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GPCR/G-Protein

GPCR/G-Protein

GPCR/G-Protein inhibitors are compounds that target G-protein coupled receptors (GPCRs) and associated G-proteins, which play critical roles in transmitting signals from the outside to the inside of cells. These inhibitors are essential for studying the signaling pathways mediated by GPCRs, which are involved in numerous physiological processes, including sensory perception, immune response, and neurotransmission. GPCR inhibitors are also important in drug development, as many therapeutic agents target these receptors. At CymitQuimica, we offer a wide range of high-quality GPCR/G-Protein inhibitors to support your research in pharmacology, cell biology, and related fields.

Subcategories of "GPCR/G-Protein"

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Found 5745 products of "GPCR/G-Protein"

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  • FAUC 346
    Targetmol
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    FAUC 346

    CAS:
    FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.
    Formula:C24H29N3O2S
    Purity:99.46%
    Color and Shape:Solid
    Molecular weight:423.57

    Ref: TM-T9081

  • Loxapine
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    Loxapine

    CAS:
    Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.
    Formula:C18H18ClN3O
    Purity:99.88%
    Color and Shape:Pale Yellowish Crystals From Petroleum Ether Solid
    Molecular weight:327.81

    Ref: TM-T21629

  • Mizagliflozin
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    Mizagliflozin

    CAS:
    Mizagliflozin is an orally active, selective SGLT1 inhibitor with a Ki value of 27 nM for human SGLT1.Cost-effective and quality-assured.
    Formula:C28H44N4O8
    Purity:98.66% - 99.67%
    Color and Shape:Solid
    Molecular weight:564.67

    Ref: TM-T16083

  • JD-5037
    Targetmol
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    JD-5037

    CAS:
    JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.
    Formula:C27H27Cl2N5O3S
    Purity:99.54% - 99.84%
    Color and Shape:Solid
    Molecular weight:572.51

    Ref: TM-T4453

  • RO 46-8443
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    RO 46-8443

    CAS:
    RO 46-8443: First non-peptide ETB receptor antagonist, >2000-fold ETB selectivity in binding and function.
    Formula:C31H35N3O8S
    Purity:98.77% - 99.77%
    Color and Shape:Solid
    Molecular weight:609.69

    Ref: TM-T3474

  • AM966
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    AM966

    CAS:
    <p>AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.</p>
    Formula:C27H23ClN2O5
    Purity:98.06% - 99.79%
    Color and Shape:Solid
    Molecular weight:490.93

    Ref: TM-T4278

  • AdipoRon
    Targetmol
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    AdipoRon

    CAS:
    AdipoRon (SC-396658) is an orally bioavailable adiponectin receptor agonist. It can combine with AdipoR1/2 (KD: 1.8/3.1 μM).
    Formula:C27H28N2O3
    Purity:97.90% - 99.86%
    Color and Shape:Solid
    Molecular weight:428.52

    Ref: TM-T2257

  • GSK189254A
    Targetmol
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    GSK189254A

    CAS:
    <p>GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).</p>
    Formula:C21H25N3O2
    Purity:98.71% - 99.858%
    Color and Shape:Solid
    Molecular weight:351.44

    Ref: TM-TQ0066

  • Ticagrelor metabolite M5
    Targetmol
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    Ticagrelor metabolite M5

    CAS:
    Ticagrelor metabolite M5 (T437700) is a metabolite of Ticagrelor, the first reversible oral antagonist of P2Y12 receptor.
    Formula:C14H22N6O4S
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:370.43

    Ref: TM-T21059

  • [Lys5,MeLeu9,Nle10]-NKA(4-10)
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    [Lys5,MeLeu9,Nle10]-NKA(4-10)

    CAS:
    Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
    Formula:C39H65N9O9
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:803.99

    Ref: TM-TP1883

  • Lurasidone hydrochloride
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    Lurasidone hydrochloride

    CAS:
    Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.
    Formula:C28H36N4O2S·HCl
    Purity:99.51%
    Color and Shape:Solid
    Molecular weight:529.14

    Ref: TM-T1735

  • Almotriptan
    Targetmol
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    Almotriptan

    CAS:
    Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.
    Formula:C17H25N3O2S
    Purity:99.85%
    Color and Shape:Light Yellow Or White Power
    Molecular weight:335.46

    Ref: TM-T21231

  • Lecirelin acetate(61012-19-9 free base)
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    Lecirelin acetate(61012-19-9 free base)

    Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts
    Formula:C61H88N16O14
    Purity:98.1%
    Color and Shape:Solid
    Molecular weight:1269.45

    Ref: TM-TP1434L

  • Neurokinin A
    Targetmol
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    Neurokinin A

    CAS:
    <p>Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.</p>
    Formula:C50H80N14O14S
    Purity:>99.99%
    Color and Shape:White To Off-White Lyophilized Solid
    Molecular weight:1133.32

    Ref: TM-TP1008

  • Nefazodone hydrochloride
    Targetmol
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    Nefazodone hydrochloride

    CAS:
    <p>Nefazodone hydrochloride (Serzone) is a serotoninergic modulating antidepressant that is used in therapy of depression, aggressive behavior and panic disorder.</p>
    Formula:C25H33Cl2N5O2
    Purity:99% - 99.86%
    Color and Shape:White Solid
    Molecular weight:506.47

    Ref: TM-T3275

  • BA 1 acetate(183241-31-8 free base)
    Targetmol
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    BA 1 acetate(183241-31-8 free base)

    <p>BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.</p>
    Formula:C59H80N14O13
    Purity:95.3%
    Color and Shape:Solid
    Molecular weight:1193.35

    Ref: TM-TP1913L1

  • Nelotanserin
    Targetmol
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    Nelotanserin

    CAS:
    Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).
    Formula:C18H15BrF2N4O2
    Purity:98.42% - 99.88%
    Color and Shape:Solid
    Molecular weight:437.24

    Ref: TM-T7350

  • Phenylbiguanide
    Targetmol
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    Phenylbiguanide

    CAS:
    <p>Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)</p>
    Formula:C8H11N5
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:177.21

    Ref: TM-T7135

  • VUF10460
    Targetmol
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    VUF10460

    CAS:
    VUF10460 is a non-imidazole histamine H4 receptor agonist.
    Formula:C15H19N5
    Purity:99.44% - 99.57%
    Color and Shape:Solid
    Molecular weight:269.34

    Ref: TM-T3963

  • Geissoschizine methyl ether
    Targetmol
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    Geissoschizine methyl ether

    CAS:
    Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.
    Formula:C22H26N2O3
    Purity:99.24% - 99.68%
    Color and Shape:Solid
    Molecular weight:366.45

    Ref: TM-TN1032