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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5963 products of "GPCR/G-Protein"

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  • CIA-1 hcl(452087-38-6 Free base)

    CAS:
    CIA-1 inhibits the nuclear receptor COUP-TFII, with IC50s ranging from 1.2 μM to 7.6 μM in prostate cancer cell lines.CIA-1 inhibits the growth of a variety of
    Formula:C17H20ClN3O2S
    Purity:99.02%
    Color and Shape:Solid
    Molecular weight:365.88

    Ref: TM-T71534

    10mg
    540.00€
    50mg
    2,252.00€
  • Q8 hydrochloride

    CAS:
    Q8 is an antagonist of cysteinyl leukotreine receptor. Q8 inhibits VEGF-independent angiogenesis.
    Formula:C17H14ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:299.75

    Ref: TM-T28481

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • AUY-954 free base

    CAS:
    AUY-954 is a selective S1P(1) modulator reducing EAN inflammation and demyelination in rats.
    Formula:C25H20F3NO2S
    Color and Shape:Solid
    Molecular weight:455.49

    Ref: TM-T30215

    1mg
    386.00€
    5mg
    1,198.00€
    500µg
    221.00€
  • Clopenthixol

    CAS:
    Clopenthixol is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics. It is an antagonist at D1 and D2 dopamine receptors.
    Formula:C22H25ClN2OS
    Color and Shape:Solid
    Molecular weight:400.96

    Ref: TM-T68193

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Paltusotine HCl

    CAS:
    Paltusotine, also known as CRN00808, is a somatostatin receptor agonist.
    Formula:C27H24Cl2F2N4O
    Color and Shape:Solid
    Molecular weight:529.41

    Ref: TM-T69836

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SC 53116 Hydrochloride

    CAS:
    SC 53116 Hydrochloride is selective agonist of the newly identified serotonin 5-HT4 receptor subtype.
    Formula:C16H23Cl2N3O2
    Color and Shape:Solid
    Molecular weight:360.28

    Ref: TM-T28696

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Pd 158771

    CAS:
    Pd 158771 is a D2 and 5-HT1A agonist.
    Formula:C22H31N5
    Color and Shape:Solid
    Molecular weight:365.52

    Ref: TM-T70081

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • WRC-0571

    CAS:
    WRC-0571 is a highly potent, selective antagonist of A1 adenosine receptors.
    Formula:C17H26N6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:330.43

    Ref: TM-T29162

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Daledalin

    CAS:
    Daledalin, an unmarketed 1970s antidepressant, is a selective norepinephrine reuptake inhibitor without serotonergic or dopaminergic effects.
    Formula:C19H24N2
    Color and Shape:Solid
    Molecular weight:280.41

    Ref: TM-T69788

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Fenspiride-d5

    CAS:
    Fenspiride-d5: internal standard for GC/LC-MS quantification, H1 antagonist, NSAID, anti-inflammatory, selective PDE4,5,3 inhibitor.
    Formula:C15H15D5N2O2
    Color and Shape:Solid
    Molecular weight:265.36

    Ref: TM-T71141

    1mg
    1,018.00€
    5mg
    3,312.00€
  • SGC agonist 2

    CAS:
    SGC agonist 2 is a potent activator for cardiovascular and fibrotic diseases, per patent WO2021219088A1, compound 031.
    Formula:C23H17F2N7O2
    Color and Shape:Solid
    Molecular weight:461.42

    Ref: TM-T62909

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Sch 33303

    CAS:
    Sch 33303 is an antiallergy agents.
    Formula:C19H16N2O3
    Color and Shape:Solid
    Molecular weight:320.34

    Ref: TM-T28714

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SLM6031434 (free base)

    CAS:
    SLM6031434 (free base) is an inhibitor of sphingosine kinase type 2 (SphK2). It consists of pedant 1-guanidino-2-phenyloxadiazolylpyrrolidine group.
    Formula:C22H30F3N5O2
    Color and Shape:Solid
    Molecular weight:453.5

    Ref: TM-T70071

    1mg
    172.00€
    5mg
    512.00€
    10mg
    750.00€
  • ChemR23-IN-4

    CAS:
    ChemR23-IN-4 is a potent inhibitor of orally active ChemR23, capable of acting on human ChemR23 (IC50: 17 nM).
    Formula:C27H26N6O3
    Color and Shape:Solid
    Molecular weight:482.53

    Ref: TM-T63195

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Cetrorelix Acetate

    CAS:
    Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.
    Formula:C70H92ClN17O14·xC2H4O2
    Purity:97.96%
    Color and Shape:Solid
    Molecular weight:1491.11

    Ref: TM-T5520

    1mg
    46.00€
    5mg
    80.00€
    10mg
    114.00€
    25mg
    236.00€
    50mg
    380.00€
    100mg
    595.00€
    1mL*10mM (DMSO)
    170.00€
  • CM304

    CAS:
    CM304 is a highly selective sigma-1 receptor antagonist.
    Formula:C18H26ClFN2OS
    Color and Shape:Solid
    Molecular weight:372.93

    Ref: TM-T71949

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Elzasonan

    CAS:
    Elzasonan is a selective 5-hydroxytryptamine 1B receptor antagonist used to treat patients with major depressive disorder and obsessive compulsive disorder.
    Formula:C22H23Cl2N3OS
    Color and Shape:Solid
    Molecular weight:448.41

    Ref: TM-T69364

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Phenoprolamine Hydrochloride

    CAS:
    Phenoprolamine HCl: α1 blocker with anti-hypertensive, brain, and heart protection; inhibits CYP2D/3A, crosses the blood-brain barrier.
    Formula:C21H30ClNO3
    Color and Shape:Solid
    Molecular weight:379.92

    Ref: TM-T28400

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Naxifylline

    CAS:
    Naxifylline is an A1 adenosine receptor blocker that increases urine and protects kidneys during edema treatment in heart failure.
    Formula:C18H24N4O3
    Color and Shape:Solid
    Molecular weight:344.41

    Ref: TM-T33600

    25mg
    2,157.00€
    50mg
    2,832.00€
    100mg
    3,800.00€
  • CAY10788

    CAS:
    CAY10788 is an antagonist of CysLT1 receptor.
    Formula:C18H15NO3
    Color and Shape:Solid
    Molecular weight:293.32

    Ref: TM-T71273

    1mg
    111.00€
    5mg
    487.00€
    10mg
    812.00€
    25mg
    1,596.00€
  • ONO-AE-248

    CAS:
    ONO-AE-248 is a selective agonist of EP3 receptor.
    Formula:C22H36O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:380.52

    Ref: TM-T28252

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • AVN-101 free base

    CAS:
    AVN-101: potent 5-HT7 antagonist, also targets 5-HT6, 5-HT2A, 5-HT2C. Aims to treat CNS disorders.
    Formula:C21H24N2
    Color and Shape:Solid
    Molecular weight:304.43

    Ref: TM-T71593

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Guanadrel Sulfate

    CAS:
    Guanadrel Sulfate, a postganglionic blocker, is stored in neurons via the norepinephrine pump.
    Formula:C10H21N3O6S
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:311.35

    Ref: TM-T9097L

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • SUN 1334H

    CAS:
    SUN 1334H is a potent, orally active, highly selective antagonist of H1 receptor(Ki of 9.7 nM).
    Formula:C23H28Cl2F2N2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:489.38

    Ref: TM-T13040

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • 2-Acetylbenzoic acid

    CAS:
    2-Acetylbenzoic acid outperforms 2-propionyloxybenzoic in hindering platelet function and PG synthesis; both similar in blocking PGI2 creation.
    Formula:C9H8O3
    Purity:99.62%
    Color and Shape:Off-White Solid
    Molecular weight:164.16

    Ref: TM-TMA0536

    1g
    34.00€
    1mL*10mM (DMSO)
    34.00€
  • WAY 629

    CAS:
    WAY 629 is a selective SR-2C agonist that also act as potent 5-HT2C receptor agonists.
    Formula:C15H18N2
    Color and Shape:Solid
    Molecular weight:226.32

    Ref: TM-T69067

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • GAT229

    CAS:
    GAT229 is a CB1 positive modulator, enhancing CB agonist activity without direct activation; influences binding, signaling, and lowers ocular pressure in mice.
    Formula:C22H18N2O2
    Color and Shape:Solid
    Molecular weight:342.39

    Ref: TM-T38204

    1mg
    379.00€
  • Pargolol

    CAS:
    Pargolol is a beta adrenergic receptor antagonist.
    Formula:C16H23NO3
    Color and Shape:Solid
    Molecular weight:277.36

    Ref: TM-T69217

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • CP-809101

    CAS:
    CP-809101 is an effective and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).
    Formula:C15H17ClN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:304.77

    Ref: TM-TQ0130

    5mg
    320.00€
    10mg
    502.00€
    25mg
    1,169.00€
    50mg
    2,185.00€
  • Colterol (free base)

    CAS:
    Colterol: short-acting β2 agonist; Bitolterol prodrug treats asthma, COPD bronchospasm.
    Formula:C12H19NO3
    Color and Shape:Solid
    Molecular weight:225.28

    Ref: TM-T70089

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • BN-81,674

    CAS:
    BN-81,674 is a bioactive chemical.
    Formula:C30H38N4
    Color and Shape:Solid
    Molecular weight:454.65

    Ref: TM-T30553

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Seprilose

    CAS:
    Seprilose, prostaglandin E2 inhibitor, inhibits prostaglandin E2 synthesis.
    Formula:C16H30O6
    Color and Shape:Solid
    Molecular weight:318.41

    Ref: TM-T28755

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CP 66713

    CAS:
    CP-66713 is an adenosine A2 receptor antagonist.
    Formula:C15H10ClN5
    Color and Shape:Solid
    Molecular weight:295.73

    Ref: TM-T31026

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • AM-211 sodium

    CAS:
    AM-211 sodium: potent DP2 receptor antagonist, active against allergic inflammation, selective, and orally bioavailable in rats and dogs.
    Formula:C27H26F3N2NaO4
    Color and Shape:Solid
    Molecular weight:522.5

    Ref: TM-T71088

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • M-25

    CAS:
    M-25 is a Smoothened antagonist and inhibitor of the Hedgehog pathway.
    Formula:C23H29N3O2
    Color and Shape:Solid
    Molecular weight:379.5

    Ref: TM-T71299

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Y2 Antagonist 36

    CAS:
    Y2 Antagonist 36 is a highly potent, soluble and selective antagonist of NPY Y2.
    Formula:C27H29ClN4O3
    Color and Shape:Solid
    Molecular weight:493

    Ref: TM-T29171

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SMM-189

    CAS:
    SMM-189 is a potent and selective CB2 inverse agonist.
    Formula:C19H12Cl2O3
    Color and Shape:Solid
    Molecular weight:359.2

    Ref: TM-T28819

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • CAY10412

    CAS:
    Anandamide (AEA) is an endocannabinoid with neural reuptake. CAY10412, an AEA analog, inhibits this reuptake without binding to CB receptors.
    Formula:C25H36O2S
    Color and Shape:Solid
    Molecular weight:400.62

    Ref: TM-T37684

    5mg
    128.00€
    10mg
    233.00€
    50mg
    945.00€
    100mg
    1,648.00€
  • A 49816

    CAS:
    A 49816 is a high-ceiling diuretic.
    Formula:C18H17Cl2NO5
    Color and Shape:Solid
    Molecular weight:398.24

    Ref: TM-T29496

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Stresson

    CAS:
    Stresson is a beta-blocking agent bunitrolol.
    Formula:C14H21ClN2O2
    Color and Shape:Solid
    Molecular weight:284.78

    Ref: TM-T34724

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • TR4161

    CAS:
    TR4161 is a prostaglandin bronchodilator of low tracheobronchial irritancy.
    Formula:C20H36O4
    Color and Shape:Solid
    Molecular weight:340.5

    Ref: TM-T34913

    1mg
    200.00€
    5mg
    828.00€
    10mg
    1,431.00€
    500µg
    112.00€
  • FK-1052 HCl

    CAS:
    FK-1052 HCl is a serotonin 3 & 4 dual receptor antagonist.
    Formula:C18H20ClN3O
    Color and Shape:Solid
    Molecular weight:329.83

    Ref: TM-T71045

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Photoregulin1

    CAS:
    Photoregulin1 modulates Nr2e3, slows photoreceptor degeneration in RhoP23H, Pde6brd1 mouse RP models.
    Formula:C21H23N3O2S
    Color and Shape:Solid
    Molecular weight:381.49

    Ref: TM-T28409

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Savoxepin mesylate

    CAS:
    Savoxepin mesylate, a tetracyclic cyano-dibenzoxepino-azepine derivative, has potent antidopaminergic activity.
    Formula:C26H30N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:466.59

    Ref: TM-T28666

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • LEQ-506

    CAS:
    LEQ506, an oral Smoothened antagonist, may inhibit cancer growth by blocking the Hedgehog signaling pathway.
    Formula:C27H29N5O
    Color and Shape:Solid
    Molecular weight:439.55

    Ref: TM-T71520

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PF-4522654

    CAS:
    PF-4522654 is a potent and selective 5-HT2C receptor agonist.
    Formula:C16H18F2N4
    Color and Shape:Solid
    Molecular weight:304.34

    Ref: TM-T71507

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • NR2F1 agonist 1

    CAS:
    NR2F1 agonist 1 activates cancer cell dormancy, suppresses growth in HNSCC, and inhibits tumor growth in mice.
    Formula:C28H30N4OS
    Color and Shape:Solid
    Molecular weight:470.63

    Ref: TM-T72776

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • Medroxalol hydrochloride

    CAS:
    Medroxalol hydrochloride is an antihypertensive agent that possesses both alpha and beta-adrenergic antagonistic properties.
    Formula:C20H25ClN2O5
    Color and Shape:Solid
    Molecular weight:408.88

    Ref: TM-T68838

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Zelandopam free base

    CAS:
    Zelandopam: dopamine D1 agonist, boosts pancreatic secretion, renal vasodilator, counters renal dysfunction.
    Formula:C15H15NO4
    Color and Shape:Solid
    Molecular weight:273.28

    Ref: TM-T29213

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Dothiepin HCl

    CAS:
    Dothiepin HCl: TCA, SNRI, with antihistamine, antiadrenergic, anticholinergic, and sodium block properties.
    Formula:C19H22ClNS
    Color and Shape:Solid
    Molecular weight:331.9

    Ref: TM-T69579

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Isamoltane

    CAS:
    Isamoltane is a serotonin 5-HT1 Receptor Antagonist
    Formula:C16H23ClN2O2
    Color and Shape:Solid
    Molecular weight:310.82

    Ref: TM-T68176

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Ro 63-0563

    CAS:
    Ro 63-0563 is a potent, 5-HT6 receptors selective antagonist.
    Formula:C13H17N5O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:307.37

    Ref: TM-T28594

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Labetalone hydrochloride

    CAS:
    Labetalone hydrochloride, a Labetalol impurity, is an orally active alpha and beta-adrenoceptor blocker.
    Formula:C19H23ClN2O3
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:362.85

    Ref: TM-T35326

    25mg
    43.00€
    50mg
    62.00€
    100mg
    92.00€
    200mg
    142.00€
    500mg
    235.00€
    1mL*10mM (DMSO)
    33.00€
  • 2-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide

    CAS:
    2-Decenoylaminoethyl cyclohexylethyl sulfide prevents stress ulcers, stabilizes phospholipase A2 and prostaglandin E2.
    Formula:C20H37NOS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:339.58

    Ref: TM-T13488

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (S)-Azelastine

    CAS:
    (S)-Azelastine is an antihistamine reducing receptors H1R, M1R, M3R, and inhibiting HNEpC cell growth.
    Formula:C22H24ClN3O
    Color and Shape:Solid
    Molecular weight:381.9

    Ref: TM-T70674

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SB 714786

    CAS:
    SB 714786 is a selective antagonist of 5-HT1D.
    Formula:C26H28N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:412.53

    Ref: TM-T28679

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Butaclamol HCl

    CAS:
    Butaclamol (AY-23,028), an unmarketed typical antipsychotic, is a research chemical that inhibits dopamine receptors.
    Formula:C25H32ClNO
    Color and Shape:Solid
    Molecular weight:397.98

    Ref: TM-T69355

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Trelanserin

    CAS:
    Trelanserin (SL-650472) is an antagonist of the serotonin receptor.
    Formula:C24H24FN5O2S
    Color and Shape:Solid
    Molecular weight:465.54

    Ref: TM-T34918

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • KY 234

    CAS:
    KY 234 is a thromboxane synthetase antagonist.
    Formula:C33H35N5O2
    Color and Shape:Solid
    Molecular weight:533.676

    Ref: TM-T70241

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • (R)-PF-06256142

    CAS:
    (R)-PF-06256142: low-activity R enantiomer of a potent, selective D1 agonist reducing receptor desensitization.
    Formula:C21H16N4O2
    Color and Shape:Solid
    Molecular weight:356.38

    Ref: TM-T72744

    25mg
    1,260.00€
    50mg
    1,639.00€
    100mg
    2,250.00€
  • APC-3316 tosylate

    CAS:
    APC-3316 tosylate is a vinyl sulfone cysteine protease inhibitor and selective CCR4 antagonist.
    Formula:C39H46N4O7S2
    Color and Shape:Solid
    Molecular weight:746.94

    Ref: TM-T69183

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • Benzoctamine

    CAS:
    Benzoctamine: oral psychoactive with tranquillizing effects; boosts catecholamine turnover; enhances rat heart [3H]noradrenaline uptake.
    Formula:C18H19N
    Color and Shape:Solid
    Molecular weight:249.35

    Ref: TM-T60368

    25mg
    1,927.00€
    50mg
    2,507.00€
    100mg
    3,168.00€
  • Efpeglenatide

    CAS:
    Efpeglenatide is a long-acting GLP-1 receptor agonist that improves insulin sensitivity, lowers blood glucose, delays weight gain, and supports metabolic disease research.
    Purity:100% - 100%
    Color and Shape:Solid

    Ref: TM-T64252

    1mg
    To inquire
    5mg
    To inquire
    10mg
    To inquire
    25mg
    1,539.00€
    50mg
    1,941.00€
    100mg
    2,451.00€
  • VPC12249

    CAS:
    VPC12249, a lysophosphatidic acid receptor type 1 (LPA1) antagonist, plays a functional role in osteoclast differentiation and bone resorption activity.
    Formula:C34H52NO6P
    Color and Shape:Solid
    Molecular weight:601.75

    Ref: TM-T29109

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • A2AAR antagonist 1

    CAS:
    Compound 21a, A2AAR antagonist with 20 nM Ki, useful in neurodegenerative disease study.
    Formula:C12H8BrN3O
    Color and Shape:Solid
    Molecular weight:290.12

    Ref: TM-T60591

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Alprenolol hydrochloride, (S)-

    CAS:
    Alprenolol hydrochloride, (S)- is a nonselective β-blocker. It is also a serotonin 5HT1A receptor antagonist.
    Formula:C15H24ClNO2
    Color and Shape:Solid
    Molecular weight:285.81

    Ref: TM-T4560L1

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Clonidine

    CAS:
    Clonidine (Kapvay): central alpha-adrenergic agonist, antihypertensive, often combined, not tied to liver issues.
    Formula:C9H9Cl2N3
    Purity:99.42% - 99.44%
    Color and Shape:Crystals Solid
    Molecular weight:230.09

    Ref: TM-T7045

    5mg
    35.00€
    10mg
    46.00€
    25mg
    64.00€
    50mg
    89.00€
    100mg
    130.00€
    500mg
    306.00€
  • CP94253 hydrochloride

    CAS:
    CP94253 hydrochloride: selective 5-HT1B agonist, Ki=2 nM; less active on 5-HT1A/D/C/2 (Ki=89/49/860/1600 nM).
    Formula:C15H20ClN3O
    Purity:99.78%
    Color and Shape:Solid
    Molecular weight:293.79

    Ref: TM-T22689

    5mg
    66.00€
    10mg
    90.00€
    25mg
    205.00€
    50mg
    334.00€
    100mg
    537.00€
    200mg
    745.00€
    1mL*10mM (DMSO)
    66.00€
  • (R)-(-)-α-Methylhistamine dihydrobromide

    CAS:
    (R)-(-)-α-Methylhistamine dihydrobromide is a potent and selective agonist of H3 histamine receptor( Kd of 50.3 nM).
    Formula:C6H13Br2N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:287

    Ref: TM-T12630

    50mg
    2,585.00€
  • Midodrine (hydrochloride)

    CAS:
    Midodrine hydrochloride ((±)-Midodrine hydrochloride) is an α1-receptor agonist used in the treatment of dysautonomia and orthostatic hypotension.
    Formula:C12H19ClN2O4
    Molecular weight:290.74

    Ref: TM-T21671

    10mg
    To inquire
    25mg
    To inquire
  • A61603

    CAS:
    A61603 is an alpha-1A adrenergic receptor.
    Formula:C14H19N3O3S
    Color and Shape:Solid
    Molecular weight:309.38

    Ref: TM-T29511

    25mg
    1,586.00€
    50mg
    2,072.00€
    100mg
    2,660.00€
  • SV293

    CAS:
    SV293 is a selective antagonist of D2 dopamine receptor.
    Formula:C22H26N2O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:382.52

    Ref: TM-T28890

    25mg
    1,444.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
  • (R)-DOI hydrochloride

    CAS:
    (R)-DOI hydrochloride is the salt form of 2,5-Dimethoxy-4-iodoamphetamine (DOI), a potent 5-HT2A and 5-HT2C receptor agonist, orally active and hallucinogenic.
    Formula:C11H17ClINO2
    Purity:99.88% - >99.99%
    Color and Shape:Solid
    Molecular weight:357.62

    Ref: TM-T68620

    1mg
    285.00€
    5mg
    692.00€
    10mg
    947.00€
    25mg
    1,458.00€
    50mg
    1,839.00€
    100mg
    2,322.00€
  • EA-230

    CAS:
    Ea-230 is an immunomodulator that may be used in the treatment of renal failure.
    Formula:C15H27N5O6
    Color and Shape:Solid
    Molecular weight:373.4

    Ref: TM-T31594

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • Amosulalol, (-)-

    CAS:
    Amosulalol, (-)-, is an adrenergic agent.
    Formula:C18H24N2O5S
    Color and Shape:Solid
    Molecular weight:380.46

    Ref: TM-T30028

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • SID7970631

    CAS:
    SID7970631 is an isoquinolinone analogue, a selective and potent submicromolar SF-1 inhibitor with an IC50 of 260 nM. SID7970631 can be used to study cancer.
    Formula:C24H24N2O7
    Color and Shape:Solid
    Molecular weight:452.46

    Ref: TM-T62757

    25mg
    690.00€
    50mg
    895.00€
    100mg
    1,404.00€
  • BGC201531

    CAS:

    BGC201531 (AP-1531) is a EP4 antagonist for the treatment of acute migraine.

    Formula:C26H28N2O6S
    Purity:98.51% - 99.33%
    Color and Shape:Solid
    Molecular weight:496.58

    Ref: TM-T8993

    1mg
    136.00€
    5mg
    320.00€
    10mg
    465.00€
    25mg
    777.00€
    50mg
    1,074.00€
    100mg
    1,454.00€
  • Lesopitron dihydrochloride

    CAS:
    Lesopitron dihydrochloride with IC50 of 125 nM in rat hippocampal membranes, is a full and selective 5-HT1A receptor agonist.
    Formula:C15H23Cl3N6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:393.74

    Ref: TM-T11839

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • L-750,667 Trihydrochloride

    CAS:
    L-750,667 Trihydrochloride is a selective D4 receptor antagonist, reverses the dopamine-induced inhibition of cAMP accumulation in the central nervous system.
    Formula:C18H22Cl3IN4
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:527.66

    Ref: TM-T27777

    1mg
    62.00€
    5mg
    130.00€
    10mg
    203.00€
    25mg
    412.00€
    50mg
    652.00€
    100mg
    1,027.00€
    200mg
    1,391.00€
  • CCX354

    CAS:
    CCX354 (CCR1 antagonist 1) is a potent small molecule CCR1 antagonist with anti-inflammatory activity for the treatment of rheumatoid arthritis.
    Formula:C22H22ClN7O2
    Purity:99.43% - 99.44%
    Color and Shape:Solid
    Molecular weight:451.91

    Ref: TM-T15253

    1mg
    250.00€
    5mg
    562.00€
    10mg
    909.00€
    25mg
    1,406.00€
    50mg
    1,882.00€
    100mg
    2,375.00€
    200mg
    3,163.00€
  • Azelastine

    CAS:
    Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.
    Formula:C22H24ClN3O
    Purity:99.35% - 99.99%
    Color and Shape:White Crystal Powder
    Molecular weight:381.90

    Ref: TM-T0211

    100mg
    52.00€
  • BI-6901

    CAS:
    BI-6901 is a CCR10 antagonist. In a mouse model of DNFB exposure hypersensitivity, BI 6901 displays its anti-inflammatory response in a dose-dependent manner.
    Formula:C23H27N5O3S
    Purity:99.83% - 99.94%
    Color and Shape:Solid
    Molecular weight:453.56

    Ref: TM-T36478

    1mg
    180.00€
  • GW 766994

    CAS:
    GW 766994 is a specific and oral chemokine receptor-3 (CCR3) antagonist. It has the potential for asthma and eosinophilic bronchitis treatment.
    Formula:C21H24Cl2N4O3
    Purity:98.77%
    Color and Shape:Solid
    Molecular weight:451.35

    Ref: TM-T11521

    25mg
    1,080.00€
    50mg
    1,404.00€
    100mg
    2,250.00€
  • Nexopamil racemate

    CAS:
    Nexopamil racemate((Rac)-Nexopamil) is a racemate of Nexopamil. The Nexopamil racemate has potential anti-asthmatic and anti-ulcer activity.
    Formula:C24H40N2O3
    Purity:98.61%
    Color and Shape:Solid
    Molecular weight:404.59

    Ref: TM-T12215

    1mg
    630.00€
    5mg
    1,620.00€
  • CCR2 antagonist 3

    CAS:
    CCR2 antagonist 3 (AZD-2927) is an antagonist of CCR2.
    Formula:C17H25FN2O2
    Purity:99.87%
    Color and Shape:Solid
    Molecular weight:308.39

    Ref: TM-T10712

    1mg
    66.00€
    5mg
    147.00€
    10mg
    225.00€
    25mg
    398.00€
    50mg
    532.00€
    100mg
    745.00€
    200mg
    982.00€
    1mL*10mM (DMSO)
    161.00€
  • NPS-2143

    CAS:
    NPS-2143 (SB 262470A) is a novel potent and selective antagonist of Ca(2+) receptor.
    Formula:C24H25ClN2O2
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:408.92

    Ref: TM-T1730

    1ml
    54.00€
    5mg
    49.00€
    10mg
    82.00€
    25mg
    145.00€
    50mg
    208.00€
    100mg
    313.00€
  • CCR1 antagonist 9

    CAS:
    CCR1 antagonist 9 (compound 19e) is a selective CCR1 antagonist based on aziridine. CCR1 inhibition in calcium flux assays.
    Formula:C20H16FN5O3S
    Purity:99.13%
    Color and Shape:Solid
    Molecular weight:425.44

    Ref: TM-T10710

    1mg
    101.00€
    5mg
    241.00€
    10mg
    402.00€
    25mg
    727.00€
    50mg
    1,046.00€
    100mg
    1,525.00€
    1mL*10mM (DMSO)
    265.00€
  • YM022

    CAS:
    YM022 is a highly effective and selective gastrin/cholecystokinin (CCK)-B receptor antagonist.
    Formula:C32H28N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:516.59

    Ref: TM-T17274

    10mg
    919.00€
    50mg
    3,771.00€
  • C-021 dihydrochloride

    CAS:
    C-021 dihydrochloride is a potent CCR4 antagonist. It potently inhibits functional chemotaxis in human and mouse with IC50s of 140 nM and 39 nM.
    Formula:C27H43Cl2N5O2
    Purity:98.67%
    Color and Shape:Solid
    Molecular weight:540.57

    Ref: TM-T10639

    1mg
    52.00€
    5mg
    97.00€
    10mg
    154.00€
    25mg
    249.00€
    50mg
    374.00€
    1mL*10mM (DMSO)
    115.00€
  • CCR4 antagonist 3-1

    CAS:

    CCR4 antagonist 3-1 is a weak inhibitor of [125I]TARC binding and CEM cell migration, with IC50 values of 1.7 μM and 6.4 μM, respectively.

    Formula:C14H12N2S
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:240.32

    Ref: TM-T60336

    1mg
    92.00€
    5mg
    216.00€
    10mg
    354.00€
    25mg
    692.00€
    50mg
    1,074.00€
    100mg
    1,454.00€
    500mg
    2,822.00€
  • Calhex 231 hydrochloride

    CAS:
    Calhex 231 hydrochloride a potent CaSR negative-conversion modulator that blocks the increase in [3H]inositol phosphate, inhibits mir-208a-mediated .
    Formula:C25H28Cl2N2O
    Purity:99.36%
    Color and Shape:Solid
    Molecular weight:443.41

    Ref: TM-T10666

    1mg
    47.00€
    5mg
    92.00€
    10mg
    152.00€
    25mg
    To inquire
    50mg
    To inquire
    1mL*10mM (DMSO)
    101.00€
  • SMANT hydrochloride

    CAS:
    SMANT hydrochloride (N-(4-bromophenyl)-3-(3,5-dimethylpiperidin-1-yl)propanamide hydrochloride) is an antagonist of Smoothened accumulation.
    Formula:C16H24BrClN2O
    Purity:99.81%
    Color and Shape:Solid
    Molecular weight:375.73

    Ref: TM-T23370

    10mg
    44.00€
    25mg
    82.00€
    50mg
    130.00€
    100mg
    213.00€
    200mg
    309.00€
  • Monatepil maleate

    CAS:
    Monatepil maleate (AJ-2615 maleate) is a Ca2+-channel and α1-adrenergic receptor antagonist, and ACAT inhibitor with antihypertensive activity.
    Formula:C32H34FN3O5S
    Purity:97.90%
    Color and Shape:Solid
    Molecular weight:591.69

    Ref: TM-T25828

    1mg
    279.00€
    5mg
    685.00€
    10mg
    938.00€
    25mg
    1,444.00€
    50mg
    1,882.00€
  • CCR1 antagonist 7

    CAS:
    CCR1 antagonist 7 (compound 16r) is an antagonist of chemokine receptor 1 (CCR1) with an IC 50 of 4 nM [1].
    Formula:C21H24ClN5O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:461.96

    Ref: TM-T10709

    25mg
    1,369.00€
    50mg
    1,783.00€
    100mg
    2,250.00€
  • PNU-177864

    CAS:
    PNU-177864 is a selective dopamine D3 receptor antagonist.
    Formula:C18H21F3N2O3S
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:402.43

    Ref: TM-T23167

    1mg
    42.00€
    5mg
    84.00€
    10mg
    93.00€
    25mg
    202.00€
    50mg
    284.00€
    100mg
    391.00€
    200mg
    545.00€
  • S 14506 hydrochloride

    CAS:
    S 14506 hydrochloride is a 5-HT1A receptor full agonist.
    Formula:C24H27ClFN3O2
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:443.94

    Ref: TM-T23285

    2mg
    47.00€
    5mg
    67.00€
    10mg
    101.00€
    25mg
    197.00€
    50mg
    304.00€
    100mg
    457.00€
    200mg
    650.00€
  • Iodophenpropit dihydrobromide

    CAS:
    Iodophenpropit dihydrobromide: selective histamine H3 antagonist, reversible binding, high affinity (KD: 0.32 nM).
    Formula:C15H20BrIN4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:495.22

    Ref: TM-T15590

    5mg
    386.00€
    10mg
    577.00€
  • PF-03654746 Tosylate

    CAS:
    PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
    Formula:C25H32F2N2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:494.6

    Ref: TM-T12416

    25mg
    828.00€
    50mg
    1,063.00€
    100mg
    1,611.00€
  • SB-277011 dihydrochloride

    CAS:
    SB-277011 dihydrochloride: potent, selective D3 antagonist; orally bioavailable; crosses blood-brain barrier; pKi 8.0 for D3 receptor.
    Formula:C28H32Cl2N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:511.49

    Ref: TM-T12861L

    1mg
    148.00€
    5mg
    384.00€
    10mg
    617.00€
    25mg
    1,378.00€
  • Taprenepag isopropyl

    CAS:
    Taprenepag isopropyl is a highly selective agonist of the EP2 receptor.
    Formula:C27H28N4O5S
    Purity:99.44%
    Color and Shape:Solid
    Molecular weight:520.6

    Ref: TM-T16988

    2mg
    47.00€