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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5964 products of "GPCR/G-Protein"

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  • MK-8133

    CAS:
    MK-8133 is an antagonist of orexin-2 selective receptor with favorable development properties.
    Formula:C23H21N5O2
    Color and Shape:Solid
    Molecular weight:399.45

    Ref: TM-T28060

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Methyldopate hydrochloride

    CAS:
    Methyldopate HCl is an agent of antihypertensive.
    Formula:C12H18ClNO4
    Color and Shape:Solid
    Molecular weight:275.73

    Ref: TM-T20133

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A-943931

    CAS:
    A-943931 is a selective histamine H4 receptor antagonist with human and rat Ki values of 4.6 and 3.8 nM respectively.inhibits the scratching response in mice.
    Formula:C17H21N5
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:295.38

    Ref: TM-T73352

    1mg
    54.00€
    5mg
    153.00€
    10mg
    241.00€
    25mg
    408.00€
    50mg
    571.00€
  • BRL 37344 sodium

    CAS:
    BRL 37344 sodium is a specific agonist of the β3-adrenergic receptor. The treatment of BRL 37344 sodium significantly lowers the bodyweight of obese mice.
    Formula:C19H22ClNNaO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.83

    Ref: TM-T10613

    1mg
    166.00€
    5mg
    384.00€
    10mg
    705.00€
    25mg
    1,513.00€
  • (Rac)-HAMI 3379

    CAS:
    HAMI 3379: potent CysLT2 receptor blocker; protects against acute/subacute brain injury; reduces microglia inflammation.
    Formula:C34H45NO8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:595.72

    Ref: TM-T15463

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Fluprostenol methyl ester

    CAS:
    Fluprostenol, a vet-approved luteolytic, has an isopropyl ester, travoprost, used as an eye pressure reducer. CAY10532 is its methyl ester form.
    Formula:C24H31F3O6
    Color and Shape:Solid
    Molecular weight:472.49

    Ref: TM-T37813

    1mg
    227.00€
    5mg
    973.00€
    10mg
    1,773.00€
  • SB 207710

    CAS:
    SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.
    Formula:C19H27IN2O4
    Color and Shape:Solid
    Molecular weight:474.33

    Ref: TM-T28672

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • QCC-374

    CAS:
    QCC-374 is a prostanoid agonist. It potentially for the treatment of pulmonary arterial hypertension.
    Formula:C28H33N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:443.58

    Ref: TM-T19660

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • UK 1745

    CAS:
    UK 1745 is a novel drug of cardiotonic.
    Formula:C16H23ClN2O2
    Color and Shape:Solid
    Molecular weight:310.82

    Ref: TM-T34987

    25mg
    1,783.00€
  • Zenidolol

    CAS:
    Zenidolol (ICI-118551) is a β2 adrenoceptor blocker with K i values: β2 (0.7 nM), β1 (49.5 nM), β3 (611 nM); used in eye disease research.
    Formula:C17H27NO2
    Color and Shape:Solid
    Molecular weight:277.4

    Ref: TM-T68385

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • CP-195543

    CAS:
    CP-195543 is an effective leukotriene B4 antagonist for the treatment of inflammatory diseases.
    Formula:C24H19F3O4
    Color and Shape:Solid
    Molecular weight:428.4

    Ref: TM-T31042

    5mg
    3,445.00€
  • LY288513

    CAS:
    Selective CCK2 receptor antagonist
    Formula:C22H18BrN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:436.3

    Ref: TM-T22949

    10mg
    1,288.00€
    50mg
    5,544.00€
  • GSK-269984B

    CAS:
    GSK-269984B is a novel antagonist of EP1 receptor.
    Formula:C20H14Cl2FNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:406.23

    Ref: TM-T27466

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Guanethidine

    CAS:
    Guanethidine sulphate, made in 1959, lowers blood pressure by disrupting neurotransmitters in sympathetic nerves.
    Formula:C10H22N4
    Color and Shape:Solid
    Molecular weight:198.31

    Ref: TM-T50109

    100mg
    To inquire
    500mg
    To inquire
  • EP4 receptor antagonist 4

    CAS:
    EP4 receptor antagonist 4 is an agonist of EP4 receptor (human pEC 50 = 6.3) [1].
    Formula:C19H14N2OS
    Color and Shape:Solid
    Molecular weight:318.39

    Ref: TM-T60840

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • 5-HT7 agonist 2

    CAS:
    Potent 5-HT7 agonist with 28.7 nM IC50; promising for CNS disorder research.
    Formula:C23H29N3O
    Color and Shape:Solid
    Molecular weight:363.5

    Ref: TM-T61375

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SKF-75670 Hydrobromide

    CAS:
    SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.
    Formula:C17H20BrNO2
    Color and Shape:Solid
    Molecular weight:350.25

    Ref: TM-T28792

    2mg
    495.00€
    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Zicronapine

    CAS:
    Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.
    Formula:C22H27ClN2
    Color and Shape:Solid
    Molecular weight:354.92

    Ref: TM-T35307

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A 55453

    CAS:
    A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.
    Formula:C25H32N6O3
    Color and Shape:Solid
    Molecular weight:464.56

    Ref: TM-T26421

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • FRG8701

    CAS:
    FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.
    Formula:C22H30N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:418.55

    Ref: TM-T11324

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • NAEPA

    CAS:
    NAEPA, an LPA mimetic, is a selective agonist of the lysophosphatidic acid-1 (LPA1) receptor.
    Formula:C20H40NO5P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:405.51

    Ref: TM-T25847

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • EP2 receptor antagonist-1

    CAS:
    EP2 receptor antagonist-1: reversible, potent, depends on agonist; anti-inflammatory.
    Formula:C24H22N4O5
    Color and Shape:Solid
    Molecular weight:446.46

    Ref: TM-T62641

    25mg
    1,260.00€
    50mg
    1,639.00€
    100mg
    2,538.00€
  • WB403

    CAS:
    WB403 activates TGR5, lowers fasting/postprandial glucose and HbA1c, enhances glucose tolerance, and normalizes pancreatic α/β-cells in diabetic mice.
    Formula:C19H19BrN2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:403.34

    Ref: TM-T29154

    5mg
    110.00€
    10mg
    168.00€
    25mg
    338.00€
    50mg
    533.00€
    100mg
    2,375.00€
  • PD-135666

    CAS:
    PD-135666 is an antagonist of CCK receptor.
    Formula:C33H39N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:557.68

    Ref: TM-T28340

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Naronapride

    CAS:
    Naronapride (ATI-7505) is a potent agonist of the prokinetic 5-HT4receptor and can be used to study gastrointestinal disorders.
    Formula:C27H41ClN4O5
    Color and Shape:Solid
    Molecular weight:537.09

    Ref: TM-T63785

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • LY 219057

    CAS:
    LY 219057 is a potent, competitive, and specific antagonist of CCK receptor on the exocrine pancreas.
    Formula:C23H17ClF3N3OS
    Color and Shape:Solid
    Molecular weight:475.91

    Ref: TM-T27900

    25mg
    1,369.00€
  • CB1R Allosteric modulator 1

    CAS:
    CB1R modulator 1 (compound 11), a potent CB1R inhibitor, decreases activity of orthosteric ligands.
    Formula:C24H24ClN3O
    Color and Shape:Solid
    Molecular weight:405.92

    Ref: TM-T62016

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • S-777469

    CAS:
    S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.
    Formula:C23H27FN2O4
    Color and Shape:Solid
    Molecular weight:414.47

    Ref: TM-T62132

    25mg
    1,108.00€
    50mg
    1,449.00€
    100mg
    2,385.00€
  • CB2 receptor agonist 3

    CAS:
    GP 2A is a selective agonist of CB2 receptor.
    Formula:C24H23Cl2N3O
    Color and Shape:Solid
    Molecular weight:440.36

    Ref: TM-T24097

    25mg
    690.00€
    50mg
    898.00€
    100mg
    1,566.00€
  • SANT-2

    CAS:
    SANT-2 is a potent inhibitor of Shh signaling pathway.
    Formula:C23H20ClN3O4
    Color and Shape:Solid
    Molecular weight:437.88

    Ref: TM-T69189

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Nivasorexant

    CAS:
    Nivasorexant is a potent antagonist of the orexin receptor.
    Formula:C23H23N7O2
    Color and Shape:Solid
    Molecular weight:429.47

    Ref: TM-T62370

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ATL-801

    CAS:
    ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.
    Formula:C24H25N7O3
    Color and Shape:Solid
    Molecular weight:459.5

    Ref: TM-T26680

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Povafonidine

    CAS:
    Povafonidine (PGE-6201204), an alpha-2 adrenoreceptor agonist, constricts vessels, reduces congestion for nasal research.
    Formula:C11H13N5
    Color and Shape:Solid
    Molecular weight:215.25

    Ref: TM-T60263

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Ziprasidone mesylate trihydrate

    CAS:
    Ziprasidone mesylate hydrate is an oral 5-HT/D2 antagonist with Ki: D2=4.8nM, 5-HT2A=0.42nM, 5-HT1A=3.4nM in rats.
    Formula:C22H31ClN4O7S2
    Color and Shape:Solid
    Molecular weight:563.08

    Ref: TM-T63979

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • Nebidrazine

    CAS:
    Nebidrazine is an alpha-adrenoceptor agonist.
    Formula:C9H8Cl2N6
    Color and Shape:Solid
    Molecular weight:271.11

    Ref: TM-T69108

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • INCB38579

    CAS:
    INCB38579: Oral, selective H4 antagonist; crosses brain barrier; IC50s - hH4R: 4.8 nM, mH4R: 42 nM, rH4R: 32 nM; anti-inflammatory and antipruritic.
    Formula:C25H34N6O
    Color and Shape:Solid
    Molecular weight:434.58

    Ref: TM-T62460

    25mg
    858.00€
    50mg
    1,116.00€
    100mg
    1,791.00€
  • Latanoprost ethyl amide

    CAS:
    Lat-NEt, a latanoprost analog, is an ocular hypotensive prodrug with slower hydrolysis, converting to free acids in corneal tissue.
    Formula:C25H39NO4
    Color and Shape:Solid
    Molecular weight:417.58

    Ref: TM-T37627

    1mg
    239.00€
    5mg
    1,018.00€
    10mg
    1,783.00€
  • BAY-u 9773

    CAS:
    BAY-u9773 is a non-selective CysLT receptor antagonist with similar IC50 for CysLT1 and CysLT2, inhibiting LT responses.
    Formula:C27H36O5S
    Color and Shape:White Oil
    Molecular weight:472.64

    Ref: TM-T21864

    25µg
    208.00€
    50µg
    389.00€
    100µg
    735.00€
    500µg
    3,222.00€
  • Remogliflozin

    CAS:
    Remogliflozin is an effective sodium-glucose transporter 2 inhibitor (Kis = 12.4 and 26 nM for human and rat SGLT2, respectively).
    Formula:C23H34N2O7
    Color and Shape:Solid
    Molecular weight:450.53

    Ref: TM-T24708

    1mg
    284.00€
    5mg
    1,288.00€
    10mg
    2,332.00€
    500µg
    157.00€
  • MAT2A-IN-3

    CAS:
    MAT2A-IN-3: potent MAT2A inhibitor, hinders MTAP-deficient cancer cell growth, potential for cancer research.
    Formula:C24H16F5N5O3
    Color and Shape:Solid
    Molecular weight:517.41

    Ref: TM-T63603

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • 5-HT2A receptor agonist-2

    CAS:
    Potent 5-HT2A receptor agonist-2 targets 5-HT2A/B/C with EC50 1.7, 0.58, 0.50 nM.
    Formula:C20H21ClN2O3
    Color and Shape:Solid
    Molecular weight:372.85

    Ref: TM-T61507

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AP-521 (Free base)

    CAS:
    AP-521, a 5-HT1A receptor antagonist, is used potentially for the treatment of anxiety.
    Formula:C20H18N2O3S
    Color and Shape:Solid
    Molecular weight:366.43

    Ref: TM-T26640

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BRD5814

    CAS:
    BRD5814 is a highly brain penetrant β-arrestin biased D2R antagonist.
    Formula:C21H23ClF3NO2
    Color and Shape:Solid
    Molecular weight:413.86

    Ref: TM-T70040

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Edivoxetine

    CAS:
    Edivoxetine (LY2216684) is a selective norepinephrine reuptake inhibitor for ADHD and depression.
    Formula:C18H26FNO4
    Color and Shape:Solid
    Molecular weight:339.4

    Ref: TM-T31604

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • ChemR23-IN-1

    CAS:
    ChemR23-IN-1 inhibits human and mouse ChemR23 (IC50: 38 nM, 100 nM) and stops CAL-1 chemotaxis induced by Chemerin in vitro.
    Formula:C28H29N7O2
    Color and Shape:Solid
    Molecular weight:495.58

    Ref: TM-T63347

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BGC-20-1531 free base

    CAS:
    BGC-20-1531 (PGN 1531) free base is a selective and potent prostaglandin EP4 receptor antagonist (pKB: 7.6) that exhibits potential for migraine research.
    Formula:C26H24N2O6S
    Color and Shape:Solid
    Molecular weight:492.54

    Ref: TM-T63316

    25mg
    1,026.00€
    50mg
    1,341.00€
    100mg
    2,197.00€
  • Medroxalol

    CAS:
    Medroxalol (RMI81968), an oral α- & β-adrenergic blocker, has antihypertensive and vasodilatory effects.
    Formula:C20H24N2O5
    Color and Shape:Solid
    Molecular weight:372.42

    Ref: TM-T61495

    25mg
    1,746.00€
    50mg
    2,800.00€
  • Bopindolol (malonate)

    CAS:
    Bopindolol is a non-selective β-adrenergic receptor antagonist.
    Formula:C26H32N2O7
    Color and Shape:Solid
    Molecular weight:484.549

    Ref: TM-T35871

    100mg
    298.00€
    500mg
    1,035.00€
  • GPR183-IN-2

    CAS:

    GPR183-IN-2 (compound 23) is an effective, orally active inhibitor of GPR183, displaying an IC50 value of 39.45 nM in Ca2+ mobilization assays. This compound has potential applications in research related to cancer, autoimmune diseases, pain, and osteoporosis.

    Formula:C19H23BrN2O3
    Color and Shape:Solid
    Molecular weight:407.3

    Ref: TM-T88500

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • DuP 734

    CAS:

    DuP 734 is a potent and selective sigma receptor antagonist, functioning as a ligand for both sigma and 5-HT2 receptors, and exhibiting weak affinity towards D2 receptors. It possesses potential antipsychotic activity, potentially devoid of the motor side effects commonly observed with neuroleptics[1][2][3].

    Formula:C17H23BrFNO
    Color and Shape:Solid
    Molecular weight:356.279

    Ref: TM-T37074

    5mg
    982.00€
    50mg
    1,941.00€
    100mg
    2,451.00€
  • GPR183 antagonist-2

    CAS:
    GPR183 antagonist-2 (compound 32), a selective antagonist of GPR183, exhibits excellent water solubility and pharmacokinetic properties. This compound effectively diminishes paw and joint swelling, and reduces gene expression of pro-inflammatory cytokines (MCP-1, MMPs, and VEGF) in a dose-dependent manner within a collagen-induced arthritis (CIA) mouse model. GPR183 antagonist-2 is applicable in researching autoimmune diseases [1].
    Formula:C20H18F2N4O5
    Color and Shape:Solid
    Molecular weight:432.38

    Ref: TM-T86519

    25mg
    1,539.00€
    50mg
    1,941.00€
    100mg
    2,451.00€
  • MoTP

    CAS:
    MoTP is a specific platelet activating factor receptor antagonist that induces ablation of melanocyte. MoTP can be used in cancer research.
    Formula:C14H21NO2S
    Color and Shape:Solid
    Molecular weight:267.39

    Ref: TM-T60451

    1mg
    111.00€
    5mg
    283.00€
    10mg
    469.00€
    25mg
    919.00€
  • MG 1

    CAS:
    MG 1 is a potent alpha-1 adrenergic receptor antagonist.
    Formula:C17H25N3O2
    Purity:98.98% - >99.99%
    Color and Shape:Solid
    Molecular weight:303.4

    Ref: TM-T12030

    1mg
    665.00€
    5mg
    1,710.00€
  • I942

    CAS:
    I942 is a novel, selective ACyclic nucleotide (NCN) EPAC1 agonist that activates exchange proteins to regulate inflammatory gene expression in human umbilical
    Formula:C20H19NO4S
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:369.43

    Ref: TM-T24154

    1mg
    89.00€
    5mg
    215.00€
    10mg
    350.00€
    25mg
    575.00€
    50mg
    793.00€
    100mg
    1,071.00€
    500mg
    2,187.00€
  • Iso-SLR 080811

    CAS:
    Iso-SLR 080811 is an isomer of SLR 080811, suitable for relevant research in the life sciences. SLR080811 is a selective SphK2 inhibitor (Ki=1.3 μM).
    Formula:C21H32ClN5O
    Purity:98.34%
    Color and Shape:Solid
    Molecular weight:405.97

    Ref: TM-T70614

    1mg
    279.00€
    5mg
    685.00€
    10mg
    938.00€
    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • CB1R Allosteric modulator 3

    CAS:
    CB1R Allosteric modulator 3 is a CB1R modulator.CB1R Allosteric modulator 3 inhibits cAMP, and can be used for the study of obesity and nicotine addiction.
    Formula:C22H17ClN2O2
    Purity:98.18%
    Color and Shape:Solid
    Molecular weight:376.84

    Ref: TM-T61562

    2mg
    39.00€
    5mg
    59.00€
    10mg
    90.00€
    25mg
    152.00€
    50mg
    219.00€
    100mg
    324.00€
    200mg
    470.00€
  • NRA-0160

    CAS:
    NRA-0160 is a selective antagonist of dopamine D4 receptor(Ki of 0.48 nM)
    Formula:C24H23F2N3OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:439.52

    Ref: TM-T12252

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • hA2AAR antagonist 1

    CAS:
    Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.
    Formula:C15H15N5O
    Color and Shape:Solid
    Molecular weight:281.31

    Ref: TM-T88549

    25mg
    1,539.00€
    50mg
    1,941.00€
    100mg
    2,451.00€
  • CJ 033466

    CAS:
    CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.
    Formula:C19H28ClN5O
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:377.91

    Ref: TM-T22671

    1mg
    48.00€
    5mg
    101.00€
    10mg
    170.00€
    25mg
    270.00€
    50mg
    386.00€
    100mg
    520.00€
    1mL*10mM (DMSO)
    124.00€
  • Eplivanserin

    CAS:
    Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.
    Formula:C19H21FN2O2
    Purity:97.04%
    Color and Shape:Solid
    Molecular weight:328.38

    Ref: TM-T11217

    1mg
    175.00€
    5mg
    394.00€
    10mg
    582.00€
    25mg
    888.00€
    50mg
    1,243.00€
    1mL*10mM (DMSO)
    399.00€
  • DOV-216,303 Free Base

    CAS:
    DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.
    Formula:C11H11Cl2N
    Purity:96.7%
    Color and Shape:Solid
    Molecular weight:228.12

    Ref: TM-T11087

    2mg
    46.00€
    5mg
    66.00€
    10mg
    97.00€
    25mg
    159.00€
    50mg
    226.00€
    100mg
    339.00€
    1mL*10mM (DMSO)
    67.00€
  • EMDT

    CAS:
    EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.
    Formula:C15H22N2O
    Purity:97.66% - 99.78%
    Color and Shape:Solid
    Molecular weight:246.35

    Ref: TM-T11183

    1mg
    87.00€
    2mg
    118.00€
    5mg
    167.00€
    10mg
    202.00€
    25mg
    449.00€
    50mg
    652.00€
    100mg
    888.00€
    500mg
    1,783.00€
    1mL*10mM (DMSO)
    166.00€
  • Chlorazanil

    CAS:
    Chlorazanil is a triazine-based, orally active diuretic that blocks Na+ and Cl– reabsorption in distal tubules, increases renal prostaglandin.
    Formula:C9H8ClN5
    Purity:98.89%
    Color and Shape:Solid
    Molecular weight:221.65

    Ref: TM-T13609L

    10mg
    33.00€
    25mg
    33.00€
    50mg
    To inquire
    1mL*10mM (DMSO)
    48.00€
  • Nedocromil

    CAS:
    Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).
    Formula:C19H17NO7
    Purity:95% - 97.34%
    Color and Shape:Solid
    Molecular weight:371.34

    Ref: TM-T16280

    5mg
    70.00€
    10mg
    96.00€
    25mg
    202.00€
    50mg
    329.00€
    100mg
    520.00€
  • Quinpirole Hydrochloride

    CAS:
    Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and mice
    Formula:C13H22ClN3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:255.79

    Ref: TM-T12606

    1mg
    100.00€
  • H3R-IN-1 Hydrochloride

    CAS:
    H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .
    Formula:C19H24ClN3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:377.86

    Ref: TM-T11531

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Org-12962

    CAS:
    Org-12962: 5-HT2C agonist (pEC50: 7.01), anti-panic in rats, affects 5-HT2A/B (pEC50: 6.38/6.28).
    Formula:C10H11ClF3N3
    Purity:98.34%
    Color and Shape:Solid
    Molecular weight:265.66

    Ref: TM-T16401

    5mg
    48.00€
    10mg
    62.00€
    25mg
    90.00€
    50mg
    111.00€
    100mg
    159.00€
    1mL*10mM (DMSO)
    52.00€
  • 5-Carboxamidotryptamine maleate

    CAS:
    5-Carboxamidotryptamine maleate (5-CT maleate) (5-CT maleate) is a receptor agonist with antihypertensive and glucose-raising effects.
    Formula:C15H17N3O5
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:319.31

    Ref: TM-T22520

    1mg
    35.00€
    5mg
    84.00€
    10mg
    119.00€
    25mg
    207.00€
    50mg
    289.00€
    100mg
    399.00€
    200mg
    555.00€
  • Mirisetron

    CAS:
    Mirisetron (WAY-100579, SEC-579) is a 5-HT3 receptor antagonist, cognitive-enhancing effects. counteracts learning deficits.
    Formula:C24H31N3O2
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:393.52

    Ref: TM-T70879

    1mg
    285.00€
    5mg
    692.00€
    10mg
    947.00€
    25mg
    1,458.00€
    50mg
    1,839.00€
    100mg
    2,322.00€
  • ICI 162,846

    CAS:
    ICI 162,846 is an orally active and potent H2 receptor antagonist that inhibits gastric secretion and may be used in the study of duodenal ulcers.
    Formula:C11H17F3N6O
    Purity:97.45%
    Color and Shape:Solid
    Molecular weight:306.29

    Ref: TM-T22848

    1mg
    34.00€
    5mg
    65.00€
    10mg
    94.00€
    25mg
    138.00€
    50mg
    197.00€
  • PRX-08066 Maleic acid

    CAS:
    PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.
    Formula:C23H21ClFN5O4S
    Purity:97.59%
    Color and Shape:Solid
    Molecular weight:517.96

    Ref: TM-T6959

    1mg
    84.00€
    5mg
    172.00€
    10mg
    233.00€
    25mg
    419.00€
    50mg
    620.00€
    100mg
    882.00€
    200mg
    1,198.00€
    1mL*10mM (DMSO)
    401.00€
  • Iprindole

    CAS:
    Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].
    Formula:C19H28N2
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:284.44

    Ref: TM-T37015

    2mg
    37.00€
    5mg
    52.00€
    10mg
    80.00€
    25mg
    154.00€
    50mg
    266.00€
    100mg
    455.00€
    200mg
    652.00€
    1mL*10mM (DMSO)
    84.00€
  • Thioproperazine

    CAS:
    Thioproperazine (RP 7843) is an orally effective antipsychotic schizophrenia and bipolar disorder, histamine and adrenergic receptor blocker.
    Formula:C22H30N4O2S2
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:446.63

    Ref: TM-T21368

    1mg
    37.00€
    5mg
    79.00€
    10mg
    114.00€
    25mg
    185.00€
    50mg
    276.00€
    100mg
    409.00€
  • LPA2 antagonist 2

    CAS:
    LPA2 antagonist 2 is an and LPA2 antagonist (IC50: 28.3 nM) with potential anticancer activity, inhibits LPA3, and can be used for cancer research.
    Formula:C20H16N2O6
    Purity:96.13%
    Color and Shape:Solid
    Molecular weight:380.35

    Ref: TM-T11875

    1mg
    96.00€
    5mg
    227.00€
    10mg
    359.00€
    25mg
    595.00€
    50mg
    838.00€
    100mg
    1,130.00€
  • (RS)-Minesapride

    CAS:
    Minesapride is a serotonin receptor agonist.
    Formula:C21H31ClN4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:454.95

    Ref: TM-T28043

    25mg
    2,043.00€
    50mg
    2,682.00€
    100mg
    3,600.00€
  • LY 206130

    CAS:
    LY 206130 is an antagonist of serotonin 5-HT1A.
    Formula:C17H24N2O2
    Color and Shape:Solid
    Molecular weight:288.38

    Ref: TM-T27894

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SDZ 205-557 hydrochloride

    CAS:
    5-HT3/5-HT4 receptor antagonist
    Formula:C14H22Cl2N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:337.24

    Ref: TM-T23342

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • RS 15385-197

    CAS:
    RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.
    Formula:C18H26N2O3S
    Color and Shape:Solid
    Molecular weight:350.48

    Ref: TM-T26134

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Alclofenac sodium

    CAS:
    Alclofenac sodium is an anti-inflammatory utilized in the treatment of rheumatoid arthritis.
    Formula:C11H11ClNaO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:249.65

    Ref: TM-T25036

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Chloracyzine

    CAS:
    Chloracyzine lowers heart oxygen use, shrinks coronary flow after brief dilation, slightly ups heart rate and arterial pressure.
    Formula:C19H21ClN2OS
    Color and Shape:Solid
    Molecular weight:360.9

    Ref: TM-T25237

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Garomefrine HCl

    CAS:
    Garomefrine HCl, a α1A-adrenoceptor agonist, is potential for the treatment of urinary incontinence.
    Formula:C9H14ClFN2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:284.73

    Ref: TM-T27401

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Viprostol

    CAS:
    Viprostol is an agent of prostaglandin antihypertensive.
    Formula:C23H36O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.53

    Ref: TM-T24938

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • GS 283

    CAS:
    GS 283 is a Ca(2+) antagonist. GS 283 is also a weak histamine and muscarinic receptor blocker in rat and guinea pig tracheal smooth muscles.
    Formula:C17H17NO3
    Color and Shape:Solid
    Molecular weight:283.32

    Ref: TM-T27435

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AHR-13268D

    CAS:
    AHR-13268D is a new agent of antiallergic/antihistaminic.
    Formula:C28H29F2NNaO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:504.53

    Ref: TM-T23679

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • R 47243

    CAS:
    R 47243 is used as a racemic alpha 2 antagonist.
    Formula:C22H25N3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:395.52

    Ref: TM-T26014

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Burimamide

    CAS:
    Burimamide is an antagonist of histamine. It appears to block both H2 and H3 histamine receptors.
    Formula:C9H16N4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:212.32

    Ref: TM-T23841

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • MS437

    CAS:
    MS437 is a potent TSH receptor agonist.
    Formula:C22H24N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:332.44

    Ref: TM-T24502

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LG 82-4-00

    CAS:
    LG 82-4-00 is an inhibitor of thromboxane.
    Formula:C10H11ClN2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:274.72

    Ref: TM-T25709

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • FR 121196

    CAS:
    FR 121196, a potential antidementia drug, ameliorates the impaired memory of rat in the Morris water maze.
    Formula:C12H16FN3O3S
    Color and Shape:Solid
    Molecular weight:301.34

    Ref: TM-T27361

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • A23887

    CAS:
    A23887 is a potentially neuroleptic tetracyclic spiro amine that has affinity for dopamine D-2 receptors.
    Formula:C22H24ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:337.89

    Ref: TM-T26472

    25mg
    1,783.00€
  • AHR-14310C

    CAS:
    AHR-14310C is a long-acting and nonsedating H1-antihistamine.
    Formula:C24H28F2N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.49

    Ref: TM-T23680

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • NNC-38-1049

    CAS:
    NNC-38-1049 is a novel selective antagonist of histamine H3.
    Formula:C19H25ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.87

    Ref: TM-T28184

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LP 20 hydrochloride

    CAS:
    ligand of the 5-HT7 receptor
    Formula:C17H21ClN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:304.81

    Ref: TM-T22930

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • LY 25648

    CAS:
    LY 25648 is an antagonist of leukotriene B4.
    Formula:C19H27NO2S
    Color and Shape:Solid
    Molecular weight:333.49

    Ref: TM-T27906

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bromperidol decanoate

    CAS:
    Bromperidol decanoate is an antipsychotic agent that is utilized for long-term maintenance treatment for schizophrenia.
    Formula:C31H41BrFNO3
    Color and Shape:Solid
    Molecular weight:574.56

    Ref: TM-T25181

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Hetramine

    CAS:
    Hetramine is a synthetic pyrimidine agent that possesses antihistamine and anti anaphylactic effects.
    Formula:C15H20N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:256.35

    Ref: TM-T25494

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Asperlicin D

    CAS:
    Asperlicin D is a cholecystokinin antagonist agent.
    Formula:C25H18N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:406.44

    Ref: TM-T25116

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JTH-601 free base

    CAS:
    JTH-601 free base is an antagonist of alpha 1 adrenergic receptor.
    Formula:C24H35NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.54

    Ref: TM-T24220

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • JNJ-7925476 HCl

    CAS:
    JNJ-7925476 HCl inhibits DAT, NET, SERT; ED(50): DAT 2.4, NET 0.09, SERT 0.18 mg/kg in rats.
    Formula:C20H20ClN
    Color and Shape:Solid
    Molecular weight:309.83

    Ref: TM-T27689

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Bragsin1

    CAS:
    Bragsin1 is a potent and selective and noncompetitive ArfGEF BRAG2 inhibitor, inhibits Arf GTPase activation(IC50 : 3 μM),and with anti-cancer activity.
    Formula:C11H6F3NO4
    Color and Shape:Solid
    Molecular weight:273.16

    Ref: TM-T14774

    5mg
    268.00€
    25mg
    888.00€
    50mg
    1,224.00€
    100mg
    1,674.00€
    1mL*10mM (DMSO)
    286.00€