
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,994 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(59 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5964 products of "GPCR/G-Protein"
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MK-8133
CAS:MK-8133 is an antagonist of orexin-2 selective receptor with favorable development properties.Formula:C23H21N5O2Color and Shape:SolidMolecular weight:399.45Methyldopate hydrochloride
CAS:Methyldopate HCl is an agent of antihypertensive.Formula:C12H18ClNO4Color and Shape:SolidMolecular weight:275.73A-943931
CAS:A-943931 is a selective histamine H4 receptor antagonist with human and rat Ki values of 4.6 and 3.8 nM respectively.inhibits the scratching response in mice.Formula:C17H21N5Purity:99.79%Color and Shape:SolidMolecular weight:295.38BRL 37344 sodium
CAS:BRL 37344 sodium is a specific agonist of the β3-adrenergic receptor. The treatment of BRL 37344 sodium significantly lowers the bodyweight of obese mice.Formula:C19H22ClNNaO4Purity:98%Color and Shape:SolidMolecular weight:386.83(Rac)-HAMI 3379
CAS:HAMI 3379: potent CysLT2 receptor blocker; protects against acute/subacute brain injury; reduces microglia inflammation.Formula:C34H45NO8Purity:98%Color and Shape:SolidMolecular weight:595.72Fluprostenol methyl ester
CAS:Fluprostenol, a vet-approved luteolytic, has an isopropyl ester, travoprost, used as an eye pressure reducer. CAY10532 is its methyl ester form.Formula:C24H31F3O6Color and Shape:SolidMolecular weight:472.49SB 207710
CAS:SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.Formula:C19H27IN2O4Color and Shape:SolidMolecular weight:474.33QCC-374
CAS:QCC-374 is a prostanoid agonist. It potentially for the treatment of pulmonary arterial hypertension.Formula:C28H33N3O2Purity:98%Color and Shape:SolidMolecular weight:443.58UK 1745
CAS:UK 1745 is a novel drug of cardiotonic.Formula:C16H23ClN2O2Color and Shape:SolidMolecular weight:310.82Zenidolol
CAS:Zenidolol (ICI-118551) is a β2 adrenoceptor blocker with K i values: β2 (0.7 nM), β1 (49.5 nM), β3 (611 nM); used in eye disease research.Formula:C17H27NO2Color and Shape:SolidMolecular weight:277.4CP-195543
CAS:CP-195543 is an effective leukotriene B4 antagonist for the treatment of inflammatory diseases.Formula:C24H19F3O4Color and Shape:SolidMolecular weight:428.4LY288513
CAS:Selective CCK2 receptor antagonistFormula:C22H18BrN3O2Purity:98%Color and Shape:SolidMolecular weight:436.3GSK-269984B
CAS:GSK-269984B is a novel antagonist of EP1 receptor.Formula:C20H14Cl2FNO3Purity:98%Color and Shape:SolidMolecular weight:406.23Guanethidine
CAS:Guanethidine sulphate, made in 1959, lowers blood pressure by disrupting neurotransmitters in sympathetic nerves.Formula:C10H22N4Color and Shape:SolidMolecular weight:198.31EP4 receptor antagonist 4
CAS:EP4 receptor antagonist 4 is an agonist of EP4 receptor (human pEC 50 = 6.3) [1].Formula:C19H14N2OSColor and Shape:SolidMolecular weight:318.395-HT7 agonist 2
CAS:Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.Formula:C23H29N3OColor and Shape:SolidMolecular weight:363.5SKF-75670 Hydrobromide
CAS:SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.Formula:C17H20BrNO2Color and Shape:SolidMolecular weight:350.25Zicronapine
CAS:Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.Formula:C22H27ClN2Color and Shape:SolidMolecular weight:354.92A 55453
CAS:A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.Formula:C25H32N6O3Color and Shape:SolidMolecular weight:464.56FRG8701
CAS:FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.Formula:C22H30N2O4SPurity:98%Color and Shape:SolidMolecular weight:418.55NAEPA
CAS:NAEPA, an LPA mimetic, is a selective agonist of the lysophosphatidic acid-1 (LPA1) receptor.Formula:C20H40NO5PPurity:98%Color and Shape:SolidMolecular weight:405.51EP2 receptor antagonist-1
CAS:EP2 receptor antagonist-1: reversible, potent, depends on agonist; anti-inflammatory.Formula:C24H22N4O5Color and Shape:SolidMolecular weight:446.46WB403
CAS:WB403 activates TGR5, lowers fasting/postprandial glucose and HbA1c, enhances glucose tolerance, and normalizes pancreatic α/β-cells in diabetic mice.Formula:C19H19BrN2OSPurity:98%Color and Shape:SolidMolecular weight:403.34PD-135666
CAS:PD-135666 is an antagonist of CCK receptor.Formula:C33H39N3O5Purity:98%Color and Shape:SolidMolecular weight:557.68Naronapride
CAS:Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.Formula:C27H41ClN4O5Color and Shape:SolidMolecular weight:537.09LY 219057
CAS:LY 219057 is a potent, competitive, and specific antagonist of CCK receptor on the exocrine pancreas.Formula:C23H17ClF3N3OSColor and Shape:SolidMolecular weight:475.91CB1R Allosteric modulator 1
CAS:CB1R modulator 1 (compound 11), a potent CB1R inhibitor, decreases activity of orthosteric ligands.Formula:C24H24ClN3OColor and Shape:SolidMolecular weight:405.92S-777469
CAS:S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.Formula:C23H27FN2O4Color and Shape:SolidMolecular weight:414.47CB2 receptor agonist 3
CAS:GP 2A is a selective agonist of CB2 receptor.Formula:C24H23Cl2N3OColor and Shape:SolidMolecular weight:440.36SANT-2
CAS:SANT-2 is a potent inhibitor of Shh signaling pathway.Formula:C23H20ClN3O4Color and Shape:SolidMolecular weight:437.88Nivasorexant
CAS:Nivasorexant is a potent antagonist of the orexin receptor.Formula:C23H23N7O2Color and Shape:SolidMolecular weight:429.47ATL-801
CAS:ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.Formula:C24H25N7O3Color and Shape:SolidMolecular weight:459.5Povafonidine
CAS:Povafonidine (PGE-6201204), an alpha-2 adrenoreceptor agonist, constricts vessels, reduces congestion for nasal research.Formula:C11H13N5Color and Shape:SolidMolecular weight:215.25Ziprasidone mesylate trihydrate
CAS:Ziprasidone mesylate hydrate is an oral 5-HT/D2 antagonist with Ki: D2=4.8nM, 5-HT2A=0.42nM, 5-HT1A=3.4nM in rats.Formula:C22H31ClN4O7S2Color and Shape:SolidMolecular weight:563.08Nebidrazine
CAS:Nebidrazine is an alpha-adrenoceptor agonist.Formula:C9H8Cl2N6Color and Shape:SolidMolecular weight:271.11INCB38579
CAS:INCB38579: Oral, selective H4 antagonist; crosses brain barrier; IC50s - hH4R: 4.8 nM, mH4R: 42 nM, rH4R: 32 nM; anti-inflammatory and antipruritic.Formula:C25H34N6OColor and Shape:SolidMolecular weight:434.58Latanoprost ethyl amide
CAS:Lat-NEt, a latanoprost analog, is an ocular hypotensive prodrug with slower hydrolysis, converting to free acids in corneal tissue.Formula:C25H39NO4Color and Shape:SolidMolecular weight:417.58BAY-u 9773
CAS:BAY-u9773 is a non-selective CysLT receptor antagonist with similar IC50 for CysLT1 and CysLT2, inhibiting LT responses.Formula:C27H36O5SColor and Shape:White OilMolecular weight:472.64Remogliflozin
CAS:Remogliflozin is an effective sodium-glucose transporter 2 inhibitor (Kis = 12.4 and 26 nM for human and rat SGLT2, respectively).Formula:C23H34N2O7Color and Shape:SolidMolecular weight:450.53MAT2A-IN-3
CAS:MAT2A-IN-3: potent MAT2A inhibitor, hinders MTAP-deficient cancer cell growth, potential for cancer research.Formula:C24H16F5N5O3Color and Shape:SolidMolecular weight:517.415-HT2A receptor agonist-2
CAS:Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.Formula:C20H21ClN2O3Color and Shape:SolidMolecular weight:372.85AP-521 (Free base)
CAS:AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.Formula:C20H18N2O3SColor and Shape:SolidMolecular weight:366.43BRD5814
CAS:BRD5814 is a highly brain penetrant β-arrestin biased D2R antagonist.Formula:C21H23ClF3NO2Color and Shape:SolidMolecular weight:413.86Edivoxetine
CAS:Edivoxetine (LY2216684) is a selective norepinephrine reuptake inhibitor for ADHD and depression.Formula:C18H26FNO4Color and Shape:SolidMolecular weight:339.4ChemR23-IN-1
CAS:ChemR23-IN-1 inhibits human and mouse ChemR23 (IC50: 38 nM, 100 nM) and stops CAL-1 chemotaxis induced by Chemerin in vitro.Formula:C28H29N7O2Color and Shape:SolidMolecular weight:495.58BGC-20-1531 free base
CAS:BGC-20-1531 (PGN 1531) free base is a selective and potent prostaglandin EP4 receptor antagonist (pKB: 7.6) that exhibits potential for migraine research.Formula:C26H24N2O6SColor and Shape:SolidMolecular weight:492.54Medroxalol
CAS:Medroxalol (RMI81968), an oral α- & β-adrenergic blocker, has antihypertensive and vasodilatory effects.Formula:C20H24N2O5Color and Shape:SolidMolecular weight:372.42Bopindolol (malonate)
CAS:Bopindolol is a non-selective β-adrenergic receptor antagonist.Formula:C26H32N2O7Color and Shape:SolidMolecular weight:484.549GPR183-IN-2
CAS:GPR183-IN-2 (compound 23) is an effective, orally active inhibitor of GPR183, displaying an IC50 value of 39.45 nM in Ca2+ mobilization assays. This compound has potential applications in research related to cancer, autoimmune diseases, pain, and osteoporosis.
Formula:C19H23BrN2O3Color and Shape:SolidMolecular weight:407.3DuP 734
CAS:DuP 734 is a potent and selective sigma receptor antagonist, functioning as a ligand for both sigma and 5-HT2 receptors, and exhibiting weak affinity towards D2 receptors. It possesses potential antipsychotic activity, potentially devoid of the motor side effects commonly observed with neuroleptics[1][2][3].
Formula:C17H23BrFNOColor and Shape:SolidMolecular weight:356.279GPR183 antagonist-2
CAS:GPR183 antagonist-2 (compound 32), a selective antagonist of GPR183, exhibits excellent water solubility and pharmacokinetic properties. This compound effectively diminishes paw and joint swelling, and reduces gene expression of pro-inflammatory cytokines (MCP-1, MMPs, and VEGF) in a dose-dependent manner within a collagen-induced arthritis (CIA) mouse model. GPR183 antagonist-2 is applicable in researching autoimmune diseases [1].Formula:C20H18F2N4O5Color and Shape:SolidMolecular weight:432.38MoTP
CAS:MoTP is a specific platelet activating factor receptor antagonist that induces ablation of melanocyte. MoTP can be used in cancer research.Formula:C14H21NO2SColor and Shape:SolidMolecular weight:267.39MG 1
CAS:MG 1 is a potent alpha-1 adrenergic receptor antagonist.Formula:C17H25N3O2Purity:98.98% - >99.99%Color and Shape:SolidMolecular weight:303.4I942
CAS:I942 is a novel, selective ACyclic nucleotide (NCN) EPAC1 agonist that activates exchange proteins to regulate inflammatory gene expression in human umbilicalFormula:C20H19NO4SPurity:99.86%Color and Shape:SolidMolecular weight:369.43Iso-SLR 080811
CAS:Iso-SLR 080811 is an isomer of SLR 080811, suitable for relevant research in the life sciences. SLR080811 is a selective SphK2 inhibitor (Ki=1.3 μM).Formula:C21H32ClN5OPurity:98.34%Color and Shape:SolidMolecular weight:405.97CB1R Allosteric modulator 3
CAS:CB1R Allosteric modulator 3 is a CB1R modulator.CB1R Allosteric modulator 3 inhibits cAMP, and can be used for the study of obesity and nicotine addiction.Formula:C22H17ClN2O2Purity:98.18%Color and Shape:SolidMolecular weight:376.84NRA-0160
CAS:NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)Formula:C24H23F2N3OSPurity:98%Color and Shape:SolidMolecular weight:439.52hA2AAR antagonist 1
CAS:Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.Formula:C15H15N5OColor and Shape:SolidMolecular weight:281.31CJ 033466
CAS:CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.Formula:C19H28ClN5OPurity:99.72%Color and Shape:SolidMolecular weight:377.91Ref: TM-T22671
1mg48.00€5mg101.00€10mg170.00€25mg270.00€50mg386.00€100mg520.00€1mL*10mM (DMSO)124.00€Eplivanserin
CAS:Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.Formula:C19H21FN2O2Purity:97.04%Color and Shape:SolidMolecular weight:328.38DOV-216,303 Free Base
CAS:DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.Formula:C11H11Cl2NPurity:96.7%Color and Shape:SolidMolecular weight:228.12EMDT
CAS:EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.Formula:C15H22N2OPurity:97.66% - 99.78%Color and Shape:SolidMolecular weight:246.35Ref: TM-T11183
1mg87.00€2mg118.00€5mg167.00€10mg202.00€25mg449.00€50mg652.00€100mg888.00€500mg1,783.00€1mL*10mM (DMSO)166.00€Chlorazanil
CAS:Chlorazanil is a triazine-based, orally active diuretic that blocks Na+ and Cl– reabsorption in distal tubules, increases renal prostaglandin.Formula:C9H8ClN5Purity:98.89%Color and Shape:SolidMolecular weight:221.65Nedocromil
CAS:Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).Formula:C19H17NO7Purity:95% - 97.34%Color and Shape:SolidMolecular weight:371.34Quinpirole Hydrochloride
CAS:Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and miceFormula:C13H22ClN3Purity:98%Color and Shape:SolidMolecular weight:255.79H3R-IN-1 Hydrochloride
CAS:H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .Formula:C19H24ClN3O3Purity:98%Color and Shape:SolidMolecular weight:377.86Org-12962
CAS:Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).Formula:C10H11ClF3N3Purity:98.34%Color and Shape:SolidMolecular weight:265.665-Carboxamidotryptamine maleate
CAS:5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.Formula:C15H17N3O5Purity:99.88%Color and Shape:SolidMolecular weight:319.31Mirisetron
CAS:Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.Formula:C24H31N3O2Purity:99.88%Color and Shape:SolidMolecular weight:393.52ICI 162,846
CAS:ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.Formula:C11H17F3N6OPurity:97.45%Color and Shape:SolidMolecular weight:306.29PRX-08066 Maleic acid
CAS:PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.Formula:C23H21ClFN5O4SPurity:97.59%Color and Shape:SolidMolecular weight:517.96Ref: TM-T6959
1mg84.00€5mg172.00€10mg233.00€25mg419.00€50mg620.00€100mg882.00€200mg1,198.00€1mL*10mM (DMSO)401.00€Iprindole
CAS:Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].Formula:C19H28N2Purity:99.54%Color and Shape:SolidMolecular weight:284.44Ref: TM-T37015
2mg37.00€5mg52.00€10mg80.00€25mg154.00€50mg266.00€100mg455.00€200mg652.00€1mL*10mM (DMSO)84.00€Thioproperazine
CAS:Thioproperazine (RP 7843) is an orally effective antipsychotic schizophrenia and bipolar disorder, histamine and adrenergic receptor blocker.Formula:C22H30N4O2S2Purity:99.45%Color and Shape:SolidMolecular weight:446.63LPA2 antagonist 2
CAS:LPA2 antagonist 2 is an and LPA2 antagonist (IC50: 28.3 nM) with potential anticancer activity, inhibits LPA3, and can be used for cancer research.Formula:C20H16N2O6Purity:96.13%Color and Shape:SolidMolecular weight:380.35(RS)-Minesapride
CAS:Minesapride is a serotonin receptor agonist.Formula:C21H31ClN4O5Purity:98%Color and Shape:SolidMolecular weight:454.95LY 206130
CAS:LY 206130 is an antagonist of serotonin 5-HT1A.Formula:C17H24N2O2Color and Shape:SolidMolecular weight:288.38SDZ 205-557 hydrochloride
CAS:5-HT3/5-HT4 receptor antagonistFormula:C14H22Cl2N2O3Purity:98%Color and Shape:SolidMolecular weight:337.24RS 15385-197
CAS:RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.Formula:C18H26N2O3SColor and Shape:SolidMolecular weight:350.48Alclofenac sodium
CAS:Alclofenac sodium is an anti-inflammatory utilized in the treatment of rheumatoid arthritis.Formula:C11H11ClNaO3Purity:98%Color and Shape:SolidMolecular weight:249.65Chloracyzine
CAS:Chloracyzine lowers heart oxygen use, shrinks coronary flow after brief dilation, slightly ups heart rate and arterial pressure.Formula:C19H21ClN2OSColor and Shape:SolidMolecular weight:360.9Garomefrine HCl
CAS:Garomefrine HCl, a α1A-adrenoceptor agonist, is potential for the treatment of urinary incontinence.Formula:C9H14ClFN2O3SPurity:98%Color and Shape:SolidMolecular weight:284.73Viprostol
CAS:Viprostol is an agent of prostaglandin antihypertensive.Formula:C23H36O5Purity:98%Color and Shape:SolidMolecular weight:392.53GS 283
CAS:GS 283 is a Ca(2+) antagonist. GS 283 is also a weak histamine and muscarinic receptor blocker in rat and guinea pig tracheal smooth muscles.Formula:C17H17NO3Color and Shape:SolidMolecular weight:283.32AHR-13268D
CAS:AHR-13268D is a new agent of antiallergic/antihistaminic.Formula:C28H29F2NNaO4Purity:98%Color and Shape:SolidMolecular weight:504.53R 47243
CAS:R 47243 is used as a racemic alpha 2 antagonist.Formula:C22H25N3O2SPurity:98%Color and Shape:SolidMolecular weight:395.52Burimamide
CAS:Burimamide is an antagonist of histamine. It appears to block both H2 and H3 histamine receptors.Formula:C9H16N4SPurity:98%Color and Shape:SolidMolecular weight:212.32MS437
CAS:MS437 is a potent TSH receptor agonist.Formula:C22H24N2OPurity:98%Color and Shape:SolidMolecular weight:332.44LG 82-4-00
CAS:LG 82-4-00 is an inhibitor of thromboxane.Formula:C10H11ClN2O3SPurity:98%Color and Shape:SolidMolecular weight:274.72FR 121196
CAS:FR 121196, a potential antidementia drug, ameliorates the impaired memory of rat in the Morris water maze.Formula:C12H16FN3O3SColor and Shape:SolidMolecular weight:301.34A23887
CAS:A23887 is a potentially neuroleptic tetracyclic spiro amine that has affinity for dopamine D-2 receptors.Formula:C22H24ClNPurity:98%Color and Shape:SolidMolecular weight:337.89AHR-14310C
CAS:AHR-14310C is a long-acting and nonsedating H1-antihistamine.Formula:C24H28F2N2O3Purity:98%Color and Shape:SolidMolecular weight:430.49NNC-38-1049
CAS:NNC-38-1049 is a novel selective antagonist of histamine H3.Formula:C19H25ClN2O2Purity:98%Color and Shape:SolidMolecular weight:348.87LP 20 hydrochloride
CAS:ligand of the 5-HT7 receptorFormula:C17H21ClN2OPurity:98%Color and Shape:SolidMolecular weight:304.81LY 25648
CAS:LY 25648 is an antagonist of leukotriene B4.Formula:C19H27NO2SColor and Shape:SolidMolecular weight:333.49Bromperidol decanoate
CAS:Bromperidol decanoate is an antipsychotic agent that is utilized for long-term maintenance treatment for schizophrenia.Formula:C31H41BrFNO3Color and Shape:SolidMolecular weight:574.56Hetramine
CAS:Hetramine is a synthetic pyrimidine agent that possesses antihistamine and anti anaphylactic effects.Formula:C15H20N4Purity:98%Color and Shape:SolidMolecular weight:256.35Asperlicin D
CAS:Asperlicin D is a cholecystokinin antagonist agent.Formula:C25H18N4O2Purity:98%Color and Shape:SolidMolecular weight:406.44JTH-601 free base
CAS:JTH-601 free base is an antagonist of alpha 1 adrenergic receptor.Formula:C24H35NO4Purity:98%Color and Shape:SolidMolecular weight:401.54JNJ-7925476 HCl
CAS:JNJ-7925476 HCl inhibits DAT, NET, SERT; ED(50): DAT 2.4, NET 0.09, SERT 0.18 mg/kg in rats.Formula:C20H20ClNColor and Shape:SolidMolecular weight:309.83Bragsin1
CAS:Bragsin1 is a potent and selective and noncompetitive ArfGEF BRAG2 inhibitor, inhibits Arf GTPase activation(IC50 : 3 μM),and with anti-cancer activity.Formula:C11H6F3NO4Color and Shape:SolidMolecular weight:273.16
