
GPCR/G-Protein
GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.
Subcategories of "GPCR/G-Protein"
- 5-HT Receptor(1,003 products)
- Adenosine Receptor(247 products)
- Adrenergic Receptor(3,010 products)
- Bombesin Receptor(33 products)
- Bradykinin Receptor(60 products)
- CXCR(153 products)
- CaSR(33 products)
- Cannabinoid Receptor(215 products)
- Cholecystokinin(1 products)
- Dopamine Receptor(435 products)
- Endothelin Receptor(83 products)
- GNRH Receptor(82 products)
- GPCR19(33 products)
- GRK(32 products)
- GTPase(22 products)
- Glucagon Receptor(190 products)
- Hedgehog/Smoothened(48 products)
- Histamine Receptor(381 products)
- LPA Receptor(21 products)
- Melatonin Receptor(26 products)
- OX Receptor(41 products)
- Opioid Receptor(321 products)
- PAFR(13 products)
- PKA(51 products)
- S1P Receptor(18 products)
- SGLT(31 products)
- Sigma receptor(46 products)
Show 19 more subcategories
Found 5838 products of "GPCR/G-Protein"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Cefaclor
CAS:Cefaclor (Panoral) is a cephalosporin antibiotic.Formula:C15H14ClN3O4SPurity:99.03% - 99.98%Color and Shape:SolidMolecular weight:367.81Antazoline phosphate
CAS:Antazoline phosphate: H1 histamine receptor antagonist with anticholinergic effects, eases allergies.Formula:C17H22N3O4PPurity:98%Color and Shape:CoaMolecular weight:363.35Ziprasidone D8
CAS:Ziprasidone D8, deuterium-labeled, is a potent antipsychotic, antagonizing 5-HT and dopamine receptors.Formula:C21H21ClN4OSPurity:98%Color and Shape:SolidMolecular weight:420.99Pimozide-d4
CAS:Pimozide D4 is a deuterium labeled Pimozide.Formula:C28H29F2N3OPurity:98%Color and Shape:SolidMolecular weight:465.57NBI-27914
CAS:<p>NBI-27914 is a selective and non-peptide CRFR1 (corticotropin-releasing factor receptor 1) antagonist with analgesic effects, capable of blocking CRF-induced anxiety.</p>Formula:C18H20Cl4N4Purity:99.47% - 99.64%Color and Shape:SolidMolecular weight:434.194,4-Diphenylbutylamine hydrochloride
CAS:4,4-Diphenylbutylamine shows affinity for the 5-HT2A and H1 receptors with Kis of 2589 and 1670 nM, respectively[1].Formula:C16H20ClNColor and Shape:SolidMolecular weight:261.79SKF-82958 hydrobromide
CAS:SKF-82958 hydrobromide is a D1/D5 receptor full agonist.Formula:C19H21BrClNO2Purity:98%Color and Shape:SolidMolecular weight:410.73Mozavaptan hydrochloride
CAS:Mozavaptan is a vasopressin receptor antagonist.Formula:C27H30ClN3O2Color and Shape:SolidMolecular weight:464ML 00253764
CAS:melanocortin MC4 receptor antagonistFormula:C18H18BrFN2OColor and Shape:SolidMolecular weight:377.25Thiethylperazine
CAS:Thiethylperazine (Tietilperazina) is a D2 receptor and H1 receptor antagonist, and an ABCC1 activator with antimicrobial and antiemetic activity.Formula:C22H29N3S2Purity:98.72%Color and Shape:SolidMolecular weight:399.62TFLLR-NH2(TFA)
CAS:TFLLR-NH2 (TFA) is a selective PAR1 agonist with an EC50 of 1.9 μM. EC50: 1.9 μM (PAR1)Formula:C33H54F3N9O8Purity:98%Color and Shape:SolidMolecular weight:761.83BMS-986020 sodium
CAS:BMS-986020 sodium (AM152 sodium) is a high-affinity LPA1 antagonist for investigating idiopathic pulmonary fibrosis.Formula:C29H25N2NaO5Purity:99.83%Color and Shape:SolidMolecular weight:504.51Nadolol-d9
CAS:<p>Nadolol D9 is the deuterium labeled Nadolol is a blocker of non-selective beta.</p>Formula:C17H27NO4Purity:98%Color and Shape:SolidMolecular weight:318.46(R)-Praziquantel-d11
CAS:(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.Formula:C19H24N2O2Purity:98%Color and Shape:SolidMolecular weight:323.47Emedastine Difumarate
CAS:Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.Formula:C25H34N4O9Color and Shape:SolidMolecular weight:534.56JNJ-10397049
CAS:OX2 receptor antagonistFormula:C19H20Br2N2O3Color and Shape:SolidMolecular weight:484.18Tiotidine
CAS:Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium).Formula:C10H16N8S2Purity:98%Color and Shape:SolidMolecular weight:312.42SB-674042
CAS:SB-674042 is a nonpeptide dual antagonist of the appetite peptides OX1 and OX2 receptors.SB-674042 is used in the treatment of depression.Formula:C24H21FN4O2SPurity:99.9%Color and Shape:SolidMolecular weight:448.51Clorprenaline
CAS:Clorprenaline is a β-adrenergic receptor agonist that activates adenylate cyclase, relaxation of bronchial smooth muscle cells. anti-inflammatory.Formula:C11H16ClNOPurity:98.9%Color and Shape:SolidMolecular weight:213.7GLP-1R modulator C16
CAS:GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.Formula:C21H26ClFN2O3Purity:99.6% - >99.99%Color and Shape:SolidMolecular weight:408.89
