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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5960 products of "GPCR/G-Protein"

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  • Tulobuterol-d9 HCl

    CAS:
    Tulobuterol-d9 HCl is a deuterated compound of Tulobuterol HCl.
    Formula:C12H10D9Cl2NO
    Color and Shape:Solid
    Molecular weight:273.25

    Ref: TM-TMIH-0589

    1mg
    200.00€
    5mg
    497.00€
    10mg
    708.00€
  • Granisetron

    CAS:

    Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.

    Formula:C18H24N4O
    Color and Shape:Solid
    Molecular weight:312.41

    Ref: TM-T22340

    5mg
    922.00€
  • MRS-3777 hemioxalate

    CAS:

    MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.

    Formula:C17H19N5OC2H2O4
    Purity:97.10%
    Color and Shape:Solid
    Molecular weight:354.39

    Ref: TM-T12107

    1mg
    82.00€
    5mg
    To inquire
  • Clothiapine

    CAS:
    Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.
    Formula:C18H18ClN3S
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:343.87

    Ref: TM-T23900

    1mg
    93.00€
  • 3-Hydroxy agomelatine

    CAS:
    3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.
    Formula:C15H17NO3
    Color and Shape:Solid
    Molecular weight:259.3

    Ref: TM-T10114

    1mg
    60.00€
  • SANT 2

    CAS:
    SANT 2 is a Hedgehog (Hh) signaling pathway antagonist with potential anti-inflammatory and anti-cancer activities.
    Formula:C26H26ClN3O4
    Purity:99.23%
    Color and Shape:Solid
    Molecular weight:479.96

    Ref: TM-T23307

    2mg
    33.00€
    5mg
    44.00€
    1mL*10mM (DMSO)
    54.00€
  • Rebamipide-d4

    CAS:
    Rebamipide D4 is deuterium labeled Rebamipide.
    Formula:C19H15ClN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:374.81

    Ref: TM-T19547

    1mg
    490.00€
    5mg
    790.00€
    10mg
    1,063.00€
  • SAR247799

    CAS:
    SAR247799 is a selective and G-protein-biased S1P1 agonist that activates downstream G-protein signaling pathways more preferentially on endothelial cells.
    Formula:C21H16ClN3O5
    Color and Shape:Solid
    Molecular weight:425.82

    Ref: TM-T38716

    5mg
    1,214.00€
  • Sumanirole maleate

    CAS:
    Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.
    Formula:C15H17N3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:319.31

    Ref: TM-TQ0140

    2mg
    72.00€
  • Quetiapine-d8 Hemifumarate

    CAS:
    Quetiapine-d8 Hemifumarate is a deuterated compound of Quetiapine Hemifumarate. Quetiapine Hemifumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.
    Formula:C25H21D8N3O6S
    Color and Shape:Solid
    Molecular weight:507.63

    Ref: TM-TMID-0025

    50mg
    4,244.00€
  • Neurotensin(8-13)

    CAS:
    Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.
    Formula:C38H64N12O8
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:816.99

    Ref: TM-T7617

    1mg
    72.00€
  • Asenapine hydrochloride

    CAS:
    Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.
    Formula:C17H17Cl2NO
    Color and Shape:Solid
    Molecular weight:322.23

    Ref: TM-T22589

    1mg
    72.00€
  • 5-HT2B antagonist-1

    CAS:
    Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.
    Formula:C11H14BrN5
    Purity:99.965%
    Color and Shape:Solid
    Molecular weight:296.17

    Ref: TM-T9842

    10mg
    43.00€
    25mg
    71.00€
    50mg
    112.00€
    100mg
    180.00€
    500mg
    444.00€
    1mL*10mM (DMSO)
    33.00€
  • GPR34 receptor antagonist 3


    Compound 5e, a GPR34 receptor antagonist, exhibits selective inhibition of lysophosphatidylserine-induced ERK1/2 phosphorylation in a dose-dependent manner,
    Color and Shape:Odour Solid

    Ref: TM-T82264

    1mg
    120.00€
    5mg
    289.00€
    10mg
    465.00€
    25mg
    888.00€
    50mg
    1,468.00€
    100mg
    1,998.00€
  • RU-SKI 43 Hydrochloride

    CAS:
    RU-SKI 43 Hydrochloride is a selective Hedgehog acyltransferase inhibitor (IC50 850 nM) with reported anticancer activity in tumor biology studies.
    Formula:C22H31ClN2O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:423.01

    Ref: TM-T12797L

    2mg
    72.00€
  • Nefazodone

    CAS:
    Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.
    Formula:C25H32ClN5O2
    Purity:99.85%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:470.01

    Ref: TM-T21451

    2mg
    42.00€
    5mg
    60.00€
    10mg
    87.00€
    25mg
    177.00€
    50mg
    276.00€
    100mg
    422.00€
    200mg
    604.00€
    1mL*10mM (DMSO)
    95.00€
  • Apraclonidine hydrochloride

    CAS:
    Apraclonidine hydrochloride (ALO 2145) is an α2-adrenergic agonist and a weak α-1 adrenergic receptor agonist.
    Formula:C9H11Cl3N4
    Purity:99.74%
    Color and Shape:Solid
    Molecular weight:281.57

    Ref: TM-T21371

    10mg
    49.00€
    25mg
    84.00€
    50mg
    110.00€
    100mg
    165.00€
    200mg
    224.00€
    1mL*10mM (DMSO)
    34.00€
  • Piribedil D8

    CAS:
    Piribedil D8 is the deuterium labeled Piribedil, which is an agent of antiparkinsonian.
    Formula:C16H18N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:306.39

    Ref: TM-T12486

    1mg
    255.00€
    5mg
    To inquire
  • Hydroxyzine D8

    CAS:
    Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.
    Formula:C21H27ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:382.95

    Ref: TM-T11592

    1mg
    379.00€
    5mg
    1,314.00€
    10mg
    2,305.00€
  • Trimethobenzamide

    CAS:
    Trimethobenzamide (Ro 2-9578) is a D2 antagonist used to prevent nausea and vomiting.
    Formula:C21H28N2O5
    Color and Shape:Solid
    Molecular weight:388.46

    Ref: TM-T38802

    5mg
    873.00€