
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,025 products)
- Adenosine Receptor(248 products)
- Adrenergic Receptor(2,999 products)
- Bombesin Receptor(35 products)
- Bradykinin Receptor(61 products)
- CXCR(154 products)
- CaSR(34 products)
- Cannabinoid Receptor(216 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(445 products)
- Endothelin Receptor(86 products)
- GNRH Receptor(84 products)
- GPCR19(33 products)
- GRK(33 products)
- GTPase(23 products)
- Glucagon Receptor(191 products)
- Hedgehog/Smoothened(49 products)
- Histamine Receptor(385 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(40 products)
- Opioid Receptor(325 products)
- PAFR(14 products)
- PKA(60 products)
- S1P Receptor(17 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5960 products of "GPCR/G-Protein"
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Tulobuterol-d9 HCl
CAS:Tulobuterol-d9 HCl is a deuterated compound of Tulobuterol HCl.Formula:C12H10D9Cl2NOColor and Shape:SolidMolecular weight:273.25Granisetron
CAS:Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.
Formula:C18H24N4OColor and Shape:SolidMolecular weight:312.41MRS-3777 hemioxalate
CAS:MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.
Formula:C17H19N5OC2H2O4Purity:97.10%Color and Shape:SolidMolecular weight:354.39Clothiapine
CAS:Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.Formula:C18H18ClN3SPurity:99.93%Color and Shape:SolidMolecular weight:343.873-Hydroxy agomelatine
CAS:3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.Formula:C15H17NO3Color and Shape:SolidMolecular weight:259.3SANT 2
CAS:SANT 2 is a Hedgehog (Hh) signaling pathway antagonist with potential anti-inflammatory and anti-cancer activities.Formula:C26H26ClN3O4Purity:99.23%Color and Shape:SolidMolecular weight:479.96Rebamipide-d4
CAS:Rebamipide D4 is deuterium labeled Rebamipide.Formula:C19H15ClN2O4Purity:98%Color and Shape:SolidMolecular weight:374.81SAR247799
CAS:SAR247799 is a selective and G-protein-biased S1P1 agonist that activates downstream G-protein signaling pathways more preferentially on endothelial cells.Formula:C21H16ClN3O5Color and Shape:SolidMolecular weight:425.82Sumanirole maleate
CAS:Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.Formula:C15H17N3O5Purity:98%Color and Shape:SolidMolecular weight:319.31Quetiapine-d8 Hemifumarate
CAS:Quetiapine-d8 Hemifumarate is a deuterated compound of Quetiapine Hemifumarate. Quetiapine Hemifumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Formula:C25H21D8N3O6SColor and Shape:SolidMolecular weight:507.63Neurotensin(8-13)
CAS:Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.Formula:C38H64N12O8Purity:99.95%Color and Shape:SolidMolecular weight:816.99Asenapine hydrochloride
CAS:Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.Formula:C17H17Cl2NOColor and Shape:SolidMolecular weight:322.235-HT2B antagonist-1
CAS:Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.Formula:C11H14BrN5Purity:99.965%Color and Shape:SolidMolecular weight:296.17GPR34 receptor antagonist 3
Compound 5e, a GPR34 receptor antagonist, exhibits selective inhibition of lysophosphatidylserine-induced ERK1/2 phosphorylation in a dose-dependent manner,Color and Shape:Odour SolidRU-SKI 43 Hydrochloride
CAS:RU-SKI 43 Hydrochloride is a selective Hedgehog acyltransferase inhibitor (IC50 850 nM) with reported anticancer activity in tumor biology studies.Formula:C22H31ClN2O2SPurity:98%Color and Shape:SolidMolecular weight:423.01Nefazodone
CAS:Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.Formula:C25H32ClN5O2Purity:99.85%Color and Shape:White To Off-White Crystalline PowderMolecular weight:470.01Ref: TM-T21451
2mg42.00€5mg60.00€10mg87.00€25mg177.00€50mg276.00€100mg422.00€200mg604.00€1mL*10mM (DMSO)95.00€Apraclonidine hydrochloride
CAS:Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.Formula:C9H11Cl3N4Purity:99.74%Color and Shape:SolidMolecular weight:281.57Piribedil D8
CAS:Piribedil D8 is the deuterium labeled Piribedil, which is an agent of antiparkinsonian.Formula:C16H18N4O2Purity:98%Color and Shape:SolidMolecular weight:306.39Hydroxyzine D8
CAS:Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.Formula:C21H27ClN2O2Purity:98%Color and Shape:SolidMolecular weight:382.95Trimethobenzamide
CAS:Trimethobenzamide (Ro 2-9578) is a D2 antagonist used to prevent nausea and vomiting.Formula:C21H28N2O5Color and Shape:SolidMolecular weight:388.46

