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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5964 products of "GPCR/G-Protein"

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  • Cirazoline (free base)

    CAS:
    Cirazoline: full α1A agonist, partial α1B/D, nonselective α2 antagonist; potential vasoconstrictor.
    Formula:C13H16N2O
    Color and Shape:Solid
    Molecular weight:216.28

    Ref: TM-T69031

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GSK-269984A

    CAS:
    GSK-269984A is an antagonist of Prostaglandin E2 Receptor 1 (EP1) (pIC50: 7.9).
    Formula:C20H14Cl2FNNaO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:429.22

    Ref: TM-T15421

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ZD 7114 hydrochloride

    CAS:
    β3-adrenoceptor agonist
    Formula:C22H31ClN2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.94

    Ref: TM-T23558

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PNU-96415E

    CAS:
    dopamine D4 and serotonergic 5-HT2A receptor antagonist
    Formula:C21H27Cl2FN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:413.36

    Ref: TM-T23170

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Adriforant hydrochloride

    CAS:
    Adriforant hydrochloride is an antagonist of histamine H4 receptor.
    Formula:C13H25Cl3N6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:371.74

    Ref: TM-T12435

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • TMPPAA

    CAS:
    TMPPAA is an allosteric agonist of 5-HT3 receptor.
    Formula:C15H21NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:247.33

    Ref: TM-T28986

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Bambuterol

    CAS:
    long acting beta-adrenoceptor agonist
    Formula:C18H29N3O5
    Purity:98%
    Color and Shape:Off-White Powder
    Molecular weight:367.44

    Ref: TM-T22599

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Landiolol

    CAS:
    Landiolol is used as a highly cardioselective ultra short-acting beta-blocker.
    Formula:C25H39N3O8
    Purity:98%
    Color and Shape:White Crystalline Powder
    Molecular weight:509.59

    Ref: TM-T5028L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SR-31747

    CAS:
    SR-31747 blocks cell proliferation by inhibiting sterol isomerase. SR-31747 is a sigma ligand. It has immunosuppressive and anti-inflammatory properties.
    Formula:C23H35Cl2N
    Purity:98%
    Color and Shape:Solid
    Molecular weight:396.44

    Ref: TM-T16926

    5mg
    873.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
    1mL*10mM (DMSO)
    962.00€
  • NBI-27914 hydrochloride

    CAS:
    corticotropin-releasing factor1 (CRF1) receptor antagonist
    Formula:C18H21Cl5N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:470.65

    Ref: TM-T23057

    10mg
    705.00€
  • Protokylol hydrochloride

    CAS:
    Protokylol hydrochloride is a β-adrenergic agonist and bronchodilator, marketed as Asmetil, Caytine, Palison, Ventaire.
    Formula:C18H22ClNO5
    Color and Shape:Solid
    Molecular weight:367.83

    Ref: TM-T70854

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • UK-9040

    CAS:
    UK-9040 inhibits gastric secretory.
    Formula:C23H31NS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:353.56

    Ref: TM-T29056

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Butaxamine

    CAS:
    Butaxamine is a beta-2 selective adrenergic antagonist used mostly in animal and tissue experiments to characterize BETA-2 adrenergic receptors.
    Formula:C15H25NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:267.36

    Ref: TM-T25186

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (1R,1'S,3'R/1R,1'R,3'S)-L-054,264

    CAS:
    somatostatin sst2 receptor agonist
    Formula:C33H41N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:539.71

    Ref: TM-T22487

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Apricoxib

    CAS:
    Apricoxib: oral NSAID with antiangiogenic, antineoplastic properties; inhibits COX-2, may reduce tumor growth and angiogenesis.
    Formula:C19H20N2O3S
    Color and Shape:Solid
    Molecular weight:356.44

    Ref: TM-T70018

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bifeprunox

    CAS:
    Bifeprunox: potent antipsychotic, partial agonist at D2-like/5-HT1A receptors; treats schizophrenia.
    Formula:C24H23N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:385.46

    Ref: TM-T10542

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Protokylol

    CAS:
    Protokylol is a β-adrenergic receptor agonist.
    Formula:C18H21NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.36

    Ref: TM-T24670

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L 741742 hydrochloride

    CAS:
    L 741742 hydrochloride is a selective, high-affinity human D4 receptor antagonist with good oral bioavailability and brain penetration.
    Formula:C23H26Cl2N2O
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:417.37

    Ref: TM-T22903

    1mg
    136.00€
    5mg
    329.00€
    10mg
    517.00€
    25mg
    947.00€
    50mg
    1,554.00€
    100mg
    2,025.00€
    200mg
    2,740.00€
  • VUF 8430

    CAS:
    VUF 8430 is a selective agonist for the H4 receptor.
    Formula:C4H11N5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:161.23

    Ref: TM-T29146

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bunaprolast

    CAS:
    Bunaprolast (U66858) is a novel and potent leukotriene B4 (LTB4) inhibitor.Bunaprolast exhibits oxidative degradation activity and inhibits lipoxygenase and
    Formula:C17H20O3
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:272.34

    Ref: TM-T17191

    1mg
    630.00€
    5mg
    1,620.00€
  • L-775,606

    CAS:
    L-775,606 is a selective agonist of 5-hydroxytryptamine 1D.
    Formula:C25H29FN6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:432.54

    Ref: TM-T27782

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • VUF 5681 dihydrobromide

    CAS:
    histamine H3 receptor silent antagonist
    Formula:C11H21Br2N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:355.11

    Ref: TM-T23519

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Verlukast

    CAS:
    Verlukast (MK-0679) is a selective, orally active leukotriene D4 receptor antagonist for use in bronchial asthma research.
    Formula:C26H27ClN2O3S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:515.09

    Ref: TM-T19674

    50mg
    723.00€
    100mg
    1,094.00€
  • JNJ-27141491

    CAS:
    JNJ-27141491 is a potent, noncompetitive antagonist of human CCR2.
    Formula:C17H15F2N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:379.38

    Ref: TM-T27674

    25mg
    1,444.00€
  • Metazosin

    CAS:
    Metazosin is an antihypertensive agent that replaces 3H-prazosin from its bond to alpha-1 receptors of the cerebral cortex.
    Formula:C18H25N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:375.42

    Ref: TM-T25793

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LY 203647

    CAS:
    LY 203647 is a antagonist of leukotriene D4 and E4 receptor.
    Formula:C21H30N8O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:442.51

    Ref: TM-T27893

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A 61603

    CAS:
    Cixutumumab (IMC-A12) is a humanized IgG monoclonal antibody targeting the IGF1R with anticancer activity.
    Formula:C14H20BrN3O3S
    Color and Shape:Solid
    Molecular weight:390.3

    Ref: TM-T21927

    1mg
    105.00€
    5mg
    325.00€
    10mg
    444.00€
  • DH97

    CAS:
    MT2 melatonin receptor antagonist
    Formula:C22H26N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:334.45

    Ref: TM-T22721

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A68930

    CAS:
    A 68930 is a dopamine D-1 receptor antagonist. A 68930 inhibits NLRP3 inflammasome activity.
    Formula:C16H17NO3
    Color and Shape:Solid
    Molecular weight:271.31

    Ref: TM-T26432

    25mg
    3,492.00€
    50mg
    5,239.00€
    100mg
    7,857.00€
  • LY 225910

    CAS:
    LY 225910 is a CCK2 receptor antagonist.
    Formula:C27H24BrN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:502.4

    Ref: TM-T22941

    10mg
    470.00€
    50mg
    1,918.00€
  • MS 245 oxalate

    CAS:
    MS 245 oxalate is a 5-HT6 antagonist.
    Formula:C21H24N2O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.49

    Ref: TM-T23029

    1mg
    124.00€
    5mg
    462.00€
    10mg
    695.00€
  • CAY10535

    CAS:
    CAY10535 is a selective TPβ antagonist (IC50 = 99 nM for TPβ vs 1970 nM for TPα), weakly affects platelets (IC50 = 985 nM).
    Formula:C18H21N3O7S
    Color and Shape:Solid
    Molecular weight:423.44

    Ref: TM-T36550

    1mg
    118.00€
    5mg
    515.00€
    10mg
    888.00€
    25mg
    1,882.00€
  • N-Salicyloyltryptamine

    CAS:
    N-Salicyloyltryptamine (STP): a tryptamine with anticonvulsant, anti-inflammatory, analgesic effects; inhibits Na+, Ca2+, K+ channels (IC50 34.6 μM).
    Formula:C17H16N2O2
    Color and Shape:Solid
    Molecular weight:280.32

    Ref: TM-T60526

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SB 235375

    CAS:
    SB 235375 is a potent and selective antagonist of neurokinin-3 receptor with a low central nervous system-penetrant.
    Formula:C27H24N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.49

    Ref: TM-T28676

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A1AR antagonist 6

    CAS:
    A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].
    Formula:C17H15N3O2
    Color and Shape:Solid
    Molecular weight:293.32

    Ref: TM-T60615

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SKF-83566 hydrobromide

    CAS:
    D1-like dopamine receptor antagonist
    Formula:C17H19BrClNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:368.7

    Ref: TM-T23362

    5mg
    200.00€
    10mg
    314.00€
    25mg
    620.00€
  • Lu AA41063

    CAS:
    Lu AA41063 is a potent and selective antagonist of the hA2A receptor.
    Formula:C16H17F2N3O2S
    Color and Shape:Solid
    Molecular weight:353.39

    Ref: TM-T24418

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Todralazine

    CAS:
    Todralazine is an anti-hypertensive agent and acts as a β2AR blocker. It also has an antioxidant and free radical scavenging activity.
    Formula:C11H12N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:232.24

    Ref: TM-T17112

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Lexipafant

    CAS:
    Lexipafant is a platelet-activating factor (PAF) receptor antagonist.
    Formula:C23H30N4O4S
    Color and Shape:Solid
    Molecular weight:458.57

    Ref: TM-T27821

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • T 82

    CAS:
    T 82 is an antagonist of 5-HT3 and inhibitor of acetylcholinesterase (AChE) and used for the treatment of Alzheimer's Disease.
    Formula:C56H62N6O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:947.146

    Ref: TM-T13239

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L-670,596

    CAS:
    L-670,596 is a thromboxane A2/prostaglandin endoperoxide receptor antagonist.
    Formula:C22H21F2NO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.47

    Ref: TM-T22897

    100mg
    2,250.00€
  • A2A receptor antagonist 3

    CAS:
    A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM).
    Formula:C26H26N6O2
    Color and Shape:Solid
    Molecular weight:454.52

    Ref: TM-T62797

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • Ro 22-9194

    CAS:
    Ro 22-9194, a class I antiarrhythmic, reduces upstroke velocity and shortens action potential in guinea-pig hearts at ≥10 μM.
    Formula:C19H27Cl2N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:384.35

    Ref: TM-T28567

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Thioperamide

    CAS:
    histamine H3 and H4 antagonist/inverse agonist
    Formula:C15H24N4S
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:292.44

    Ref: TM-T23456

    10mg
    502.00€
    50mg
    2,070.00€
  • (Rac)-Upacicalcet

    CAS:
    (Rac)-Upacicalcet, a racemate, is an IV calcimimetic targeting parathyroid receptors to lower PTH, possibly treating SHPT.
    Formula:C11H14ClN3O6S
    Color and Shape:Solid
    Molecular weight:351.76

    Ref: TM-T61232

    25mg
    1,314.00€
  • BFE-55

    CAS:
    BFE-55 is derivative of befunolol (a beta-adrenergic partial agonist). BFE-55 interacts with only the high affinity sites in beta-adrenoceptors
    Formula:C14H19NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:249.31

    Ref: TM-T26783

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AR-A 2

    CAS:
    AR-A 2, a selective 5-HT1B antagonist; high guinea pig 5-HT1B/1D affinity (Ki: 0.24, 0.47 nM); 10x less for 5-HT1D (Ki: 5 nM).
    Formula:C27H36N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.6

    Ref: TM-T10360

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • NVS-CRF38

    CAS:
    NVS-CRF38 is an antagonist of corticotropin-releasing factor receptor 1 (CRF1).
    Formula:C19H21N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.4

    Ref: TM-T12276

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • SB 206553 hydrochloride

    CAS:
    SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disorders
    Formula:C17H17ClN4O
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:328.8

    Ref: TM-T23314

    1mg
    58.00€
    5mg
    124.00€
    10mg
    192.00€
    25mg
    386.00€
    50mg
    556.00€
  • Levemopamil HCl

    CAS:
    Levemopamil HCl is used as a calcium channel blocker.
    Formula:C23H31ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:370.96

    Ref: TM-T25692L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Alaproclate (hydrochloride)

    CAS:
    Alaproclate, an SSRI, enhances serotonin and SIRT1, hinders NMDA and K+ currents in neurons, and shows antidepressant-like effects in rats.
    Formula:C13H19Cl2NO2
    Color and Shape:Solid
    Molecular weight:292.2

    Ref: TM-T36521

    5mg
    230.00€
    10mg
    399.00€
  • γ-Linolenic acid ethyl ester

    CAS:
    γ-Linolenic acid ethyl ester (Ethyl γ-linolenate) is a leukotriene B 4 receptor 4 (LTB 4 ) antagonist which has a potential anti-inflammatory effect[1].
    Formula:C20H34O2
    Color and Shape:Solid
    Molecular weight:306.48

    Ref: TM-T41235

    1g
    1,288.00€
    50mg
    114.00€
    100mg
    208.00€
    250mg
    489.00€
  • Benzatropine

    CAS:
    Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.
    Formula:C21H25NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:307.43

    Ref: TM-T23781

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (RS)-Butyryltimolol

    CAS:
    (RS)-Butyryltimolol, a racemic prodrug of Timolol, enhances its corneal absorption and acts as a β-adrenergic blocker.
    Formula:C17H30N4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.51

    Ref: TM-T13439

    2mg
    63.00€
  • Remoxipride

    CAS:
    Remoxipride is an antipsychotic agent. Remoxipride is specific for dopamine D2 receptors.
    Formula:C16H23BrN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:371.27

    Ref: TM-T28514

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PF-4479745

    CAS:
    PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.
    Formula:C17H22N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:282.38

    Ref: TM-T28384

    1mg
    427.00€
  • MRS1186

    CAS:
    MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).
    Formula:C16H12ClN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:341.75

    Ref: TM-T16138

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • L-Alprenolol

    CAS:
    L-Alprenolol is a non-selective beta-blocker and a 5-HT1A and 5-HT1B receptor antagonist.
    Formula:C15H23NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:249.35

    Ref: TM-T24386

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Carcinine

    CAS:
    Carcinine ditrifluoroacetate is a H3 receptor antagonist.
    Formula:C8H14N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:182.22

    Ref: TM-T22624

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ro 60-0175 fumarate

    CAS:
    5-HT2 receptor agonist
    Formula:C15H16ClFN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:342.75

    Ref: TM-T23246

    1mg
    105.00€
    5mg
    268.00€
  • MRS2298

    CAS:
    MRS2298, a potent antagonists of the P2Y 1 receptor, has antiaggregatory activity in human platelets.
    Formula:C10H16ClN5O8P2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.66

    Ref: TM-T28100

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MAT2A-IN-1

    CAS:
    MAT2A-IN-1 suppresses MAT2A, key for MTAP-deficient cancer cell growth; studied for gastric, colon, liver, pancreatic cancers.
    Formula:C29H28F2N6O4
    Color and Shape:Solid
    Molecular weight:562.57

    Ref: TM-T63975

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • GW848687X

    CAS:
    GW848687X, a potent and selective prostaglandin EP1 receptor antagonist, is used for the treatment of inflammatory pain.
    Formula:C24H18ClF2NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.85

    Ref: TM-T27517

    1mg
    537.00€
    5mg
    2,277.00€
    500µg
    290.00€
  • GR 196429

    CAS:
    GR 196429: MT1-selective melatonin receptor agonist; induces sleep, alters circadian rhythm, stimulates melatonin in mice.
    Formula:C14H18N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:246.3

    Ref: TM-T27430

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CID1792197

    CAS:
    CID1792197 is a selective agonist of GPR55.
    Formula:C24H23N3O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.59

    Ref: TM-T27017

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Setastine HCl

    CAS:
    Setastine HCl is a potent antagonist of histamine H1-receptor mediated responses.
    Formula:C22H29Cl2NO
    Color and Shape:Solid
    Molecular weight:394.38

    Ref: TM-T71791

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PM226

    CAS:
    CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.
    Formula:C22H31NO3
    Color and Shape:Solid
    Molecular weight:357.49

    Ref: TM-T37815

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L-817,818

    CAS:
    somatostatin sst5 receptor agonist
    Formula:C33H36N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:536.66

    Ref: TM-T22907

    10mg
    1,279.00€
  • TC 1

    CAS:
    σ1 receptor ligand
    Formula:C19H20FNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.37

    Ref: TM-T23423

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • threo Ifenprodil hemitartrate

    CAS:
    σ receptor agonist and NR2B subunit-selective NMDA receptor antagonist
    Formula:C21H27NO2C4H6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:400.49

    Ref: TM-T23457

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Vasopressin V2 receptor antagonist 1

    CAS:
    Vasopressin V2 receptor antagonist 1 (Compound 4g) is a vasopressin V2receptor (V2R) antagonist (Ki: 3.8 nM). dominant polycystic kidney disease (ADPKD).
    Formula:C33H37ClN4O4
    Color and Shape:Solid
    Molecular weight:589.12

    Ref: TM-T64174

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • PA-9

    CAS:
    PA-9 is the first small-molecule PAC1 receptor antagonist.
    Formula:C17H18N6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:338.36

    Ref: TM-T24585

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MRS1177

    CAS:
    MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).
    Formula:C20H12ClN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:389.79

    Ref: TM-T16137

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Vicagrel

    CAS:
    Vicagrel, an oral antiplatelet, boosts aspirin's effect, targeting P2Y12 and fights clots in heart and vessel diseases.
    Formula:C18H18ClNO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:379.86

    Ref: TM-T17231

    2mg
    217.00€
    25mg
    888.00€
    50mg
    1,224.00€
    100mg
    1,674.00€
  • Ibodutant

    CAS:
    Ibodutant is an effective and selective tachykinin NK2 receptor antagonist (pKi: 10.1).
    Formula:C37H48N4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:644.87

    Ref: TM-T16039

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • S20928

    CAS:
    S20928 is an antagonist of melatonin receptor.
    Formula:C17H19NO
    Color and Shape:Solid
    Molecular weight:253.34

    Ref: TM-T28644

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DV 7028 hydrochloride

    CAS:
    DV 7028 hydrochloride is a 5-HT2A receptor antagonist.
    Formula:C21H26ClFN4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:436.91

    Ref: TM-T22753

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • hA2A/hCA XII modulator 1

    CAS:
    Potent hA2AAR antagonist & hCA XII inhibitor; Ki: hA2AAR 6.4 nM, hCA XII 6.2 nM. Possible cancer research use.
    Formula:C24H19N7O4S
    Color and Shape:Solid
    Molecular weight:501.52

    Ref: TM-T63400

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Carbinoxamine

    CAS:
    Carbinoxamine: antihistamine for hay fever, angioedema, rhinitis, mild urticaria, dermatographism, allergic conjunctivitis; an H1-antagonist.
    Formula:C16H19ClN2O
    Purity:98%
    Color and Shape:Liquid
    Molecular weight:290.79

    Ref: TM-T21247

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • EGIS-7625

    CAS:
    EGIS-7625 is a selective and competitive antagonist of 5-HT2B receptor.
    Formula:C18H24Cl2N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.32

    Ref: TM-T27249

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GR-203040 HCl

    CAS:
    GR203040 inhibits cyclophosphamide-induced damage in the rat and ferret bladder. GR-203040 is a selective NK1 receptor antagonist.
    Formula:C20H26Cl2N6O
    Color and Shape:Solid
    Molecular weight:437.37

    Ref: TM-T24102

    25mg
    1,738.00€
  • HEMADO

    CAS:
    HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).
    Formula:C17H23N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:361.4

    Ref: TM-T15468

    1mg
    112.00€
    5mg
    388.00€
  • PF-592379

    CAS:
    PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).
    Formula:C13H21N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:235.33

    Ref: TM-T10080

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Centanafadine

    CAS:
    Centanafadine inhibits NE/DA transporters and serotonin transporter (IC50: NE=6 nM, DA=38 nM, 5-HT=83 nM).
    Formula:C15H15N
    Purity:98%
    Color and Shape:Solid
    Molecular weight:209.29

    Ref: TM-T10758

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • UCSF678

    CAS:
    UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.
    Formula:C15H18N2O2S
    Color and Shape:Solid
    Molecular weight:290.38

    Ref: TM-T60597

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • S(-)-Bisoprolol

    CAS:
    S(-)-Bisoprolol, a β1-blocker, may aid in researching hypertension and heart diseases.
    Formula:C18H31NO4
    Color and Shape:Solid
    Molecular weight:325.44

    Ref: TM-T60901

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Spirendolol

    CAS:
    Spirendolol is an antagonist of β adrenergic receptor.
    Formula:C21H31NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:345.48

    Ref: TM-T16919

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • UP202-56

    CAS:
    UP202-56 is an adenosinergic agonist and is an adenosine analog.
    Formula:C33H37N7O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:595.69

    Ref: TM-T13256

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • A331440

    CAS:
    A331440 is an modulator of L-histidine and histamine H3 receptor.
    Formula:C22H27N3O
    Color and Shape:Solid
    Molecular weight:349.47

    Ref: TM-T26480

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TCS-OX2-29 HCl

    CAS:
    TCS-OX2-29 is a selective orexin-2 receptor antagonist (IC50 = 40 nM), which plays an important role in pain modulation.
    Formula:C23H32ClN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.97

    Ref: TM-T4965L

    5mg
    316.00€
    10mg
    600.00€
    50mg
    2,502.00€
  • (R,R)-Reboxetine mesylate

    CAS:
    (R,R)-Reboxetine mesylate: Antidepressant, high bioavailability, (R,R) enantiomer, selective for noradrenaline, low toxicity.
    Formula:C20H27NO6S
    Color and Shape:Solid
    Molecular weight:409.5

    Ref: TM-T72209

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AZD5213

    CAS:
    AZD5213: selective human H3 receptor antagonist, pKi 9.3, for sleep/cognition research.
    Formula:C19H25N3O2
    Color and Shape:Solid
    Molecular weight:327.42

    Ref: TM-T71423

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PF-06256142

    CAS:
    PF-06256142 is a potent and selective orthosteric D1 receptor agonist(D1 EC50=30 nM ).
    Formula:C21H16N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.38

    Ref: TM-T12423

    25mg
    1,260.00€
    50mg
    1,639.00€
    100mg
    2,250.00€
  • MRS 1334

    CAS:
    antagonist for the human adenosine A3 receptor
    Formula:C31H26N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:522.55

    Ref: TM-T23017

    25mg
    2,232.00€
  • SB357134

    CAS:
    SB357134 is a potent, selective and orally active antagonist of 5-HT6 receptor and shows nootropic effects in animal studies.
    Formula:C17H18Br2FN3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:523.21

    Ref: TM-T28689

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AChE-IN-14

    CAS:
    AChE-IN-14 inhibits eeAChE, hAChE, eqBuChE (IC50: 0.46-0.48 μM) and binds to H3R (Ki: 159.8 nM), useful for Alzheimer's research.
    Formula:C28H35NO3
    Color and Shape:Solid
    Molecular weight:433.58

    Ref: TM-T62441

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • YQA14

    CAS:
    YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.
    Formula:C23H27ClN4O3
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:442.94

    Ref: TM-T29195

    1mg
    77.00€
    5mg
    170.00€
    10mg
    262.00€
    25mg
    546.00€
    50mg
    855.00€
    100mg
    1,170.00€
  • WIN 62,577

    CAS:
    WIN 62,577 is a allosteric antagonist of mAChR.
    Formula:C29H31N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:437.58

    Ref: TM-T29158

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LUF6000

    CAS:
    LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR).
    Formula:C22H20Cl2N4
    Color and Shape:Solid
    Molecular weight:411.33

    Ref: TM-T15791

    5mg
    294.00€
    25mg
    690.00€
    50mg
    898.00€
    100mg
    1,575.00€
    1mL*10mM (DMSO)
    323.00€
  • Tacitin

    CAS:
    Tacitin (Benzoctamine Hydrochloride) shows sedative and anti-anxiety properties. Tacitin blocks the central postsynaptic serotonin receptors.
    Formula:C18H20ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:285.81

    Ref: TM-T26772

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€