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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5838 products of "GPCR/G-Protein"

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  • Doxazosin D8

    CAS:
    Doxazosin D8, a deuterium-labeled version, is a selective AP1 adrenergic antagonist and a quinazoline derivative.
    Formula:C23H25N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:459.52
  • Propranolol-d7 hydrochloride

    CAS:
    Propranolol D7 HCl: deuterium-labeled, nonselective βAR antagonist.
    Formula:C16H22ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.85
  • Metipranolol hydrochloride

    CAS:
    Metipranolol hydrochloride is a non-selective β-adrenergic receptor blocking agent.
    Formula:C17H28ClNO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:345.86
  • Lysosphingomyelin (d18:1)

    CAS:
    <p>Sphingomyelins are phosphorylcholine, sphingosine, and fatty acid. Lysosphingomyelin, missing the fatty acid, activates diverse cellular pathways.</p>
    Formula:C23H49N2O5P
    Color and Shape:Solid
    Molecular weight:464.628
  • Thioridazine

    CAS:
    Thioridazine: an antipsychotic, anti-anxiety drug, blocks dopamine D2, PI3K-Akt-mTOR; halts angiogenesis, kills cancer cells, targets CSCs.
    Formula:C21H26N2S2
    Color and Shape:Solid
    Molecular weight:370.57
  • Bombesin

    CAS:
    Bombesin: 14-amino acid peptide from toad skin with two mammalian homologs, neuromedin B and gastrin-releasing peptide.
    Formula:C71H110N24O18S
    Color and Shape:While Lyophilized Powder
    Molecular weight:1619.85
  • Lanreotide

    CAS:
    Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.
    Formula:C54H69N11O10S2
    Color and Shape:Solid
    Molecular weight:1096.32
  • 5-HT2B antagonist-1

    CAS:
    Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.
    Formula:C11H14BrN5
    Purity:99.965%
    Color and Shape:Solid
    Molecular weight:296.17
  • β2AR/M-receptor agonist-2

    CAS:
    <p>β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).</p>
    Formula:C36H49ClN4O7S
    Color and Shape:Solid
    Molecular weight:717.31
  • Ceralifimod

    CAS:
    Ceralifimod (ONO-4641) is a potent agonist for sphingosine 1-phosphate receptors 1 and 5 (EC50s: 27.3, 334 pM for human S1P receptor 1 and 5).
    Formula:C27H33NO4
    Color and Shape:Solid
    Molecular weight:435.56
  • GLP-1 receptor agonist 2

    CAS:
    GLP-1 receptor agonist 2 is a glucagon-like peptide-1 receptor (GLP-1R) agonist.
    Formula:C30H31ClFN5O4
    Color and Shape:Solid
    Molecular weight:580.05
  • Cetirizine D8

    CAS:
    Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.
    Formula:C21H25ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:396.94
  • MK-761 TFA


    MK-761 TFA is an effective, orally active β2-adrenergic receptor blocker. It exhibits antihypertensive properties and positive inotropic effects, along with vasodilatory activity.
    Formula:C15H20F3N3O4
    Color and Shape:Solid
    Molecular weight:363.332
  • Mozavaptan hydrochloride

    CAS:
    Mozavaptan is a vasopressin receptor antagonist.
    Formula:C27H30ClN3O2
    Color and Shape:Solid
    Molecular weight:464
  • GB-88

    CAS:
    GB-88 is an selective , oral non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 μM.
    Formula:C32H42N4O4
    Color and Shape:Solid
    Molecular weight:546.7
  • Bradykinin (1-5)

    CAS:
    Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.
    Formula:C27H40N8O6
    Color and Shape:Solid
    Molecular weight:572.66
  • (S)-ZINC-3573

    CAS:
    (S)-ZINC 3573 is a negative control for (R)-ZINC 3573. (S)-ZINC 3573 displays no activity at MRGPRX2 at concentrations below 100 μM.
    Formula:C18H21N5
    Color and Shape:Solid
    Molecular weight:307.401
  • Endothelin-3 (Rat,Human) (TFA)


    <p>Endothelin-3 (Rat, Human) (TFA) is a 21-amino acid vasoactive peptide of endothelial origi, an agonist for the endothelin receptor type B (EDNRB).</p>
    Formula:C123H169F3N26O35S4·xC2HF3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2757.07 (free base)
  • 3-Hydroxy agomelatine D3

    CAS:
    3-Hydroxy agomelatine D3 is a deuterated metabolite of Agomelatine and a 5-HT2C antagonist (IC50: 3.2 μM, Ki: 1.8 μM).
    Formula:C15H17NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:262.32
  • Ozagrel Sodium

    CAS:
    Ozagrel Sodium is a thromboxane A2 synthase inhibitor. It is used to treat cerebrovascular diseases.
    Formula:C13H12N2NaO2
    Purity:98%
    Color and Shape:White Or Off-White Crystalline Powder
    Molecular weight:251.24