GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,024 products)
- Adenosine Receptor(249 products)
- Adrenergic Receptor(3,029 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(159 products)
- CaSR(34 products)
- Cannabinoid Receptor(217 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(443 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(83 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(22 products)
- Glucagon Receptor(195 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(42 products)
- Opioid Receptor(326 products)
- PAFR(14 products)
- PKA(52 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5972 products of "GPCR/G-Protein"
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Acreozast
CAS:Acreozast, a histamine release inhibitor, is used potentially for the treatment of asthma and atopic dermatitis.Formula:C15H14ClN3O6Color and Shape:SolidMolecular weight:367.74LASSBio-1359
CAS:LASSBio-1359 is an adenosine receptor agonist. It acts by inducing relaxation of the corpus cavernosum. It also acts as a novel selective phosphodiesterase.Formula:C17H18N2O3Purity:98%Color and Shape:SolidMolecular weight:298.34LP44 hydrochloride
CAS:LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.Formula:C27H38ClN3OSPurity:98.06%Color and Shape:SolidMolecular weight:488.13Phenindamine
CAS:Phenindamine (Nu 1504) is an H1-receptor antagonist which is antihistamine[1].Formula:C19H19NColor and Shape:SolidMolecular weight:261.36CM398
CAS:CM398, a sigma-2 receptor selective ligand (Ki=0.43 nM), also binds dopamine and serotonin transporters, shows anti-inflammatory analgesic effects.Formula:C23H29N3O3Color and Shape:SolidMolecular weight:395.49Eplivanserin hemifumarate
CAS:Eplivanserin is an inverse agonist of 5-HT2A.Formula:C23H25FN2O6Color and Shape:SolidMolecular weight:444.45Rp-cAMPS sodium
CAS:Rp-cAMPS sodium is a phosphorothioate analog of cAMP, a PKA inhibitor and cAMP antagonist that inhibits cAMP-dependent protein kinases.Formula:C10H11N5NaO5PSPurity:99.71%Color and Shape:SolidMolecular weight:367.25VUF-10497
CAS:VUF-10497: H4 receptor inverse agonist, anti-inflammatory in rats, binds human H1 receptor (pKi=7.57).Formula:C18H20ClN5SPurity:98%Color and Shape:SolidMolecular weight:373.9LY 334370 hydrochloride
CAS:5-HT1F receptor agonistFormula:C21H23ClFN3OPurity:98%Color and Shape:SolidMolecular weight:387.88BMS CCR2 22
CAS:BMS CCR2 22 is a potent and selective antagonist of CCR2 with calcium flux IC50 of 18 nM, chemotaxis IC50 of 1 nM, and binding IC50 of 5.1 nM.Formula:C28H34F3N5O4SPurity:99.65%Color and Shape:SolidMolecular weight:593.66Ref: TM-T14688
1mg58.00€5mg116.00€10mg183.00€25mg368.00€50mg562.00€100mg758.00€200mg1,017.00€1mL*10mM (DMSO)156.00€CYM5181
CAS:<p>CYM5181 is related to the body's immune system and can be used to study multiple sclerosis, transplant rejection, and adult respiratory distress syndrome.</p>Formula:C17H17N3O3Purity:99.51%Color and Shape:SolidMolecular weight:311.34Rezatomidine
CAS:Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.Formula:C13H16N2SPurity:98.34%Color and Shape:SolidMolecular weight:232.34Adoprazine
CAS:<p>Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.</p>Formula:C24H24FN3O2Purity:99.83%Color and Shape:SolidMolecular weight:405.46Halopemide
CAS:Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).Formula:C21H22ClFN4O2Purity:96.57%Color and Shape:SolidMolecular weight:416.88BL-1020 Mesylate
CAS:BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.Formula:C28H45ClN4O11S4Purity:>99.99%Color and Shape:SolidMolecular weight:777.39Pipoxazole
CAS:Pipoxazole, an adrenergic receptor antagonist, is used potentially for the treatment of depression.Formula:C14H20N4OPurity:98.58% - 99.53%Color and Shape:SolidMolecular weight:260.33SCH-336
CAS:<p>SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 preference, reduces leukocyte migration and eosinophilia.</p>Formula:C23H25NO8S3Purity:95.01%Color and Shape:SolidMolecular weight:539.64Ticalopride
CAS:Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.Formula:C14H20ClN3O3Purity:99.51%Color and Shape:SolidMolecular weight:313.78A2A receptor antagonist 1
CAS:A2A receptor antagonist 1 (CPI-444 analog) is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.Formula:C16H12FN5OPurity:99.52% - 99.93%Color and Shape:SolidMolecular weight:309.3Ref: TM-T37792
2mgTo inquire5mg62.00€10mg87.00€25mg183.00€50mg280.00€100mg416.00€200mgTo inquire1mL*10mM (DMSO)47.00€Isbogrel
CAS:Isbogrel (CV4151) is a TXA2 synthase inhibitor for researching arrhythmias, ischemic attacks, and thrombosis.Formula:C18H19NO2Purity:99.58%Color and Shape:SolidMolecular weight:281.35NNC 92-1687
CAS:NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.Formula:C15H12N2O3SPurity:98.70% - 99.96%Color and Shape:SolidMolecular weight:300.33BMS-817399
CAS:BMS-817399: oral CCR1 antagonist with binding and chemotaxis inhibition IC50s, potential for rheumatoid arthritis research.Formula:C23H36ClN3O4Purity:99.7%Color and Shape:SolidMolecular weight:454Ref: TM-T26861
1mg160.00€5mg338.00€10mg512.00€25mg812.00€50mg1,093.00€100mg1,473.00€1mL*10mM (DMSO)376.00€Lesopitron
CAS:Lesopitron: anxiolytic, 5-HT1A agonist, treats rodent anxiety, counters benzodiazepine withdrawal, low toxicity, no alcohol/barbiturate interaction.Formula:C15H21ClN6Purity:99.33% - 99.46%Color and Shape:SolidMolecular weight:320.82Ref: TM-T25672
1mg140.00€5mg343.00€10mg504.00€25mg817.00€50mg1,121.00€100mg1,510.00€500mg3,030.00€1mL*10mM (DMSO)340.00€LTB4-IN-1
CAS:LTB4-IN-1 (Anti-inflammatory agent 2) with IC50 of 70 nM is an inhibitor of leukotriene synthesis (LTB4).Formula:C26H30N2O4SPurity:99.93%Color and Shape:SolidMolecular weight:466.59Ref: TM-T10917
1mg276.00€5mg545.00€10mg924.00€25mg1,359.00€50mg1,853.00€100mg2,490.00€1mL*10mM (DMSO)690.00€DA-6886
CAS:DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.Formula:C19H28Cl2N6O2Purity:99.91% - 99.99%Color and Shape:SolidMolecular weight:443.37R 59-022 hydrochloride
CAS:<p>R 59-022 hydrochloride is a 5-HT antagonist, PKC activator, DGK inhibitor (IC50: 2.8 µM), and modulates lipid production in platelets and neutrophils.</p>Formula:C27H27ClFN3OSPurity:97.7%Color and Shape:SolidMolecular weight:496.04Bavisant
CAS:Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.Formula:C19H27N3O2Purity:99.21% - 99.65%Color and Shape:SolidMolecular weight:329.44Ref: TM-TQ0046
1mg43.00€5mg96.00€10mg134.00€25mg221.00€50mg325.00€100mg465.00€500mgTo inquire1mL*10mM (DMSO)94.00€Clemastine
CAS:Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.Formula:C21H26ClNOPurity:99.21%Color and Shape:SolidMolecular weight:343.89Egis-11150
CAS:Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.Formula:C19H21ClFN5O2Purity:97.49% - >99.99%Color and Shape:SolidMolecular weight:405.85Rafabegron
CAS:Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.Formula:C21H23ClN2O4Purity:99.81%Color and Shape:SolidMolecular weight:402.87PPTN hydrochloride
CAS:<p>PPTN hydrochloride is a potent, high-affinity, competitive, highly selective P2Y14 receptor antagonist (KB: 434 pM), but no agonist or antagonist activity at</p>Formula:C29H25ClF3NO2Purity:99.80%Color and Shape:SolidMolecular weight:511.96Nemazoline Free Base
CAS:Nemazoline Free Base: a long-lasting nasal decongestant, better than oxymetazoline, with no systemic effects or toxicity in dogs and rats.Formula:C10H11Cl2N3Purity:98.06% - 98.83%Color and Shape:SolidMolecular weight:244.12BMY-14802 hydrochloride
CAS:BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.Formula:C18H23ClF2N4OPurity:99.97%Color and Shape:SolidMolecular weight:384.85A-437203
CAS:A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.Formula:C20H27F3N6OSPurity:98.80%Color and Shape:SolidMolecular weight:456.53Ref: TM-T10213
1mg89.00€5mg198.00€10mg279.00€25mg434.00€50mg562.00€100mg780.00€200mg1,035.00€1mL*10mM (DMSO)227.00€N-[(4-Aminophenyl)methyl]adenosine
CAS:N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).Formula:C17H20N6O4Purity:98.75%Color and Shape:SolidMolecular weight:372.38Ref: TM-T16166
1mg55.00€5mg117.00€10mg170.00€25mg335.00€50mg532.00€100mg848.00€1mL*10mM (DMSO)149.00€SB 699551 dihydrochloride
CAS:SB 699551 dihydrochloride is a 5-ht5a receptor antagonist.Formula:C34H47Cl2N3OPurity:99.83%Color and Shape:SolidMolecular weight:584.66Ref: TM-T23325
1mg52.00€5mg111.00€10mg180.00€25mg311.00€50mg449.00€100mg615.00€1mL*10mM (DMSO)150.00€Amosulalol
CAS:<p>Amosulalol is a combined alpha and beta adrenoceptor antagonist.</p>Formula:C18H24N2O5SPurity:99.5%Color and Shape:SolidMolecular weight:380.46Dabelotine
CAS:<p>Dabelotine (UNII-6RY56RB98P) is an adrenergic agonist used in the study of dementia.</p>Formula:C15H22N2O2Purity:98.55%Color and Shape:SolidMolecular weight:262.35Milenperone
CAS:Milenperone (R 34009) is a novel anti-invasive compound for the control of behavioral disorders in patients with epilepsy and alcoholism.Formula:C22H23ClFN3O2Purity:98.09% - 99.84%Color and Shape:SolidMolecular weight:415.89Femoxetine hydrochloride
CAS:Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.Formula:C20H26ClNO2Purity:99.63%Color and Shape:SolidMolecular weight:347.88FK-453
CAS:FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.Formula:C23H25N3O2Purity:99.44%Color and Shape:SolidMolecular weight:375.46K6PC-5
CAS:K6PC-5 is a ceramide derivative that acts as an activator of sphingosine kinase 1 (SPHK1), inducing a swift and temporary rise in intracellular calcium levels.Formula:C19H37NO4Purity:99.9%Color and Shape:SolidMolecular weight:343.5Compound C108
CAS:<p>Compound C108 is an inhibitor of GTPase-activating protein SH3 domain-binding protein 2 (G3BP2).</p>Formula:C15H14N2O3Purity:99.77%Color and Shape:SolidMolecular weight:270.28BMS-470539 dihydrochloride
CAS:BMS-470539 dihydrochloride is a MC-1 R agonist with anti-inflammatory activity.Formula:C32H43Cl2N5O4Purity:>99.99%Color and Shape:SolidMolecular weight:632.62Selodenoson
CAS:Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.Formula:C17H24N6O4Purity:99.39%Color and Shape:SolidMolecular weight:376.41ANR 94
CAS:ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.Formula:C9H13N5OPurity:98.9%Color and Shape:SolidMolecular weight:207.23Ref: TM-T22031
5mg48.00€10mg74.00€25mg137.00€50mg230.00€100mg325.00€200mg457.00€1mL*10mM (DMSO)48.00€Neldazosin
CAS:Neldazosin is used as a potent α1-adrenoceptor antagonist.Formula:C18H25N5O4Purity:99.76% - 99.97%Color and Shape:SolidMolecular weight:375.42LY266097 hydrochloride
CAS:<p>LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.</p>Formula:C21H24Cl2N2O2Purity:98.58%Color and Shape:SolidMolecular weight:407.33Rocepafant
CAS:Rocepafant (LAU8080), a PAF antagonist, reduces neonatal rat brain damage and inhibits TNF-α toxicity in L929 cells.Formula:C26H23ClN6OS2Purity:97.31% - 98.95%Color and Shape:SolidMolecular weight:535.088-OH-Dpat
CAS:<p>8-OH-Dpat (8-Hydroxy-DPAT) is a serotonin 1A-receptor agonist that is used experimentally to test the effects of serotonin.</p>Formula:C16H25NOPurity:98%Color and Shape:SolidMolecular weight:247.38Milveterol HCl
CAS:Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).Formula:C25H30ClN3O4Purity:99.9%Color and Shape:SolidMolecular weight:471.98AM-1235
CAS:AM-1235 is a potent and selective cannabinoid receptor CB1 agonist.Formula:C24H21FN2O3Purity:99.92%Color and Shape:SolidMolecular weight:404.43SDZ-62-434
CAS:SDZ-62-434 is a platelet-activating factor inhibitor with antitumor activity and may be used in the study of leukemia.Formula:C23H27Cl2N3Purity:98.38%Color and Shape:SolidMolecular weight:416.39Quinupramine
CAS:Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.Formula:C21H24N2Purity:99.77%Color and Shape:SolidMolecular weight:304.43ML 10302 hydrochloride
CAS:ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.Formula:C15H22Cl2N2O3Purity:99.99%Color and Shape:SolidMolecular weight:349.25(Z)-Thiothixene
CAS:<p>(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.</p>Formula:C23H29N3O2S2Purity:99.21%Color and Shape:Yellow To Yellow With A Tan Cast PowderMolecular weight:443.63Lorglumide sodium salt
CAS:Lorglumide sodium salt (CR-1409 sodium salt) is an antagonist of cholecystokinin receptors (CCK).Formula:C22H31Cl2N2NaO4Purity:99.32%Color and Shape:SolidMolecular weight:481.39APNEA
CAS:APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.Formula:C18H22N6O4Purity:99.88%Color and Shape:SolidMolecular weight:386.41Roxindole
CAS:Roxindole: dopamine agonist, serotonin reuptake inhibitor, 5-HT1A agonist, developed for schizophrenia.Formula:C23H26N2OPurity:98.03% - 98.93%Color and Shape:SolidMolecular weight:346.4748740 RP
CAS:48740 RP (RP 55779) is an antagonist of platelet-activating factor.Formula:C12H11N3OSPurity:99.79%Color and Shape:SolidMolecular weight:245.3Ref: TM-T10159
1mg356.00€5mg567.00€10mg907.00€25mg1,339.00€50mg1,815.00€100mg2,432.00€1mL*10mM (DMSO)567.00€Spizofurone
CAS:Spizofurone (Espizofurona) has anti-ulcer activity, protective effect on the gastric mucosa of rats and can increase alkaline secretion.Formula:C12H10O3Purity:>99.99%Color and Shape:SolidMolecular weight:202.21Oxyfedrine L-form HCl
CAS:Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent.Formula:C19H24ClNO3Purity:99.5% - 99.57%Color and Shape:SolidMolecular weight:349.85Ref: TM-T24579
1mg96.00€5mg188.00€10mg329.00€25mg512.00€50mg740.00€100mg944.00€200mg1,264.00€1mL*10mM (DMSO)215.00€Ecopipam
CAS:Ecopipam: orally active, selective dopamine D1/D5 antagonist (Ki: 1.2 nM/2.0 nM). 40x more selective over D2/D4/5-HT/α2a. For schizophrenia, obesity research.Formula:C19H20ClNOPurity:99.68%Color and Shape:SolidMolecular weight:313.82Butofilolol
CAS:Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.Formula:C17H26FNO3Purity:98.96% - >99.99%Color and Shape:SolidMolecular weight:311.392Xamoterol hemifumarate
CAS:Xamoterol hemifumarate is a potent and selective β1-adrenoceptor agonist.Xamoterol hemifumarate is a potential compound for the study of the relationshipFormula:C36H54N6O14Purity:99.79%Color and Shape:White SolidMolecular weight:794.37Ecastolol
CAS:Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.Formula:C26H33N3O6Purity:99.89%Color and Shape:SolidMolecular weight:483.56Ref: TM-T11148
1mg369.00€5mg735.00€10mg938.00€25mg1,473.00€50mg1,882.00€100mg2,670.00€1mL*10mM (DMSO)929.00€NCGC00135472
CAS:NCGC00135472: DRV1 agonist with pro-catabolic effects, activates DRV1/GPR32, EC50: 0.37 uM (beta-blocker), 0.05 uM (cAMP), enhances phagocytosis.Formula:C20H14F2N4OPurity:99.41% - 99.48%Color and Shape:SolidMolecular weight:364.35Ref: TM-T33613
1mg333.00€5mg787.00€10mg1,074.00€25mg1,510.00€50mg1,882.00€100mg2,375.00€500mg4,655.00€Goxalapladib
CAS:Goxalapladib（GSK 677116） is a small molecule compound that can be used to treat cardiovascular risks associated with atherosclerosis.Formula:C40H39F5N4O3Purity:99.64% - 99.93%Color and Shape:SolidMolecular weight:718.75UNC0006
CAS:<p>UNC0006 is a β-arrestin-biased dopamine D2 ligand.</p>Formula:C24H29Cl2N3O2Purity:99.35% - 99.97%Color and Shape:SolidMolecular weight:462.415-HT2 antagonist 1
CAS:5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.Formula:C22H29FN4O2Purity:99.76%Color and Shape:SolidMolecular weight:400.49Ref: TM-T12597
1mg678.00€5mg1,359.00€10mg1,833.00€25mg2,727.00€50mg3,676.00€100mg4,969.00€1mL*10mM (DMSO)1,605.00€Proxyfan
CAS:Proxyfan is a high-affinity protean antagonist/agonist of H3 receptors from full agonist to full inverse agonist, depending on given tissue or brain region.Formula:C13H16N2OPurity:99.68%Color and Shape:SolidMolecular weight:216.28Noberastine
CAS:Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.Formula:C17H21N5OPurity:99.72% - >99.99%Color and Shape:SolidMolecular weight:311.38Masilukast
CAS:Masilukast(MCC-847) is an oral leukotriene D4 (LTD4) receptor antagonist for the study of diseases associated with inflammation.Formula:C31H32F3N3O5SPurity:99.23% - 99.62%Color and Shape:SolidMolecular weight:615.66NP10679
CAS:NP10679 is a N-methyl-D-aspartate (NMDA) receptor inhibitor of the GluN2B subunit that inhibits histamine H1, hERG channels, and CYPase.Formula:C23H26F3N3O3Purity:99.43%Color and Shape:SolidMolecular weight:449.47Nonabine
CAS:Nonabine is a compound with strong antiemetic properties that can be used to prevent nausea and vomiting associated with cancer chemotherapy.Formula:C25H33NO2Purity:99.82% - 99.94%Color and Shape:SolidMolecular weight:379.54L-693,403 maleate
CAS:L-693,403 maleate has analgesic activity.Formula:C24H27NO4Purity:99.88%Color and Shape:SolidMolecular weight:393.48Ref: TM-T22899
1mg333.00€5mg787.00€10mg1,074.00€25mg1,510.00€50mg1,882.00€100mg2,375.00€500mg4,655.00€Lensiprazine
CAS:Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder andFormula:C24H27FN4O2Purity:97.86%Color and Shape:SolidMolecular weight:422.5CP 96021
CAS:<p>"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."</p>Formula:C29H21FN4OSPurity:97.81% - 99.62%Color and Shape:SoildMolecular weight:492.57Evodenoson
CAS:Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.Formula:C23H29N7O6Purity:99.75% - 99.83%Color and Shape:SolidMolecular weight:499.52LX-2931
CAS:LX-2931(LX-3305) is a sphingosine-1-phosphate cleavage enzyme (S1P) inhibitor for the treatment of rheumatoid arthritis.Formula:C9H15N3O5Purity:98.85% - 99.83%Color and Shape:SolidMolecular weight:245.23cis-Urocanic acid
CAS:cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).Formula:C6H6N2O2Purity:99.81%Color and Shape:SolidMolecular weight:138.12SLP9101555
<p>SLP9101555 is a potent and selective sphingosine kinase 2 (SphK2) inhibitor with a Ki of 90 nM.SLP9101555 has a high affinity for SphK2, which is 200-fold</p>Formula:C16H22BrClN2Purity:99.45%Color and Shape:SolidMolecular weight:357.72Ref: TM-T63047
1mg333.00€5mg787.00€10mg1,074.00€25mg1,510.00€50mg1,882.00€100mg2,375.00€500mg4,655.00€Tedatioxetine
CAS:Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.Formula:C18H21NSPurity:99.76% - >99.99%Color and Shape:SolidMolecular weight:283.43ReN-1869
CAS:ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseasesFormula:C24H27NO2Purity:99.83% - 99.98%Color and Shape:SolidMolecular weight:361.48CMF019
CAS:CMF019 is a potent agonist of the Apelin receptor (APJ) with G protein bias. CMF019 binds to APJ (pKis: 8.58, 8.49, and 8.71 for the human, rat, and mouse).Formula:C25H33N3O3SPurity:99.5%Color and Shape:SolidMolecular weight:455.61CCR1 antagonist 6
CAS:<p>CCR1 antagonist 6 is a CCR1 antagonist (IC50: 3 nM).</p>Formula:C21H23ClN4O3SPurity:99.02% - 99.15%Color and Shape:SolidMolecular weight:446.95SMO-IN-2
CAS:SMO-IN-2 is a SMO inhibitor with antiproliferative activity and anticancer activity and inhibits Hh signaling.SMO-IN-2 can be used in the study of cancer.Formula:C25H25F4N5O2Purity:98.64%Color and Shape:SolidMolecular weight:503.49BMS 182874
CAS:BMS 182874: Oral ETA antagonist, IC50=0.150 μM, Ki=0.055 μM, lowers hypertension in rats.Formula:C17H19N3O3SPurity:99.73%Color and Shape:SolidMolecular weight:345.42KSK94
CAS:KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value of 75.2 nM, and can be used to study injurious pain.Formula:C25H26N4OPurity:99.60%Color and Shape:SolidMolecular weight:398.5Sinitrodil
CAS:Sinitrodil (ITF-296) is a guanylate cyclase stimulant that may be used in the treatment of myocardial ischemia and angina pectoris.Formula:C10H10N2O5Purity:97.03%Color and Shape:SolidMolecular weight:238.2Ref: TM-T34648
1mg139.00€5mg333.00€10mg504.00€25mg817.00€50mg1,121.00€100mg1,510.00€500mg3,030.00€1mL*10mM (DMSO)401.00€Landipirdine
CAS:Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.Formula:C18H19FN2O3SPurity:97.61% - 99.99%Color and Shape:SolidMolecular weight:362.42Thonzylamine hydrochloride
CAS:Thonzylamine hydrochloride (Resistab) is an anticholinergic and antihistamine used as an antipruritic.Formula:C16H23ClN4OPurity:99.67%Color and Shape:White Crystalline PowderMolecular weight:322.83Enerisant hydrochloride
CAS:Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteinsFormula:C22H31ClN4O3Purity:99.95%Color and Shape:SolidMolecular weight:434.96OPC-51803
CAS:OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.Formula:C26H32ClN3O2Purity:98.93% - >99.99%Color and Shape:SolidMolecular weight:454JTE-907
CAS:JTE-907 是一种具有高度选择性和口服活性的 CB2 受体反向激动剂。JTE-907在体内展现出抗炎活性。Formula:C24H26N2O6Purity:99.93%Color and Shape:SolidMolecular weight:438.47Ref: TM-T19705
1mg56.00€5mg126.00€10mg187.00€25mg329.00€50mg490.00€100mg700.00€1mL*10mM (DMSO)150.00€E6801
CAS:E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.Formula:C17H18ClN5O2S2Purity:96.32% - 97.24%Color and Shape:SolidMolecular weight:423.94KSK68
CAS:KSK68 is a sigma-1 and histamine H3 receptor antagonist with analgesic activity, inhibits H3 receptors and can be used to study pain.Formula:C23H28N2O2Purity:99.11%Color and Shape:SolidMolecular weight:364.48CCG 203769
CAS:CCG 203769 (Thiadiazolidinone (TDZD) deriv. 6) is a selective inhibitor of RGS4 with an IC50 of 17 nM for the RGS4-Gαo protein-protein interaction.Formula:C8H14N2O2SPurity:99.88%Color and Shape:SolidMolecular weight:202.27Ref: TM-T10705
1mg88.00€5mg187.00€10mg264.00€25mg469.00€50mg657.00€100mg944.00€500mg1,882.00€1mL*10mM (DMSO)207.00€Abt-288
CAS:ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.Formula:C23H24N4OPurity:98.17% - 98.49%Color and Shape:SolidMolecular weight:372.46Irdabisant
CAS:Irdabisant (CEP-26401) is an H3R antagonist/inverse agonist, BBB permeable, with cognition-enhancing effects for schizophrenia/cognitive research.Formula:C18H23N3O2Purity:99.96%Color and Shape:SolidMolecular weight:313.39
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