tetrasodium) is a nucleotide agonist of the purinergic P2Y2 and P2Y4 receptors. It can induce the accumulation of inositol phosphate in 1321N1 cells expressing P2Y2 or P2Y4, with EC50 values of 5.4 and 27 μM, respectively.
Color and Shape:Odour Solid
Ref: TM-T212478
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Mapenterol hydrochloride
CAS:
- 54238-51-6
Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.
Formula:C₁₄H₂₁Cl₂F₃N₂O
Purity:98.11% - 99.98%
Color and Shape:Solid
Molecular weight:361.23
Ref: TM-T40622
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SB236057
CAS:
- 180083-49-2
SB236057: potent selective inverse agonist at 5-HT autoreceptors; increases brain 5-HT; teratogen causing musculoskeletal defects in rodents.
Formula:C₃₃H₃₄N₄O₃
Purity:98%
Color and Shape:Solid
Molecular weight:534.65
Ref: TM-T28685
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Vedaprofen
CAS:
- 71109-09-6
Vedaprofen (PM 150) is a COX-1 inhibitor with anti-inflammatory effects, blocking E. coli clamp at IC50 222 μM, Ki 131 μM.
Formula:C₁₉H₂₂O₂
Purity:99.24% - 99.70%
Color and Shape:Solid
Molecular weight:282.38
Ref: TM-T36683
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Guanylin (mouse, rat)
CAS:
- 145257-03-0
Guanylin (mouse, rat), a peptide consisting of 15 amino acids, acts as an activator of intestinal guanylate cyclase and is utilized in diarrhea research [1].
Formula:C₆₀H₉₀N₁₆O₂₂S₄
Purity:98%
Color and Shape:Solid
Molecular weight:1515.71
Ref: TM-T80150
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GEP44
GEP44 is a peptide-biased triple agonist targeting the glucagon-like peptide-1 receptor (GLP-1R), neuropeptide Y1 receptor (Y1-R), and neuropeptide Y2 receptor (Y2-R). It induces GLP-1R-dependent insulin secretion in rat and human islets by offsetting the actions of Y1-R and GLP-1R agonism, controlled by Y1-R antagonists. Additionally, GEP44 enhances glucose uptake in muscle tissue through Y1-R mediation independent of insulin and significantly reduces food intake and body weight in diet-induced obese rat models. GEP44 is utilized in studies related to obesity and type 2 diabetes.
Color and Shape:Odour Solid
Ref: TM-TP3915
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2,3-dinor Thromboxane B1
CAS:
- 196493-76-2
TXB2 released from platelets becomes 11-dehydro and 2,3-dinor TXB2. Rats excrete 2,3-dinor TXB1, a reliable thromboxane biosynthesis marker.
Formula:C₁₈H₃₂O₆
Color and Shape:Solid
Molecular weight:344.448
Ref: TM-T36220
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SR 142948 TFA
SR 142948 TFA is an orally active, selective non-peptide neurotensin receptor (NT) antagonist, displaying IC50 values of 1.19 nM in h-NTR1-CHO cells, 0.32 nM in HT-29 cells, and 3.96 nM in adult rat brain. In HT-29 cells, it counteracts NT-induced inositol monophosphate formation with an IC50 of 3.9 nM. It blocks NT-induced hypothermia, analgesia, and turning behavior in vivo and can cross the blood-brain barrier, making it useful for research in psychiatric disorders.
Color and Shape:Odour Solid
Ref: TM-T211341
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NF546 hydrate
NF546 (hydrate), a selective non-nucleotide P2Y11 agonist, exhibits a pEC50 value of 6.27 and induces interleukin-8 secretion from human monocyte-derived
Formula:C₄₇H₄₄N₆Na₄O₁₇P₄·5H₂O
Purity:98%
Color and Shape:Solid
Molecular weight:1424.01
Ref: TM-T78079
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D3R ligand 1
D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template.
Formula:C₂₇H₃₇NO₅
Purity:98%
Color and Shape:Solid
Molecular weight:455.59
Ref: TM-T78736
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Tamsolusin Hydrochloride
CAS:
- 80223-99-0
Tamsolusin Hydrochloride (YM 12617) is a highly selective alpha-1A adrenergic receptor antagonist used in the treatment of benign prostatic hypertrophy.
Formula:C₂₀H₂₉ClN₂O₅S
Purity:99.92%
Color and Shape:Soild
Molecular weight:444.97
Ref: TM-T83965
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ZM 253270
CAS:
- 169340-04-9
ZM 253270 is an nonpeptide neurokinin A antagonist.
Formula:C₂₂H₂₆ClN₇O₃
Purity:98%
Color and Shape:Solid
Molecular weight:471.95
Ref: TM-T29234
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rGHRH(1-29)NH2
RGHRH (1-29)NH2 is a synthetic peptide that stimulates the secretion of growth hormone (GH).
Formula:C₁₅₅H₂₅₁N₄₉O₄₀S
Purity:98%
Color and Shape:Solid
Molecular weight:3473.02
Ref: TM-TP1393
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c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm
CAS:
- 1647119-71-8
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm: potent, selective V2R agonist; EC50: 0.25 nM (hV2R), 0.05 nM (rV2R).
Formula:C₄₇H₆₉ClN₁₂O₉S₂
Purity:98%
Color and Shape:Solid
Molecular weight:1045.71
Ref: TM-TP1560
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γ-2-MSH (41-58), amide
CAS:
- 799841-81-9
Melanocortin (MC) 3-MSH (Melanocyte-Stimulating Hormone) is believed to signal through the MC 3 receptor.
Formula:C₇₄H₁₀₀N₂₂O₁₅S
Purity:98%
Color and Shape:Solid
Molecular weight:1569.79
Ref: TM-TP1532
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Ornipressin
CAS:
- 3397-23-7
Ornipressin is a vasoconstrictor, haemostatic and renal agent.
Formula:C₄₅H₆₃N₁₃O₁₂S₂
Purity:98%
Color and Shape:White Powder
Molecular weight:1042.19
Ref: TM-TP1049
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SC 45694
CAS:
- 120772-66-9
SC 45694 is a leukotriene B4 (LTB4) analog.
Formula:C₂₂H₃₂LiO₄
Color and Shape:Solid
Molecular weight:367.43
Ref: TM-T34555
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RS 56812
CAS:
- 143137-37-5
RS 56812 is a 5-HT3 receptor antagonist and agonist used in the study of cognitive disorders.
Formula:C₁₈H₂₁N₃O₂
Purity:99.38%
Color and Shape:Soild
Molecular weight:311.38
Ref: TM-T23264L
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Beraprost
CAS:
- 88430-50-6
Beraprost is a stable prostacyclin analog.
Formula:C₂₄H₃₀O₅
Color and Shape:Solid
Molecular weight:398.49
Ref: TM-T30426
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BE-24566B
CAS:
- 149466-04-6
BE-24566B, a polyketide from S. violaceusniger, inhibits various bacteria and blocks ET receptors (ETA IC50=11 μM, ETB=3.9 μM).
Formula:C₂₇H₂₄O₇
Color and Shape:Solid
Molecular weight:460.482
Ref: TM-T38167
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Zenagamtide sodium
Zenagamtide is an agonist for both glucagon-like peptide-1 (GLP-1) and amylin receptors.
Color and Shape:Odour Solid
Ref: TM-TP3862
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Cannabinol methyl ether
CAS:
- 41935-92-6
Cannabinol methyl ether, a phytocannabinoid, serves as an analytical reference standard. This compound can be obtained through isolation from Cannabis plants, derived from cannabinol, or synthesized. The physiological and toxicological properties of cannabinol methyl ether remain unknown. It is designed exclusively for research and forensic applications.
Formula:C₂₂H₂₈O₂
Color and Shape:Solid
Molecular weight:324.5
Ref: TM-TN7267
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CCR6 antagonist 2
CCR6 antagonist2 (Compound 20c) acts as a CCR6 antagonist with a Ki of 1.1 nM. It inhibits CCL20-induced calcium influx with an IC50 of 4.9 nM and suppresses the chemotactic migration of CCR6+ T cells with an IC50 of 190 nM.
Formula:C₁₉H₂₄N₄O₄
Color and Shape:Solid
Molecular weight:372.42
Ref: TM-T205072
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Methimepip dihydrobromide
CAS:
- 817636-54-7
Methimepip dihydrobromide is a selective H3R agonist.
Formula:C₁₀H₁₉Br₂N₃
Color and Shape:Solid
Molecular weight:341.091
Ref: TM-T37727
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Exendin-3/4 (59-86)
Exendin-3/4 (59-86) is a Exendin-4 peptide derivative.
Formula:NA
Purity:98%
Color and Shape:Solid
Molecular weight:3055.49
Ref: TM-TP1366
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PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM for
Formula:C₁₈H₂₀N₅O₇S₂·NH₄·75H₂O
Purity:98%
Color and Shape:Solid
Molecular weight:532.09
Ref: TM-T78084
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CB1R antagonist 2
CB1R antagonist 2 (Compound 11g) functions as an antagonist of the cannabinoid receptor 1 (CB1R), inhibiting the MAPK/NF-κB signaling pathway and exhibiting anti-inflammatory properties. In RAW264.7 cells, it suppresses LPS-induced expression of IL-6, IL-1β, and TNF-α. In murine models, it improves OVA-induced allergic rhinitis.
Formula:C₂₄H₂₆N₄O
Color and Shape:Solid
Molecular weight:386.49
Ref: TM-T205110
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Bimatoprost cyclohexyl amide
Bimatoprostcyclohexyl amide (N-Cyclohexyl-desamethyl bimatoprost; 17-Phenyl trinor prostaglandin F2α cyclohexyl amide) is an analogue of Bimatoprost. This compound acts as an agonist of the prostaglandin F2α receptor (FP receptor) and can be utilized for research in lowering intraocular pressure and in studies of glaucoma.
Color and Shape:Odour Solid
Ref: TM-T211826
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Luprostiol
CAS:
- 67110-79-6
Luprostiol is a prostaglandin analog.
Formula:C₂₁H₂₉ClO₆S
Color and Shape:Solid
Molecular weight:444.97
Ref: TM-T32978
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6β-Prostaglandin I1
CAS:
- 62770-50-7
6β-PGI1 is a stable PGI2 analog resistant to hydrolysis in aqueous solutions.
Formula:C₂₀H₃₄O₅
Color and Shape:Solid
Molecular weight:354.487
Ref: TM-T36239
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Cetamolol hydrochloride
CAS:
- 77590-95-5
Cetamolol hydrochloride is a biochemical.
Formula:C₁₆H₂₇ClN₂O₄
Color and Shape:Solid
Molecular weight:346.85
Ref: TM-T30799
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GPR61 Inverse agonist 1
Compound 1, identified as a GPR61 inverse agonist, exhibits an IC50 of 11 nM, rendering it suitable for metabolism and body weight disorder research, including
Color and Shape:Odour Solid
Ref: TM-T82263
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Quinazosin hydrochloride
CAS:
- 7262-00-2
Quinazosin hydrochloride is an antihypertensive agent.
Formula:C₁₇H₂₅Cl₂N₅O₂
Color and Shape:Solid
Molecular weight:402.32
Ref: TM-T28486
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Astressin
CAS:
- 170809-51-5
Astressin is a truncated CRF analog; binds strongly to receptor's extracellular domain, likely acting as a neutral competitive antagonist.
Formula:C₁₆₁H₂₆₉N₄₉O₄₂
Purity:98%
Color and Shape:Solid
Molecular weight:3563.16
Ref: TM-TP1448
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PACAP-Related Peptide (PRP), human
PRP, human: 29-amino-acid PACAP precursor segment, synthesized for biological/structural research.
Formula:C₁₃₉H₂₂₉N₄₁O₄₂
Purity:98%
Color and Shape:Solid
Molecular weight:3146.57
Ref: TM-TP1850
+ Info
ALD1910
ALD1910 is a humanized monoclonal antibody targeting PACAP38 and PACAP27. It inhibits PACAP signaling through pituitary adenylate cyclase-activating peptide type I receptor (PAC1-R), vasoactive intestinal peptide receptor 1 (VPAC1-R), and VPAC2-R. ALD1910 recognizes a non-linear epitope within PACAP and prevents its binding to cell surfaces. It is useful for studying PACAP-mediated migraines.
Color and Shape:Odour Liquid
Ref: TM-T9901A-1636
+ Info
JPC0323
JPC0323 is a dual positive allosteric modulator of the 5-HT2C and 5-HT2A receptors, featuring on-target properties, acceptable plasma exposure, and adequate
Formula:C₂₂H₄₃NO₄
Purity:98%
Color and Shape:Solid
Molecular weight:385.58
Ref: TM-T79524
+ Info
Human follicular gonadotropin releasing peptide
CAS:
- 107873-08-5
Human Follicular Gonadotropin Releasing Peptide (hF-GRP) is a hormonal peptide that, in vitro, can induce the secretion of pituitary luteinizing hormone (LH)
Formula:C₆₈H₉₄N₂₂O₂₇
Molecular weight:1651.61
Ref: TM-T82162
+ Info
Cholecystokinin Octapeptide, desulfated TFA
CAS:
- 171486-94-5
Cholecystokinin Octapeptide, desulfated TFA, is a synthetic octapeptide derived from Cholecystokinin (CCK) that has undergone desulfation.
Formula:C₅₁H₆₃F₃N₁₀O₁₅S₂
Molecular weight:1177.24
Ref: TM-T39170
+ Info
CMKLR1 antagonist 1
CMKLR1 antagonist 1 (compound S-26d) is a potent, orally active antagonist of the chemokine-like receptor 1 (CMKLR1), exhibiting a pIC50 of 7.44 in hCMKLR1-
Color and Shape:Odour Solid
Ref: TM-T82703
+ Info
Filimelnotide
CAS:
- 2093087-54-6
Filimelnotide is an agonist of the melanocortin receptor.
Formula:C₄₇H₆₉N₁₅O₉S₂
Color and Shape:Solid
Molecular weight:1052.28
Ref: TM-TP3737
+ Info
AM-0466
CAS:
- 1642113-59-4
AM-0466 has a wide range of applications in life science related research.
Formula:C₂₇H₁₉F₃N₄O₄S
Color and Shape:Solid
Molecular weight:552.52
Ref: TM-T71696
+ Info
L803
CAS:
- 348089-28-1
L803 is a selective somatostatin receptor type 4 (SST4) agonist that can inhibit L-type calcium channel currents (ICa). It holds potential for research into degenerative diseases of retinal ganglion cells (RGC), such as glaucoma.
Formula:C₅₀H₈₀N₁₃O₁₉P
Color and Shape:Solid
Molecular weight:1198.22
Ref: TM-TP3907
+ Info
Dp[Tyr(methyl)2,Arg8]-Vasopressin
CAS:
- 67269-08-3
Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].
Formula:C₄₉H₇₀N₁₄O₁₂S₂
Purity:98%
Color and Shape:Solid
Molecular weight:1111.3
Ref: TM-T80073
+ Info
Tiaspirone hydrochloride
CAS:
- 87691-92-7
Tiaspirone hydrochloride (BMY-13859 hydrochloride) exhibits antipsychotic activity and influences the electrophysiological activity of dopaminergic neurons.
Formula:C₂₄H₃₃ClN₄O₂S
Purity:99.87%
Color and Shape:Soild
Molecular weight:477.06
Ref: TM-T24885L
+ Info
4-Thiouridine 5′-triphosphate disodium
CAS:
- 68507-49-3
4-Thiouridine 5′-triphosphate (4-Thio-UTP) tetrasodium functions as a potent agonist at P2Y 2 and P2Y 4 receptors, with half-maximal effective concentrations (
Formula:C₉H₁₁N₂Na₂O₁₄P₃S
Purity:98%
Color and Shape:Solid
Molecular weight:546.19
Ref: TM-T79197
+ Info
5-HT6R antagonist 1
Compound 8 (5-HT6R antagonist 1), a 5-HT6R antagonist (K i : 5 nM), not only demonstrates inhibition of platelet aggregation and excellent metabolic stability
Formula:C₁₇H₂₂F₂N₆O
Purity:98%
Color and Shape:Solid
Molecular weight:364.39
Ref: TM-T79684
+ Info
CB2 PET Radioligand 1
CB2 PET Radioligand 1 (compound [18F]9) is a positron emission tomography (PET) radioligand with high affinity for the human cannabinoid receptor 2 (hCB2, Ki=7.
Formula:C₂₀H₁₉F₃N₄O
Purity:98%
Color and Shape:Solid
Molecular weight:388.39
Ref: TM-T79577
+ Info
BQ-3020 ammonium
BQ-3020 ammonium, a selective endothelin receptor (ET B receptor) agonist, demonstrates inhibition of [125 I] ET-1 binding to ET B receptors with an IC50 of 0.2
Formula:C₉₆H₁₄₀N₂₀O₂₅S·xNH₃
Purity:98%
Color and Shape:Solid
Molecular weight:2006.32 (free base)
Ref: TM-T78096
+ Info
TCMCB07 TFA
TCMCB07 TFA is a cyclic nonapeptide and an orally active, brain-penetrating antagonist of the melanocortin receptor 4 (MC4R), playing a significant role in
Formula:C₆₃H₈₇N₁₅O₁₁·xC₂HF₃O₂
Purity:98%
Color and Shape:Solid
Molecular weight:1230.46 (free base)
Ref: TM-T80541
+ Info
Khusimol
CAS:
- 16223-63-5
Khusimol is a vasopressin V1a receptors non-peptide ligand that acts by inhibiting the binding of vasopressin.
Formula:C₁₅H₂₄O
Purity:98%
Color and Shape:Solid
Molecular weight:220.35
Ref: TM-T25577
+ Info
LCKLSL
CAS:
- 533902-29-3
LCKLSL, an N-terminal hexapeptide, inhibits AnxA2 and tPA binding, reduces plasmin, and exhibits anti-angiogenic effects.
Formula:C₃₀H₅₇N₇O₈S
Molecular weight:675.89
Ref: TM-T40614
+ Info
Anaritide
CAS:
- 95896-08-5
Anaritide, a synthetic form of atrial natriuretic peptide (ANP) composed of 25 amino acids, enhances the glomerular filtration rate by dilating afferent arterioles and constricting efferent arterioles. It is utilized for studying its effects on patients with acute tubular necrosis, with a focus on improving dialysis-free survival rates.
Formula:C₁₁₂H₁₇₅N₃₉O₃₅S₃
Molecular weight:2724.02
Ref: TM-TP2664
+ Info
Ghrelin receptor full agonist-2
CAS:
- 2602452-73-1
Ghrelin receptor full agonist-2 is a highly potent Ghrelin receptor full agonist.
Formula:C₂₆H₂₈ClN₅O₅S
Color and Shape:Solid
Molecular weight:558.05
Ref: TM-T40234
+ Info
Prolactin-Releasing Peptide (1-31), bovine
Prolactin-Releasing Peptide (1-31), bovine, is a fragment of prolactin-releasing peptide (PrRP).
Formula:C₄₄H₈₀N₁₄O₁₅
Molecular weight:1044.59276
Ref: TM-TP3385
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Oxopurpureine
CAS:
- 32845-27-5
Oxopurpureine, classified as an oxoaporphine compound, functions to inhibit plant pathogens.
Formula:C₂₁H₁₉NO₆
Molecular weight:381.38
Ref: TM-T202909
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OXA(17-33)
CAS:
- 343268-91-7
Potent and selective peptide orexin OX1 receptor agonist (EC50 values are 8.29 and 187 nM for OX1 and OX2 receptors respectively). Truncated form of orexin A.
Formula:C₇₉H₁₂₅N₂₃O₂₂
Purity:98%
Color and Shape:Solid
Molecular weight:1749
Ref: TM-TP1973
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CCK (27-33) (non-sulfated)
CAS:
- 47910-79-2
CCK (27-33), a non-sulfated peptide, inhibits [3H]naloxone binding (IC50=4uM) and guinea pig ileum contractions (IC50=17uM), reversed by naloxone.
Formula:C₄₅H₅₇N₉O₁₀S₂
Molecular weight:948.12
Ref: TM-T37206
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(Leu31,Pro34)-Peptide YY (human)
CAS:
- 179986-95-9
(Leu31,Pro34)-Peptide YY (human) is a derivative of Peptide YY, acting as a potent and selective Y1 receptor agonist with a dissociation constant (KD) of 1.0 nM
Formula:C₁₉₅H₂₉₆N₅₄O₅₆
Molecular weight:4292.75
Ref: TM-T76442
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[D-Phe2,6, Pro3]-LH-RH
CAS:
- 64789-67-9
[D-Phe2,6, Pro3]-LH-RH is a potent antagonist of luteinizing hormone-releasing hormone (LHRH).
Formula:C₅₉H₈₀N₁₄O₁₃
Molecular weight:1193.35
Ref: TM-T83499
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Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP (1-7)-GRF (8-27)
CAS:
- 202463-00-1
Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP(1-7)-GRF(8-27) is a selective antagonist [1] for the vasoactive intestinal peptide 1 (VIP 1) receptor.
Formula:C₁₅₀H₂₄₆N₄₄O₃₈
Molecular weight:3273.83
Ref: TM-T83195
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15(S)-Latanoprost
CAS:
- 145773-22-4
15(S)-Latanoprost, a latanoprost analog with inverted hydroxyl at C-15, has an IC50 of 24 nM and reduces IOP by 1 mmHg at 3 μg.
Formula:C₂₆H₄₀O₅
Color and Shape:Solid
Molecular weight:432.59
Ref: TM-T37931
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Desmethyl Mirtazapine (hydrochloride)
CAS:
- 1188265-41-9
Desmethyl mirtazapine is a metabolite of the antidepressant mirtazapine.1It is formed from mirtazapine by the cytochrome P450 (CYP) isoform CYP3A4.
Formula:C₁₆H₁₈ClN₃
Color and Shape:Solid
Molecular weight:287.79
Ref: TM-T37352
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N,N′-Diferuloylputrescine
CAS:
- 42369-86-8
N,N′-Diferuloylputrescine acts as a pigment inhibitor, showing a 57% reduction in pigmentation.
Formula:C₂₄H₂₈N₂O₆
Purity:98%
Color and Shape:Solid
Molecular weight:440.49
Ref: TM-T79996
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Biotinyl-neuropeptide W-23 (human)
CAS:
- 1815618-09-7
Biotinyl-neuropeptide W-23 (human) is a biotinylated form of neuropeptide W-23 (human), which functions as an agonist for the NPBW1 (GPR7) and NPBW2 (GPR8)
Formula:C₁₂₉H₁₉₇N₃₇O₃₀S₂
Molecular weight:2810.3
Ref: TM-T82862
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DD202-114
CAS:
- 2886728-09-0
DD202-114 is an effective and selective agonist of GLP1R. It promotes the accumulation of cAMP, reduces blood glucose levels, and decreases food intake. Additionally, DD202-114 holds potential for research in type 2 diabetes mellitus (T2DM) and obesity studies.
Formula:C₃₃H₃₅FN₄O₅
Molecular weight:586.65
Ref: TM-T200392
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KB-5492 FA
KB-5492 FA is a selective sigma receptor inhibitor with antiulcerogenic effects.CAS 번호128-52-56-8
Formula:C₂₄H₃₂N₂O₈
Purity:98.12%
Color and Shape:Solid
Molecular weight:476.52
Ref: TM-T62396L
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Men 10208
CAS:
- 129781-07-3
Men 10208 is an antagonist of the neurokinin A receptor.
Formula:C₆₁H₇₅N₁₅O₁₂
Purity:98%
Color and Shape:Solid
Molecular weight:1210.36
Ref: TM-T24447
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hNTS1R agonist-1
Compound 10, an hNTS1R agonist-1, acts as a full agonist with a strong affinity for hNTS1R (K i: 6.9 nM), showing the ability to cross the blood-brain barrier (
Formula:C₃₇H₆₂N₁₀O₉
Purity:98%
Color and Shape:Solid
Molecular weight:790.95
Ref: TM-T78954
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CAY10597
CAS:
- 916046-55-4
PGD2 effects via DP1/CRTH2/DP2 receptors; CAY10597 blocks CRTH2/DP2 (Ki=37nM), R enantiomer stronger (Ki=23-22nM), inhibits eosinophil migration (IC50=40nM).
Formula:C₂₀H₁₄ClFN₂O₅
Color and Shape:Solid
Molecular weight:416.79
Ref: TM-T38365
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Galanin-Like Peptide (porcine)
CAS:
- 245114-96-9
Galanin-Like Peptide (porcine) is a 60 amino acid neuropeptide originally isolated from the porcine hypothalamus.
Formula:C₂₈₁H₄₄₃N₈₁O₇₈
Purity:98%
Color and Shape:Solid
Molecular weight:6204.02
Ref: TM-T80145
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ent-Prostaglandin E2
CAS:
- 65085-69-0
Enzymatic PGE2 is optically pure; radical peroxidation makes it racemic. In oxidative stress, rac-PGE2 forms via 15-E2t-isoprostane.
Formula:C₂₀H₃₂O₅
Color and Shape:Solid
Molecular weight:352.471
Ref: TM-T35991
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17-trifluoromethylphenyl trinor Prostaglandin F2α ethyl amide
CAS:
- 1621369-73-0
Prostaglandin F2α (PGF2α), acting through the FP receptor, causes smooth muscle contraction and exhibits potent luteolytic activity.
Formula:C₂₆H₃₆F₃NO₄
Color and Shape:Solid
Molecular weight:483.572
Ref: TM-T37777
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Nolomirole
CAS:
- 90060-42-7
Nolomirole is a dopamine receptor agonist that reduces symptoms of congestive heart failure caused by monoclinine.
Formula:C₁₉H₂₇NO₄
Color and Shape:Solid
Molecular weight:333.42
Ref: TM-T33711
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GW-328267
CAS:
- 210237-78-8
GW-328267 is an agonist of the adenosine A2 receptor.
Formula:C₂₁H₂₆N₁₀O₄
Color and Shape:Solid
Molecular weight:482.5
Ref: TM-T24120
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AP 811
CAS:
- 124833-45-0
AP 811: Selective NPR3 antagonist, Ki of 0.48 nM, >20,000x selective over NPR1, blocks ANP-induced pump stimulation.
Formula:C₄₆H₆₆N₁₂O₈
Molecular weight:915.11
Ref: TM-T38641
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1,2,3-Trilinoelaidoyl-rac-glycerol
CAS:
- 5188-25-0
1,2,3-Trilinoelaidoyl-glycerol is a TAG with linoelaidic acid; reduces rat serum thromboxane B2, PGF2, and PGE.
Formula:C₅₇H₉₈O₆
Color and Shape:Solid
Molecular weight:879.405
Ref: TM-T37383
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N-Desmethyl Pimavanserin
CAS:
- 639863-77-7
N-Desmethyl Pimavanserin (AC-279) is the active metabolite of Pimavanserin and is used in the treatment of insomnia and other sleep disorders.
Formula:C₂₄H₃₂FN₃O₂
Purity:98.02%
Color and Shape:Solid
Molecular weight:413.53
Ref: TM-T37979
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IRL-1038 TFA
IRL-1038 TFA is an ETB receptor antagonist used in the study of cardiovascular disease.
Formula:C₇₀H₉₃F₃N₁₄O₁₇S₂
Purity:98.79%
Color and Shape:Solid
Molecular weight:1523.7
Ref: TM-TP2262L1
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(R)-Citalopram oxalate
CAS:
- 219861-53-7
(R)-Citalopram oxalate is a weak selective serotonin reuptake inhibitor (SSRI) that antagonises its S-isomer (escitalopram), anticonvulsant and antidepressant
Formula:C₂₂H₂₃FN₂O₅
Purity:99.76%
Color and Shape:White Solid
Molecular weight:414.43
Ref: TM-T6493L
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JMV-1645
CAS:
- 284037-77-0
JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.
Formula:C₄₉H₆₉N₁₃O₁₂S
Purity:98%
Color and Shape:Solid
Molecular weight:1064.23
Ref: TM-T25555
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Azaline
CAS:
- 134457-26-4
Azaline is a gonadorelin antagonist.
Formula:C₇₄H₁₀₆ClN₂₃O₁₂
Purity:98%
Color and Shape:Solid
Molecular weight:1545.26
Ref: TM-T25129
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Metipranolol
CAS:
- 22664-55-7
Metipranolol (Betamann) is a type of β- Adrenergic receptors（ β- A potent antagonist of adrenergic receptor on guinea pig atria β 1- Adrenergic receptors and rat uterus β The 2-adrenergic receptor exhibited the beta blocking potentials (pA2) of 8.3 and 8.4, respectively. It is also a potent substituent in the 3H DHA binding assay, with a ligand concentration of 0.7 nM and a Ki of 39 ± 24 nM.
Formula:C₁₇H₂₇NO₄
Purity:98.37%
Color and Shape:Solid
Molecular weight:309.4
Ref: TM-T8899
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3F6-9G5
3F6-9G5 is a humanized monoclonal antibody targeting AA2AR/Adenosine A2aR, used in neurodegenerative disease research.
Purity:>95%
Color and Shape:Odour Liquid
Ref: TM-T9901A-228