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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5964 products of "GPCR/G-Protein"

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  • PA-9

    CAS:
    PA-9 is the first small-molecule PAC1 receptor antagonist.
    Formula:C17H18N6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:338.36

    Ref: TM-T24585

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Mivazerol

    CAS:
    Mivazerol is an alpha 2-adrenoceptor agonist.
    Formula:C11H11N3O2
    Color and Shape:Solid
    Molecular weight:217.22

    Ref: TM-T71114

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Vasopressin V2 receptor antagonist 1

    CAS:
    Vasopressin V2 receptor antagonist 1 (Compound 4g) is a vasopressin V2receptor (V2R) antagonist (Ki: 3.8 nM). dominant polycystic kidney disease (ADPKD).
    Formula:C33H37ClN4O4
    Color and Shape:Solid
    Molecular weight:589.12

    Ref: TM-T64174

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • 5-OxoETE methyl ester

    CAS:
    5-OxoETE methyl ester is a 5-oxoETE ester, an OXER1 agonist with stronger β-arrestin response, EC50 = 1.54 μM.
    Formula:C21H32O3
    Color and Shape:Solid
    Molecular weight:332.48

    Ref: TM-T37304

    25µg
    305.00€
    50µg
    577.00€
    100µg
    1,063.00€
    250µg
    2,395.00€
  • threo Ifenprodil hemitartrate

    CAS:
    σ receptor agonist and NR2B subunit-selective NMDA receptor antagonist
    Formula:C21H27NO2C4H6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:400.49

    Ref: TM-T23457

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ethiazide

    CAS:
    Ethiazide is a benzothiadiazine sulfonamide derivative belonging to the class of the thiazide diuretics.
    Formula:C9H12ClN3O4S2
    Color and Shape:Solid
    Molecular weight:325.79

    Ref: TM-T31697

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 4-Chloro Trazodone hydrochloride

    CAS:
    4-Chloro Trazodone HCl is a Trazodone isomer, an antidepressant for anxiety disorders.
    Formula:C19H23Cl2N5O
    Color and Shape:Solid
    Molecular weight:408.32

    Ref: TM-T72119

    1mg
    96.00€
    5mg
    261.00€
    10mg
    480.00€
  • PF 10040

    CAS:
    PF 10040 is an antagonist of platelet activating factor (PAF).
    Formula:C20H24ClNO2
    Color and Shape:Solid
    Molecular weight:345.86

    Ref: TM-T28359

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Noberastine maleate

    CAS:
    Noberastine maleate, a fast-acting furan-derived H1 antagonist, peaks at 4 hours with minimal CNS effects and maximal efficacy at 30 mg/day.
    Formula:C25H29N5O9
    Color and Shape:Solid
    Molecular weight:543.53

    Ref: TM-T71425

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TC 1

    CAS:
    σ1 receptor ligand
    Formula:C19H20FNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.37

    Ref: TM-T23423

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L-817,818

    CAS:
    somatostatin sst5 receptor agonist
    Formula:C33H36N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:536.66

    Ref: TM-T22907

    10mg
    1,279.00€
  • Fertirelin acetate

    CAS:
    Fertirelin acetate is a gonadotropin-releasing hormone (GnRH) agonist.
    Formula:C55H74N16O13
    Color and Shape:Solid
    Molecular weight:1167.29

    Ref: TM-T68915

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Oxypertine

    CAS:
    Oxypertine, an indole-derived antipsychotic, treats psychoses like mania, schizophrenia, and severe anxiety, akin to chlorpromazine.
    Formula:C23H29N3O2
    Color and Shape:Solid
    Molecular weight:379.5

    Ref: TM-T28282

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PM226

    CAS:
    CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.
    Formula:C22H31NO3
    Color and Shape:Solid
    Molecular weight:357.49

    Ref: TM-T37815

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Anitrazafen

    CAS:
    Anitrazafen is a locally effective anti-inflammatory agent that has been shown to have COX-2 inhibitor activity.
    Formula:C18H17N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:307.35

    Ref: TM-T14292

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Usmarapride free base

    CAS:
    Usmarapride free base (SUVN-D4010 free base) is a partial agonist of 5-HT4 receptors, used in Alzheimer's disease research.
    Formula:C21H29N5O2
    Purity:99.91% - 99.91%
    Color and Shape:Solid
    Molecular weight:383.49

    Ref: TM-T34751

    1mg
    194.00€
  • Way 100135

    CAS:
    WAY-100135: research drug, phenylpiperazine, potent 5-HT1A antagonist, partial 5-HT1D agonist, minor 5-HT1B activity.
    Formula:C24H33N3O2
    Color and Shape:Solid
    Molecular weight:395.54

    Ref: TM-T35104

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Tiamenidine hydrochloride

    CAS:
    Tiamenidine hydrochloride is a centrally-acting alpha1 adrenergic receptor antagonist.
    Formula:C8H11Cl2N3S
    Color and Shape:Solid
    Molecular weight:252.16

    Ref: TM-T69169

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CIA-1 hcl(452087-38-6 Free base)

    CAS:
    CIA-1 inhibits the nuclear receptor COUP-TFII, with IC50s ranging from 1.2 μM to 7.6 μM in prostate cancer cell lines.CIA-1 inhibits the growth of a variety of
    Formula:C17H20ClN3O2S
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:365.88

    Ref: TM-T71534

    10mg
    540.00€
    50mg
    2,252.00€
  • Q8 hydrochloride

    CAS:
    Q8 is an antagonist of cysteinyl leukotreine receptor. Q8 inhibits VEGF-independent angiogenesis.
    Formula:C17H14ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:299.75

    Ref: TM-T28481

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Setastine HCl

    CAS:
    Setastine HCl is a potent antagonist of histamine H1-receptor mediated responses.
    Formula:C22H29Cl2NO
    Color and Shape:Solid
    Molecular weight:394.38

    Ref: TM-T71791

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Clopenthixol

    CAS:
    Clopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.
    Formula:C22H25ClN2OS
    Color and Shape:Solid
    Molecular weight:400.96

    Ref: TM-T68193

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Paltusotine HCl

    CAS:
    Paltusotine, also known as CRN00808, is a somatostatin receptor agonist.
    Formula:C27H24Cl2F2N4O
    Color and Shape:Solid
    Molecular weight:529.41

    Ref: TM-T69836

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CID1792197

    CAS:
    CID1792197 is a selective agonist of GPR55.
    Formula:C24H23N3O4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:481.59

    Ref: TM-T27017

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SC 53116 Hydrochloride

    CAS:
    SC 53116 Hydrochloride is selective agonist of the newly identified serotonin 5-HT4 receptor subtype.
    Formula:C16H23Cl2N3O2
    Color and Shape:Solid
    Molecular weight:360.28

    Ref: TM-T28696

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Pd 158771

    CAS:
    Pd 158771 is a D2 and 5-HT1A agonist.
    Formula:C22H31N5
    Color and Shape:Solid
    Molecular weight:365.52

    Ref: TM-T70081

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • WRC-0571

    CAS:
    WRC-0571 is a highly potent, selective antagonist of A1 adenosine receptors.
    Formula:C17H26N6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:330.43

    Ref: TM-T29162

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GR 196429

    CAS:
    GR 196429: MT1-selective melatonin receptor agonist; induces sleep, alters circadian rhythm, stimulates melatonin in mice.
    Formula:C14H18N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:246.3

    Ref: TM-T27430

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Daledalin

    CAS:
    Daledalin, an unmarketed 1970s antidepressant, is a selective norepinephrine reuptake inhibitor without serotonergic or dopaminergic effects.
    Formula:C19H24N2
    Color and Shape:Solid
    Molecular weight:280.41

    Ref: TM-T69788

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Fenspiride-d5

    CAS:
    Fenspiride-d5: internal standard for GC/LC-MS quantification, H1 antagonist, NSAID, anti-inflammatory, selective PDE4,5,3 inhibitor.
    Formula:C15H15D5N2O2
    Color and Shape:Solid
    Molecular weight:265.36

    Ref: TM-T71141

    1mg
    1,018.00€
    5mg
    3,312.00€
  • SGC agonist 2

    CAS:
    SGC agonist 2 is a potent activator for cardiovascular and fibrotic diseases, per patent WO2021219088A1, compound 031.
    Formula:C23H17F2N7O2
    Color and Shape:Solid
    Molecular weight:461.42

    Ref: TM-T62909

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Sch 33303

    CAS:
    Sch 33303 is an antiallergy agents.
    Formula:C19H16N2O3
    Color and Shape:Solid
    Molecular weight:320.34

    Ref: TM-T28714

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GW848687X

    CAS:
    GW848687X, a potent and selective prostaglandin EP1 receptor antagonist, is used for the treatment of inflammatory pain.
    Formula:C24H18ClF2NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:441.85

    Ref: TM-T27517

    1mg
    537.00€
    5mg
    2,277.00€
    500µg
    290.00€
  • SLM6031434 (free base)

    CAS:
    SLM6031434 (free base) is an inhibitor of sphingosine kinase type 2 (SphK2). It consists of pedant 1-guanidino-2-phenyloxadiazolylpyrrolidine group.
    Formula:C22H30F3N5O2
    Color and Shape:Solid
    Molecular weight:453.5

    Ref: TM-T70071

    1mg
    172.00€
    5mg
    512.00€
    10mg
    750.00€
  • ChemR23-IN-4

    CAS:
    ChemR23-IN-4 is a potent inhibitor of orally active ChemR23, capable of acting on human ChemR23 (IC50: 17 nM).
    Formula:C27H26N6O3
    Color and Shape:Solid
    Molecular weight:482.53

    Ref: TM-T63195

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Cetrorelix Acetate

    CAS:
    Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.
    Formula:C70H92ClN17O14·xC2H4O2
    Purity:97.96%
    Color and Shape:Solid
    Molecular weight:1491.11

    Ref: TM-T5520

    1mg
    46.00€
    5mg
    80.00€
    10mg
    114.00€
    25mg
    236.00€
    50mg
    380.00€
    100mg
    595.00€
    1mL*10mM (DMSO)
    170.00€
  • MAT2A-IN-1

    CAS:
    MAT2A-IN-1 suppresses MAT2A, key for MTAP-deficient cancer cell growth; studied for gastric, colon, liver, pancreatic cancers.
    Formula:C29H28F2N6O4
    Color and Shape:Solid
    Molecular weight:562.57

    Ref: TM-T63975

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • MRS2298

    CAS:
    MRS2298, a potent antagonists of the P2Y 1 receptor, has antiaggregatory activity in human platelets.
    Formula:C10H16ClN5O8P2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:431.66

    Ref: TM-T28100

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ro 60-0175 fumarate

    CAS:
    5-HT2 receptor agonist
    Formula:C15H16ClFN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:342.75

    Ref: TM-T23246

    1mg
    105.00€
    5mg
    268.00€
  • Carcinine

    CAS:
    Carcinine ditrifluoroacetate is a H3 receptor antagonist.
    Formula:C8H14N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:182.22

    Ref: TM-T22624

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L-Alprenolol

    CAS:
    L-Alprenolol is a non-selective beta-blocker and a 5-HT1A and 5-HT1B receptor antagonist.
    Formula:C15H23NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:249.35

    Ref: TM-T24386

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MRS1186

    CAS:
    MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).
    Formula:C16H12ClN5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:341.75

    Ref: TM-T16138

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Phenoprolamine Hydrochloride

    CAS:
    Phenoprolamine HCl: α1 blocker with anti-hypertensive, brain, and heart protection; inhibits CYP2D/3A, crosses the blood-brain barrier.
    Formula:C21H30ClNO3
    Color and Shape:Solid
    Molecular weight:379.92

    Ref: TM-T28400

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PF-4479745

    CAS:
    PF-4479745 ia a potent and selective agonist of 5-HT2C receptor.
    Formula:C17H22N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:282.38

    Ref: TM-T28384

    1mg
    427.00€
  • Remoxipride

    CAS:
    Remoxipride is an antipsychotic agent. Remoxipride is specific for dopamine D2 receptors.
    Formula:C16H23BrN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:371.27

    Ref: TM-T28514

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (RS)-Butyryltimolol

    CAS:
    (RS)-Butyryltimolol, a racemic prodrug of Timolol, enhances its corneal absorption and acts as a β-adrenergic blocker.
    Formula:C17H30N4O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.51

    Ref: TM-T13439

    2mg
    63.00€
  • Guanadrel Sulfate

    CAS:
    Guanadrel Sulfate, a postganglionic blocker, is stored in neurons via the norepinephrine pump.
    Formula:C10H21N3O6S
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:311.35

    Ref: TM-T9097L

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • 2-Acetylbenzoic acid

    CAS:
    2-Acetylbenzoic acid outperforms 2-propionyloxybenzoic in hindering platelet function and PG synthesis; both similar in blocking PGI2 creation.
    Formula:C9H8O3
    Purity:99.62%
    Color and Shape:Off-White Solid
    Molecular weight:164.16

    Ref: TM-TMA0536

    1g
    34.00€
    1mL*10mM (DMSO)
    34.00€
  • WAY 629

    CAS:
    WAY 629 is a selective SR-2C agonist that also act as potent 5-HT2C receptor agonists.
    Formula:C15H18N2
    Color and Shape:Solid
    Molecular weight:226.32

    Ref: TM-T69067

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Benzatropine

    CAS:
    Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.
    Formula:C21H25NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:307.43

    Ref: TM-T23781

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GAT229

    CAS:
    GAT229 is a CB1 positive modulator, enhancing CB agonist activity without direct activation; influences binding, signaling, and lowers ocular pressure in mice.
    Formula:C22H18N2O2
    Color and Shape:Solid
    Molecular weight:342.39

    Ref: TM-T38204

    1mg
    379.00€
  • Pargolol

    CAS:
    Pargolol is a beta adrenergic receptor antagonist.
    Formula:C16H23NO3
    Color and Shape:Solid
    Molecular weight:277.36

    Ref: TM-T69217

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Colterol (free base)

    CAS:
    Colterol: short-acting β2 agonist; Bitolterol prodrug treats asthma, COPD bronchospasm.
    Formula:C12H19NO3
    Color and Shape:Solid
    Molecular weight:225.28

    Ref: TM-T70089

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BN-81,674

    CAS:
    BN-81,674 is a bioactive chemical.
    Formula:C30H38N4
    Color and Shape:Solid
    Molecular weight:454.65

    Ref: TM-T30553

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • BMY-25271

    CAS:
    BMY-25271 is an antagonist of histamine H2 receptor.
    Formula:C12H19N5O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.44

    Ref: TM-T10575

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • γ-Linolenic acid ethyl ester

    CAS:
    γ-Linolenic acid ethyl ester (Ethyl γ-linolenate) is a leukotriene B 4 receptor 4 (LTB 4 ) antagonist which has a potential anti-inflammatory effect[1].
    Formula:C20H34O2
    Color and Shape:Solid
    Molecular weight:306.48

    Ref: TM-T41235

    1g
    1,288.00€
    50mg
    114.00€
    100mg
    208.00€
    250mg
    489.00€
  • Alaproclate (hydrochloride)

    CAS:
    Alaproclate, an SSRI, enhances serotonin and SIRT1, hinders NMDA and K+ currents in neurons, and shows antidepressant-like effects in rats.
    Formula:C13H19Cl2NO2
    Color and Shape:Solid
    Molecular weight:292.2

    Ref: TM-T36521

    5mg
    230.00€
    10mg
    399.00€
  • CP 66713

    CAS:
    CP-66713 is an adenosine A2 receptor antagonist.
    Formula:C15H10ClN5
    Color and Shape:Solid
    Molecular weight:295.73

    Ref: TM-T31026

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • AM-211 sodium

    CAS:
    AM-211 sodium: potent DP2 receptor antagonist, active against allergic inflammation, selective, and orally bioavailable in rats and dogs.
    Formula:C27H26F3N2NaO4
    Color and Shape:Solid
    Molecular weight:522.5

    Ref: TM-T71088

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Levemopamil HCl

    CAS:
    Levemopamil HCl is used as a calcium channel blocker.
    Formula:C23H31ClN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:370.96

    Ref: TM-T25692L

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SB 206553 hydrochloride

    CAS:
    SB 206553 hydrochloride is a 5-HT2C inverse agonist and a 5-HT2C/5-HT2B receptor antagonist with anxiolytic activity, useful for studying neurological disorders
    Formula:C17H17ClN4O
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:328.8

    Ref: TM-T23314

    1mg
    58.00€
    5mg
    124.00€
    10mg
    192.00€
    25mg
    386.00€
    50mg
    556.00€
  • M-25

    CAS:
    M-25 is a Smoothened antagonist and inhibitor of the Hedgehog pathway.
    Formula:C23H29N3O2
    Color and Shape:Solid
    Molecular weight:379.5

    Ref: TM-T71299

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • NVS-CRF38

    CAS:
    NVS-CRF38 is an antagonist of corticotropin-releasing factor receptor 1 (CRF1).
    Formula:C19H21N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.4

    Ref: TM-T12276

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • AR-A 2

    CAS:
    AR-A 2, a selective 5-HT1B antagonist; high guinea pig 5-HT1B/1D affinity (Ki: 0.24, 0.47 nM); 10x less for 5-HT1D (Ki: 5 nM).
    Formula:C27H36N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.6

    Ref: TM-T10360

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • BFE-55

    CAS:
    BFE-55 is derivative of befunolol (a beta-adrenergic partial agonist). BFE-55 interacts with only the high affinity sites in beta-adrenoceptors
    Formula:C14H19NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:249.31

    Ref: TM-T26783

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (Rac)-Upacicalcet

    CAS:
    (Rac)-Upacicalcet, a racemate, is an IV calcimimetic targeting parathyroid receptors to lower PTH, possibly treating SHPT.
    Formula:C11H14ClN3O6S
    Color and Shape:Solid
    Molecular weight:351.76

    Ref: TM-T61232

    25mg
    1,314.00€
  • Thioperamide

    CAS:
    histamine H3 and H4 antagonist/inverse agonist
    Formula:C15H24N4S
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:292.44

    Ref: TM-T23456

    10mg
    502.00€
    50mg
    2,070.00€
  • Y2 Antagonist 36

    CAS:
    Y2 Antagonist 36 is a highly potent, soluble and selective antagonist of NPY Y2.
    Formula:C27H29ClN4O3
    Color and Shape:Solid
    Molecular weight:493

    Ref: TM-T29171

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ro 22-9194

    CAS:
    Ro 22-9194, a class I antiarrhythmic, reduces upstroke velocity and shortens action potential in guinea-pig hearts at ≥10 μM.
    Formula:C19H27Cl2N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:384.35

    Ref: TM-T28567

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • A2A receptor antagonist 3

    CAS:
    A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM).
    Formula:C26H26N6O2
    Color and Shape:Solid
    Molecular weight:454.52

    Ref: TM-T62797

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • SMM-189

    CAS:
    SMM-189 is a potent and selective CB2 inverse agonist.
    Formula:C19H12Cl2O3
    Color and Shape:Solid
    Molecular weight:359.2

    Ref: TM-T28819

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L-670,596

    CAS:
    L-670,596 is a thromboxane A2/prostaglandin endoperoxide receptor antagonist.
    Formula:C22H21F2NO4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.47

    Ref: TM-T22897

    100mg
    2,250.00€
  • T 82

    CAS:
    T 82 is an antagonist of 5-HT3 and inhibitor of acetylcholinesterase (AChE) and used for the treatment of Alzheimer's Disease.
    Formula:C56H62N6O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:947.146

    Ref: TM-T13239

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Lexipafant

    CAS:
    Lexipafant is a platelet-activating factor (PAF) receptor antagonist.
    Formula:C23H30N4O4S
    Color and Shape:Solid
    Molecular weight:458.57

    Ref: TM-T27821

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Todralazine

    CAS:
    Todralazine is an anti-hypertensive agent and acts as a β2AR blocker. It also has an antioxidant and free radical scavenging activity.
    Formula:C11H12N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:232.24

    Ref: TM-T17112

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Lu AA41063

    CAS:
    Lu AA41063 is a potent and selective antagonist of the hA2A receptor.
    Formula:C16H17F2N3O2S
    Color and Shape:Solid
    Molecular weight:353.39

    Ref: TM-T24418

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SKF-83566 hydrobromide

    CAS:
    D1-like dopamine receptor antagonist
    Formula:C17H19BrClNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:368.7

    Ref: TM-T23362

    5mg
    200.00€
    10mg
    314.00€
    25mg
    620.00€
  • A1AR antagonist 6

    CAS:
    A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].
    Formula:C17H15N3O2
    Color and Shape:Solid
    Molecular weight:293.32

    Ref: TM-T60615

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SB 235375

    CAS:
    SB 235375 is a potent and selective antagonist of neurokinin-3 receptor with a low central nervous system-penetrant.
    Formula:C27H24N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.49

    Ref: TM-T28676

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • N-Salicyloyltryptamine

    CAS:
    N-Salicyloyltryptamine (STP): a tryptamine with anticonvulsant, anti-inflammatory, analgesic effects; inhibits Na+, Ca2+, K+ channels (IC50 34.6 μM).
    Formula:C17H16N2O2
    Color and Shape:Solid
    Molecular weight:280.32

    Ref: TM-T60526

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CAY10535

    CAS:
    CAY10535 is a selective TPβ antagonist (IC50 = 99 nM for TPβ vs 1970 nM for TPα), weakly affects platelets (IC50 = 985 nM).
    Formula:C18H21N3O7S
    Color and Shape:Solid
    Molecular weight:423.44

    Ref: TM-T36550

    1mg
    118.00€
    5mg
    515.00€
    10mg
    888.00€
    25mg
    1,882.00€
  • MS 245 oxalate

    CAS:
    MS 245 oxalate is a 5-HT6 antagonist.
    Formula:C21H24N2O7S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:448.49

    Ref: TM-T23029

    1mg
    124.00€
    5mg
    462.00€
    10mg
    695.00€
  • LY 225910

    CAS:
    LY 225910 is a CCK2 receptor antagonist.
    Formula:C27H24BrN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:502.4

    Ref: TM-T22941

    10mg
    470.00€
    50mg
    1,918.00€
  • A68930

    CAS:
    A 68930 is a dopamine D-1 receptor antagonist. A 68930 inhibits NLRP3 inflammasome activity.
    Formula:C16H17NO3
    Color and Shape:Solid
    Molecular weight:271.31

    Ref: TM-T26432

    25mg
    3,492.00€
    50mg
    5,239.00€
    100mg
    7,857.00€
  • DH97

    CAS:
    MT2 melatonin receptor antagonist
    Formula:C22H26N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:334.45

    Ref: TM-T22721

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A 61603

    CAS:
    Cixutumumab (IMC-A12) is a humanized IgG monoclonal antibody targeting the IGF1R with anticancer activity.
    Formula:C14H20BrN3O3S
    Color and Shape:Solid
    Molecular weight:390.3

    Ref: TM-T21927

    1mg
    105.00€
    5mg
    325.00€
    10mg
    444.00€
  • Bemesetron

    CAS:
    Bemesetron (MDL 72222) is a selective antagonist of 5-HT3 (IC50 = 0.33 nM) with neuroprotective effects.
    Formula:C15H17Cl2NO2
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:314.21

    Ref: TM-T14526

    10mg
    52.00€
    25mg
    66.00€
    50mg
    89.00€
  • LY 203647

    CAS:
    LY 203647 is a antagonist of leukotriene D4 and E4 receptor.
    Formula:C21H30N8O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:442.51

    Ref: TM-T27893

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Metazosin

    CAS:
    Metazosin is an antihypertensive agent that replaces 3H-prazosin from its bond to alpha-1 receptors of the cerebral cortex.
    Formula:C18H25N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:375.42

    Ref: TM-T25793

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JNJ-27141491

    CAS:
    JNJ-27141491 is a potent, noncompetitive antagonist of human CCR2.
    Formula:C17H15F2N3O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:379.38

    Ref: TM-T27674

    25mg
    1,444.00€
  • A 49816

    CAS:
    A 49816 is a high-ceiling diuretic.
    Formula:C18H17Cl2NO5
    Color and Shape:Solid
    Molecular weight:398.24

    Ref: TM-T29496

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Verlukast

    CAS:
    Verlukast (MK-0679) is a selective, orally active leukotriene D4 receptor antagonist for use in bronchial asthma research.
    Formula:C26H27ClN2O3S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:515.09

    Ref: TM-T19674

    50mg
    723.00€
    100mg
    1,094.00€
  • Fallypride

    CAS:
    Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.
    Formula:C20H29FN2O3
    Purity:98.97% - >99.99%
    Color and Shape:Solid
    Molecular weight:364.45

    Ref: TM-T70302

    1mg
    359.00€
    5mg
    842.00€
    10mg
    1,035.00€
    25mg
    1,663.00€
    50mg
    2,072.00€
    100mg
    2,660.00€
    1mL*10mM (DMSO)
    677.00€
  • Stresson

    CAS:
    Stresson is a beta-blocking agent bunitrolol.
    Formula:C14H21ClN2O2
    Color and Shape:Solid
    Molecular weight:284.78

    Ref: TM-T34724

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • VUF 5681 dihydrobromide

    CAS:
    histamine H3 receptor silent antagonist
    Formula:C11H21Br2N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:355.11

    Ref: TM-T23519

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TR4161

    CAS:
    TR4161 is a prostaglandin bronchodilator of low tracheobronchial irritancy.
    Formula:C20H36O4
    Color and Shape:Solid
    Molecular weight:340.5

    Ref: TM-T34913

    1mg
    200.00€
    5mg
    828.00€
    10mg
    1,431.00€
    500µg
    112.00€
  • L-775,606

    CAS:
    L-775,606 is a selective agonist of 5-hydroxytryptamine 1D.
    Formula:C25H29FN6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:432.54

    Ref: TM-T27782

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • FK-1052 HCl

    CAS:
    FK-1052 HCl is a serotonin 3 & 4 dual receptor antagonist.
    Formula:C18H20ClN3O
    Color and Shape:Solid
    Molecular weight:329.83

    Ref: TM-T71045

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Photoregulin1

    CAS:
    Photoregulin1 modulates Nr2e3, slows photoreceptor degeneration in RhoP23H, Pde6brd1 mouse RP models.
    Formula:C21H23N3O2S
    Color and Shape:Solid
    Molecular weight:381.49

    Ref: TM-T28409

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Savoxepin mesylate

    CAS:
    Savoxepin mesylate, a tetracyclic cyano-dibenzoxepino-azepine derivative, has potent antidopaminergic activity.
    Formula:C26H30N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:466.59

    Ref: TM-T28666

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€