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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5957 products of "GPCR/G-Protein"

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  • CCX777

    CAS:
    CCX777 is a partial agonist recruited to ACKR3 by β-arrestin-2 and is used in cancer research.
    Formula:C31H43N7O3S
    Purity:98.73%
    Color and Shape:Solid
    Molecular weight:593.78

    Ref: TM-T23866

    1mg
    269.00€
  • SB-277011 dihydrochloride

    CAS:
    SB-277011 dihydrochloride: potent, selective D3 antagonist; orally bioavailable; crosses blood-brain barrier; pKi 8.0 for D3 receptor.
    Formula:C28H32Cl2N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:511.49

    Ref: TM-T12861L

    1mg
    148.00€
    5mg
    384.00€
    10mg
    617.00€
    25mg
    1,378.00€
  • DOV-216,303 Free Base

    CAS:
    DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.
    Formula:C11H11Cl2N
    Purity:96.7%
    Color and Shape:Solid
    Molecular weight:228.12

    Ref: TM-T11087

    2mg
    46.00€
    5mg
    66.00€
    10mg
    97.00€
    25mg
    159.00€
    50mg
    226.00€
    100mg
    339.00€
    1mL*10mM (DMSO)
    67.00€
  • Neladenoson dalanate HCl

    CAS:
    Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).
    Formula:C35H35Cl2N7O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:752.73

    Ref: TM-T24526

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Chlorazanil

    CAS:
    Chlorazanil is a triazine-based, orally active diuretic that blocks Na+ and Cl– reabsorption in distal tubules, increases renal prostaglandin.
    Formula:C9H8ClN5
    Purity:98.89%
    Color and Shape:Solid
    Molecular weight:221.65

    Ref: TM-T13609L

    10mg
    36.00€
    25mg
    36.00€
    50mg
    To inquire
    1mL*10mM (DMSO)
    48.00€
  • PF-03654746 Tosylate

    CAS:
    PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
    Formula:C25H32F2N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:494.6

    Ref: TM-T12416

    25mg
    828.00€
    50mg
    1,063.00€
    100mg
    1,611.00€
  • Sortilin antagonist 1

    CAS:
    Sortilin antagonist 1 blocks Neurotensin binding with 20 nM IC50, useful in neurological disease research.
    Formula:C20H24N2O4
    Color and Shape:Solid
    Molecular weight:356.42

    Ref: TM-T72410

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Dicarbine

    CAS:
    Double carbene blocks dopamine receptors, aiding schizophrenia and alcoholism research; it maintains defense reflexes despite mid-brain stimulation.
    Formula:C13H18N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:202.3

    Ref: TM-T13652

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PNU-177864

    CAS:
    PNU-177864 is a selective dopamine D3 receptor antagonist.
    Formula:C18H21F3N2O3S
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:402.43

    Ref: TM-T23167

    1mg
    42.00€
    5mg
    84.00€
    10mg
    93.00€
    25mg
    202.00€
    50mg
    284.00€
    100mg
    391.00€
    200mg
    545.00€
  • Quinpirole Hydrochloride

    CAS:
    Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and mice
    Formula:C13H22ClN3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:255.79

    Ref: TM-T12606

    1mg
    100.00€
  • YQA14

    CAS:
    YQA14 is a selective, high-affinity dopamine D3 receptor antagonist that inhibits cocaine self-administration in rats and mice, opioid addiction research.
    Formula:C23H27ClN4O3
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:442.94

    Ref: TM-T29195

    1mg
    77.00€
    5mg
    170.00€
    10mg
    262.00€
    25mg
    546.00€
    50mg
    855.00€
    100mg
    1,170.00€
  • Antiplatelet agent 1

    CAS:
    Antiplatelet agent 1 is a ticagrelor analogue that exhibits anti-platelet effects and can be used in platelet agglutination studies.
    Formula:C21H24F2N6O4S
    Color and Shape:Solid
    Molecular weight:494.51

    Ref: TM-T63334

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • Aligeron

    CAS:
    Aligeron is a non-selective prostaglandin (PG) antagonist that inhibits PGF2α- and PGE2-induced decreases in blood pressure in cats, and can be used to inhibit
    Formula:C20H24N2
    Purity:99.09% - >99.99%
    Color and Shape:Solid
    Molecular weight:292.42

    Ref: TM-T36619

    1mg
    630.00€
    5mg
    1,620.00€
  • BMS-466442

    CAS:
    BMS-466442 is the first selective amino acid transporter alanine serine cysteine transporter-1 inhibitor.
    Formula:C31H30N4O5
    Color and Shape:Solid
    Molecular weight:538.59

    Ref: TM-T23806

    10mg
    884.00€
  • CP 59430

    CAS:
    CP 59430 is an azide analogue of prazosin. Prazosin is a highly selective α 1-adrenergic receptor antagonist.
    Formula:C21H22N8O3
    Color and Shape:Solid
    Molecular weight:434.45

    Ref: TM-T31022

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Aganepag

    CAS:
    Aganepag: Potent EP2 agonist, EC50 0.19 nM, inactive at EP4, used in wound healing and scar/wrinkle treatment research.
    Formula:C24H31NO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:429.57

    Ref: TM-T14139

    25mg
    2,043.00€
    50mg
    2,682.00€
    100mg
    3,600.00€
  • AChE-IN-14

    CAS:
    AChE-IN-14 inhibits eeAChE, hAChE, eqBuChE (IC50: 0.46-0.48 μM) and binds to H3R (Ki: 159.8 nM), useful for Alzheimer's research.
    Formula:C28H35NO3
    Color and Shape:Solid
    Molecular weight:433.58

    Ref: TM-T62441

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • RUSKI-201 dihydrochloride

    CAS:
    RUSKI-201 dihydrochloride: potent Hhat inhibitor (IC50: 0.20 μM), blocks Hh signaling, and inhibits Hh palmitoylation.
    Formula:C20H29Cl2N3OS
    Color and Shape:Solid
    Molecular weight:430.43

    Ref: TM-T62388

    1mg
    197.00€
    5mg
    862.00€
    10mg
    1,521.00€
  • RS 64459-193

    CAS:
    RS 64459-193 has a high affinity for the 5-HT1A binding site.
    Formula:C26H36Cl2N2O2
    Color and Shape:Solid
    Molecular weight:479.48

    Ref: TM-T34415

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Vapitadine dihydrochloride

    CAS:
    Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.
    Formula:C17H22Cl2N4O
    Purity:98.28% - 99.30%
    Color and Shape:Solid
    Molecular weight:369.29

    Ref: TM-T29096

    1mg
    245.00€
    5mg
    610.00€
    10mg
    868.00€
    25mg
    1,301.00€
    50mg
    1,758.00€
  • Monatepil maleate

    CAS:
    Monatepil maleate (AJ-2615 maleate) is a Ca2+-channel and α1-adrenergic receptor antagonist, and ACAT inhibitor with antihypertensive activity.
    Formula:C32H34FN3O5S
    Purity:97.90%
    Color and Shape:Solid
    Molecular weight:591.69

    Ref: TM-T25828

    1mg
    279.00€
    5mg
    685.00€
    10mg
    938.00€
    25mg
    1,444.00€
    50mg
    1,882.00€
  • 5-Carboxamidotryptamine maleate

    CAS:
    5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.
    Formula:C15H17N3O5
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:319.31

    Ref: TM-T22520

    1mg
    35.00€
    5mg
    84.00€
    10mg
    119.00€
    25mg
    207.00€
    50mg
    289.00€
    100mg
    399.00€
    200mg
    555.00€
  • Mirisetron

    CAS:
    Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.
    Formula:C24H31N3O2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:393.52

    Ref: TM-T70879

    1mg
    285.00€
    5mg
    692.00€
    10mg
    947.00€
    25mg
    1,458.00€
    50mg
    1,839.00€
    100mg
    2,322.00€
  • Atrasentan hydrochloride

    CAS:
    Atrasentan hydrochloride (ABT-627 hydrochloride) is an antagonist of the endothelin receptor(IC50 = 55.1 μM for ETA).
    Formula:C29H39ClN2O6
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:547.08

    Ref: TM-TQ0270

    1mg
    47.00€
    5mg
    92.00€
    10mg
    130.00€
    25mg
    250.00€
    50mg
    356.00€
    1mL*10mM (DMSO)
    110.00€
  • Sigma-LIGAND-1

    CAS:
    Sigma-LIGAND-1 is a selective Sigma Receptor ligand with an IC50s of 16 nM, 19 nM at the DTG site and the PPP site, respectively.
    Formula:C27H33NO4
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:435.56

    Ref: TM-T13510

    1mg
    48.00€
    5mg
    104.00€
    10mg
    156.00€
    25mg
    235.00€
    50mg
    316.00€
    100mg
    434.00€
    200mg
    585.00€
    1mL*10mM (DMSO)
    119.00€
  • ICI 162,846

    CAS:
    ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.
    Formula:C11H17F3N6O
    Purity:97.45%
    Color and Shape:Solid
    Molecular weight:306.29

    Ref: TM-T22848

    1mg
    34.00€
    5mg
    65.00€
    10mg
    94.00€
    25mg
    138.00€
    50mg
    197.00€
  • A2AR-agonist-1

    CAS:
    A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).
    Formula:C20H22N6O4
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:410.43

    Ref: TM-T10212

    1mg
    90.00€
    2mg
    127.00€
    5mg
    178.00€
    10mg
    269.00€
    25mg
    427.00€
    50mg
    610.00€
    100mg
    820.00€
    500mg
    1,603.00€
    1mL*10mM (DMSO)
    207.00€
  • RXFP3/4 agonist 2

    CAS:
    RXFP3/4 agonist 2 is a nonpeptide bis-RXFP3/4 agonist used in the study of diseases caused by metabolic abnormalities.
    Formula:C22H22N6O2
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:402.45

    Ref: TM-T61964

    1mg
    284.00€
  • CCR4 antagonist 3-1

    CAS:

    CCR4 antagonist 3-1 is a weak inhibitor of [125I]TARC binding and CEM cell migration, with IC50 values of 1.7 μM and 6.4 μM, respectively.

    Formula:C14H12N2S
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:240.32

    Ref: TM-T60336

    1mg
    92.00€
    5mg
    216.00€
    10mg
    354.00€
    25mg
    692.00€
    50mg
    1,074.00€
    100mg
    1,454.00€
    500mg
    2,822.00€
  • PRX-08066 Maleic acid

    CAS:
    PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.
    Formula:C23H21ClFN5O4S
    Purity:97.59%
    Color and Shape:Solid
    Molecular weight:517.96

    Ref: TM-T6959

    1mg
    79.00€
    5mg
    168.00€
    10mg
    220.00€
    25mg
    398.00€
    50mg
    587.00€
    100mg
    835.00€
    200mg
    1,134.00€
    1mL*10mM (DMSO)
    380.00€
  • C-021 dihydrochloride

    CAS:
    C-021 dihydrochloride is a potent CCR4 antagonist. It potently inhibits functional chemotaxis in human and mouse with IC50s of 140 nM and 39 nM.
    Formula:C27H43Cl2N5O2
    Purity:98.67%
    Color and Shape:Solid
    Molecular weight:540.57

    Ref: TM-T10639

    1mg
    52.00€
    5mg
    97.00€
    10mg
    154.00€
    25mg
    249.00€
    50mg
    374.00€
    1mL*10mM (DMSO)
    115.00€
  • NPEC-caged-dopamine

    CAS:
    Dopamine receptor agonist
    Formula:C17H18N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:346.33

    Ref: TM-T23082

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MRGPRX1 agonist 2

    CAS:
    MRGPRX1 agonist 2 is a potent modulator with 0.48 μM EC50, potential for neuropathic pain research.
    Formula:C15H14N2OS
    Color and Shape:Solid
    Molecular weight:270.35

    Ref: TM-T60466

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SB357134

    CAS:
    SB357134 is a potent, selective and orally active antagonist of 5-HT6 receptor and shows nootropic effects in animal studies.
    Formula:C17H18Br2FN3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:523.21

    Ref: TM-T28689

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SSTR4 agonist 3

    CAS:
    SSTR4 agonist 3 activates SSTR4 in the hippocampus and neocortex, aiding memory and learning, and shows potent pain relief in rodents.
    Formula:C18H24N4OS
    Color and Shape:Solid
    Molecular weight:344.47

    Ref: TM-T61130

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bemesetron

    CAS:
    Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.
    Formula:C15H17Cl2NO2
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:314.21

    Ref: TM-T14526

    10mg
    52.00€
    25mg
    66.00€
    50mg
    89.00€
  • SB-269970

    CAS:
    SB-269970 is a antagonist of 5-HT7 receptor(pKi of 8.3).
    Formula:C18H28N2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.49

    Ref: TM-T12842

    25mg
    2,178.00€
    50mg
    3,042.00€
    100mg
    4,140.00€
  • Isamoltane hemifumarate

    CAS:
    5-HT1B antagonist
    Formula:C16H22N202C4H404
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.4

    Ref: TM-T22872

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • WS 009A

    CAS:
    WS 009A is an antagonist of the endothelin receptor.
    Formula:C24H25NO10S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:519.52

    Ref: TM-T24053

    25mg
    1,369.00€
  • Fallypride

    CAS:
    Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.
    Formula:C20H29FN2O3
    Purity:98.97% - >99.99%
    Color and Shape:Solid
    Molecular weight:364.45

    Ref: TM-T70302

    1mg
    359.00€
    5mg
    842.00€
    10mg
    1,035.00€
    25mg
    1,663.00€
    50mg
    2,072.00€
    100mg
    2,660.00€
    1mL*10mM (DMSO)
    677.00€
  • VNA-932

    CAS:
    VNA-932 is an agonist of the vasopressin V2-receptor (IC50: 80.3 nM and 778 nM in human-V2 binding and V1a binding assay).
    Formula:C23H19ClN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:402.88

    Ref: TM-T17251

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MRS 1334

    CAS:
    antagonist for the human adenosine A3 receptor
    Formula:C31H26N2O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:522.55

    Ref: TM-T23017

    25mg
    2,232.00€
  • Thioproperazine

    CAS:
    Thioproperazine (RP 7843) is an orally effective antipsychotic schizophrenia and bipolar disorder, histamine and adrenergic receptor blocker.
    Formula:C22H30N4O2S2
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:446.63

    Ref: TM-T21368

    1mg
    37.00€
    5mg
    79.00€
    10mg
    114.00€
    25mg
    185.00€
    50mg
    276.00€
    100mg
    409.00€
  • 5-HT3 antagonist 3

    CAS:
    5-HT3 antagonist 3 (Compound 15b) is a high-affinity 5-HT3 receptor antagonist. It binds to 5-HT3 receptors in rat brain cortical membranes (Ki: 0.25 nM).
    Formula:C20H21N3O
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:319.4

    Ref: TM-T10162

    1mg
    109.00€
    2mg
    163.00€
    5mg
    243.00€
    10mg
    355.00€
    25mg
    532.00€
    50mg
    750.00€
    100mg
    1,009.00€
    500mg
    To inquire
  • PF-06256142

    CAS:
    PF-06256142 is a potent and selective orthosteric D1 receptor agonist(D1 EC50=30 nM ).
    Formula:C21H16N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:356.38

    Ref: TM-T12423

    25mg
    1,260.00€
    50mg
    1,639.00€
    100mg
    2,250.00€
  • CCR1 antagonist 9

    CAS:
    CCR1 antagonist 9 (compound 19e) is a selective CCR1 antagonist based on aziridine. CCR1 inhibition in calcium flux assays.
    Formula:C20H16FN5O3S
    Purity:99.13%
    Color and Shape:Solid
    Molecular weight:425.44

    Ref: TM-T10710

    1mg
    101.00€
    5mg
    241.00€
    10mg
    402.00€
    25mg
    727.00€
    50mg
    1,046.00€
    100mg
    1,525.00€
    1mL*10mM (DMSO)
    265.00€
  • AZD5213

    CAS:
    AZD5213: selective human H3 receptor antagonist, pKi 9.3, for sleep/cognition research.
    Formula:C19H25N3O2
    Color and Shape:Solid
    Molecular weight:327.42

    Ref: TM-T71423

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (R,R)-Reboxetine mesylate

    CAS:
    (R,R)-Reboxetine mesylate: Antidepressant, high bioavailability, (R,R) enantiomer, selective for noradrenaline, low toxicity.
    Formula:C20H27NO6S
    Color and Shape:Solid
    Molecular weight:409.5

    Ref: TM-T72209

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Amgen-23

    CAS:
    Amgen-23 is a selective and highly potent sphingosine kinase 1 (SPHK1) inhibitor that inhibits SPHK2 and can be used in anticancer research.
    Formula:C23H25Cl2N3O2S
    Purity:97.31%
    Color and Shape:Solid
    Molecular weight:478.44

    Ref: TM-T63132

    1mg
    84.00€
    5mg
    177.00€
    10mg
    281.00€
    25mg
    510.00€
    50mg
    790.00€
    1mL*10mM (DMSO)
    178.00€
  • TCS-OX2-29 HCl

    CAS:
    TCS-OX2-29 is a selective orexin-2 receptor antagonist (IC50 = 40 nM), which plays an important role in pain modulation.
    Formula:C23H32ClN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.97

    Ref: TM-T4965L

    5mg
    316.00€
    10mg
    600.00€
    50mg
    2,502.00€
  • TC-C 14G

    CAS:
    CB1 receptor inverse agonist
    Formula:C24H17Cl2F2NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:492.3

    Ref: TM-T23427

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • NPS-2143

    CAS:
    NPS-2143 (SB 262470A) is a novel potent and selective antagonist of Ca(2+) receptor.
    Formula:C24H25ClN2O2
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:408.92

    Ref: TM-T1730

    1ml
    54.00€
    5mg
    49.00€
    10mg
    82.00€
    25mg
    145.00€
    50mg
    208.00€
    100mg
    313.00€
  • A331440

    CAS:
    A331440 is an modulator of L-histidine and histamine H3 receptor.
    Formula:C22H27N3O
    Color and Shape:Solid
    Molecular weight:349.47

    Ref: TM-T26480

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CCR2 antagonist 3

    CAS:
    CCR2 antagonist 3 (AZD-2927) is an antagonist of CCR2.
    Formula:C17H25FN2O2
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:308.39

    Ref: TM-T10712

    1mg
    66.00€
    5mg
    147.00€
    10mg
    225.00€
    25mg
    398.00€
    50mg
    532.00€
    100mg
    745.00€
    200mg
    982.00€
    1mL*10mM (DMSO)
    161.00€
  • GW 766994

    CAS:
    GW 766994 is a specific and oral chemokine receptor-3 (CCR3) antagonist. It has the potential for asthma and eosinophilic bronchitis treatment.
    Formula:C21H24Cl2N4O3
    Purity:98.77%
    Color and Shape:Solid
    Molecular weight:451.35

    Ref: TM-T11521

    25mg
    1,080.00€
    50mg
    1,404.00€
    100mg
    2,250.00€
  • UP202-56

    CAS:
    UP202-56 is an adenosinergic agonist and is an adenosine analog.
    Formula:C33H37N7O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:595.69

    Ref: TM-T13256

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Spirendolol

    CAS:
    Spirendolol is an antagonist of β adrenergic receptor.
    Formula:C21H31NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:345.48

    Ref: TM-T16919

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LPA2 antagonist 2

    CAS:
    LPA2 antagonist 2 is an and LPA2 antagonist (IC50: 28.3 nM) with potential anticancer activity, inhibits LPA3, and can be used for cancer research.
    Formula:C20H16N2O6
    Purity:96.13%
    Color and Shape:Solid
    Molecular weight:380.35

    Ref: TM-T11875

    1mg
    96.00€
    5mg
    227.00€
    10mg
    359.00€
    25mg
    595.00€
    50mg
    838.00€
    100mg
    1,130.00€
  • S(-)-Bisoprolol

    CAS:
    S(-)-Bisoprolol, a β1-blocker, may aid in researching hypertension and heart diseases.
    Formula:C18H31NO4
    Color and Shape:Solid
    Molecular weight:325.44

    Ref: TM-T60901

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • AM404

    CAS:
    AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.
    Formula:C26H37NO2
    Color and Shape:Solid
    Molecular weight:395.58

    Ref: TM-T39281

    5mg
    65.00€
    10mg
    105.00€
    50mg
    419.00€
    100mg
    713.00€
  • UCSF678

    CAS:
    UCSF678: selective 42 nM partial agonist at 5-HT5AR, fewer off-target effects, and lower assay risks than SB-699551.
    Formula:C15H18N2O2S
    Color and Shape:Solid
    Molecular weight:290.38

    Ref: TM-T60597

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Centanafadine

    CAS:
    Centanafadine inhibits NE/DA transporters and serotonin transporter (IC50: NE=6 nM, DA=38 nM, 5-HT=83 nM).
    Formula:C15H15N
    Purity:98%
    Color and Shape:Solid
    Molecular weight:209.29

    Ref: TM-T10758

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PF-592379

    CAS:
    PF-592379 is a potent agonist of dopamine D3 receptor (EC50: 21 nM).
    Formula:C13H21N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:235.33

    Ref: TM-T10080

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GR 113808

    CAS:
    GR 113808 is a 5-HT4 receptor antagonist that inhibits 5-HT1B and 5-HT3 receptors and attenuates morphine-stimulated dopamine release in the rat striatum.
    Formula:C19H27N3O4S
    Purity:98.16% - 99.96%
    Color and Shape:Solid
    Molecular weight:393.5

    Ref: TM-T15414

    1mg
    35.00€
    5mg
    79.00€
  • HEMADO

    CAS:
    HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).
    Formula:C17H23N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:361.4

    Ref: TM-T15468

    1mg
    112.00€
    5mg
    388.00€
  • GR-203040 HCl

    CAS:
    GR203040 inhibits cyclophosphamide-induced damage in the rat and ferret bladder. GR-203040 is a selective NK1 receptor antagonist.
    Formula:C20H26Cl2N6O
    Color and Shape:Solid
    Molecular weight:437.37

    Ref: TM-T24102

    25mg
    1,738.00€
  • GBR 13069 dihydrochloride

    CAS:
    GBR 13069 dihydrochloride is a dopamine uptake inhibitor.
    Formula:C28H32Cl2F2N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:521.47

    Ref: TM-T22799

    5mg
    259.00€
    10mg
    500.00€
    25mg
    1,161.00€
  • (R)-SLV 319

    CAS:
    (R)-SLV 319: potent CB1 antagonist, K i of 894 nM, dextrorotatory isomer.
    Formula:C23H20Cl2N4O2S
    Color and Shape:Solid
    Molecular weight:487.4

    Ref: TM-T22140

    5mg
    1,018.00€
    10mg
    1,513.00€
  • Loratadine N-oxide

    CAS:
    Loratadine N-oxide is a metabolite of the histamine H1 receptor inverse agonist loratadine.
    Formula:C22H23ClN2O3
    Color and Shape:Solid
    Molecular weight:398.88

    Ref: TM-T70306

    1mg
    101.00€
    5mg
    314.00€
    10mg
    437.00€
  • 2-Methylthioadenosine diphosphate trisodium

    CAS:
    2-Methylthioadenosine diphosphate trisodium(2-MeS-ADP) is a purinergic P2Y receptor agonist that agonizes P2Y13 and P2Y12, induces platelet aggregation.
    Formula:C11H14N5Na3O10P2S
    Color and Shape:Solid
    Molecular weight:539.24

    Ref: TM-T23581

    1mg
    144.00€
    5mg
    607.00€
    10mg
    933.00€
  • SCH-23390 maleate

    CAS:
    SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,
    Formula:C21H22ClNO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:403.86

    Ref: TM-T12865

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • DS-3801b

    CAS:
    DS-3801b is a non-macrolide GPR38 agonist with an N-methylaniline structure for the study of functional gastrointestinal disorders.
    Formula:C28H39N3O3
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:465.63

    Ref: TM-T62973

    1mg
    167.00€
    5mg
    425.00€
    10mg
    691.00€
    25mg
    1,377.00€
    50mg
    1,941.00€
    1mL*10mM (DMSO)
    435.00€
  • EGIS-7625

    CAS:
    EGIS-7625 is a selective and competitive antagonist of 5-HT2B receptor.
    Formula:C18H24Cl2N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:399.32

    Ref: TM-T27249

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Carbinoxamine

    CAS:
    Carbinoxamine: antihistamine for hay fever, angioedema, rhinitis, mild urticaria, dermatographism, allergic conjunctivitis; an H1-antagonist.
    Formula:C16H19ClN2O
    Purity:98%
    Color and Shape:Liquid
    Molecular weight:290.79

    Ref: TM-T21247

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L-750,667 Trihydrochloride

    CAS:
    L-750,667 Trihydrochloride is a selective D4 receptor antagonist, reverses the dopamine-induced inhibition of cAMP accumulation in the central nervous system.
    Formula:C18H22Cl3IN4
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:527.66

    Ref: TM-T27777

    1mg
    62.00€
    5mg
    130.00€
    10mg
    203.00€
    25mg
    412.00€
    50mg
    652.00€
    100mg
    1,027.00€
    200mg
    1,391.00€
  • 5-HT3 antagonist 2

    CAS:
    5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.
    Formula:C18H21N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:295.38

    Ref: TM-T12988

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • hA2A/hCA XII modulator 1

    CAS:
    Potent hA2AAR antagonist & hCA XII inhibitor; Ki: hA2AAR 6.4 nM, hCA XII 6.2 nM. Possible cancer research use.
    Formula:C24H19N7O4S
    Color and Shape:Solid
    Molecular weight:501.52

    Ref: TM-T63400

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • DV 7028 hydrochloride

    CAS:
    DV 7028 hydrochloride is a 5-HT2A receptor antagonist.
    Formula:C21H26ClFN4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:436.91

    Ref: TM-T22753

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (RS)-Minesapride

    CAS:
    Minesapride is a serotonin receptor agonist.
    Formula:C21H31ClN4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.95

    Ref: TM-T28043

    25mg
    2,043.00€
    50mg
    2,682.00€
    100mg
    3,600.00€
  • S20928

    CAS:
    S20928 is an antagonist of melatonin receptor.
    Formula:C17H19NO
    Color and Shape:Solid
    Molecular weight:253.34

    Ref: TM-T28644

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LY 206130

    CAS:
    LY 206130 is an antagonist of serotonin 5-HT1A.
    Formula:C17H24N2O2
    Color and Shape:Solid
    Molecular weight:288.38

    Ref: TM-T27894

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Afurolol Hydrochloride

    CAS:
    Afurolol Hydrochloride (DL 071-IT) is a non-selective β-adrenergic receptor antagonist. DL 071 IT exhibits intrinsic sympathomimetic activity.
    Formula:C15H22ClNO4
    Purity:98.86%
    Color and Shape:Solid
    Molecular weight:315.79

    Ref: TM-T5450

    1mg
    95.00€
    5mg
    195.00€
    10mg
    293.00€
    25mg
    519.00€
    50mg
    750.00€
    100mg
    1,046.00€
    200mg
    1,410.00€
  • RS 15385-197

    CAS:
    RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.
    Formula:C18H26N2O3S
    Color and Shape:Solid
    Molecular weight:350.48

    Ref: TM-T26134

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Lesopitron dihydrochloride

    CAS:
    Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.
    Formula:C15H23Cl3N6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:393.74

    Ref: TM-T11839

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Alclofenac sodium

    CAS:
    Alclofenac sodium is an anti-inflammatory utilized in the treatment of rheumatoid arthritis.
    Formula:C11H11ClNaO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:249.65

    Ref: TM-T25036

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Chloracyzine

    CAS:
    Chloracyzine lowers heart oxygen use, shrinks coronary flow after brief dilation, slightly ups heart rate and arterial pressure.
    Formula:C19H21ClN2OS
    Color and Shape:Solid
    Molecular weight:360.9

    Ref: TM-T25237

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Garomefrine HCl

    CAS:
    Garomefrine HCl, a α1A-adrenoceptor agonist, is potential for the treatment of urinary incontinence.
    Formula:C9H14ClFN2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:284.73

    Ref: TM-T27401

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Viprostol

    CAS:
    Viprostol is an agent of prostaglandin antihypertensive.
    Formula:C23H36O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.53

    Ref: TM-T24938

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GS 283

    CAS:
    GS 283 is a Ca(2+) antagonist. GS 283 is also a weak histamine and muscarinic receptor blocker in rat and guinea pig tracheal smooth muscles.
    Formula:C17H17NO3
    Color and Shape:Solid
    Molecular weight:283.32

    Ref: TM-T27435

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LBP-1

    CAS:
    LBP-1 is a cannabinoid receptor type 1 (CB1) agonist.
    Formula:C23H29ClN6O3
    Color and Shape:Solid
    Molecular weight:472.97

    Ref: TM-T27803

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Seproxetine HCl

    CAS:
    Seproxetine HCl, a more active enantiomer of N-desmethyl metabolite fluoxetine, works by selectively inhibiting the serotonin uptake carrier.
    Formula:C16H17ClF3NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:331.76

    Ref: TM-T26184

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GSK1059865

    CAS:
    GSK1059865 is a potent antagonist of the orexin 1 receptor.
    Formula:C20H23BrFN3O2
    Color and Shape:Solid
    Molecular weight:436.32

    Ref: TM-T11477

    2mg
    101.00€
    25mg
    662.00€
    50mg
    860.00€
    100mg
    1,521.00€
  • PNU-96391

    CAS:
    PNU-96391 (OSU-6162) is an antagonist of dopamine D2 and a partial agonist of 5-HT2A. PNU-96391 can be used in research on the treatment of chronic diseases.
    Formula:C15H23NO2S
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:281.41

    Ref: TM-T28435

    1mg
    77.00€
    5mg
    155.00€
    10mg
    221.00€
    25mg
    338.00€
    50mg
    472.00€
    100mg
    632.00€
    200mg
    843.00€
    1mL*10mM (DMSO)
    145.00€
  • MS437

    CAS:
    MS437 is a potent TSH receptor agonist.
    Formula:C22H24N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.44

    Ref: TM-T24502

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LG 82-4-00

    CAS:
    LG 82-4-00 is an inhibitor of thromboxane.
    Formula:C10H11ClN2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:274.72

    Ref: TM-T25709

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BGC201531

    CAS:

    BGC201531 (AP-1531) is a EP4 antagonist for the treatment of acute migraine.

    Formula:C26H28N2O6S
    Purity:98.51% - 99.33%
    Color and Shape:Solid
    Molecular weight:496.58

    Ref: TM-T8993

    1mg
    136.00€
    5mg
    320.00€
    10mg
    465.00€
    25mg
    777.00€
    50mg
    1,074.00€
    100mg
    1,454.00€
  • LY 163443

    CAS:
    LY 163443 is an dual receptor antagonist of LTD4 and LTE4.
    Formula:C20H22N4O3
    Color and Shape:Solid
    Molecular weight:366.41

    Ref: TM-T27877

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • FR 121196

    CAS:
    FR 121196, a potential antidementia drug, ameliorates the impaired memory of rat in the Morris water maze.
    Formula:C12H16FN3O3S
    Color and Shape:Solid
    Molecular weight:301.34

    Ref: TM-T27361

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A23887

    CAS:
    A23887 is a potentially neuroleptic tetracyclic spiro amine that has affinity for dopamine D-2 receptors.
    Formula:C22H24ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:337.89

    Ref: TM-T26472

    25mg
    1,783.00€
  • SID7970631

    CAS:
    SID7970631 is an isoquinolinone analogue, a selective and potent submicromolar SF-1 inhibitor with an IC50 of 260 nM. SID7970631 can be used to study cancer.
    Formula:C24H24N2O7
    Color and Shape:Solid
    Molecular weight:452.46

    Ref: TM-T62757

    25mg
    690.00€
    50mg
    895.00€
    100mg
    1,404.00€