
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,997 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5957 products of "GPCR/G-Protein"
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CCX777
CAS:CCX777 is a partial agonist recruited to ACKR3 by β-arrestin-2 and is used in cancer research.Formula:C31H43N7O3SPurity:98.73%Color and Shape:SolidMolecular weight:593.78SB-277011 dihydrochloride
CAS:SB-277011 dihydrochloride: potent, selective D3 antagonist; orally bioavailable; crosses blood-brain barrier; pKi 8.0 for D3 receptor.Formula:C28H32Cl2N4OPurity:98%Color and Shape:SolidMolecular weight:511.49DOV-216,303 Free Base
CAS:DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.Formula:C11H11Cl2NPurity:96.7%Color and Shape:SolidMolecular weight:228.12Neladenoson dalanate HCl
CAS:Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).Formula:C35H35Cl2N7O4S2Purity:98%Color and Shape:SolidMolecular weight:752.73Chlorazanil
CAS:Chlorazanil is a triazine-based, orally active diuretic that blocks Na+ and Cl– reabsorption in distal tubules, increases renal prostaglandin.Formula:C9H8ClN5Purity:98.89%Color and Shape:SolidMolecular weight:221.65PF-03654746 Tosylate
CAS:PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.Formula:C25H32F2N2O4SPurity:98%Color and Shape:SolidMolecular weight:494.6Sortilin antagonist 1
CAS:Sortilin antagonist 1 blocks Neurotensin binding with 20 nM IC50, useful in neurological disease research.Formula:C20H24N2O4Color and Shape:SolidMolecular weight:356.42Dicarbine
CAS:Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.Formula:C13H18N2Purity:98%Color and Shape:SolidMolecular weight:202.3PNU-177864
CAS:PNU-177864 is a selective dopamine D3 receptor antagonist.Formula:C18H21F3N2O3SPurity:99.92%Color and Shape:SolidMolecular weight:402.43Quinpirole Hydrochloride
CAS:Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and miceFormula:C13H22ClN3Purity:98%Color and Shape:SolidMolecular weight:255.79YQA14
CAS:YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.Formula:C23H27ClN4O3Purity:99.52%Color and Shape:SolidMolecular weight:442.94Antiplatelet agent 1
CAS:Antiplatelet agent 1 is a ticagrelor analogue that exhibits anti-platelet effects and can be used in platelet agglutination studies.Formula:C21H24F2N6O4SColor and Shape:SolidMolecular weight:494.51Aligeron
CAS:Aligeron is a non-selective prostaglandin (PG) antagonist that inhibits PGF2α- and PGE2-induced decreases in blood pressure in cats, and can be used to inhibitFormula:C20H24N2Purity:99.09% - >99.99%Color and Shape:SolidMolecular weight:292.42BMS-466442
CAS:BMS-466442 is the first selective amino acid transporter alanine serine cysteine transporter-1 inhibitor.Formula:C31H30N4O5Color and Shape:SolidMolecular weight:538.59CP 59430
CAS:CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist.Formula:C21H22N8O3Color and Shape:SolidMolecular weight:434.45Aganepag
CAS:Aganepag: Potent EP2 agonist, EC50 0.19 nM, inactive at EP4, used in wound healing and scar/wrinkle treatment research.Formula:C24H31NO4SPurity:98%Color and Shape:SolidMolecular weight:429.57AChE-IN-14
CAS:AChE-IN-14 inhibits eeAChE, hAChE, eqBuChE (IC50: 0.46-0.48 μM) and binds to H3R (Ki: 159.8 nM), useful for Alzheimer's research.Formula:C28H35NO3Color and Shape:SolidMolecular weight:433.58RUSKI-201 dihydrochloride
CAS:RUSKI-201 dihydrochloride: potent Hhat inhibitor (IC50: 0.20 μM), blocks Hh signaling, and inhibits Hh palmitoylation.Formula:C20H29Cl2N3OSColor and Shape:SolidMolecular weight:430.43RS 64459-193
CAS:RS 64459-193 has a high affinity for the 5-HT1A binding site.Formula:C26H36Cl2N2O2Color and Shape:SolidMolecular weight:479.48Vapitadine dihydrochloride
CAS:Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.Formula:C17H22Cl2N4OPurity:98.28% - 99.30%Color and Shape:SolidMolecular weight:369.29Monatepil maleate
CAS:Monatepil maleate (AJ-2615 maleate) is a Ca2+-channel and α1-adrenergic receptor antagonist, and ACAT inhibitor with antihypertensive activity.Formula:C32H34FN3O5SPurity:97.90%Color and Shape:SolidMolecular weight:591.695-Carboxamidotryptamine maleate
CAS:5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.Formula:C15H17N3O5Purity:99.88%Color and Shape:SolidMolecular weight:319.31Mirisetron
CAS:Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.Formula:C24H31N3O2Purity:99.88%Color and Shape:SolidMolecular weight:393.52Atrasentan hydrochloride
CAS:Atrasentan hydrochloride (ABT-627 hydrochloride) is an antagonist of the endothelin receptor(IC50 = 55.1 μM for ETA).Formula:C29H39ClN2O6Purity:99.75%Color and Shape:SolidMolecular weight:547.08Sigma-LIGAND-1
CAS:Sigma-LIGAND-1 is a selective Sigma Receptor ligand with an IC50s of 16 nM, 19 nM at the DTG site and the PPP site, respectively.Formula:C27H33NO4Purity:99.89%Color and Shape:SolidMolecular weight:435.56Ref: TM-T13510
1mg48.00€5mg104.00€10mg156.00€25mg235.00€50mg316.00€100mg434.00€200mg585.00€1mL*10mM (DMSO)119.00€ICI 162,846
CAS:ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.Formula:C11H17F3N6OPurity:97.45%Color and Shape:SolidMolecular weight:306.29A2AR-agonist-1
CAS:A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).Formula:C20H22N6O4Purity:99.9%Color and Shape:SolidMolecular weight:410.43Ref: TM-T10212
1mg90.00€2mg127.00€5mg178.00€10mg269.00€25mg427.00€50mg610.00€100mg820.00€500mg1,603.00€1mL*10mM (DMSO)207.00€RXFP3/4 agonist 2
CAS:RXFP3/4 agonist 2 is a nonpeptide bis-RXFP3/4 agonist used in the study of diseases caused by metabolic abnormalities.Formula:C22H22N6O2Purity:99.82%Color and Shape:SolidMolecular weight:402.45CCR4 antagonist 3-1
CAS:CCR4 antagonist 3-1 is a weak inhibitor of [125I]TARC binding and CEM cell migration, with IC50 values of 1.7 μM and 6.4 μM, respectively.
Formula:C14H12N2SPurity:99.53%Color and Shape:SolidMolecular weight:240.32PRX-08066 Maleic acid
CAS:PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.Formula:C23H21ClFN5O4SPurity:97.59%Color and Shape:SolidMolecular weight:517.96Ref: TM-T6959
1mg79.00€5mg168.00€10mg220.00€25mg398.00€50mg587.00€100mg835.00€200mg1,134.00€1mL*10mM (DMSO)380.00€C-021 dihydrochloride
CAS:C-021 dihydrochloride is a potent CCR4 antagonist. It potently inhibits functional chemotaxis in human and mouse with IC50s of 140 nM and 39 nM.Formula:C27H43Cl2N5O2Purity:98.67%Color and Shape:SolidMolecular weight:540.57NPEC-caged-dopamine
CAS:Dopamine receptor agonistFormula:C17H18N2O6Purity:98%Color and Shape:SolidMolecular weight:346.33MRGPRX1 agonist 2
CAS:MRGPRX1 agonist 2 is a potent modulator with 0.48 μM EC50, potential for neuropathic pain research.Formula:C15H14N2OSColor and Shape:SolidMolecular weight:270.35SB357134
CAS:SB357134 is a potent, selective and orally active antagonist of 5-HT6 receptor and shows nootropic effects in animal studies.Formula:C17H18Br2FN3O3SPurity:98%Color and Shape:SolidMolecular weight:523.21SSTR4 agonist 3
CAS:SSTR4 agonist 3 activates SSTR4 in the hippocampus and neocortex, aiding memory and learning, and shows potent pain relief in rodents.Formula:C18H24N4OSColor and Shape:SolidMolecular weight:344.47Bemesetron
CAS:Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.Formula:C15H17Cl2NO2Purity:99.77%Color and Shape:SolidMolecular weight:314.21SB-269970
CAS:SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).Formula:C18H28N2O3SPurity:98%Color and Shape:SolidMolecular weight:352.49Isamoltane hemifumarate
CAS:5-HT1B antagonistFormula:C16H22N202C4H404Purity:98%Color and Shape:SolidMolecular weight:332.4WS 009A
CAS:WS 009A is an antagonist of the endothelin receptor.Formula:C24H25NO10SPurity:98%Color and Shape:SolidMolecular weight:519.52Fallypride
CAS:Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.Formula:C20H29FN2O3Purity:98.97% - >99.99%Color and Shape:SolidMolecular weight:364.45Ref: TM-T70302
1mg359.00€5mg842.00€10mg1,035.00€25mg1,663.00€50mg2,072.00€100mg2,660.00€1mL*10mM (DMSO)677.00€VNA-932
CAS:VNA-932 is an agonist of the vasopressin V2-receptor (IC50: 80.3 nM and 778 nM in human-V2 binding and V1a binding assay).Formula:C23H19ClN4OPurity:98%Color and Shape:SolidMolecular weight:402.88MRS 1334
CAS:antagonist for the human adenosine A3 receptorFormula:C31H26N2O6Purity:98%Color and Shape:SolidMolecular weight:522.55Thioproperazine
CAS:Thioproperazine (RP 7843) is an orally effective antipsychotic schizophrenia and bipolar disorder, histamine and adrenergic receptor blocker.Formula:C22H30N4O2S2Purity:99.45%Color and Shape:SolidMolecular weight:446.635-HT3 antagonist 3
CAS:5-HT3 antagonist 3 (Compound 15b) is a high-affinity 5-HT3 receptor antagonist. It binds to 5-HT3 receptors in rat brain cortical membranes (Ki: 0.25 nM).Formula:C20H21N3OPurity:99.9%Color and Shape:SolidMolecular weight:319.4Ref: TM-T10162
1mg109.00€2mg163.00€5mg243.00€10mg355.00€25mg532.00€50mg750.00€100mg1,009.00€500mgTo inquirePF-06256142
CAS:PF-06256142 is a potent and selective orthosteric D1 receptor agonist(D1 EC50=30 nM ).Formula:C21H16N4O2Purity:98%Color and Shape:SolidMolecular weight:356.38CCR1 antagonist 9
CAS:CCR1 antagonist 9 (compound 19e) is a selective CCR1 antagonist based on aziridine. CCR1 inhibition in calcium flux assays.Formula:C20H16FN5O3SPurity:99.13%Color and Shape:SolidMolecular weight:425.44Ref: TM-T10710
1mg101.00€5mg241.00€10mg402.00€25mg727.00€50mg1,046.00€100mg1,525.00€1mL*10mM (DMSO)265.00€AZD5213
CAS:AZD5213: selective human H3 receptor antagonist, pKi 9.3, for sleep/cognition research.Formula:C19H25N3O2Color and Shape:SolidMolecular weight:327.42(R,R)-Reboxetine mesylate
CAS:(R,R)-Reboxetine mesylate: Antidepressant, high bioavailability, (R,R) enantiomer, selective for noradrenaline, low toxicity.Formula:C20H27NO6SColor and Shape:SolidMolecular weight:409.5Amgen-23
CAS:Amgen-23 is a selective and highly potent sphingosine kinase 1 (SPHK1) inhibitor that inhibits SPHK2 and can be used in anticancer research.Formula:C23H25Cl2N3O2SPurity:97.31%Color and Shape:SolidMolecular weight:478.44TCS-OX2-29 HCl
CAS:TCS-OX2-29 is a selective orexin-2 receptor antagonist (IC50 = 40 nM), which plays an important role in pain modulation.Formula:C23H32ClN3O3Purity:98%Color and Shape:SolidMolecular weight:433.97TC-C 14G
CAS:CB1 receptor inverse agonistFormula:C24H17Cl2F2NO4Purity:98%Color and Shape:SolidMolecular weight:492.3NPS-2143
CAS:NPS-2143 (SB 262470A) is a novel potent and selective antagonist of Ca(2+) receptor.Formula:C24H25ClN2O2Purity:99.56%Color and Shape:SolidMolecular weight:408.92A331440
CAS:A331440 is an modulator of L-histidine and histamine H3 receptor.Formula:C22H27N3OColor and Shape:SolidMolecular weight:349.47CCR2 antagonist 3
CAS:CCR2 antagonist 3 (AZD-2927) is an antagonist of CCR2.Formula:C17H25FN2O2Purity:99.87%Color and Shape:SolidMolecular weight:308.39Ref: TM-T10712
1mg66.00€5mg147.00€10mg225.00€25mg398.00€50mg532.00€100mg745.00€200mg982.00€1mL*10mM (DMSO)161.00€GW 766994
CAS:GW 766994 is a specific and oral chemokine receptor-3 (CCR3) antagonist. It has the potential for asthma and eosinophilic bronchitis treatment.Formula:C21H24Cl2N4O3Purity:98.77%Color and Shape:SolidMolecular weight:451.35UP202-56
CAS:UP202-56 is an adenosinergic agonist and is an adenosine analog.Formula:C33H37N7O4Purity:98%Color and Shape:SolidMolecular weight:595.69Spirendolol
CAS:Spirendolol is an antagonist of β adrenergic receptor.Formula:C21H31NO3Purity:98%Color and Shape:SolidMolecular weight:345.48LPA2 antagonist 2
CAS:LPA2 antagonist 2 is an and LPA2 antagonist (IC50: 28.3 nM) with potential anticancer activity, inhibits LPA3, and can be used for cancer research.Formula:C20H16N2O6Purity:96.13%Color and Shape:SolidMolecular weight:380.35S(-)-Bisoprolol
CAS:S(-)-Bisoprolol, a β1-blocker, may aid in researching hypertension and heart diseases.Formula:C18H31NO4Color and Shape:SolidMolecular weight:325.44AM404
CAS:AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.Formula:C26H37NO2Color and Shape:SolidMolecular weight:395.58UCSF678
CAS:UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.Formula:C15H18N2O2SColor and Shape:SolidMolecular weight:290.38Centanafadine
CAS:Centanafadine inhibits NE/DA transporters and serotonin transporter (IC50: NE=6 nM, DA=38 nM, 5-HT=83 nM).Formula:C15H15NPurity:98%Color and Shape:SolidMolecular weight:209.29PF-592379
CAS:PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).Formula:C13H21N3OPurity:98%Color and Shape:SolidMolecular weight:235.33GR 113808
CAS:GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.Formula:C19H27N3O4SPurity:98.16% - 99.96%Color and Shape:SolidMolecular weight:393.5HEMADO
CAS:HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).Formula:C17H23N5O4Purity:98%Color and Shape:SolidMolecular weight:361.4GR-203040 HCl
CAS:GR203040 inhibits cyclophosphamide-induced damage in the rat and ferret bladder. GR-203040 is a selective NK1 receptor antagonist.Formula:C20H26Cl2N6OColor and Shape:SolidMolecular weight:437.37GBR 13069 dihydrochloride
CAS:GBR 13069 dihydrochloride is a dopamine uptake inhibitor.Formula:C28H32Cl2F2N2OPurity:98%Color and Shape:SolidMolecular weight:521.47(R)-SLV 319
CAS:(R)-SLV 319: potent CB1 antagonist, K i of 894 nM, dextrorotatory isomer.Formula:C23H20Cl2N4O2SColor and Shape:SolidMolecular weight:487.4Loratadine N-oxide
CAS:Loratadine N-oxide is a metabolite of the histamine H1 receptor inverse agonist loratadine.Formula:C22H23ClN2O3Color and Shape:SolidMolecular weight:398.882-Methylthioadenosine diphosphate trisodium
CAS:2-Methylthioadenosine diphosphate trisodium(2-MeS-ADP) is a purinergic P2Y receptor agonist that agonizes P2Y13 and P2Y12, induces platelet aggregation.Formula:C11H14N5Na3O10P2SColor and Shape:SolidMolecular weight:539.24SCH-23390 maleate
CAS:SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,Formula:C21H22ClNO5Purity:98%Color and Shape:SolidMolecular weight:403.86DS-3801b
CAS:DS-3801b is a non-macrolide GPR38 agonist with an N-methylaniline structure for the study of functional gastrointestinal disorders.Formula:C28H39N3O3Purity:99.21%Color and Shape:SolidMolecular weight:465.63EGIS-7625
CAS:EGIS-7625 is a selective and competitive antagonist of 5-HT2B receptor.Formula:C18H24Cl2N4O2Purity:98%Color and Shape:SolidMolecular weight:399.32Carbinoxamine
CAS:Carbinoxamine: antihistamine for hay fever, angioedema, rhinitis, mild urticaria, dermatographism, allergic conjunctivitis; an H1-antagonist.Formula:C16H19ClN2OPurity:98%Color and Shape:LiquidMolecular weight:290.79L-750,667 Trihydrochloride
CAS:L-750,667 Trihydrochloride is a selective D4 receptor antagonist, reverses the dopamine-induced inhibition of cAMP accumulation in the central nervous system.Formula:C18H22Cl3IN4Purity:99.63%Color and Shape:SolidMolecular weight:527.665-HT3 antagonist 2
CAS:5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.Formula:C18H21N3OPurity:98%Color and Shape:SolidMolecular weight:295.38hA2A/hCA XII modulator 1
CAS:Potent hA2AAR antagonist & hCA XII inhibitor; Ki: hA2AAR 6.4 nM, hCA XII 6.2 nM. Possible cancer research use.Formula:C24H19N7O4SColor and Shape:SolidMolecular weight:501.52DV 7028 hydrochloride
CAS:DV 7028 hydrochloride is a 5-HT2A receptor antagonist.Formula:C21H26ClFN4O3Purity:98%Color and Shape:SolidMolecular weight:436.91(RS)-Minesapride
CAS:Minesapride is a serotonin receptor agonist.Formula:C21H31ClN4O5Purity:98%Color and Shape:SolidMolecular weight:454.95S20928
CAS:S20928 is an antagonist of melatonin receptor.Formula:C17H19NOColor and Shape:SolidMolecular weight:253.34LY 206130
CAS:LY 206130 is an antagonist of serotonin 5-HT1A.Formula:C17H24N2O2Color and Shape:SolidMolecular weight:288.38Afurolol Hydrochloride
CAS:Afurolol Hydrochloride (DL 071-IT) is a non-selective β-adrenergic receptor antagonist. DL 071 IT exhibits intrinsic sympathomimetic activity.Formula:C15H22ClNO4Purity:98.86%Color and Shape:SolidMolecular weight:315.79RS 15385-197
CAS:RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.Formula:C18H26N2O3SColor and Shape:SolidMolecular weight:350.48Lesopitron dihydrochloride
CAS:Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.Formula:C15H23Cl3N6Purity:98%Color and Shape:SolidMolecular weight:393.74Alclofenac sodium
CAS:Alclofenac sodium is an anti-inflammatory utilized in the treatment of rheumatoid arthritis.Formula:C11H11ClNaO3Purity:98%Color and Shape:SolidMolecular weight:249.65Chloracyzine
CAS:Chloracyzine lowers heart oxygen use, shrinks coronary flow after brief dilation, slightly ups heart rate and arterial pressure.Formula:C19H21ClN2OSColor and Shape:SolidMolecular weight:360.9Garomefrine HCl
CAS:Garomefrine HCl, a α1A-adrenoceptor agonist, is potential for the treatment of urinary incontinence.Formula:C9H14ClFN2O3SPurity:98%Color and Shape:SolidMolecular weight:284.73Viprostol
CAS:Viprostol is an agent of prostaglandin antihypertensive.Formula:C23H36O5Purity:98%Color and Shape:SolidMolecular weight:392.53GS 283
CAS:GS 283 is a Ca(2+) antagonist. GS 283 is also a weak histamine and muscarinic receptor blocker in rat and guinea pig tracheal smooth muscles.Formula:C17H17NO3Color and Shape:SolidMolecular weight:283.32LBP-1
CAS:LBP-1 is a cannabinoid receptor type 1 (CB1) agonist.Formula:C23H29ClN6O3Color and Shape:SolidMolecular weight:472.97Seproxetine HCl
CAS:Seproxetine HCl, a more active enantiomer of N-desmethyl metabolite fluoxetine, works by selectively inhibiting the serotonin uptake carrier.Formula:C16H17ClF3NOPurity:98%Color and Shape:SolidMolecular weight:331.76GSK1059865
CAS:GSK1059865 is a potent antagonist of the orexin 1 receptor.Formula:C20H23BrFN3O2Color and Shape:SolidMolecular weight:436.32PNU-96391
CAS:PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.Formula:C15H23NO2SPurity:99.53%Color and Shape:SolidMolecular weight:281.41Ref: TM-T28435
1mg77.00€5mg155.00€10mg221.00€25mg338.00€50mg472.00€100mg632.00€200mg843.00€1mL*10mM (DMSO)145.00€MS437
CAS:MS437 is a potent TSH receptor agonist.Formula:C22H24N2OPurity:98%Color and Shape:SolidMolecular weight:332.44LG 82-4-00
CAS:LG 82-4-00 is an inhibitor of thromboxane.Formula:C10H11ClN2O3SPurity:98%Color and Shape:SolidMolecular weight:274.72BGC201531
CAS:BGC201531 (AP-1531) is a EP4 antagonist for the treatment of acute migraine.
Formula:C26H28N2O6SPurity:98.51% - 99.33%Color and Shape:SolidMolecular weight:496.58LY 163443
CAS:LY 163443 is an dual receptor antagonist of LTD4 and LTE4.Formula:C20H22N4O3Color and Shape:SolidMolecular weight:366.41FR 121196
CAS:FR 121196, a potential antidementia drug, ameliorates the impaired memory of rat in the Morris water maze.Formula:C12H16FN3O3SColor and Shape:SolidMolecular weight:301.34A23887
CAS:A23887 is a potentially neuroleptic tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Formula:C22H24ClNPurity:98%Color and Shape:SolidMolecular weight:337.89SID7970631
CAS:SID7970631 is an isoquinolinone analogue, a selective and potent submicromolar SF-1 inhibitor with an IC50 of 260 nM. SID7970631 can be used to study cancer.Formula:C24H24N2O7Color and Shape:SolidMolecular weight:452.46
